Compile Data Set for Download or QSAR
maximum 50k data
Found 155 with Last Name = 'zhang' and Initial = 'xk'
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM78433(2-[4-[3-[2-(trifluoromethyl)-10-phenothiazinyl]pro...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM82475(ACETOPHENAZINE | CAS_5714-00-1 | NSC_17676 | med.2...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50346422(10-(3-(4-hydroxypiperidin-1-yl)propyl)-10H-phenoth...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataIC50:  4nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataIC50:  5nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataIC50:  5nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151228(6-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50:  6nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  8nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50:  10nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151230(6-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50:  11nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151229(4-[Cyclopropylidene-(3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataIC50:  21nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataIC50:  29nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  31nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  60nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  73nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  85nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  117nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151231(4-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50376214(CHEMBL263660)
Affinity DataIC50:  250nMAssay Description:Inhibition of wild type androgen receptor expressed in CV1 cells assessed as dihydrotestosterone-stimulated transactivation by CAT reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151227(4-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50:  270nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50:  371nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11 [205-593](Homo sapiens (Human))
Burnham Institute For Medical Research

LigandPNGBDBM25127((2E)-3-{3-chloro-4-[3-(3,3-dimethylbut-1-yn-1-yl)-...)
Affinity DataIC50:  450nMpH: 6.0 T: 2°CAssay Description:The phosphatase-catalyzed hydrolysis of 6,8-difluoro-4-methylumbelliferyl phosphate was assayed in the presence of each test compound. The fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151226(4-[(3-Butyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular retinoic acid-binding protein 1(Gallus gallus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataIC50:  600nMAssay Description:Inhibition of binding to chick skin Cytoplasmic retinoic acid binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor RXR-beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  640nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular retinoic acid-binding protein 1(Gallus gallus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50:  700nMAssay Description:Inhibition of binding to chick skin Cytoplasmic retinoic acid binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50:  708nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular retinoic acid-binding protein 1(Gallus gallus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataIC50:  900nMAssay Description:Inhibition of binding to chick skin Cytoplasmic retinoic acid binding proteinMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50:  900nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCellular retinoic acid-binding protein 1(Gallus gallus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of binding to chick skin Cytoplasmic retinoic acid binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50407395(CHEMBL2111557)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031459((2Z,4E6E,8E)-3,7-dimethyl-9-(2,6,6-trimethylcycloh...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of murine Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Burnham Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50212333(5-[3'-(1-adamantyl)-2-chloro-4'-hydroxy-4-biphenyl...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of CD45 PTP by fluorescence spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
Burnham Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50212333(5-[3'-(1-adamantyl)-2-chloro-4'-hydroxy-4-biphenyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of SHP2 PTP by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of binding to murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031457((2Z,5E)-3-{(E)-3-[3-Ethyl-2-isopropyl-cyclohex-2-e...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of binding to murine Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50430582(CHEMBL2337792)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H]-9-cis-RA from human GST-tagged N-terminal truncated RXRalpha after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11 [205-593](Homo sapiens (Human))
Burnham Institute For Medical Research

LigandPNGBDBM25124((2E)-3-{4-[3-(adamantan-1-yl)-4-aminophenyl]-3-chl...)
Affinity DataIC50:  1.83E+3nMpH: 6.0 T: 2°CAssay Description:The phosphatase-catalyzed hydrolysis of 6,8-difluoro-4-methylumbelliferyl phosphate was assayed in the presence of each test compound. The fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50110164((Z)-2-(3-(4-(methylthio)benzylidene)-6-fluoro-2-me...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11 [205-593](Homo sapiens (Human))
Burnham Institute For Medical Research

LigandPNGBDBM25122((2E)-3-{4-[3-(adamantan-1-yl)-4-hydroxyphenyl]-3-c...)
Affinity DataIC50:  2.10E+3nMpH: 6.0 T: 2°CAssay Description:The phosphatase-catalyzed hydrolysis of 6,8-difluoro-4-methylumbelliferyl phosphate was assayed in the presence of each test compound. The fluorescen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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