Affinity DataKi: 0.150nMAssay Description:Inhibition constant determined against Acetylcholinesterase (AChE) receptor.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+4nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+5nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+5nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+5nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+5nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+6nMAssay Description:Inhibition of choline acetyltransferase isolated from squid head gangliaMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+6nMAssay Description:Binding affinity of the compound towards AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 6.40E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 6.40E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 7.20E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 7.60E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataKi: 8.70E+6nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis of acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+7nMAssay Description:Enzyme inhibition dissociation constant for choline acetyl transferase (ChAcT) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(competitive)More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(com)More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+7nMAssay Description:Enzyme inhibition dissociation constant for choline acetyl transferase (ChAcT) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(com)More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+7nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(com)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+8nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(com)More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+8nMAssay Description:Compound was evaluated for reversible inhibition of hydrolysis acetylcholine by acetylcholinesterase and represented as KI(noncompetitive)More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:In vitro inhibitory activity of the compound against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Compound was tested for the competitive inhibition of acetylcholinesterase (AChE)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Compound was tested for the competitive inhibition of acetylcholinesterase (AChE)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Compound was tested for the competitive inhibition of acetylcholinesterase (AChE)More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against chick optic lobe choline acetyltransferase (ChAT)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against rat choline acetyltransferase (ChAT)More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against chick optic lobe choline acetyltransferase (ChAT)More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against chick optic lobe choline acetyltransferase (ChAT)More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against chick choline acetyltransferase (ChAT)More data for this Ligand-Target Pair
Affinity DataIC50: 1.85E+5nMAssay Description:Compound was tested for the competitive inhibition of acetylcholinesterase (AChE)More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+5nMAssay Description:Compound was tested for the competitive inhibition of acetylcholinesterase (AChE)More data for this Ligand-Target Pair