Compile Data Set for Download or QSAR
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Found 11 Enz. Inhib. hit(s) with Target = 'G1/S-specific cyclin-E1'
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50246253(4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-(me...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Cyclin E/CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50:  220nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50:  230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50:  330nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50:  410nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50:  430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50319619(4-(2,4-Dimethylthiazol-5-yl)-N-(4-morpholinophenyl...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed