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Found 5 Enz. Inhib. hit(s) with Target = 'Dimer of Prostaglandin G/H synthase 2'
TargetDimer of Prostaglandin G/H synthase 2(Homo sapiens (Human))
University Of Michigan Medical School

LigandPNGBDBM209868(3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17...)
Affinity DataKd:  130nMpH: 8.0Assay Description:POX reactions were conducted in 2 ml of filtered and degassed 50 mM Tris-HCl, pH 8.0, containing 50 mM NaCl, 0.1 mM H2O2, 4.5 mM guaiacol, and the in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Prostaglandin G/H synthase 2 [Y385F](Homo sapiens (Human))
University Of Michigan Medical School

LigandPNGBDBM209868(3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17...)
Affinity DataKd:  1.60E+3nMpH: 8.0Assay Description:POX reactions were conducted in 2 ml of filtered and degassed 50 mM Tris-HCl, pH 8.0, containing 50 mM NaCl, 0.1 mM H2O2, 4.5 mM guaiacol, and the in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Prostaglandin G/H synthase 2 [S530A](Homo sapiens (Human))
University Of Michigan Medical School

LigandPNGBDBM209868(3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17...)
Affinity DataKd:  190nMpH: 8.0Assay Description:POX reactions were conducted in 2 ml of filtered and degassed 50 mM Tris-HCl, pH 8.0, containing 50 mM NaCl, 0.1 mM H2O2, 4.5 mM guaiacol, and the in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Prostaglandin G/H synthase 2 [R120A](Homo sapiens (Human))
University Of Michigan Medical School

LigandPNGBDBM209868(3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17...)
Affinity DataKd:  750nMpH: 8.0Assay Description:POX reactions were conducted in 2 ml of filtered and degassed 50 mM Tris-HCl, pH 8.0, containing 50 mM NaCl, 0.1 mM H2O2, 4.5 mM guaiacol, and the in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Prostaglandin G/H synthase 2 [R120Q](Homo sapiens (Human))
University Of Michigan Medical School

LigandPNGBDBM209868(3-[18-(2-carboxyethyl)-8,13-bis(ethenyl)-3,7,12,17...)
Affinity DataKd:  220nMpH: 8.0Assay Description:POX reactions were conducted in 2 ml of filtered and degassed 50 mM Tris-HCl, pH 8.0, containing 50 mM NaCl, 0.1 mM H2O2, 4.5 mM guaiacol, and the in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed