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Found 42 Enz. Inhib. hit(s) with Target = 'Histidine kinase'
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453878(CHEMBL371380)
Affinity DataKi:  3.80E+3nMAssay Description:Competitive inhibition of Caulobacter vibrioides full length wild type cell cycle histidine kinase CckA deltaTM Escherichia coli BL21-AI in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM15364(4-chloro-6-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453878(CHEMBL371380)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50409992(CHEMBL364882)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453882(CHEMBL4218027)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453881(CCT018159 | CHEBI:41656 | CHEMBL399530)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50409996(CHEMBL191228)
Affinity DataIC50:  3.23E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453884(CHEMBL4217100)
Affinity DataIC50:  3.27E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453883(CHEMBL4204469)
Affinity DataIC50:  3.36E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM15365(3-(2,4-Dihydroxyphenyl)-4-(4-methoxyphenyl)-5-meth...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453887(CHEMBL1551662)
Affinity DataIC50:  5.69E+4nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Streptococcus pneumoniae PCS8203)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453885(CHEMBL4209595)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of Streptococcus pneumoniae VicK preincubated for 30 mins followed by [gamma-33P]ATP addition after 30 mins by SDS-PAGE methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Caulobacter vibrioides)
Williams College

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataIC50:  1.84E+5nMAssay Description:Inhibition of recombinant Caulobacter vibrioides cell cycle histidine kinase CckA deltaTM mutant DHp domain (70 to 691 residues) expressed in Escheri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase(Streptococcus pneumoniae PCS8203)
Williams College

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50:  2.16E+5nMAssay Description:Inhibition of Streptococcus pneumoniae VicK preincubated for 30 mins followed by [gamma-33P]ATP addition after 30 mins by SDS-PAGE methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274506(3-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4843...)
Affinity DataEC50:  1.30E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274507(4-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4843...)
Affinity DataEC50:  1.65E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274548(2-chloro-N-(2-methoxyphenyl)-9H-purin-6-amine | CH...)
Affinity DataEC50:  3.30E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274549(2-Chloro-6-(3-methoxyanilino)purine | CHEMBL484383)
Affinity DataEC50:  2.10E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274550(2-chloro-N-(4-methoxyphenyl)-9H-purin-6-amine | CH...)
Affinity DataEC50:  3.31E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM59843((3-methoxyphenyl)-(7H-purin-6-yl)amine | CHEMBL484...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274552(2-Fluoro-6-(3-methoxyanilino)purine | CHEMBL483378)
Affinity DataEC50:  1.90E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50267036((2E)-2-methyl-4-(9H-purin-6-ylamino)but-2-en-1-ol ...)
Affinity DataEC50:  700nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274591(CHEMBL505661 | Thidiazuron)
Affinity DataEC50:  950nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274501(2-chloro-N-(3-chlorophenyl)-9H-purin-6-amine | CHE...)
Affinity DataEC50:  7.50E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274502(2-Chloro-6-(4-chloroanilino)purine | CHEMBL448763)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274505(2-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4855...)
Affinity DataEC50:  1.90E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274504(2-chloro-N-(4-fluorophenyl)-9H-purin-6-amine | CHE...)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274503(2-chloro-N-(3-fluorophenyl)-9H-purin-6-amine | CHE...)
Affinity DataEC50:  6.00E+3nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274502(2-Chloro-6-(4-chloroanilino)purine | CHEMBL448763)
Affinity DataEC50:  1.51E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274501(2-chloro-N-(3-chlorophenyl)-9H-purin-6-amine | CHE...)
Affinity DataEC50:  1.07E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274469(2-Chloro-6-anilinopurine | CHEMBL519852)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 3(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50240929(6-anilinopurine | CHEMBL359730 | Phenyl-(9H-purin-...)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Arabidopsis thaliana AHK3 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274591(CHEMBL505661 | Thidiazuron)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50267036((2E)-2-methyl-4-(9H-purin-6-ylamino)but-2-en-1-ol ...)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274552(2-Fluoro-6-(3-methoxyanilino)purine | CHEMBL483378)
Affinity DataEC50:  1.90E+4nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM59843((3-methoxyphenyl)-(7H-purin-6-yl)amine | CHEMBL484...)
Affinity DataEC50:  3.10E+4nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274549(2-Chloro-6-(3-methoxyanilino)purine | CHEMBL484383)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274507(4-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4843...)
Affinity DataEC50:  4.60E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274506(3-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4843...)
Affinity DataEC50:  3.75E+3nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274503(2-chloro-N-(3-fluorophenyl)-9H-purin-6-amine | CHE...)
Affinity DataEC50:  2.48E+4nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine kinase 4(Arabidopsis thaliana)
Ieb As Cr & Palacký

Curated by ChEMBL
LigandPNGBDBM50274505(2-(2-chloro-9H-purin-6-ylamino)phenol | CHEMBL4855...)
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Arabidopsis thaliana AHK4/CRE1 receptor expressed in Escherichia coli KMI001 by beta-galactosidase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed