TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 4.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 4.90E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Inhibition of Rattus norvegicus Wistar (rat) rat Gamma-glutamyltranspeptidase using L-gamma-glutamyl-p-nitroanilide as substrate incubated for 15 min...More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+4nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 6.10E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 8.70E+4nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 8.80E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 1.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 1.73E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.02E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.20E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+5nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.54E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.60E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 3.43E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 3.56E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 5.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+5nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 5.89E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.15E+6nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+6nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+6nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
Affinity DataKi: 2.69E+7nMpH: 8.0Assay Description:Compound tested for the inhibition of Gamma-glutamyltranspeptidase in rat kidney at pH 8.0 at 37 degree C (Competitive inhibition)More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of gamma-glutamyltranspeptidase (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
TargetGlutathione hydrolase 1 proenzyme(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataIC50: 2.63E+4nMAssay Description:Inhibition of recombinant GGT1 (unknown origin) using GGPP as substrate preincubated for 5 mins followed by protein addition measured over 20 mins by...More data for this Ligand-Target Pair