Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with Target = 'Sensor protein kinase WalK'
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50368125(ADENOSINE DIPHOSPHATE | ADP)
Affinity DataIC50:  7.19E+3nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453880(CHEMBL3343945)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant Staphylococcus epidermidis ATCC 35984 N-terminal GB1-tagged YycG expressed in Escherichia coli BL21 (DE3) preincubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453886(CHEMBL4215525)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant Staphylococcus epidermidis ATCC 35984 N-terminal GB1-tagged YycG expressed in Escherichia coli BL21 (DE3) preincubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM15759(4,7 Diazaindole 22 | 4-[7-(4-fluorophenyl)-5H-pyrr...)
Affinity DataIC50:  9.33E+4nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM27434(11,13-dimethyl-8-thia-3,5,10-triazatricyclo[7.4.0....)
Affinity DataIC50:  9.55E+4nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus aureus subsp. aureus CN1)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453879(CHEMBL4202687)
Affinity DataIC50:  2.12E+5nMAssay Description:Inhibition of Staphylococcus aureus DHp-catalytic domain PhoR autophosphorylation expressed in Escherichia coli RIL in presence of gamma-32P-ATP by S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM18134(({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataIC50:  2.28E+5nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM153747(ROCHE screening, 65)
Affinity DataIC50:  8.83E+8nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed