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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1 [852-1142]'
TargetTyrosine-protein kinase JAK1 [852-1142](Homo sapiens (Human))
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US Patent
LigandPNGBDBM185700(US10875847, Compound Oclacitinib | US9161939, 1a |...)
Affinity DataIC50:  9.53nMpH: 7.4Assay Description:Methods: A peptide mobility shift assay was used to quantify the phosphorylation of the JAKtide (JAK-2 and JAK-3) or the IRS-1 peptide (JAK-1 and Tyk...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1 [852-1142](Homo sapiens (Human))
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US Patent
LigandPNGBDBM185701(US9161939, 2 | US9271981, 2)
Affinity DataIC50:  45nMpH: 7.4Assay Description:Methods: A peptide mobility shift assay was used to quantify the phosphorylation of the JAKtide (JAK-2 and JAK-3) or the IRS-1 peptide (JAK-1 and Tyk...More data for this Ligand-Target Pair
In DepthDetails US Patent