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Found 7 Enz. Inhib. hit(s) with Target = 'Cadherin-1 [819-873]/Catenin beta-1 [138-686]'
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  1.17E+4nM ΔG°:  -28.2kJ/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM213748(US9284299, PKF115-584 | US9738628, Compound PKF115...)
Affinity DataKi:  1.30E+4nM ΔG°:  -27.9kJ/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  1.33E+4nM ΔG°:  -27.8kJ/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  1.44E+4nM ΔG°:  -27.6kJ/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  1.99E+4nM ΔG°:  -26.8kJ/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM213761(US9284299, 12 | US9738628, Compound 12)
Affinity DataKi:  1.04E+5nM ΔG°:  -22.7kJ/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCadherin-1 [819-873]/Catenin beta-1 [138-686](Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM213761(US9284299, 12 | US9738628, Compound 12)
Affinity DataKi:  1.05E+5nM ΔG°:  -22.7kJ/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent