TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 328nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Dixon and ...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Cheng-Prus...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Dixon and ...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.59E+3nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.07E+4nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Competitive inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 15 mins by Dixo...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.57E+4nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of rat CD39 expressed in CHO cells using ATP as substrate incubated for 10 mins by UV absorbance methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of rat NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of human NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+4nMAssay Description:Tested for inhibition of Nucleoside Triphosphate Diphosphohydrolase (NTPDase) from bovine spleen.More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 4.60E+4nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 4.91E+4nMAssay Description:Inhibition of rat NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 5.52E+4nMAssay Description:Inhibition of human NTPDase 1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: >1.50E+5nMAssay Description:Inhibition of rat NTPdase1 by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.54E+5nMAssay Description:Inhibition of human NTPDase 1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.61E+5nMAssay Description:Inhibition of human NTPDase 1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 1.82E+5nMAssay Description:Inhibition of human NTPDase 1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 3.00E+5nMAssay Description:Inhibition of rat NTPDase 1More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 3.00E+5nMAssay Description:Inhibition of rat recombinant NTPDase1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 7.86E+5nMAssay Description:Inhibition of human NTPDase 1 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of CD39 (unknown origin)More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Mus musculus)
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of mouse CD39More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Mus musculus)
Ningxia Medical University
Curated by ChEMBL
Ningxia Medical University
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of mouse CD39More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human CD39 expressed in green monkey Cos-7 cells using ATP as substrate preincubated for 3 mins followed by substrate addition by malac...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Malachite ...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 6.21E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 9.02E+3nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CD39 expressed in CHO cells incubated for 4 hrs before addition of AMP and further incubated for 60 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human CD39 expressed in green monkey Cos-7 cells using ATP as substrate preincubated for 3 mins followed by substrate addition by malac...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of human NTPDase1 expressed in African green monkey COS7 cell membrane fraction using ATP as substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human NTPDase1 expressed in CHO cells using ADP as substrate incubated for 10 mins by capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CD39 expressed in CHO cells using ATP as substrate preincubated for 1 hr followed by substrate addition and measured after 50 min...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Rattus norvegicus)
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of rat NTPDase1 expressed in CHO cells using ATP as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
TargetEctonucleoside triphosphate diphosphohydrolase 1(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human CD39 using ATP as substrate preincubated for 3 mins followed by substrate addition and measured after 10 to 15 mins by Malachite ...More data for this Ligand-Target Pair