Compile Data Set for Download or QSAR
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Found 768 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform alpha'
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)
Affinity DataKi:  501nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKi:  650nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50463484(CHEMBL4248525)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50463483(CHEMBL4245242)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50224883(7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,1...)
Affinity DataKi: >6.92E+3nMAssay Description:Inhibition of CK1alpha1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataKi:  3.83E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataKi:  3.83E+4nM ΔG°:  -25.6kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM92607(H-88)
Affinity DataKi:  6.07E+4nM ΔG°:  -24.5kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50375645(CHEMBL219301 | US11542290, Compound A-3)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50331612(CHEMBL1290072 | N-(4-methoxybenzyl)benzofuro[2,3-b...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human CK1-alpha1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50395892(CHEMBL2163772)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Ck1alpha1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625246(2-(4-fluorophenyl)-N-[4-(4-oxo-3-phenyl-4,5,6,7-te...)
Affinity DataIC50:  0.660nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625275(2-(4-fluorophenyl)-N-[4-(5-methyl-4-oxo-3-phenyl-4...)
Affinity DataIC50:  0.710nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629242((−)-N-{4-[5-fluoro-6-methyl-3-(pyridin-2-yl)...)
Affinity DataIC50:  0.739nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625179(2-(4-fluorophenyl)-N-[4-(5-methyl-4-oxo-3-phenyl-4...)
Affinity DataIC50:  0.860nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625180(4,4-difluoro-2-(4-fluorophenyl)-N-[4-(5-methyl-4-o...)
Affinity DataIC50:  0.940nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629261(N-{4-[5-chloro-3-(pyridin-2-yl)-1H-pyrrolo[3,2-b]p...)
Affinity DataIC50:  0.941nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629245((+)-2-(4-fluorophenyl)-N-{4-[3-(pyridin-2-yl)-1H-p...)
Affinity DataIC50:  0.949nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625331(N-[4-(5-cyclopropyl-4-oxo-3-phenyl-4,5-dihydro-1H-...)
Affinity DataIC50:  0.960nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629241((+)-2-(4-fluorophenyl)-N-{4-[5-fluoro-3-(pyridin-2...)
Affinity DataIC50:  1nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625274((+)-2-(4-fluorophenyl)-N-{4-[3-(4-fluorophenyl)-5-...)
Affinity DataIC50:  1nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629257(2-(4-fluorophenyl)-N-{4-[7-(pyridin-2-yl)-5H-pyrro...)
Affinity DataIC50:  1.02nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629252(2-(4-fluorophenyl)-N-[4-(3-phenyl-1H-pyrrolo[3,2-b...)
Affinity DataIC50:  1.04nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629243(2-(4-fluorophenyl)-N-{4-[3-(pyridin-2-yl)-1H-pyrro...)
Affinity DataIC50:  1.06nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625176(4,4-difluoro-2-(4-fluorophenyl)-N-[4-(5-methyl-4-o...)
Affinity DataIC50:  1.10nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625216(N-[4-(7,7-dimethyl-4-oxo-3-phenyl-4,5,6,7-tetrahyd...)
Affinity DataIC50:  1.20nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629280(US20230339939, Example 42)
Affinity DataIC50:  1.23nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625266(2-(4-fluorophenyl)-N-{4-[3-(4-fluorophenyl)-6,6-di...)
Affinity DataIC50:  1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629258(2-(4-fluorophenyl)-N-[4-(7-phenyl-5H-pyrrolo[3,2-c...)
Affinity DataIC50:  1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625175(2-(4-fluorophenyl)-N-[4-(5-methyl-4-oxo-3-phenyl-4...)
Affinity DataIC50:  1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625325((Rac)-N-[4-(5-methyl-4-oxo-3-phenyl-4,5,6,7-tetrah...)
Affinity DataIC50:  1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625254(N-[4-(6,6-dimethyl-4-oxo-3-phenyl-4,5,6,7-tetrahyd...)
Affinity DataIC50:  1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629288(N-{4-[5-fluoro-3-(5-fluoropyridin-2-yl)-1H-pyrrolo...)
Affinity DataIC50:  1.42nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM636432(N-{4-[3-anilino-7-ethyl-4-oxo-4,5,6,7-tetrahydro-1...)
Affinity DataIC50:  1.5nMAssay Description:CSNK1A1-inhibitory activity of compounds of the present invention in presence of 1 μM adenosine-tri-phosphate (ATP) was quantified employing the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629265(N-{4-[5-fluoro-6-methyl-3-(pyridin-2-yl)-1H-pyrrol...)
Affinity DataIC50:  1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629260(N-{4-[7-chloro-3-(pyridin-2-yl)-1H-pyrrolo[3,2-b]p...)
Affinity DataIC50:  1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625248(2-(4-fluorophenyl)-N-[4-(4-oxo-3-phenyl-4,5,6,7-te...)
Affinity DataIC50:  1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625312(4-[2-({4-[3-(4-fluorophenyl)-5-methyl-4-oxo-4,5,6,...)
Affinity DataIC50:  1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625228((+)-2-(4-fluorophenyl)-N-[4-(5′-methyl-4R...)
Affinity DataIC50:  1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629259(2-(4-fluorophenyl)-N-{4-[7-(pyridin-2-yl)-5H-pyrro...)
Affinity DataIC50:  1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629251((+)-2-(4-fluorophenyl)-N-[4-(3-phenyl-1H-pyrrolo[3...)
Affinity DataIC50:  1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629239(2-(4-fluorophenyl)-N-{4-[5-fluoro-3-(pyridin-2-yl)...)
Affinity DataIC50:  1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629247(2-(4-fluorophenyl)-N-{4-[6-fluoro-3-(pyridin-2-yl)...)
Affinity DataIC50:  1.68nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629286((+)-N-{4-[5-fluoro-3-(5-fluoropyridin-2-yl)-1H-pyr...)
Affinity DataIC50:  1.69nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629268(US20230339939, Example 30)
Affinity DataIC50:  1.69nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625243(N-{4-[3-(2,4-difluorophenyl)-5-methyl-4-oxo-4,5,6,...)
Affinity DataIC50:  1.70nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625176(4,4-difluoro-2-(4-fluorophenyl)-N-[4-(5-methyl-4-o...)
Affinity DataIC50:  1.70nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM629244(2-(4-fluorophenyl)-N-{4-[3-(pyridin-2-yl)-1H-pyrro...)
Affinity DataIC50:  1.73nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM625220(N-[4-(7,7-dimethyl-4-oxo-3-phenyl-4,5,6,7-tetrahyd...)
Affinity DataIC50:  1.80nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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