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Found 115 Enz. Inhib. hit(s) with Target = 'Follicle-stimulating hormone receptor'
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410306(CHEMBL436481)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410307(CHEMBL360981)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410303(CHEMBL361847)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410309(CHEMBL365545)
Affinity DataIC50:  9nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of maximum response evoked by cAMP on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410304(CHEMBL195469)
Affinity DataIC50:  25nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410302(CHEMBL361167)
Affinity DataIC50:  27nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410308(CHEMBL192868)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410298(CHEMBL178980)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335479((R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynylo...)
Affinity DataIC50:  39nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410294(CHEMBL195347)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410292(CHEMBL192334)
Affinity DataIC50:  54nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410300(CHEMBL179505)
Affinity DataIC50:  76nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410297(CHEMBL372649)
Affinity DataIC50:  166nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410299(CHEMBL426824)
Affinity DataIC50:  170nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410296(CHEMBL363164)
Affinity DataIC50:  240nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335480((R)-N-(1-acetyl-4-(4-((1-(2-(2-(2-azidoethoxy)etho...)
Affinity DataIC50:  324nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Rattus norvegicus)
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  540nMAssay Description:In vitro inhibition against maximum response evoked by cAMP in rat GFSHR-17 granulosa cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410301(CHEMBL372506)
Affinity DataIC50:  580nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335470((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataIC50:  920nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410291(CHEMBL194996)
Affinity DataIC50:  930nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335472((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataIC50:  1.02E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335471((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataIC50:  1.66E+3nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410293(CHEMBL195321)
Affinity DataIC50:  1.88E+3nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410295(CHEMBL371595)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50:  8.03E+3nMAssay Description:Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50505783(CHEMBL4458424)
Affinity DataIC50: >1.60E+4nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50: >1.60E+4nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50505793(CHEMBL4593222)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50505789(CHEMBL4471621)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50505788(CHEMBL4449797)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  48nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142676((3S,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity of the compound was determined in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142675(1-Butyl-1-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-di...)
Affinity DataEC50:  9.5nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142662(1-Butyl-1-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-di...)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142672(Butyl-[4'-((2S,5S)-1,5-dimethyl-4-octyl-3,6-dioxo-...)
Affinity DataEC50:  2.70nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142657((3S,6S)-1-Heptyl-4,6-dimethyl-3-(3',4',5'-trimetho...)
Affinity DataEC50:  32nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142661(CHEMBL47059 | N-Butyl-N-[4'-((2S,5S)-1,5-dimethyl-...)
Affinity DataEC50:  35nMAssay Description:Agonistic activity of the compound was determined in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142656(Butyl-[4'-((2S,5S)-4-hexyl-1,5-dimethyl-3,6-dioxo-...)
Affinity DataEC50:  8.90nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142655(2-{4-[4'-(1-Butyl-3-methyl-ureidomethyl)-biphenyl-...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonistic activity against Follicle stimulating hormone receptor expressed in chinese hamster ovary cells(CHO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142651(CHEMBL300022 | N-Hexyl-2-[(S)-4-methyl-2,5-dioxo-3...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonistic activity against Follicle stimulating hormone receptor expressed in chinese hamster ovary cells(CHO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142654(2-{(S)-3-[3'-(1-Butyl-3-methyl-ureidomethyl)-biphe...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonistic activity against Follicle stimulating hormone receptor expressed in chinese hamster ovary cells(CHO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142652(CHEMBL47120 | {2'-[(Acetyl-butyl-amino)-methyl]-bi...)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonistic activity against Follicle stimulating hormone receptor expressed in chinese hamster ovary cells(CHO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142653(3'-(1-Butyl-3-methyl-ureidomethyl)-biphenyl-4-carb...)
Affinity DataEC50:  260nMAssay Description:Agonistic activity against Follicle stimulating hormone receptor expressed in chinese hamster ovary cells(CHO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142673((3R,6S)-1,3-Dimethyl-4-octyl-6-(3',4',5'-trimethox...)
Affinity DataEC50:  120nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142651(CHEMBL300022 | N-Hexyl-2-[(S)-4-methyl-2,5-dioxo-3...)
Affinity DataEC50:  3nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142678(CHEMBL44663 | N-Butyl-N-[4'-((2S,5S)-4-hexyl-1,5-d...)
Affinity DataEC50:  150nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50142665((3S,6S)-1-Hexyl-4,6-dimethyl-3-(3',4',5'-trimethox...)
Affinity DataEC50:  100nMAssay Description:Agonistic activity against human follicle stimulating hormone receptor in CHO-hFSHR-luciferase assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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