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Found 1110 Enz. Inhib. hit(s) with Target = 'Urease'
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50493380(CHEMBL2425469)
Affinity DataKi:  14nMAssay Description:Mixed-type competitive inhibition of Helicobacter pylori ATCC 43504 urease using urea as substrate by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223161(1-cyclohexyl-1-isopropyl-3,3-dimethylselenourea | ...)
Affinity DataKi:  25nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50462868(CHEMBL4251246)
Affinity DataKi:  43nMAssay Description:Mixed-type inhibition of Helicobacter pylori ATCC 43504 urease assessed as enzyme-inhibitor complex using urea as substrate preincubated for 1.5 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50493373(CHEMBL2425478)
Affinity DataKi:  45nMAssay Description:Mixed-type competitive inhibition of Helicobacter pylori ATCC 43504 urease using urea as substrate by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50462868(CHEMBL4251246)
Affinity DataKi:  54nMAssay Description:Mixed-type inhibition of Helicobacter pylori ATCC 43504 urease assessed as enzyme-substrate-inhibitor complex using urea as substrate preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50449762(CHEMBL4172924)
Affinity DataKi:  60.2nMAssay Description:Mixed type non-competitive inhibition of urease in Helicobacter pylori ATCC 43504 assessed as enzyme-substrate-inhibitor complex constant preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50602006(CHEMBL5209436)
Affinity DataKi:  65nMAssay Description:Mixed type inhibition of Helicobacter pyroli urease assessed as dissociation constant for EI complex by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356190(CHEMBL193474)
Affinity DataKi:  90nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223158((S)-1,1-dimethyl-3-(1-(naphthalen-1-yl)ethyl)selen...)
Affinity DataKi:  94nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356195(CHEMBL241902)
Affinity DataKi:  122nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223159(3-dodecyl-1,1-dimethylthiourea | CHEMBL251521)
Affinity DataKi:  124nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM53627(1-[[(E)-(5-oxidanyl-6-oxidanylidene-cyclohexa-2,4-...)
Affinity DataKi:  127nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356192(CHEMBL241894)
Affinity DataKi:  127nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356201(CHEMBL1910224)
Affinity DataKi:  134nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223157(3-(4-bromobenzyl)-1,1-dimethylselenourea | CHEMBL3...)
Affinity DataKi:  135nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50449754(CHEMBL4167553)
Affinity DataKi:  152nMAssay Description:Mixed type non-competitive inhibition of urease in Helicobacter pylori ATCC 43504 assessed as enzyme-substrate-inhibitor complex constant preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356197(CHEMBL1910221)
Affinity DataKi:  152nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit alpha/beta/gamma(Bacillus pasteurii)
Wroclaw University Of Technology

LigandPNGBDBM24969([(2-{[(benzyloxy)carbonyl]amino}acetamido)methyl](...)
Affinity DataKi:  170nM ΔG°:  -39.3kJ/mole IC50:  1.80E+3nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356186(CHEMBL239452)
Affinity DataKi:  170nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50534783(CHEMBL4575318)
Affinity DataKi:  184nMAssay Description:Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 after 120 mins by Berthelot colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356198(CHEMBL1910222)
Affinity DataKi:  191nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488912(CHEMBL2298033)
Affinity DataKi:  200nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  226nMAssay Description:Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 after 120 mins by Berthelot colorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50223160(3-(4-bromophenyl)-1,1-dimethylthiourea | CHEMBL249...)
Affinity DataKi:  255nMAssay Description:Inhibition of jack bean ureaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50449763(CHEMBL4176964)
Affinity DataKi:  314nMAssay Description:Mixed type non-competitive inhibition of urease in Helicobacter pylori ATCC 43504 assessed as enzyme-substrate-inhibitor complex constant preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50534504(CHEMBL4590676)
Affinity DataKi:  372nMAssay Description:Inhibition of Helicobacter pylori urease using urea as substrate assessed as inhibition constant for enzyme-urea-inhibitor complex by non-linear fitt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356199(CHEMBL242113)
Affinity DataKi:  391nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356188(CHEMBL391982)
Affinity DataKi:  398nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50534504(CHEMBL4590676)
Affinity DataKi:  404nMAssay Description:Inhibition of Helicobacter pylori urease using urea as substrate assessed as inhibition constant for enzyme-inhibitor complex by non-linear fitting a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356196(CHEMBL1276230)
Affinity DataKi:  407nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356202(CHEMBL1910225)
Affinity DataKi:  430nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488911(CHEMBL2298025)
Affinity DataKi:  440nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50449762(CHEMBL4172924)
Affinity DataKi:  441nMAssay Description:Mixed type non-competitive inhibition of urease in Helicobacter pylori ATCC 43504 assessed as reduction in ammonia production preincubated for 1.5 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit alpha [F36L]/beta/gamma(Proteus vulgaris)
Wroclaw University Of Technology

LigandPNGBDBM24969([(2-{[(benzyloxy)carbonyl]amino}acetamido)methyl](...)
Affinity DataKi:  450nM ΔG°:  -36.8kJ/mole IC50:  3.10E+3nMpH: 7.0 T: 2°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488920(CHEMBL2298019)
Affinity DataKi:  450nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356191(CHEMBL193804)
Affinity DataKi:  497nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356187(CHEMBL1269725)
Affinity DataKi:  625nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50491169(CHEMBL2377164)
Affinity DataKi:  641nMAssay Description:Competitive inhibition of Helicobacter pylori ATCC 43504 urease using urea as substrate by Lineweaver-Burk/Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488905(CHEMBL2298023)
Affinity DataKi:  650nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50197347(Ebselen Diselenide)
Affinity DataKi:  651nMAssay Description:Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 after 120 mins by Berthelot colorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50114665(2-(trifluoromethyl)benzaldehyde thiosemicarbazone ...)
Affinity DataKi:  670nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356189(CHEMBL1910220)
Affinity DataKi:  770nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356193(CHEMBL398206)
Affinity DataKi:  807nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488918(CHEMBL2298024)
Affinity DataKi:  820nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488919(CHEMBL2298022)
Affinity DataKi:  890nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50356194(CHEMBL499789)
Affinity DataKi:  910nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50534782(CHEMBL4471428)
Affinity DataKi:  915nMAssay Description:Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 after 120 mins by Berthelot colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50488914(CHEMBL1370012)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibition of Canavalia ensiformis (jack bean) urease assessed as release of ammonia after 30 min by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails Article
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50602006(CHEMBL5209436)
Affinity DataKi:  1.20E+3nMAssay Description:Mixed type inhibition of Helicobacter pyroli urease assessed as dissociation constant for ESI complex by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University

Curated by ChEMBL
LigandPNGBDBM50493364(CHEMBL2425480)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of Helicobacter pylori urease using urea as substrate assessed as inhibition constant for enzyme-urea-inhibitor complex by non-linear fitt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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