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Found 258 Enz. Inhib. hit(s) with Target = 'Seed linoleate 13S-lipoxygenase-1'
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50282770(CHEMBL2296824)
Affinity DataKi:  192nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM192766(4-MMPB)
Affinity DataKi:  198nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM192766(4-MMPB)
Affinity DataKi:  204nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50489108(CHEMBL2296821)
Affinity DataKi:  486nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50489109(CHEMBL2296820)
Affinity DataKi:  662nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50304296(CHEMBL594396 | Oleyl sulfate)
Affinity DataKi:  700nMAssay Description:Binding affinity to soybean LO1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50489110(CHEMBL2296823)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50489112(CHEMBL2296819)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280213((E)-11-(3-Pentyl-thiiranyl)-undec-9-enoic acid | C...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50489111(CHEMBL2296822)
Affinity DataKi:  2.01E+3nMAssay Description:Inhibition of Glycine max (soybean) 15-lipoxygenase activity assessed as decrease in peroxide formation using linoleic acid as substrate preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280211(11-(3-Pentyl-thiiranyl)-undecanoic acid | CHEMBL28...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50401193(CHEMBL1934604)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of soyabean lipoxygenase-1 assessed as inhibition constant for enzyme-inhibitor complex by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50401193(CHEMBL1934604)
Affinity DataKi:  1.57E+4nMAssay Description:Inhibition of soyabean lipoxygenase-1 assessed as inhibition constant for enzyme-substrate-inhibitor complex by Lineweaver-Burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50445691(CHEMBL243677)
Affinity DataKi:  1.80E+4nMAssay Description:Uncompetitive inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM7461(5,7-dihydroxy-2-phenyl-4H-chromen-4-one | 5,7-dihy...)
Affinity DataKi:  1.94E+4nMAssay Description:Mixed noncompetitive type inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Line...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50150484((Z)-9-octadecenoic acid | (Z)-Octadec-9-enoic acid...)
Affinity DataKi:  2.20E+4nMAssay Description:Binding affinity to soybean LO1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50157555(2-(3,4-dihydroxyphenyl)-4H-chromen-4-one | 3',4'-d...)
Affinity DataKi:  8.45E+4nMAssay Description:Mixed noncompetitive type inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Line...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50445690(CHEMBL457821)
Affinity DataKi:  9.54E+4nMAssay Description:Uncompetitive inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280214(8-(3-Octyl-oxiranyl)-octanoic acid | CHEMBL27918)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280207(11-(3-Pentyl-oxiranyl)-undecanoic acid | CHEMBL281...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280208((E)-11-(3-Pentyl-oxiranyl)-undec-9-enoic acid | CH...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280209(8-(3-Octyl-thiiranyl)-octanoic acid | CHEMBL28539)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280210(8-[((E)-3-Oct-2-enyl)-oxiranyl]-octanoic acid | CH...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50280212(8-[((E)-3-Oct-2-enyl)-thiiranyl]-octanoic acid | C...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of the compound against Soyabean type 1 Lipoxygenase (SBLO) was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50312650(5,4'-dihydroxyflavone | 5-hydroxy-2-(4-hydroxyphen...)
Affinity DataKi:  1.03E+5nMAssay Description:Mixed noncompetitive type inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Line...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKi:  1.07E+5nMAssay Description:Uncompetitive inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKi:  1.22E+5nMAssay Description:Uncompetitive inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50304295(CHEMBL611951 | Palmitoleyl sulfate)
Affinity DataKi:  1.40E+5nMAssay Description:Binding affinity to allosteric site of soybean LO1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  1.78E+5nMAssay Description:Mixed noncompetitive type inhibition of soybean LOX-1 using linoleic acid as substrate preincubated for 5 mins followed by substrate addition by Line...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50114094(4-bromo-5-[(2R,3S)-4-(2-bromo-4,5-dihydroxyphenyl)...)
Affinity DataIC50:  57nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50114093(4-chloro-5-[(2R,3S)-4-(2-chloro-4,5-dihydroxypheny...)
Affinity DataIC50:  65nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22364(1,3-Diarylprop-2-yn-1-one, 23a | 1-(4-hydroxy-3-me...)
Affinity DataIC50:  100nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22364(1,3-Diarylprop-2-yn-1-one, 23a | 1-(4-hydroxy-3-me...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity against 15-lipoxygenase obtained from soybeanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50114096(4-ethyl-5-[4-(2-ethyl-4,5-dihydroxyphenyl)-2,3-dim...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50114097(4-[4-(2,2-dimethylbenzo[d][1,3]dioxol-5-yl)-2,3-di...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50065996(4-[(2S,3R)-4-(4-Hydroxy-3-methoxy-phenyl)-2,3-dime...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against soybean 1-lipoxygenase (SLO)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22365(1,3-Diarylprop-2-yn-1-one, 23b | 1-(3-hydroxy-4-me...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against 15-lipoxygenase obtained from soybeanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22363(1,3-Diarylprop-2-yn-1-one, 17c | 3-(4-methanesulfo...)
Affinity DataIC50:  300nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22365(1,3-Diarylprop-2-yn-1-one, 23b | 1-(3-hydroxy-4-me...)
Affinity DataIC50:  300nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22354(1,3-Diarylprop-2-yn-1-one, 13k | 1-(4-hydroxypheny...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase obtained from potatoMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22356(1,3-Diarylprop-2-yn-1-one, 13m | 1-(3-hydroxypheny...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase obtained from potatoMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22354(1,3-Diarylprop-2-yn-1-one, 13k | 1-(4-hydroxypheny...)
Affinity DataIC50:  320nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22354(1,3-Diarylprop-2-yn-1-one, 13k | 1-(4-hydroxypheny...)
Affinity DataIC50:  320nMAssay Description:In vitro inhibitory activity against 15-lipoxygenase obtained from soybeanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22348(1,3-Diarylprop-2-yn-1-one, 13e | 3-(4-methanesulfo...)
Affinity DataIC50:  360nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22370(1,3-Diarylprop-2-yn-1-one, 27 | 3-(4-methanesulfon...)
Affinity DataIC50:  360nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM50135282(CHEMBL3746867)
Affinity DataIC50:  400nMAssay Description:Inhibition of soybean LOX1 assessed as reduction in linoleic acid oxidation measured every 10 s for 10 mins by spectrophotometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22352(1,3-Diarylprop-2-yn-1-one, 13i | 1-(3,4-difluoroph...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase obtained from potatoMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22356(1,3-Diarylprop-2-yn-1-one, 13m | 1-(3-hydroxypheny...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory activity against 15-lipoxygenase obtained from soybeanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))TBA
LigandPNGBDBM22356(1,3-Diarylprop-2-yn-1-one, 13m | 1-(3-hydroxypheny...)
Affinity DataIC50:  500nMAssay Description:The lipoxygenase inhibitor screening assay detects and measures the hydroperoxides produced in the lipoxygenation reaction using a purified lipoxygen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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