BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID of Ligand	PubChem SID of Ligand	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence	PDB ID(s) of Target Chain	UniProt (SwissProt) Recommended Name of Target Chain	UniProt (SwissProt) Entry Name of Target Chain	UniProt (SwissProt) Primary ID of Target Chain	UniProt (SwissProt) Secondary ID(s) of Target Chain	UniProt (SwissProt) Alternative ID(s) of Target Chain	UniProt (TrEMBL) Submitted Name of Target Chain	UniProt (TrEMBL) Entry Name of Target Chain	UniProt (TrEMBL) Primary ID of Target Chain	UniProt (TrEMBL) Secondary ID(s) of Target Chain	UniProt (TrEMBL) Alternative ID(s) of Target Chain
385318	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(Cc3ccccc3)c(Cl)c2c1	InChI=1S/C27H20Cl3N3O/c1-33-16-31-15-24(33)27(34,18-7-10-20(28)11-8-18)19-9-12-23-21(14-19)25(29)22(26(30)32-23)13-17-5-3-2-4-6-17/h2-12,14-16,34H,13H2,1H3	IGBFRJGBHUMYIT-UHFFFAOYSA-N	50058844	CHEMBL3325741::US9290476, 1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 18				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50058844	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50058844&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221196	103954746		CHEMBL3325741				ZINC26168793	1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385319	OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(Cc3ccc(Cl)cc3)c(Cl)c2c1	InChI=1S/C28H18Cl4N2O/c29-21-9-6-17(7-10-21)13-24-26(31)23-15-19(8-11-25(23)34-27(24)32)28(35,20-4-2-12-33-16-20)18-3-1-5-22(30)14-18/h1-12,14-16,35H,13H2	OXQXJWJVGWJASD-UHFFFAOYSA-N	220159	US9290476, 2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 17				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220159&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221198	329995278							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385320	OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(Cc3ccc(F)cc3)c(Cl)c2c1	InChI=1S/C28H18Cl3FN2O/c29-21-5-1-3-18(14-21)28(35,20-4-2-12-33-16-20)19-8-11-25-23(15-19)26(30)24(27(31)34-25)13-17-6-9-22(32)10-7-17/h1-12,14-16,35H,13H2	SBTJHLXFEXNJQZ-UHFFFAOYSA-N	220160	US9290476, 3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 32				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220160&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221199	329995279							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385321	OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(Cc3cccc(Cl)c3)c(Cl)c2c1	InChI=1S/C28H18Cl4N2O/c29-21-7-1-4-17(12-21)13-24-26(31)23-15-19(9-10-25(23)34-27(24)32)28(35,20-6-3-11-33-16-20)18-5-2-8-22(30)14-18/h1-12,14-16,35H,13H2	JQYWKIHBVLDXCM-UHFFFAOYSA-N	220161	US9290476, 4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 7.7				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220161&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221259	329995280							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385322	OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C31H21Cl3N4O/c32-24-6-1-4-21(17-24)31(39,23-5-2-13-35-19-23)22-9-12-28-26(18-22)29(33)27(30(34)37-28)16-20-7-10-25(11-8-20)38-15-3-14-36-38/h1-15,17-19,39H,16H2	CLYKYJUSPRHKQB-UHFFFAOYSA-N	220162	US9290476, 5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 11				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220162&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221197	329995281							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385323	COc1ccc(Cc2c(Cl)nc3ccc(cc3c2Cl)C(O)(c2cccnc2)c2cccc(Cl)c2)cc1	InChI=1S/C29H21Cl3N2O2/c1-36-23-10-7-18(8-11-23)14-25-27(31)24-16-20(9-12-26(24)34-28(25)32)29(35,21-5-3-13-33-17-21)19-4-2-6-22(30)15-19/h2-13,15-17,35H,14H2,1H3	KGSQNIJWCOLAGX-UHFFFAOYSA-N	220163	US9290476, 6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 15				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220163	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220163&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221260	329995282							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385324	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(F)cc1)C(O)(c1cccnc1)c1cccc(Cl)c1	InChI=1S/C29H21Cl2FN2O2/c1-36-28-25(14-18-7-10-23(32)11-8-18)27(31)24-16-20(9-12-26(24)34-28)29(35,21-5-3-13-33-17-21)19-4-2-6-22(30)15-19/h2-13,15-17,35H,14H2,1H3	YXIRACZJKCHFAQ-UHFFFAOYSA-N	220164	US9290476, 7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 40				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220164&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221261	329995283							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385325	CS(=O)(=O)c1ccc(Cc2c(Cl)nc3ccc(cc3c2Cl)C(O)(c2cccnc2)c2cccc(Cl)c2)cc1	InChI=1S/C29H21Cl3N2O3S/c1-38(36,37)23-10-7-18(8-11-23)14-25-27(31)24-16-20(9-12-26(24)34-28(25)32)29(35,21-5-3-13-33-17-21)19-4-2-6-22(30)15-19/h2-13,15-17,35H,14H2,1H3	IHXQNZCYYBOBRQ-UHFFFAOYSA-N	220165	US9290476, 8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 43				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220165&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221262	329995284							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385326	OC(c1cncs1)(c1cccnc1)c1ccc2nc(Cl)c(Cc3ccc(Cl)cc3)c(Cl)c2c1	InChI=1S/C25H16Cl3N3OS/c26-18-6-3-15(4-7-18)10-20-23(27)19-11-16(5-8-21(19)31-24(20)28)25(32,22-13-30-14-33-22)17-2-1-9-29-12-17/h1-9,11-14,32H,10H2	CMXRSYSPKWFPNL-UHFFFAOYSA-N	220166	US9290476, 9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.83				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220166&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221325	329995285							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385327	OC(c1cncs1)(c1cccnc1)c1ccc2nc(Cl)c(Cc3cccc(Cl)c3)cc2c1	InChI=1S/C25H17Cl2N3OS/c26-21-5-1-3-16(10-21)9-18-11-17-12-19(6-7-22(17)30-24(18)27)25(31,23-14-29-15-32-23)20-4-2-8-28-13-20/h1-8,10-15,31H,9H2	ZEZHVKIBNFEYRX-UHFFFAOYSA-N	220167	US9290476, 10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 99				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220167&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117880572	329995286							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385328	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H22Cl3N5O/c1-37-18-34-17-27(37)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(16-21)28(32)25(29(33)36-26)15-19-3-10-23(11-4-19)38-14-2-13-35-38/h2-14,16-18,39H,15H2,1H3	TUVOSORVOJMOFI-UHFFFAOYSA-N	220168	US9290476, 11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 75				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220168	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220168&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221327	329995287							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385329	COc1ccc(Cc2c(Cl)nc3ccc(cc3c2Cl)C(O)(c2cncn2C)c2ccc(Cl)cc2)cc1	InChI=1S/C28H22Cl3N3O2/c1-34-16-32-15-25(34)28(35,18-5-8-20(29)9-6-18)19-7-12-24-22(14-19)26(30)23(27(31)33-24)13-17-3-10-21(36-2)11-4-17/h3-12,14-16,35H,13H2,1-2H3	TZAHYKIEXMAZMN-UHFFFAOYSA-N	220169	US9290476, 12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 16				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220169&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221326	329995288							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385330	COc1ccc(Cc2c(OC)nc3ccc(cc3c2Cl)C(O)(c2cncn2C)c2ccc(Cl)cc2)cc1	InChI=1S/C29H25Cl2N3O3/c1-34-17-32-16-26(34)29(35,19-6-9-21(30)10-7-19)20-8-13-25-23(15-20)27(31)24(28(33-25)37-3)14-18-4-11-22(36-2)12-5-18/h4-13,15-17,35H,14H2,1-3H3	VNRDASGWMIPLHO-UHFFFAOYSA-N	220170	US9290476, 13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 31				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220170&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117880633	329995289							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385331	CCOc1nc2ccc(cc2c(Cl)c1Cc1ccccc1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H25Cl2N3O2/c1-3-36-28-24(15-19-7-5-4-6-8-19)27(31)23-16-21(11-14-25(23)33-28)29(35,26-17-32-18-34(26)2)20-9-12-22(30)13-10-20/h4-14,16-18,35H,3,15H2,1-2H3	PAENGSSCLOGLRS-UHFFFAOYSA-N	220171	US9290476, 14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 91				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220171&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221329	329995290							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385332	Cn1cncc1C(O)(c1cncs1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C27H20Cl2N6OS/c1-34-15-30-13-23(34)27(36,24-14-31-16-37-24)18-5-8-22-20(12-18)25(28)21(26(29)33-22)11-17-3-6-19(7-4-17)35-10-2-9-32-35/h2-10,12-16,36H,11H2,1H3	YQWCFUBFHBRRQZ-UHFFFAOYSA-N	220172	US9290476, 15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.3				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220172	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220172&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117880575	329995291							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385333	CCOc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncs1)c1cncn1C	InChI=1S/C29H25ClN6O2S/c1-3-38-28-23(13-19-5-8-21(9-6-19)36-12-4-11-33-36)27(30)22-14-20(7-10-24(22)34-28)29(37,26-16-32-18-39-26)25-15-31-17-35(25)2/h4-12,14-18,37H,3,13H2,1-2H3	VMARLUAGWLOMAY-UHFFFAOYSA-N	220173	US9290476, 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.6				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220173	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220173&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221392	329995292							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385334	CCN(C)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C33H30Cl2N6O/c1-4-39(2)32-28(18-22-6-13-26(14-7-22)41-17-5-16-37-41)31(35)27-19-24(10-15-29(27)38-32)33(42,30-20-36-21-40(30)3)23-8-11-25(34)12-9-23/h5-17,19-21,42H,4,18H2,1-3H3	ABVIJTLJNLQKEH-UHFFFAOYSA-N	220174	US9290476, 17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 310				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220174&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221393	329995293							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385335	COc1ccc(cn1)C(O)(c1cncs1)c1ccc2nc(Cl)c(Cc3ccccc3)c(Cl)c2c1	InChI=1S/C26H19Cl2N3O2S/c1-33-23-10-8-18(13-30-23)26(32,22-14-29-15-34-22)17-7-9-21-19(12-17)24(27)20(25(28)31-21)11-16-5-3-2-4-6-16/h2-10,12-15,32H,11H2,1H3	WVLGOQBSBKHESG-UHFFFAOYSA-N	220175	US9290476, 18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220175	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220175&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221394	329995294							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385336	CCOc1nc2ccc(cc2c(Cl)c1Cc1ccccc1)C(O)(c1cncs1)c1ccc(OC)nc1	InChI=1S/C28H24ClN3O3S/c1-3-35-27-22(13-18-7-5-4-6-8-18)26(29)21-14-19(9-11-23(21)32-27)28(33,24-16-30-17-36-24)20-10-12-25(34-2)31-15-20/h4-12,14-17,33H,3,13H2,1-2H3	FNAYGXXYFPNBPF-UHFFFAOYSA-N	220176	US9290476, 19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.7				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220176	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220176&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221395	329995295							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385337	COc1ccc(cn1)C(O)(c1cncs1)c1ccc2nc(OC)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H24ClN5O3S/c1-38-27-11-7-21(16-33-27)30(37,26-17-32-18-40-26)20-6-10-25-23(15-20)28(31)24(29(35-25)39-2)14-19-4-8-22(9-5-19)36-13-3-12-34-36/h3-13,15-18,37H,14H2,1-2H3	HESKYEVXASVNSF-UHFFFAOYSA-N	220177	US9290476, 20A::US9290476, 20B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 3.8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220177	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220177&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715663	329995296							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385338	COc1ccc(cn1)C(O)(c1cncs1)c1ccc2nc(OC)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H24ClN5O3S/c1-38-27-11-7-21(16-33-27)30(37,26-17-32-18-40-26)20-6-10-25-23(15-20)28(31)24(29(35-25)39-2)14-19-4-8-22(9-5-19)36-13-3-12-34-36/h3-13,15-18,37H,14H2,1-2H3	HESKYEVXASVNSF-UHFFFAOYSA-N	220177	US9290476, 20A::US9290476, 20B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220177	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220177&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715663	329995296							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385339	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H25Cl2N3O4S/c1-34-17-32-16-26(34)29(35,19-6-9-21(30)10-7-19)20-8-13-25-23(15-20)27(31)24(28(33-25)38-2)14-18-4-11-22(12-5-18)39(3,36)37/h4-13,15-17,35H,14H2,1-3H3	LHVHXPSNXCRUBJ-UHFFFAOYSA-N	220188	US9290476, 31	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 5.3				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220188	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220188&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220544	329995307							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385340	COc1ccc(cn1)C(O)(c1cncn1C)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H24Cl2N6O2/c1-37-18-33-17-26(37)30(39,21-7-11-27(40-2)34-16-21)20-6-10-25-23(15-20)28(31)24(29(32)36-25)14-19-4-8-22(9-5-19)38-13-3-12-35-38/h3-13,15-18,39H,14H2,1-2H3	FVLQPFTUUNLGLJ-UHFFFAOYSA-N	220178	US9290476, 21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.1				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220178	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220178&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221461	329995297							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385341	COc1ccc(cn1)C(O)(c1cncn1C)c1ccc2nc(OC)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C31H27ClN6O3/c1-37-19-33-18-27(37)31(39,22-8-12-28(40-2)34-17-22)21-7-11-26-24(16-21)29(32)25(30(36-26)41-3)15-20-5-9-23(10-6-20)38-14-4-13-35-38/h4-14,16-19,39H,15H2,1-3H3	HRPPXVZQHFXSFY-UHFFFAOYSA-N	220179	US9290476, 22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221462	329995298							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385342	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H21Cl2F3N6O/c1-40-17-36-16-26(40)29(42,20-6-10-25(37-15-20)30(33,34)35)19-5-9-24-22(14-19)27(31)23(28(32)39-24)13-18-3-7-21(8-4-18)41-12-2-11-38-41/h2-12,14-17,42H,13H2,1H3	RNGIRHRQNXVNGK-UHFFFAOYSA-N	220180	US9290476, 23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221463	329995299							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385343	CCOc1nc2ccc(cc2cc1Cc1ccc(OC)cc1)C(O)(c1cncs1)c1cncn1C	InChI=1S/C27H26N4O3S/c1-4-34-26-20(11-18-5-8-22(33-3)9-6-18)12-19-13-21(7-10-23(19)30-26)27(32,25-15-29-17-35-25)24-14-28-16-31(24)2/h5-10,12-17,32H,4,11H2,1-3H3	VZNCGBQJXQQBTL-UHFFFAOYSA-N	220181	US9290476, 24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 750				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220181&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221464	329995300							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385344	CN(C)c1ccc(cc1)C(O)(c1cncn1C)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C32H28Cl2N6O/c1-38(2)24-12-7-22(8-13-24)32(41,29-19-35-20-39(29)3)23-9-14-28-26(18-23)30(33)27(31(34)37-28)17-21-5-10-25(11-6-21)40-16-4-15-36-40/h4-16,18-20,41H,17H2,1-3H3	XJIYGWJODWNNBE-UHFFFAOYSA-N	220182	US9290476, 25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 440				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220182&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221527	329995301							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385345	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(cc1)N(C)C	InChI=1S/C33H31ClN6O2/c1-38(2)25-13-8-23(9-14-25)33(41,30-20-35-21-39(30)3)24-10-15-29-27(19-24)31(34)28(32(37-29)42-4)18-22-6-11-26(12-7-22)40-17-5-16-36-40/h5-17,19-21,41H,18H2,1-4H3	HTRJODMUEHDFAM-UHFFFAOYSA-N	220183	US9290476, 26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 220				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220183	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220183&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221528	329995302							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385346	Cc1cc(cc2c(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)nc12)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C31H24Cl3N5O/c1-19-14-22(31(40,27-17-35-18-38(27)2)21-6-8-23(32)9-7-21)16-25-28(33)26(30(34)37-29(19)25)15-20-4-10-24(11-5-20)39-13-3-12-36-39/h3-14,16-18,40H,15H2,1-2H3	KARDQPKYJHATDW-UHFFFAOYSA-N	220184	US9290476, 27::US9290476, 85	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 85				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220184	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220184&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221529	329995303							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385347	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C32H27Cl2N5O2/c1-20-15-23(32(40,28-18-35-19-38(28)2)22-7-9-24(33)10-8-22)17-26-29(34)27(31(41-3)37-30(20)26)16-21-5-11-25(12-6-21)39-14-4-13-36-39/h4-15,17-19,40H,16H2,1-3H3	HPZHEYVXVBLMSC-UHFFFAOYSA-N	220185	US9290476, 28A::US9290476, 28B::US9290476, 28C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 53				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220185&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221530	329995304							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385348	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C32H27Cl2N5O2/c1-20-15-23(32(40,28-18-35-19-38(28)2)22-7-9-24(33)10-8-22)17-26-29(34)27(31(41-3)37-30(20)26)16-21-5-11-25(12-6-21)39-14-4-13-36-39/h4-15,17-19,40H,16H2,1-3H3	HPZHEYVXVBLMSC-UHFFFAOYSA-N	220185	US9290476, 28A::US9290476, 28B::US9290476, 28C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1600				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220185&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221530	329995304							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385349	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C32H27Cl2N5O2/c1-20-15-23(32(40,28-18-35-19-38(28)2)22-7-9-24(33)10-8-22)17-26-29(34)27(31(41-3)37-30(20)26)16-21-5-11-25(12-6-21)39-14-4-13-36-39/h4-15,17-19,40H,16H2,1-3H3	HPZHEYVXVBLMSC-UHFFFAOYSA-N	220185	US9290476, 28A::US9290476, 28B::US9290476, 28C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 5.8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220185&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221530	329995304							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385350	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H26ClF3N6O2/c1-19-13-22(31(43,27-17-37-18-41(27)2)21-7-10-26(38-16-21)32(34,35)36)15-24-28(33)25(30(44-3)40-29(19)24)14-20-5-8-23(9-6-20)42-12-4-11-39-42/h4-13,15-18,43H,14H2,1-3H3	NTMKNDJXPHULDI-UHFFFAOYSA-N	220186	US9290476, 29A::US9290476, 29B::US9290476, 29C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220186&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715664	329995305							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385351	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H26ClF3N6O2/c1-19-13-22(31(43,27-17-37-18-41(27)2)21-7-10-26(38-16-21)32(34,35)36)15-24-28(33)25(30(44-3)40-29(19)24)14-20-5-8-23(9-6-20)42-12-4-11-39-42/h4-13,15-18,43H,14H2,1-3H3	NTMKNDJXPHULDI-UHFFFAOYSA-N	220186	US9290476, 29A::US9290476, 29B::US9290476, 29C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 93				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220186&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715664	329995305							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385352	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H26ClF3N6O2/c1-19-13-22(31(43,27-17-37-18-41(27)2)21-7-10-26(38-16-21)32(34,35)36)15-24-28(33)25(30(44-3)40-29(19)24)14-20-5-8-23(9-6-20)42-12-4-11-39-42/h4-13,15-18,43H,14H2,1-3H3	NTMKNDJXPHULDI-UHFFFAOYSA-N	220186	US9290476, 29A::US9290476, 29B::US9290476, 29C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.9				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220186&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715664	329995305							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385353	Cn1cncc1C(O)(c1cncn1C)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C28H23Cl2N7O/c1-35-16-31-14-24(35)28(38,25-15-32-17-36(25)2)19-6-9-23-21(13-19)26(29)22(27(30)34-23)12-18-4-7-20(8-5-18)37-11-3-10-33-37/h3-11,13-17,38H,12H2,1-2H3	ILXMOCXUQZGNDQ-UHFFFAOYSA-N	220187	US9290476, 30	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.2				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220187	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220187&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221531	329995306							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385354	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H25Cl2N3O4S/c1-34-17-32-16-26(34)29(35,19-6-9-21(30)10-7-19)20-8-13-25-23(15-20)27(31)24(28(33-25)38-2)14-18-4-11-22(12-5-18)39(3,36)37/h4-13,15-17,35H,14H2,1-3H3	LHVHXPSNXCRUBJ-UHFFFAOYSA-N	220188	US9290476, 31	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 64				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220188	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220188&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220544	329995307							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385355	OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(Cc3cccs3)c(Cl)c2c1	InChI=1S/C26H17Cl3N2OS/c27-19-6-1-4-16(12-19)26(32,18-5-2-10-30-15-18)17-8-9-23-21(13-17)24(28)22(25(29)31-23)14-20-7-3-11-33-20/h1-13,15,32H,14H2	IYKQSHIBZGMMBS-UHFFFAOYSA-N	220189	US9290476, 32	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 33				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220189	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220189&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220545	329995308							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385356	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C31H25Cl2N5O2/c1-37-19-34-18-28(37)31(39,21-6-9-23(32)10-7-21)22-8-13-27-25(17-22)29(33)26(30(36-27)40-2)16-20-4-11-24(12-5-20)38-15-3-14-35-38/h3-15,17-19,39H,16H2,1-2H3	UWOBQISTECYGOP-UHFFFAOYSA-N	220190	US9290476, 33A::US9290476, 33B::US9290476, 33C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 43				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220190&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	8A4	5UHI	74220546	329995309							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385357	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C31H25Cl2N5O2/c1-37-19-34-18-28(37)31(39,21-6-9-23(32)10-7-21)22-8-13-27-25(17-22)29(33)26(30(36-27)40-2)16-20-4-11-24(12-5-20)38-15-3-14-35-38/h3-15,17-19,39H,16H2,1-2H3	UWOBQISTECYGOP-UHFFFAOYSA-N	220190	US9290476, 33A::US9290476, 33B::US9290476, 33C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 810				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220190&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	8A4	5UHI	74220546	329995309							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385358	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C31H25Cl2N5O2/c1-37-19-34-18-28(37)31(39,21-6-9-23(32)10-7-21)22-8-13-27-25(17-22)29(33)26(30(36-27)40-2)16-20-4-11-24(12-5-20)38-15-3-14-35-38/h3-15,17-19,39H,16H2,1-2H3	UWOBQISTECYGOP-UHFFFAOYSA-N	220190	US9290476, 33A::US9290476, 33B::US9290476, 33C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 20				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220190&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	8A4	5UHI	74220546	329995309							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385359	COc1nc2ccc(cc2c(OC)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C32H28ClN5O3/c1-37-20-34-19-29(37)32(39,22-7-10-24(33)11-8-22)23-9-14-28-26(18-23)30(40-2)27(31(36-28)41-3)17-21-5-12-25(13-6-21)38-16-4-15-35-38/h4-16,18-20,39H,17H2,1-3H3	XDDWQFIEJOPHLL-UHFFFAOYSA-N	220191	US9290476, 34	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 250				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220191	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220191&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220547	329995310							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385360	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C31H24ClF3N6O2/c1-40-18-36-17-27(40)30(42,21-7-11-26(37-16-21)31(33,34)35)20-6-10-25-23(15-20)28(32)24(29(39-25)43-2)14-19-4-8-22(9-5-19)41-13-3-12-38-41/h3-13,15-18,42H,14H2,1-2H3	LZOGZAYEBDXEJA-UHFFFAOYSA-N	220192	US9290476, 35A::US9290476, 35B::US9290476, 35C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220192&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WA	5W4V	74220611	329995311							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385361	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C31H24ClF3N6O2/c1-40-18-36-17-27(40)30(42,21-7-11-26(37-16-21)31(33,34)35)20-6-10-25-23(15-20)28(32)24(29(39-25)43-2)14-19-4-8-22(9-5-19)41-13-3-12-38-41/h3-13,15-18,42H,14H2,1-2H3	LZOGZAYEBDXEJA-UHFFFAOYSA-N	220192	US9290476, 35A::US9290476, 35B::US9290476, 35C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 70				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220192&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WA	5W4V	74220611	329995311							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385362	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C31H24ClF3N6O2/c1-40-18-36-17-27(40)30(42,21-7-11-26(37-16-21)31(33,34)35)20-6-10-25-23(15-20)28(32)24(29(39-25)43-2)14-19-4-8-22(9-5-19)41-13-3-12-38-41/h3-13,15-18,42H,14H2,1-2H3	LZOGZAYEBDXEJA-UHFFFAOYSA-N	220192	US9290476, 35A::US9290476, 35B::US9290476, 35C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220192&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WA	5W4V	74220611	329995311							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385363	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H23Cl2N3O2S/c1-35-17-33-16-27(35)30(36,19-7-10-21(31)11-8-19)20-9-12-25-23(14-20)28(32)24(29(34-25)37-2)15-22-13-18-5-3-4-6-26(18)38-22/h3-14,16-17,36H,15H2,1-2H3	QBHBKTAEUVNENV-UHFFFAOYSA-N	220193	US9290476, 36A::US9290476, 36B::US9290476, 36C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 40				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220193&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220612	329995312							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385364	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H23Cl2N3O2S/c1-35-17-33-16-27(35)30(36,19-7-10-21(31)11-8-19)20-9-12-25-23(14-20)28(32)24(29(34-25)37-2)15-22-13-18-5-3-4-6-26(18)38-22/h3-14,16-17,36H,15H2,1-2H3	QBHBKTAEUVNENV-UHFFFAOYSA-N	220193	US9290476, 36A::US9290476, 36B::US9290476, 36C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 400				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220193&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220612	329995312							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385365	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H23Cl2N3O2S/c1-35-17-33-16-27(35)30(36,19-7-10-21(31)11-8-19)20-9-12-25-23(14-20)28(32)24(29(34-25)37-2)15-22-13-18-5-3-4-6-26(18)38-22/h3-14,16-17,36H,15H2,1-2H3	QBHBKTAEUVNENV-UHFFFAOYSA-N	220193	US9290476, 36A::US9290476, 36B::US9290476, 36C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 11				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220193&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220612	329995312							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385366	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C30H22ClF3N4O2S/c1-38-16-35-15-26(38)29(39,19-8-10-25(36-14-19)30(32,33)34)18-7-9-23-21(12-18)27(31)22(28(37-23)40-2)13-20-11-17-5-3-4-6-24(17)41-20/h3-12,14-16,39H,13H2,1-2H3	HERRXBWYJBLMNI-UHFFFAOYSA-N	220194	US9290476, 37A::US9290476, 37B::US9290476, 37C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 7.8				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220194&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220613	329995313							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385367	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C30H22ClF3N4O2S/c1-38-16-35-15-26(38)29(39,19-8-10-25(36-14-19)30(32,33)34)18-7-9-23-21(12-18)27(31)22(28(37-23)40-2)13-20-11-17-5-3-4-6-24(17)41-20/h3-12,14-16,39H,13H2,1-2H3	HERRXBWYJBLMNI-UHFFFAOYSA-N	220194	US9290476, 37A::US9290476, 37B::US9290476, 37C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 44				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220194&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220613	329995313							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385368	COc1nc2ccc(cc2c(Cl)c1Cc1cc2ccccc2s1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C30H22ClF3N4O2S/c1-38-16-35-15-26(38)29(39,19-8-10-25(36-14-19)30(32,33)34)18-7-9-23-21(12-18)27(31)22(28(37-23)40-2)13-20-11-17-5-3-4-6-24(17)41-20/h3-12,14-16,39H,13H2,1-2H3	HERRXBWYJBLMNI-UHFFFAOYSA-N	220194	US9290476, 37A::US9290476, 37B::US9290476, 37C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 3.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220194&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220613	329995313							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385369	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccc(F)cc1	InChI=1S/C34H32ClFN4O3/c1-22(41)39-18-14-25(15-19-39)34(42,24-6-9-27(36)10-7-24)26-8-13-31-29(21-26)32(35)30(33(38-31)43-2)20-23-4-11-28(12-5-23)40-17-3-16-37-40/h3-13,16-17,21,25,42H,14-15,18-20H2,1-2H3	YBHGNUBDICQAPT-UHFFFAOYSA-N	220195	US9290476, 38	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 3.9				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220195&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117870100	329995314							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385370	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1ccc(F)cc1)c1cccnc1	InChI=1S/C32H24ClFN4O2/c1-40-31-28(18-21-5-12-26(13-6-21)38-17-3-16-36-38)30(33)27-19-23(9-14-29(27)37-31)32(39,24-4-2-15-35-20-24)22-7-10-25(34)11-8-22/h2-17,19-20,39H,18H2,1H3	GZTHRAHREHCGTD-UHFFFAOYSA-N	220196	US9290476, 39	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 21				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220196&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220680	329995315							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385371	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1ccc(cc1)C(F)(F)F)c1cccnc1	InChI=1S/C33H24ClF3N4O2/c1-43-31-28(18-21-5-12-26(13-6-21)41-17-3-16-39-41)30(34)27-19-24(11-14-29(27)40-31)32(42,25-4-2-15-38-20-25)22-7-9-23(10-8-22)33(35,36)37/h2-17,19-20,42H,18H2,1H3	JMLXMIANXQQSCL-UHFFFAOYSA-N	220197	US9290476, 40	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 20				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220197&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220681	329995316							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385372	COc1ccc(cc1OC)C(O)(c1cccnc1)c1ccc2nc(OC)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C34H29ClN4O4/c1-41-30-14-10-24(20-31(30)42-2)34(40,25-6-4-15-36-21-25)23-9-13-29-27(19-23)32(35)28(33(38-29)43-3)18-22-7-11-26(12-8-22)39-17-5-16-37-39/h4-17,19-21,40H,18H2,1-3H3	GIHDYAPDDPIGSP-UHFFFAOYSA-N	220198	US9290476, 41	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 29				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220198&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220682	329995317							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385373	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1ccc(cc1)N(C)C)c1cccnc1	InChI=1S/C34H30ClN5O2/c1-39(2)27-14-9-24(10-15-27)34(41,26-6-4-17-36-22-26)25-11-16-31-29(21-25)32(35)30(33(38-31)42-3)20-23-7-12-28(13-8-23)40-19-5-18-37-40/h4-19,21-22,41H,20H2,1-3H3	HZSPACMDRJFYPA-UHFFFAOYSA-N	220199	US9290476, 42	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 360				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220199&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220683	329995318							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385374	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cn(C)cn1)c1ccc(F)cc1	InChI=1S/C31H25ClFN5O2/c1-37-18-28(34-19-37)31(39,21-6-9-23(33)10-7-21)22-8-13-27-25(17-22)29(32)26(30(36-27)40-2)16-20-4-11-24(12-5-20)38-15-3-14-35-38/h3-15,17-19,39H,16H2,1-2H3	GIWGIKUMDUOHFI-UHFFFAOYSA-N	220200	US9290476, 43	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 49				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220200	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220200&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117880636	329995319							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385375	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cccnc1)c1ccc(Cl)c(Cl)c1	InChI=1S/C32H23Cl3N4O2/c1-41-31-26(16-20-5-9-24(10-6-20)39-15-3-14-37-39)30(35)25-17-21(8-12-29(25)38-31)32(40,23-4-2-13-36-19-23)22-7-11-27(33)28(34)18-22/h2-15,17-19,40H,16H2,1H3	LQFGBIOOUDUOQX-UHFFFAOYSA-N	220201	US9290476, 44	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 15				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220201	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220201&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715665	329995320							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385376	OC(c1ccc(Cl)cc1)(c1cccnc1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C31H21Cl3N4O/c32-24-9-6-21(7-10-24)31(39,23-3-1-14-35-19-23)22-8-13-28-26(18-22)29(33)27(30(34)37-28)17-20-4-11-25(12-5-20)38-16-2-15-36-38/h1-16,18-19,39H,17H2	BQMOPYYISMUQTP-UHFFFAOYSA-N	220202	US9290476, 45	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 68				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220202	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220202&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220747	329995321							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385377	OC(c1ccc(F)cc1)(c1cccnc1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C31H21Cl2FN4O/c32-29-26-18-22(31(39,23-3-1-14-35-19-23)21-6-9-24(34)10-7-21)8-13-28(26)37-30(33)27(29)17-20-4-11-25(12-5-20)38-16-2-15-36-38/h1-16,18-19,39H,17H2	WBPIYJZVIVKTPY-UHFFFAOYSA-N	220203	US9290476, 46	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 22				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220203&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220748	329995322							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385378	COc1ccc(cc1)C(O)(c1cccnc1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C32H24Cl2N4O2/c1-40-26-12-7-22(8-13-26)32(39,24-4-2-15-35-20-24)23-9-14-29-27(19-23)30(33)28(31(34)37-29)18-21-5-10-25(11-6-21)38-17-3-16-36-38/h2-17,19-20,39H,18H2,1H3	DRTOSBOXBLMTTF-UHFFFAOYSA-N	220204	US9290476, 47	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 140				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220204&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220749	329995323							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385379	OC(c1cccnc1)(c1cccc(F)c1)c1ccc2nc(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C31H21Cl2FN4O/c32-29-26-18-22(31(39,23-5-2-13-35-19-23)21-4-1-6-24(34)17-21)9-12-28(26)37-30(33)27(29)16-20-7-10-25(11-8-20)38-15-3-14-36-38/h1-15,17-19,39H,16H2	AQZPGYVCTUUSQF-UHFFFAOYSA-N	220205	US9290476, 48	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 10				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220205&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220811	329995324							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385380	Cn1cc(cn1)C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(Cc3ccccc3)c(Cl)c2c1	InChI=1S/C27H20Cl3N3O/c1-33-16-20(15-31-33)27(34,18-7-10-21(28)11-8-18)19-9-12-24-22(14-19)25(29)23(26(30)32-24)13-17-5-3-2-4-6-17/h2-12,14-16,34H,13H2,1H3	OOVDWIGQIZNEQZ-UHFFFAOYSA-N	220206	US9290476, 49	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 330				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220206&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220813	329995325							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385381	Cc1nc2ccc(cc2c(C)c1Cc1ccccc1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H26ClN3O/c1-19-25(15-21-7-5-4-6-8-21)20(2)32-27-14-11-23(16-26(19)27)29(34,28-17-31-18-33(28)3)22-9-12-24(30)13-10-22/h4-14,16-18,34H,15H2,1-3H3	KNOQLBHGAGDFRW-UHFFFAOYSA-N	220207	US9290476, 50	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 320				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220207&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220812	329995326							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385382	CNC(=O)c1nc2ccc(cc2c(c1Cc1ccccc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(F)cc1	InChI=1S/C30H24F4N4O2/c1-35-28(39)27-23(14-18-6-4-3-5-7-18)26(30(32,33)34)22-15-20(10-13-24(22)37-27)29(40,25-16-36-17-38(25)2)19-8-11-21(31)12-9-19/h3-13,15-17,40H,14H2,1-2H3,(H,35,39)	JGMPJTKMSBWZSG-UHFFFAOYSA-N	220208	US9290476, 51	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1100				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220208&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220814	329995327							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385383	COc1ccc(Cc2cc3cc(ccc3nc2Cl)C(O)(c2cncs2)c2cncn2C)cc1	InChI=1S/C25H21ClN4O2S/c1-30-14-27-12-22(30)25(31,23-13-28-15-33-23)19-5-8-21-17(11-19)10-18(24(26)29-21)9-16-3-6-20(32-2)7-4-16/h3-8,10-15,31H,9H2,1-2H3	QTXZNSNYEMLLNM-UHFFFAOYSA-N	220209	US9290476, 52	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1900				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220209&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220815	329995328							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385384	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C29H24ClF3N4O4S/c1-37-16-34-15-25(37)28(38,19-7-11-24(35-14-19)29(31,32)33)18-6-10-23-21(13-18)26(30)22(27(36-23)41-2)12-17-4-8-20(9-5-17)42(3,39)40/h4-11,13-16,38H,12H2,1-3H3	BUNRTAJYWAGDHW-UHFFFAOYSA-N	220210	US9290476, 53	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 37				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220210&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220878	329995329							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385385	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(F)cc1	InChI=1S/C29H25ClFN3O4S/c1-34-17-32-16-26(34)29(35,19-6-9-21(31)10-7-19)20-8-13-25-23(15-20)27(30)24(28(33-25)38-2)14-18-4-11-22(12-5-18)39(3,36)37/h4-13,15-17,35H,14H2,1-3H3	JGBXDXWRYBFJMF-UHFFFAOYSA-N	220294	US9290476, 54B::US9290476, 54C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 840				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220294&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220879	329995356							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385386	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(F)cc1	InChI=1S/C29H25ClFN3O4S/c1-34-17-32-16-26(34)29(35,19-6-9-21(31)10-7-19)20-8-13-25-23(15-20)27(30)24(28(33-25)38-2)14-18-4-11-22(12-5-18)39(3,36)37/h4-13,15-17,35H,14H2,1-3H3	JGBXDXWRYBFJMF-UHFFFAOYSA-N	220294	US9290476, 54B::US9290476, 54C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 23				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220294&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220879	329995356							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385387	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(O)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H23Cl2N5O2/c1-36-18-33-17-27(36)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(16-21)28(32)25(29(38)35-26)15-19-3-10-23(11-4-19)37-14-2-13-34-37/h2-14,16-18,39H,15H2,1H3,(H,35,38)	SFTBOBKNJDXTPR-UHFFFAOYSA-N	220212	US9290476, 55A::US9290476, 55B::US9290476, 55C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 7600				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715667	329995330							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385388	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(O)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H23Cl2N5O2/c1-36-18-33-17-27(36)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(16-21)28(32)25(29(38)35-26)15-19-3-10-23(11-4-19)37-14-2-13-34-37/h2-14,16-18,39H,15H2,1H3,(H,35,38)	SFTBOBKNJDXTPR-UHFFFAOYSA-N	220212	US9290476, 55A::US9290476, 55B::US9290476, 55C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				>81000				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715667	329995330							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385389	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(O)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C30H23Cl2N5O2/c1-36-18-33-17-27(36)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(16-21)28(32)25(29(38)35-26)15-19-3-10-23(11-4-19)37-14-2-13-34-37/h2-14,16-18,39H,15H2,1H3,(H,35,38)	SFTBOBKNJDXTPR-UHFFFAOYSA-N	220212	US9290476, 55A::US9290476, 55B::US9290476, 55C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 3500				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715667	329995330							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385390	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1cncn1C	InChI=1S/C30H28ClN7O2/c1-19-12-21(30(39,25-15-32-17-36(25)2)26-16-33-18-37(26)3)14-23-27(31)24(29(40-4)35-28(19)23)13-20-6-8-22(9-7-20)38-11-5-10-34-38/h5-12,14-18,39H,13H2,1-4H3	JDQYMOPCYYLDBR-UHFFFAOYSA-N	220213	US9290476, 56	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.29				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220213&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220881	329995331							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385391	COc1nc2c(C)cc(cc2c(Cl)c1Cc1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1cncn1C	InChI=1S/C28H28ClN5O4S/c1-17-10-19(28(35,23-13-30-15-33(23)2)24-14-31-16-34(24)3)12-21-25(29)22(27(38-4)32-26(17)21)11-18-6-8-20(9-7-18)39(5,36)37/h6-10,12-16,35H,11H2,1-5H3	WXTGFUGCKDNKFL-UHFFFAOYSA-N	220214	US9290476, 57	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 8.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220214&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220882	329995332							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385392	COc1nc2c(F)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C31H23ClF4N6O2/c1-41-17-37-16-26(41)30(43,19-6-9-25(38-15-19)31(34,35)36)20-13-22-27(32)23(29(44-2)40-28(22)24(33)14-20)12-18-4-7-21(8-5-18)42-11-3-10-39-42/h3-11,13-17,43H,12H2,1-2H3	MEAKHLIUQZPPED-UHFFFAOYSA-N	220298	US9290476, 58B::US9290476, 58C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 14				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220298&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869579	329995357							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385393	COc1nc2c(F)cc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C31H23ClF4N6O2/c1-41-17-37-16-26(41)30(43,19-6-9-25(38-15-19)31(34,35)36)20-13-22-27(32)23(29(44-2)40-28(22)24(33)14-20)12-18-4-7-21(8-5-18)42-11-3-10-39-42/h3-11,13-17,43H,12H2,1-2H3	MEAKHLIUQZPPED-UHFFFAOYSA-N	220298	US9290476, 58B::US9290476, 58C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 270				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220298&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869579	329995357							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385394	COc1cc(cc2c(Cl)c(Cc3ccc(cc3)-n3cccn3)c(OC)nc12)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H26ClF3N6O3/c1-41-18-37-17-27(41)31(43,20-7-10-26(38-16-20)32(34,35)36)21-14-23-28(33)24(30(45-3)40-29(23)25(15-21)44-2)13-19-5-8-22(9-6-19)42-12-4-11-39-42/h4-12,14-18,43H,13H2,1-3H3	YZSPDKGJSASVGJ-UHFFFAOYSA-N	220300	US9290476, 59B::US9290476, 59C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220300&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220945	329995358							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385395	COc1cc(cc2c(Cl)c(Cc3ccc(cc3)-n3cccn3)c(OC)nc12)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H26ClF3N6O3/c1-41-18-37-17-27(41)31(43,20-7-10-26(38-16-20)32(34,35)36)21-14-23-28(33)24(30(45-3)40-29(23)25(15-21)44-2)13-19-5-8-22(9-6-19)42-12-4-11-39-42/h4-12,14-18,43H,13H2,1-3H3	YZSPDKGJSASVGJ-UHFFFAOYSA-N	220300	US9290476, 59B::US9290476, 59C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 220				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220300&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220945	329995358							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385396	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1cncn1C	InChI=1S/C32H33ClN6O3/c1-21(40)38-15-11-23(12-16-38)32(41,29-19-34-20-37(29)2)24-7-10-28-26(18-24)30(33)27(31(36-28)42-3)17-22-5-8-25(9-6-22)39-14-4-13-35-39/h4-10,13-14,18-20,23,41H,11-12,15-17H2,1-3H3	MAJOOHMQVBMIGI-UHFFFAOYSA-N	220217	US9290476, 60A::US9290476, 60B::US9290476, 60C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 18				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WD	5W4R	86715668	329995333							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385397	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1cncn1C	InChI=1S/C32H33ClN6O3/c1-21(40)38-15-11-23(12-16-38)32(41,29-19-34-20-37(29)2)24-7-10-28-26(18-24)30(33)27(31(36-28)42-3)17-22-5-8-25(9-6-22)39-14-4-13-35-39/h4-10,13-14,18-20,23,41H,11-12,15-17H2,1-3H3	MAJOOHMQVBMIGI-UHFFFAOYSA-N	220217	US9290476, 60A::US9290476, 60B::US9290476, 60C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 33				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WD	5W4R	86715668	329995333							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385398	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1cncn1C	InChI=1S/C32H33ClN6O3/c1-21(40)38-15-11-23(12-16-38)32(41,29-19-34-20-37(29)2)24-7-10-28-26(18-24)30(33)27(31(36-28)42-3)17-22-5-8-25(9-6-22)39-14-4-13-35-39/h4-10,13-14,18-20,23,41H,11-12,15-17H2,1-3H3	MAJOOHMQVBMIGI-UHFFFAOYSA-N	220217	US9290476, 60A::US9290476, 60B::US9290476, 60C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 20				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	9WD	5W4R	86715668	329995333							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385399	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cnnn1C)c1cnnn1C	InChI=1S/C27H24ClN9O2/c1-35-23(15-29-33-35)27(38,24-16-30-34-36(24)2)18-7-10-22-20(14-18)25(28)21(26(32-22)39-3)13-17-5-8-19(9-6-17)37-12-4-11-31-37/h4-12,14-16,38H,13H2,1-3H3	UWUFHIQABBLHMZ-UHFFFAOYSA-N	220218	US9290476, 61	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74220947	329995334							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385400	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C29H21ClF6N4O2/c1-40-15-37-14-24(40)27(41,19-8-10-23(38-13-19)29(34,35)36)18-7-9-22-20(12-18)25(30)21(26(39-22)42-2)11-16-3-5-17(6-4-16)28(31,32)33/h3-10,12-15,41H,11H2,1-2H3	YKOCDXNRGRBHBI-UHFFFAOYSA-N	220219	US9290476, 62A::US9290476, 62B::US9290476, 62C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 9.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221008	329995335							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385401	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C29H21ClF6N4O2/c1-40-15-37-14-24(40)27(41,19-8-10-23(38-13-19)29(34,35)36)18-7-9-22-20(12-18)25(30)21(26(39-22)42-2)11-16-3-5-17(6-4-16)28(31,32)33/h3-10,12-15,41H,11H2,1-2H3	YKOCDXNRGRBHBI-UHFFFAOYSA-N	220219	US9290476, 62A::US9290476, 62B::US9290476, 62C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 33				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221008	329995335							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385402	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C29H21ClF6N4O2/c1-40-15-37-14-24(40)27(41,19-8-10-23(38-13-19)29(34,35)36)18-7-9-22-20(12-18)25(30)21(26(39-22)42-2)11-16-3-5-17(6-4-16)28(31,32)33/h3-10,12-15,41H,11H2,1-2H3	YKOCDXNRGRBHBI-UHFFFAOYSA-N	220219	US9290476, 62A::US9290476, 62B::US9290476, 62C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221008	329995335							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385403	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C#N)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H22Cl2N4O2/c1-35-17-33-16-26(35)29(36,20-7-10-22(30)11-8-20)21-9-12-25-23(14-21)27(31)24(28(34-25)37-2)13-18-3-5-19(15-32)6-4-18/h3-12,14,16-17,36H,13H2,1-2H3	KSSJZMDSSDTJJP-UHFFFAOYSA-N	220220	US9290476, 63A::US9290476, 63B::US9290476, 63C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 37				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221009	329995336							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385404	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C#N)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H22Cl2N4O2/c1-35-17-33-16-26(35)29(36,20-7-10-22(30)11-8-20)21-9-12-25-23(14-21)27(31)24(28(34-25)37-2)13-18-3-5-19(15-32)6-4-18/h3-12,14,16-17,36H,13H2,1-2H3	KSSJZMDSSDTJJP-UHFFFAOYSA-N	220220	US9290476, 63A::US9290476, 63B::US9290476, 63C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 350				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221009	329995336							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385405	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C#N)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H22Cl2N4O2/c1-35-17-33-16-26(35)29(36,20-7-10-22(30)11-8-20)21-9-12-25-23(14-21)27(31)24(28(34-25)37-2)13-18-3-5-19(15-32)6-4-18/h3-12,14,16-17,36H,13H2,1-2H3	KSSJZMDSSDTJJP-UHFFFAOYSA-N	220220	US9290476, 63A::US9290476, 63B::US9290476, 63C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.2				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221009	329995336							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385406	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cncn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H24Cl2N6O2/c1-37-17-33-15-27(37)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(14-21)28(32)25(29(36-26)40-2)13-19-3-10-23(11-4-19)38-18-34-16-35-38/h3-12,14-18,39H,13H2,1-2H3	BCPPJFGMAGRVIG-UHFFFAOYSA-N	220221	US9290476, 64A::US9290476, 64B::US9290476, 64C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 63				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221010	329995337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385407	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cncn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H24Cl2N6O2/c1-37-17-33-15-27(37)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(14-21)28(32)25(29(36-26)40-2)13-19-3-10-23(11-4-19)38-18-34-16-35-38/h3-12,14-18,39H,13H2,1-2H3	BCPPJFGMAGRVIG-UHFFFAOYSA-N	220221	US9290476, 64A::US9290476, 64B::US9290476, 64C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 450				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221010	329995337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385408	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cncn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C30H24Cl2N6O2/c1-37-17-33-15-27(37)30(39,20-5-8-22(31)9-6-20)21-7-12-26-24(14-21)28(32)25(29(36-26)40-2)13-19-3-10-23(11-4-19)38-18-34-16-35-38/h3-12,14-18,39H,13H2,1-2H3	BCPPJFGMAGRVIG-UHFFFAOYSA-N	220221	US9290476, 64A::US9290476, 64B::US9290476, 64C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 16				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221010	329995337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385409	Cc1cc(cc2c(C#N)c(Cc3ccc(cc3)-n3cccn3)c(nc12)C#N)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C33H23F3N8O/c1-20-12-23(32(45,30-18-39-19-43(30)2)22-6-9-29(40-17-22)33(34,35)36)14-26-27(15-37)25(28(16-38)42-31(20)26)13-21-4-7-24(8-5-21)44-11-3-10-41-44/h3-12,14,17-19,45H,13H2,1-2H3	BPIQJYCCGCVYPU-UHFFFAOYSA-N	220310	US9290476, 65B::US9290476, 65C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 140				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220310	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220310&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117868755	329995359							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385410	Cc1cc(cc2c(C#N)c(Cc3ccc(cc3)-n3cccn3)c(nc12)C#N)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C33H23F3N8O/c1-20-12-23(32(45,30-18-39-19-43(30)2)22-6-9-29(40-17-22)33(34,35)36)14-26-27(15-37)25(28(16-38)42-31(20)26)13-21-4-7-24(8-5-21)44-11-3-10-41-44/h3-12,14,17-19,45H,13H2,1-2H3	BPIQJYCCGCVYPU-UHFFFAOYSA-N	220310	US9290476, 65B::US9290476, 65C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.2				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220310	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220310&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117868755	329995359							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385411	Cc1cc(cc2c(C#N)c(Cc3ccc(cc3)-n3cccn3)c(nc12)C#N)C(O)(c1cncn1C)c1ccc(cc1)C#N	InChI=1S/C34H24N8O/c1-22-14-26(34(43,32-20-38-21-41(32)2)25-8-4-24(17-35)5-9-25)16-29-30(18-36)28(31(19-37)40-33(22)29)15-23-6-10-27(11-7-23)42-13-3-12-39-42/h3-14,16,20-21,43H,15H2,1-2H3	PMHUAAAZNHFYTO-UHFFFAOYSA-N	220312	US9290476, 66B::US9290476, 66C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 270				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220312	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220312&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221012	329995360							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385412	Cc1cc(cc2c(C#N)c(Cc3ccc(cc3)-n3cccn3)c(nc12)C#N)C(O)(c1cncn1C)c1ccc(cc1)C#N	InChI=1S/C34H24N8O/c1-22-14-26(34(43,32-20-38-21-41(32)2)25-8-4-24(17-35)5-9-25)16-29-30(18-36)28(31(19-37)40-33(22)29)15-23-6-10-27(11-7-23)42-13-3-12-39-42/h3-14,16,20-21,43H,15H2,1-2H3	PMHUAAAZNHFYTO-UHFFFAOYSA-N	220312	US9290476, 66B::US9290476, 66C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 7.9				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220312	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220312&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221012	329995360							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385413	CON(C)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H27ClF3N7O2/c1-41-19-37-18-28(41)31(44,22-8-12-27(38-17-22)32(34,35)36)21-7-11-26-24(16-21)29(33)25(30(40-26)42(2)45-3)15-20-5-9-23(10-6-20)43-14-4-13-39-43/h4-14,16-19,44H,15H2,1-3H3	RKRDETFUPDVSLB-UHFFFAOYSA-N	220224	US9290476, 67A::US9290476, 67B::US9290476, 67C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 18				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220224&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221073	329995338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385414	CON(C)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H27ClF3N7O2/c1-41-19-37-18-28(41)31(44,22-8-12-27(38-17-22)32(34,35)36)21-7-11-26-24(16-21)29(33)25(30(40-26)42(2)45-3)15-20-5-9-23(10-6-20)43-14-4-13-39-43/h4-14,16-19,44H,15H2,1-3H3	RKRDETFUPDVSLB-UHFFFAOYSA-N	220224	US9290476, 67A::US9290476, 67B::US9290476, 67C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.3				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220224&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221073	329995338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385415	CON(C)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H27ClF3N7O2/c1-41-19-37-18-28(41)31(44,22-8-12-27(38-17-22)32(34,35)36)21-7-11-26-24(16-21)29(33)25(30(40-26)42(2)45-3)15-20-5-9-23(10-6-20)43-14-4-13-39-43/h4-14,16-19,44H,15H2,1-3H3	RKRDETFUPDVSLB-UHFFFAOYSA-N	220224	US9290476, 67A::US9290476, 67B::US9290476, 67C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 57				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220224&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221073	329995338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385416	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C33H27ClF3N7O/c1-42-20-38-19-29(42)32(45,23-7-11-28(39-18-23)33(35,36)37)22-6-10-27-25(17-22)30(34)26(31(41-27)43-13-3-14-43)16-21-4-8-24(9-5-21)44-15-2-12-40-44/h2,4-12,15,17-20,45H,3,13-14,16H2,1H3	WOJSAHWKHXGTSC-UHFFFAOYSA-N	220225	US9290476, 68A::US9290476, 68B::US9290476, 68C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 8.3				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221074	329995339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385417	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C33H27ClF3N7O/c1-42-20-38-19-29(42)32(45,23-7-11-28(39-18-23)33(35,36)37)22-6-10-27-25(17-22)30(34)26(31(41-27)43-13-3-14-43)16-21-4-8-24(9-5-21)44-15-2-12-40-44/h2,4-12,15,17-20,45H,3,13-14,16H2,1H3	WOJSAHWKHXGTSC-UHFFFAOYSA-N	220225	US9290476, 68A::US9290476, 68B::US9290476, 68C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.1				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221074	329995339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385418	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1	InChI=1S/C33H27ClF3N7O/c1-42-20-38-19-29(42)32(45,23-7-11-28(39-18-23)33(35,36)37)22-6-10-27-25(17-22)30(34)26(31(41-27)43-13-3-14-43)16-21-4-8-24(9-5-21)44-15-2-12-40-44/h2,4-12,15,17-20,45H,3,13-14,16H2,1H3	WOJSAHWKHXGTSC-UHFFFAOYSA-N	220225	US9290476, 68A::US9290476, 68B::US9290476, 68C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 30				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221074	329995339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385419	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C32H25ClN6O2/c1-38-20-35-19-30(38)32(40,22-6-9-24(33)10-7-22)23-8-13-29-26(17-23)28(18-34)27(31(37-29)41-2)16-21-4-11-25(12-5-21)39-15-3-14-36-39/h3-15,17,19-20,40H,16H2,1-2H3	VEARGWNSFNEBEE-UHFFFAOYSA-N	220226	US9290476, 69	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 50				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220226&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221075	329995340							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385420	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)cc2c1	InChI=1S/C31H22F3N7O/c1-40-19-36-18-29(40)30(42,24-6-10-28(37-17-24)31(32,33)34)23-5-9-26-22(15-23)14-21(27(16-35)39-26)13-20-3-7-25(8-4-20)41-12-2-11-38-41/h2-12,14-15,17-19,42H,13H2,1H3	WQJCGKMRMLYQHD-UHFFFAOYSA-N	220318	US9290476, 70B::US9290476, 70C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1100				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220318	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220318&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869754	329995361							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385421	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)cc2c1	InChI=1S/C31H22F3N7O/c1-40-19-36-18-29(40)30(42,24-6-10-28(37-17-24)31(32,33)34)23-5-9-26-22(15-23)14-21(27(16-35)39-26)13-20-3-7-25(8-4-20)41-12-2-11-38-41/h2-12,14-15,17-19,42H,13H2,1H3	WQJCGKMRMLYQHD-UHFFFAOYSA-N	220318	US9290476, 70B::US9290476, 70C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 16000				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220318	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220318&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869754	329995361							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385422	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)c(C#N)c2c1	InChI=1S/C32H22ClN7O/c1-39-20-36-19-31(39)32(41,22-5-8-24(33)9-6-22)23-7-12-29-27(16-23)28(17-34)26(30(18-35)38-29)15-21-3-10-25(11-4-21)40-14-2-13-37-40/h2-14,16,19-20,41H,15H2,1H3	PLTOQAMSCRJXOS-UHFFFAOYSA-N	220320	US9290476, 71B::US9290476, 71C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.6				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220320&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221136	329995362							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385423	Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)c(C#N)c2c1	InChI=1S/C32H22ClN7O/c1-39-20-36-19-31(39)32(41,22-5-8-24(33)9-6-22)23-7-12-29-27(16-23)28(17-34)26(30(18-35)38-29)15-21-3-10-25(11-4-21)40-14-2-13-37-40/h2-14,16,19-20,41H,15H2,1H3	PLTOQAMSCRJXOS-UHFFFAOYSA-N	220320	US9290476, 71B::US9290476, 71C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 130				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220320	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220320&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221136	329995362							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385424	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)c(C#N)c2c1	InChI=1S/C32H21F3N8O/c1-42-19-38-18-30(42)31(44,22-6-10-29(39-17-22)32(33,34)35)21-5-9-27-25(14-21)26(15-36)24(28(16-37)41-27)13-20-3-7-23(8-4-20)43-12-2-11-40-43/h2-12,14,17-19,44H,13H2,1H3	WHRLSFGQEUBSBY-UHFFFAOYSA-N	50058934	CHEMBL3325743::US9290476, 72C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.71				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50058934	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50058934&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117870010	103954836		CHEMBL3325743				ZINC03918823	1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385425	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)c(C#N)c2c1	InChI=1S/C32H21F3N8O/c1-42-19-38-18-30(42)31(44,22-6-10-29(39-17-22)32(33,34)35)21-5-9-27-25(14-21)26(15-36)24(28(16-37)41-27)13-20-3-7-23(8-4-20)43-12-2-11-40-43/h2-12,14,17-19,44H,13H2,1H3	WHRLSFGQEUBSBY-UHFFFAOYSA-N	50058934	CHEMBL3325743::US9290476, 72C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 7.1				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50058934	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50058934&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117870010	103954836		CHEMBL3325743				ZINC03918823	1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385426	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H24F3N7O2/c1-41-19-37-18-29(41)31(43,22-7-11-28(38-17-22)32(33,34)35)21-6-10-27-24(15-21)26(16-36)25(30(40-27)44-2)14-20-4-8-23(9-5-20)42-13-3-12-39-42/h3-13,15,17-19,43H,14H2,1-2H3	GSSYPDAFZTWCGW-UHFFFAOYSA-N	220322	US9290476, 73B::US9290476, 73C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220322&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869284	329995363							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385427	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C32H24F3N7O2/c1-41-19-37-18-29(41)31(43,22-7-11-28(38-17-22)32(33,34)35)21-6-10-27-24(15-21)26(16-36)25(30(40-27)44-2)14-20-4-8-23(9-5-20)42-13-3-12-39-42/h3-13,15,17-19,43H,14H2,1-2H3	GSSYPDAFZTWCGW-UHFFFAOYSA-N	220322	US9290476, 73B::US9290476, 73C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 34				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220322	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220322&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869284	329995363							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385428	CCN(CC)c1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C35H31F3N8O/c1-4-45(5-2)33-28(17-23-7-11-26(12-8-23)46-16-6-15-42-46)29(19-39)27-18-24(9-13-30(27)43-33)34(47,32-21-40-22-44(32)3)25-10-14-31(41-20-25)35(36,37)38/h6-16,18,20-22,47H,4-5,17H2,1-3H3	LAKFKZPLUGDRPT-UHFFFAOYSA-N	220324	US9290476, 74B::US9290476, 74C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1300				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220324&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221139	329995364							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385429	CCN(CC)c1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C35H31F3N8O/c1-4-45(5-2)33-28(17-23-7-11-26(12-8-23)46-16-6-15-42-46)29(19-39)27-18-24(9-13-30(27)43-33)34(47,32-21-40-22-44(32)3)25-10-14-31(41-20-25)35(36,37)38/h6-16,18,20-22,47H,4-5,17H2,1-3H3	LAKFKZPLUGDRPT-UHFFFAOYSA-N	220324	US9290476, 74B::US9290476, 74C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 21000				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220324	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220324&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221139	329995364							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385430	CCN(CC)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C34H32Cl2N6O/c1-4-41(5-2)33-29(19-23-7-14-27(15-8-23)42-18-6-17-38-42)32(36)28-20-25(11-16-30(28)39-33)34(43,31-21-37-22-40(31)3)24-9-12-26(35)13-10-24/h6-18,20-22,43H,4-5,19H2,1-3H3	OWZFUIWCUAGNIT-UHFFFAOYSA-N	220326	US9290476, 75B::US9290476, 75C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 8600				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220326&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221201	329995365							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385431	CCN(CC)c1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C34H32Cl2N6O/c1-4-41(5-2)33-29(19-23-7-14-27(15-8-23)42-18-6-17-38-42)32(36)28-20-25(11-16-30(28)39-33)34(43,31-21-37-22-40(31)3)24-9-12-26(35)13-10-24/h6-18,20-22,43H,4-5,19H2,1-3H3	OWZFUIWCUAGNIT-UHFFFAOYSA-N	220326	US9290476, 75B::US9290476, 75C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 150				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220326	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220326&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221201	329995365							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385432	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(cc1)[N+]#[C-]	InChI=1S/C33H25N7O2/c1-35-25-10-7-23(8-11-25)33(41,31-20-36-21-39(31)2)24-9-14-30-27(18-24)29(19-34)28(32(38-30)42-3)17-22-5-12-26(13-6-22)40-16-4-15-37-40/h4-16,18,20-21,41H,17H2,2-3H3	XXRVRLIGBBWOTK-UHFFFAOYSA-N	220328	US9290476, 76B::US9290476, 76C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 76				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220328&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123879658	329995366							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385433	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(cc1)[N+]#[C-]	InChI=1S/C33H25N7O2/c1-35-25-10-7-23(8-11-25)33(41,31-20-36-21-39(31)2)24-9-14-30-27(18-24)29(19-34)28(32(38-30)42-3)17-22-5-12-26(13-6-22)40-16-4-15-37-40/h4-16,18,20-21,41H,17H2,2-3H3	XXRVRLIGBBWOTK-UHFFFAOYSA-N	220328	US9290476, 76B::US9290476, 76C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 15				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220328	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220328&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123879658	329995366							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385434	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C29H25ClF3N5O2/c1-16-5-11-23(17(2)35-16)28(39,25-15-34-37-38(25)3)20-10-12-24-21(14-20)26(30)22(27(36-24)40-4)13-18-6-8-19(9-7-18)29(31,32)33/h5-12,14-15,39H,13H2,1-4H3	HVSWHSCHDKSPHW-UHFFFAOYSA-N	220233	US9290476, 77A::US9290476, 77B::US9290476, 77C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.1				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221202	329995341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385435	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C29H25ClF3N5O2/c1-16-5-11-23(17(2)35-16)28(39,25-15-34-37-38(25)3)20-10-12-24-21(14-20)26(30)22(27(36-24)40-4)13-18-6-8-19(9-7-18)29(31,32)33/h5-12,14-15,39H,13H2,1-4H3	HVSWHSCHDKSPHW-UHFFFAOYSA-N	220233	US9290476, 77A::US9290476, 77B::US9290476, 77C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 320				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221202	329995341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385436	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C29H25ClF3N5O2/c1-16-5-11-23(17(2)35-16)28(39,25-15-34-37-38(25)3)20-10-12-24-21(14-20)26(30)22(27(36-24)40-4)13-18-6-8-19(9-7-18)29(31,32)33/h5-12,14-15,39H,13H2,1-4H3	HVSWHSCHDKSPHW-UHFFFAOYSA-N	220233	US9290476, 77A::US9290476, 77B::US9290476, 77C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.14				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221202	329995341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385437	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C30H25F3N6O2/c1-17-5-11-25(18(2)36-17)29(40,27-16-35-38-39(27)3)21-10-12-26-22(14-21)24(15-34)23(28(37-26)41-4)13-19-6-8-20(9-7-19)30(31,32)33/h5-12,14,16,40H,13H2,1-4H3	ULPKMRDWGSOKMR-UHFFFAOYSA-N	220234	US9290476, 78A::US9290476, 78B::US9290476, 78C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.52				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715671	329995342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385438	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C30H25F3N6O2/c1-17-5-11-25(18(2)36-17)29(40,27-16-35-38-39(27)3)21-10-12-26-22(14-21)24(15-34)23(28(37-26)41-4)13-19-6-8-20(9-7-19)30(31,32)33/h5-12,14,16,40H,13H2,1-4H3	ULPKMRDWGSOKMR-UHFFFAOYSA-N	220234	US9290476, 78A::US9290476, 78B::US9290476, 78C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 120				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715671	329995342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385439	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C30H25F3N6O2/c1-17-5-11-25(18(2)36-17)29(40,27-16-35-38-39(27)3)21-10-12-26-22(14-21)24(15-34)23(28(37-26)41-4)13-19-6-8-20(9-7-19)30(31,32)33/h5-12,14,16,40H,13H2,1-4H3	ULPKMRDWGSOKMR-UHFFFAOYSA-N	220234	US9290476, 78A::US9290476, 78B::US9290476, 78C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.28				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			86715671	329995342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385440	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1sc(C)nc1C	InChI=1S/C27H23ClF3N5O2S/c1-14-24(39-15(2)33-14)26(37,22-13-32-35-36(22)3)18-9-10-21-19(12-18)23(28)20(25(34-21)38-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-13,37H,11H2,1-4H3	XWZQGKUMJPPPFZ-UHFFFAOYSA-N	50058935	CHEMBL3358455::US9290476, 79C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 57				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50058935	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50058935&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221204	103954837		CHEMBL3358455				ZINC34633720	1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385441	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1sc(C)nc1C	InChI=1S/C27H23ClF3N5O2S/c1-14-24(39-15(2)33-14)26(37,22-13-32-35-36(22)3)18-9-10-21-19(12-18)23(28)20(25(34-21)38-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-13,37H,11H2,1-4H3	XWZQGKUMJPPPFZ-UHFFFAOYSA-N	50058935	CHEMBL3358455::US9290476, 79C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.024				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50058935	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50058935&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221204	103954837		CHEMBL3358455				ZINC34633720	1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385442	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C27H24ClF3N6O2/c1-15-32-13-22(36(15)2)26(38,23-14-33-35-37(23)3)18-9-10-21-19(12-18)24(28)20(25(34-21)39-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-14,38H,11H2,1-4H3	GPIRADWERUVWAO-UHFFFAOYSA-N	220235	US9290476, 80A::US9290476, 80B::US9290476, 80C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.14				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221264	329995343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385443	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C27H24ClF3N6O2/c1-15-32-13-22(36(15)2)26(38,23-14-33-35-37(23)3)18-9-10-21-19(12-18)24(28)20(25(34-21)39-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-14,38H,11H2,1-4H3	GPIRADWERUVWAO-UHFFFAOYSA-N	220235	US9290476, 80A::US9290476, 80B::US9290476, 80C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.11				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221264	329995343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385444	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C27H24ClF3N6O2/c1-15-32-13-22(36(15)2)26(38,23-14-33-35-37(23)3)18-9-10-21-19(12-18)24(28)20(25(34-21)39-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-14,38H,11H2,1-4H3	GPIRADWERUVWAO-UHFFFAOYSA-N	220235	US9290476, 80A::US9290476, 80B::US9290476, 80C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.026				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221264	329995343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385445	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C28H24F3N7O2/c1-16-33-14-24(37(16)2)27(39,25-15-34-36-38(25)3)19-9-10-23-20(12-19)22(13-32)21(26(35-23)40-4)11-17-5-7-18(8-6-17)28(29,30)31/h5-10,12,14-15,39H,11H2,1-4H3	NDGQZEJMZFDFKZ-UHFFFAOYSA-N	220236	US9290476, 81A::US9290476, 81B::US9290476, 81C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.12				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73442863	329995344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385446	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C28H24F3N7O2/c1-16-33-14-24(37(16)2)27(39,25-15-34-36-38(25)3)19-9-10-23-20(12-19)22(13-32)21(26(35-23)40-4)11-17-5-7-18(8-6-17)28(29,30)31/h5-10,12,14-15,39H,11H2,1-4H3	NDGQZEJMZFDFKZ-UHFFFAOYSA-N	220236	US9290476, 81A::US9290476, 81B::US9290476, 81C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.05				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73442863	329995344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385447	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C	InChI=1S/C28H24F3N7O2/c1-16-33-14-24(37(16)2)27(39,25-15-34-36-38(25)3)19-9-10-23-20(12-19)22(13-32)21(26(35-23)40-4)11-17-5-7-18(8-6-17)28(29,30)31/h5-10,12,14-15,39H,11H2,1-4H3	NDGQZEJMZFDFKZ-UHFFFAOYSA-N	220236	US9290476, 81A::US9290476, 81B::US9290476, 81C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.12				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73442863	329995344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385448	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1oc(C)nc1C	InChI=1S/C27H23ClF3N5O3/c1-14-24(39-15(2)33-14)26(37,22-13-32-35-36(22)3)18-9-10-21-19(12-18)23(28)20(25(34-21)38-4)11-16-5-7-17(8-6-16)27(29,30)31/h5-10,12-13,37H,11H2,1-4H3	KBUXIDBMMOYBNJ-UHFFFAOYSA-N	220237	US9290476, 82	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.63				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220237&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221466	329995345							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385449	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1	InChI=1S/C34H33ClN4O3/c1-23(40)38-19-15-26(16-20-38)34(41,25-7-4-3-5-8-25)27-11-14-31-29(22-27)32(35)30(33(37-31)42-2)21-24-9-12-28(13-10-24)39-18-6-17-36-39/h3-14,17-18,22,26,41H,15-16,19-21H2,1-2H3	QBIGUDRHHJTXKG-UHFFFAOYSA-N	220238	US9290476, 83A::US9290476, 83B::US9290476, 83C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 12				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220238&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221465	329995346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385450	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1	InChI=1S/C34H33ClN4O3/c1-23(40)38-19-15-26(16-20-38)34(41,25-7-4-3-5-8-25)27-11-14-31-29(22-27)32(35)30(33(37-31)42-2)21-24-9-12-28(13-10-24)39-18-6-17-36-39/h3-14,17-18,22,26,41H,15-16,19-21H2,1-2H3	QBIGUDRHHJTXKG-UHFFFAOYSA-N	220238	US9290476, 83A::US9290476, 83B::US9290476, 83C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 4.7				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220238&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221465	329995346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385451	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1	InChI=1S/C34H33ClN4O3/c1-23(40)38-19-15-26(16-20-38)34(41,25-7-4-3-5-8-25)27-11-14-31-29(22-27)32(35)30(33(37-31)42-2)21-24-9-12-28(13-10-24)39-18-6-17-36-39/h3-14,17-18,22,26,41H,15-16,19-21H2,1-2H3	QBIGUDRHHJTXKG-UHFFFAOYSA-N	220238	US9290476, 83A::US9290476, 83B::US9290476, 83C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 77				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220238&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221465	329995346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385452	Cc1cc(cc2c(Cl)c(Cc3ccc(cc3)-n3cccn3)c(Cl)nc12)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C31H24Cl3N5O/c1-19-14-22(31(40,27-17-35-18-38(27)2)21-6-8-23(32)9-7-21)16-25-28(33)26(30(34)37-29(19)25)15-20-4-10-24(11-5-20)39-13-3-12-36-39/h3-14,16-18,40H,15H2,1-2H3	KARDQPKYJHATDW-UHFFFAOYSA-N	220184	US9290476, 27::US9290476, 85	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 85				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220184	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220184&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221529	329995303							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385453	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(N)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C29H26ClF3N6O/c1-16-5-11-23(17(2)36-16)28(34,25-15-35-38-39(25)3)20-10-12-24-21(14-20)26(30)22(27(37-24)40-4)13-18-6-8-19(9-7-18)29(31,32)33/h5-12,14-15H,13,34H2,1-4H3	LGFQVTOJZNKMSP-UHFFFAOYSA-N	220340	US9290476, 87B::US9290476, 87C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2300				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220340&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221397	329995367							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385454	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(N)(c1cnnn1C)c1ccc(C)nc1C	InChI=1S/C29H26ClF3N6O/c1-16-5-11-23(17(2)36-16)28(34,25-15-35-38-39(25)3)20-10-12-24-21(14-20)26(30)22(27(37-24)40-4)13-18-6-8-19(9-7-18)29(31,32)33/h5-12,14-15H,13,34H2,1-4H3	LGFQVTOJZNKMSP-UHFFFAOYSA-N	220340	US9290476, 87B::US9290476, 87C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.3				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220340&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221397	329995367							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385455	Cc1ccc(c(C)n1)C(O)(c1cnnn1C)c1ccc2nc(C#N)c(Cc3ccc(cc3)C(F)(F)F)c(C#N)c2c1	InChI=1S/C30H22F3N7O/c1-17-4-10-25(18(2)37-17)29(41,28-16-36-39-40(28)3)21-9-11-26-23(13-21)24(14-34)22(27(15-35)38-26)12-19-5-7-20(8-6-19)30(31,32)33/h4-11,13,16,41H,12H2,1-3H3	UTHVPEXNFLOKBS-UHFFFAOYSA-N	220342	US9290476, 88B::US9290476, 88C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 29				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220342&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869378	329995368							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385456	Cc1ccc(c(C)n1)C(O)(c1cnnn1C)c1ccc2nc(C#N)c(Cc3ccc(cc3)C(F)(F)F)c(C#N)c2c1	InChI=1S/C30H22F3N7O/c1-17-4-10-25(18(2)37-17)29(41,28-16-36-39-40(28)3)21-9-11-26-23(13-21)24(14-34)22(27(15-35)38-26)12-19-5-7-20(8-6-19)30(31,32)33/h4-11,13,16,41H,12H2,1-3H3	UTHVPEXNFLOKBS-UHFFFAOYSA-N	220342	US9290476, 88B::US9290476, 88C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.04				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220342&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			117869378	329995368							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385457	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(=O)OC(C)(C)C)c1cnnn1C	InChI=1S/C31H33ClF3N5O3/c1-6-24-22(13-18-7-9-19(10-8-18)31(33,34)35)27(32)23-14-20(11-12-25(23)37-24)30(42,26-15-36-38-39(26)5)21-16-40(17-21)28(41)43-29(2,3)4/h7-12,14-15,21,42H,6,13,16-17H2,1-5H3	BSGJTFNOQZUTJX-UHFFFAOYSA-N	220244	US9290476, 89	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.77				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220244&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221334	329995347							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385458	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C28H27ClF3N5O2/c1-4-23-21(11-17-5-7-18(8-6-17)28(30,31)32)26(29)22-12-19(9-10-24(22)34-23)27(39,25-13-33-35-36(25)3)20-14-37(15-20)16(2)38/h5-10,12-13,20,39H,4,11,14-15H2,1-3H3	MYGPDLVYCIXIBI-UHFFFAOYSA-N	220245	US9290476, 90A::US9290476, 90B::US9290476, 90C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.44				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221333	329995348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385459	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C28H27ClF3N5O2/c1-4-23-21(11-17-5-7-18(8-6-17)28(30,31)32)26(29)22-12-19(9-10-24(22)34-23)27(39,25-13-33-35-36(25)3)20-14-37(15-20)16(2)38/h5-10,12-13,20,39H,4,11,14-15H2,1-3H3	MYGPDLVYCIXIBI-UHFFFAOYSA-N	220245	US9290476, 90A::US9290476, 90B::US9290476, 90C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.56				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221333	329995348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385460	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C28H27ClF3N5O2/c1-4-23-21(11-17-5-7-18(8-6-17)28(30,31)32)26(29)22-12-19(9-10-24(22)34-23)27(39,25-13-33-35-36(25)3)20-14-37(15-20)16(2)38/h5-10,12-13,20,39H,4,11,14-15H2,1-3H3	MYGPDLVYCIXIBI-UHFFFAOYSA-N	220245	US9290476, 90A::US9290476, 90B::US9290476, 90C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.32				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221333	329995348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385461	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)S(C)(=O)=O)c1cnnn1C	InChI=1S/C27H27ClF3N5O3S/c1-4-22-20(11-16-5-7-17(8-6-16)27(29,30)31)25(28)21-12-18(9-10-23(21)33-22)26(37,24-13-32-34-35(24)2)19-14-36(15-19)40(3,38)39/h5-10,12-13,19,37H,4,11,14-15H2,1-3H3	MUXPDVKFLJRDSN-UHFFFAOYSA-N	220246	US9290476, 91A::US9290476, 91B::US9290476, 91C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.25				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221332	329995349							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385462	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)S(C)(=O)=O)c1cnnn1C	InChI=1S/C27H27ClF3N5O3S/c1-4-22-20(11-16-5-7-17(8-6-16)27(29,30)31)25(28)21-12-18(9-10-23(21)33-22)26(37,24-13-32-34-35(24)2)19-14-36(15-19)40(3,38)39/h5-10,12-13,19,37H,4,11,14-15H2,1-3H3	MUXPDVKFLJRDSN-UHFFFAOYSA-N	220246	US9290476, 91A::US9290476, 91B::US9290476, 91C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.1				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221332	329995349							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385463	CCc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)S(C)(=O)=O)c1cnnn1C	InChI=1S/C27H27ClF3N5O3S/c1-4-22-20(11-16-5-7-17(8-6-16)27(29,30)31)25(28)21-12-18(9-10-23(21)33-22)26(37,24-13-32-34-35(24)2)19-14-36(15-19)40(3,38)39/h5-10,12-13,19,37H,4,11,14-15H2,1-3H3	MUXPDVKFLJRDSN-UHFFFAOYSA-N	220246	US9290476, 91A::US9290476, 91B::US9290476, 91C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.23				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221332	329995349							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385464	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)C(F)(F)F)c(Cl)c2c1	InChI=1S/C31H24ClF6N5O/c1-42-17-39-16-26(42)29(44,21-8-10-25(40-15-21)31(36,37)38)20-7-9-24-22(14-20)27(32)23(28(41-24)43-11-2-12-43)13-18-3-5-19(6-4-18)30(33,34)35/h3-10,14-17,44H,2,11-13H2,1H3	WWSUFOUIFRLOTO-UHFFFAOYSA-N	220247	US9290476, 92A::US9290476, 92B::US9290476, 92C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221331	329995350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385465	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)C(F)(F)F)c(Cl)c2c1	InChI=1S/C31H24ClF6N5O/c1-42-17-39-16-26(42)29(44,21-8-10-25(40-15-21)31(36,37)38)20-7-9-24-22(14-20)27(32)23(28(41-24)43-11-2-12-43)13-18-3-5-19(6-4-18)30(33,34)35/h3-10,14-17,44H,2,11-13H2,1H3	WWSUFOUIFRLOTO-UHFFFAOYSA-N	220247	US9290476, 92A::US9290476, 92B::US9290476, 92C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 12				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221331	329995350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385466	Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(Cc3ccc(cc3)C(F)(F)F)c(Cl)c2c1	InChI=1S/C31H24ClF6N5O/c1-42-17-39-16-26(42)29(44,21-8-10-25(40-15-21)31(36,37)38)20-7-9-24-22(14-20)27(32)23(28(41-24)43-11-2-12-43)13-18-3-5-19(6-4-18)30(33,34)35/h3-10,14-17,44H,2,11-13H2,1H3	WWSUFOUIFRLOTO-UHFFFAOYSA-N	220247	US9290476, 92A::US9290476, 92B::US9290476, 92C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221331	329995350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385467	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C	InChI=1S/C29H27ClF3N5O2/c1-16-34-14-24(37(16)3)28(39,25-15-35-17(2)38(25)4)20-10-11-23-21(13-20)26(30)22(27(36-23)40-5)12-18-6-8-19(9-7-18)29(31,32)33/h6-11,13-15,39H,12H2,1-5H3	ABUOQYHVERJAKF-UHFFFAOYSA-N	220248	US9290476, 93	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.017				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220248&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221330	329995351							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385468	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(nc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C28H20ClF6N5O2/c1-40-14-36-13-23(40)26(41,17-5-8-22(38-12-17)28(33,34)35)16-4-6-20-18(10-16)24(29)19(25(39-20)42-2)9-15-3-7-21(37-11-15)27(30,31)32/h3-8,10-14,41H,9H2,1-2H3	RTUAJPWIBYTPMS-UHFFFAOYSA-N	220249	US9290476, 94A::US9290476, 94B::US9290476, 94C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 12				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221268	329995352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385469	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(nc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C28H20ClF6N5O2/c1-40-14-36-13-23(40)26(41,17-5-8-22(38-12-17)28(33,34)35)16-4-6-20-18(10-16)24(29)19(25(39-20)42-2)9-15-3-7-21(37-11-15)27(30,31)32/h3-8,10-14,41H,9H2,1-2H3	RTUAJPWIBYTPMS-UHFFFAOYSA-N	220249	US9290476, 94A::US9290476, 94B::US9290476, 94C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 98				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221268	329995352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385470	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(nc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F	InChI=1S/C28H20ClF6N5O2/c1-40-14-36-13-23(40)26(41,17-5-8-22(38-12-17)28(33,34)35)16-4-6-20-18(10-16)24(29)19(25(39-20)42-2)9-15-3-7-21(37-11-15)27(30,31)32/h3-8,10-14,41H,9H2,1-2H3	RTUAJPWIBYTPMS-UHFFFAOYSA-N	220249	US9290476, 94A::US9290476, 94B::US9290476, 94C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 6.5				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221268	329995352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385471	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(Cl)cc1	InChI=1S/C29H22Cl2F3N3O2/c1-37-16-35-15-25(37)28(38,18-7-10-21(30)11-8-18)20-9-12-24-22(14-20)26(31)23(27(36-24)39-2)13-17-3-5-19(6-4-17)29(32,33)34/h3-12,14-16,38H,13H2,1-2H3	KCRUKFRIJDAXFC-UHFFFAOYSA-N	220250	US9290476, 95	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 18				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220250&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221267	329995353							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385472	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(cc1)C#N	InChI=1S/C31H22F3N5O2/c1-39-18-37-17-28(39)30(40,21-7-5-20(15-35)6-8-21)23-11-12-27-24(14-23)26(16-36)25(29(38-27)41-2)13-19-3-9-22(10-4-19)31(32,33)34/h3-12,14,17-18,40H,13H2,1-2H3	OLPSSDGMICICNG-UHFFFAOYSA-N	220251	US9290476, 96A::US9290476, 96B::US9290476, 96C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.9				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220251&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221266	329995354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385473	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(cc1)C#N	InChI=1S/C31H22F3N5O2/c1-39-18-37-17-28(39)30(40,21-7-5-20(15-35)6-8-21)23-11-12-27-24(14-23)26(16-36)25(29(38-27)41-2)13-19-3-9-22(10-4-19)31(32,33)34/h3-12,14,17-18,40H,13H2,1-2H3	OLPSSDGMICICNG-UHFFFAOYSA-N	220251	US9290476, 96A::US9290476, 96B::US9290476, 96C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 48				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220251&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221266	329995354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385474	COc1nc2ccc(cc2c(C#N)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(cc1)C#N	InChI=1S/C31H22F3N5O2/c1-39-18-37-17-28(39)30(40,21-7-5-20(15-35)6-8-21)23-11-12-27-24(14-23)26(16-36)25(29(38-27)41-2)13-19-3-9-22(10-4-19)31(32,33)34/h3-12,14,17-18,40H,13H2,1-2H3	OLPSSDGMICICNG-UHFFFAOYSA-N	220251	US9290476, 96A::US9290476, 96B::US9290476, 96C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 2.2				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220251	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220251&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221266	329995354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385475	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C27H25ClF3N5O3/c1-15(37)36-13-19(14-36)26(38,23-12-32-34-35(23)2)18-8-9-22-20(11-18)24(28)21(25(33-22)39-3)10-16-4-6-17(7-5-16)27(29,30)31/h4-9,11-12,19,38H,10,13-14H2,1-3H3	WTWRESCNHUYFQH-UHFFFAOYSA-N	220252	US9290476, 97A::US9290476, 97B::US9290476, 97C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221265	329995355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385476	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C27H25ClF3N5O3/c1-15(37)36-13-19(14-36)26(38,23-12-32-34-35(23)2)18-8-9-22-20(11-18)24(28)21(25(33-22)39-3)10-16-4-6-17(7-5-16)27(29,30)31/h4-9,11-12,19,38H,10,13-14H2,1-3H3	WTWRESCNHUYFQH-UHFFFAOYSA-N	220252	US9290476, 97A::US9290476, 97B::US9290476, 97C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 1.4				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221265	329995355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
385477	COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C	InChI=1S/C27H25ClF3N5O3/c1-15(37)36-13-19(14-36)26(38,23-12-32-34-35(23)2)18-8-9-22-20(11-18)24(28)21(25(33-22)39-3)10-16-4-6-17(7-5-16)27(29,30)31/h4-9,11-12,19,38H,10,13-14H2,1-3H3	WTWRESCNHUYFQH-UHFFFAOYSA-N	220252	US9290476, 97A::US9290476, 97B::US9290476, 97C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)				 0.64				7	1.00 C	US Patent		10.7270/Q2M61J3M		aid1802530	US9290476	Leonard, KA; Barbay, K; Edwards, JP; Kreutter, KD; Kummer, DA; Maharoof, U; Nishimura, R; Urbanski, M; Venkatesan, H; Wang, A; Wolin, RL; Woods, CR; Pierce, J; Goldberg, S; Fourie, A; Xue, X	Janssen Pharmaceutica NV	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			74221265	329995355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446759	CN(C)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C25H21ClF3N3O4/c1-31(2)22(33)15-10-11-16-19(12-15)32(30-21(16)13-6-8-14(9-7-13)24(35)36)23(34)20-17(25(27,28)29)4-3-5-18(20)26/h3-6,10-12,14H,7-9H2,1-2H3,(H,35,36)	YGFLUSDKSFGRBP-UHFFFAOYSA-N	256337	US9487490, 1A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 18					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256337	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256337&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293430	347916139							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446760	CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O	InChI=1S/C23H17ClF4N2O3/c1-22(21(32)33)10-8-12(9-11-22)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-8H,9-11H2,1H3,(H,32,33)	ICXVPFPYYBKMTL-UHFFFAOYSA-N	256338	US9487490, 1B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 21					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256338	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256338&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	4Y6	5C4T	118219039	347916140							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446761	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H15ClF4N2O3/c23-14-4-1-3-13(22(25,26)27)17(14)20(30)29-16-6-2-5-15(24)18(16)19(28-29)11-7-9-12(10-8-11)21(31)32/h1-7,12H,8-10H2,(H,31,32)	JAWOLYIAGCXUQG-UHFFFAOYSA-N	256339	US9487490, 1C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 13					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256339&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293431	347916141							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446762	OCCNC(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C25H21ClF3N3O5/c26-18-3-1-2-17(25(27,28)29)20(18)23(35)32-19-12-15(22(34)30-10-11-33)8-9-16(19)21(31-32)13-4-6-14(7-5-13)24(36)37/h1-4,8-9,12,14,33H,5-7,10-11H2,(H,30,34)(H,36,37)	FHYRSAPXHJHYJO-UHFFFAOYSA-N	256340	US9487490, 1D	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 774					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256340	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256340&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293432	347916142					C04080		1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446763	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12	InChI=1S/C21H15ClF3N3O3/c22-14-4-1-3-13(21(23,24)25)16(14)19(29)28-15-5-2-10-26-18(15)17(27-28)11-6-8-12(9-7-11)20(30)31/h1-6,10,12H,7-9H2,(H,30,31)	PSTVSHJRDIVFDL-UHFFFAOYSA-N	256341	US9487490, 1E	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 76					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256341	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256341&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293433	347916143							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446764	CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12)C(O)=O	InChI=1S/C22H17ClF3N3O3/c1-21(20(31)32)9-7-12(8-10-21)17-18-15(6-3-11-27-18)29(28-17)19(30)16-13(22(24,25)26)4-2-5-14(16)23/h2-7,11H,8-10H2,1H3,(H,31,32)	SRNRFQGJGFHEGN-UHFFFAOYSA-N	256342	US9487490, 1F	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 170					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256342	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256342&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293600	347916144							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446765	CC1C=C(CCC1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12	InChI=1S/C22H17ClF3N3O3/c1-11-10-12(7-8-13(11)21(31)32)18-19-16(6-3-9-27-19)29(28-18)20(30)17-14(22(24,25)26)4-2-5-15(17)23/h2-6,9-11,13H,7-8H2,1H3,(H,31,32)	RPNORSIVSACOLA-UHFFFAOYSA-N	256343	US9487490, 1G	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 182					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256343	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256343&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293601	347916145							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446766	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12	InChI=1S/C22H16ClF3N2O3/c23-16-6-3-5-15(22(24,25)26)18(16)20(29)28-17-7-2-1-4-14(17)19(27-28)12-8-10-13(11-9-12)21(30)31/h1-8,13H,9-11H2,(H,30,31)	WAZYMFVBHLCPOF-UHFFFAOYSA-N	256344	US9487490, 1H	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256344	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256344&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73293602	347916146							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446767	CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(Cl)c12)C(O)=O	InChI=1S/C23H17Cl2F3N2O3/c1-22(21(32)33)10-8-12(9-11-22)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-8H,9-11H2,1H3,(H,32,33)	OYBATLGLEZTBDT-UHFFFAOYSA-N	256345	US9487490, 1I	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 14					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256345	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256345&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387702	347916147							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446768	CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12)C(O)=O	InChI=1S/C25H22ClFN2O3/c1-25(24(31)32)12-10-15(11-13-25)22-21-18(27)6-3-7-19(21)29(28-22)23(30)20-16(14-8-9-14)4-2-5-17(20)26/h2-7,10,14H,8-9,11-13H2,1H3,(H,31,32)	VOVNWNVFKASLLY-UHFFFAOYSA-N	256346	US9487490, 1J	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256346	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256346&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387703	347916148							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446769	Cc1cccc(Cl)c1C(=O)n1nc(C2=CCC(CC2)C(O)=O)c2c(F)cccc12	InChI=1S/C22H18ClFN2O3/c1-12-4-2-5-15(23)18(12)21(27)26-17-7-3-6-16(24)19(17)20(25-26)13-8-10-14(11-9-13)22(28)29/h2-8,14H,9-11H2,1H3,(H,28,29)	FTKZZUUQKBDHIQ-UHFFFAOYSA-N	256347	US9487490, 1K	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256347&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387704	347916149							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446770	Cc1cccc(Cl)c1C(=O)n1nc(C2=CCC(CC2)C(O)=O)c2ncccc12	InChI=1S/C21H18ClN3O3/c1-12-4-2-5-15(22)17(12)20(26)25-16-6-3-11-23-19(16)18(24-25)13-7-9-14(10-8-13)21(27)28/h2-7,11,14H,8-10H2,1H3,(H,27,28)	WGVKQEUIMVZKMX-UHFFFAOYSA-N	256348	US9487490, 1L	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 123					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256348	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256348&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387705	347916150							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446771	COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2c1)C1=CC[C@@H](CC1)C(O)=O	InChI=1S/C29H28ClN3O5/c1-38-20-14-32(15-20)27(34)19-11-12-22-24(13-19)33(31-26(22)17-7-9-18(10-8-17)29(36)37)28(35)25-21(16-5-6-16)3-2-4-23(25)30/h2-4,7,11-13,16,18,20H,5-6,8-10,14-15H2,1H3,(H,36,37)/t18-/m0/s1	LELXANQYKFVMDB-SFHVURJKSA-N	256349	US9487490, 2A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256349	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256349&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90041564	347916151							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446772	COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2c1)C1=CC[C@H](CC1)C(O)=O	InChI=1S/C29H28ClN3O5/c1-38-20-14-32(15-20)27(34)19-11-12-22-24(13-19)33(31-26(22)17-7-9-18(10-8-17)29(36)37)28(35)25-21(16-5-6-16)3-2-4-23(25)30/h2-4,7,11-13,16,18,20H,5-6,8-10,14-15H2,1H3,(H,36,37)/t18-/m1/s1	LELXANQYKFVMDB-GOSISDBHSA-N	256393	US9487490, 2B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256393	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256393&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90041798	347916195							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446773	COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2c1)C1=CC[C@@](C)(CC1)C(O)=O	InChI=1S/C30H30ClN3O5/c1-30(29(37)38)12-10-18(11-13-30)26-22-9-8-19(27(35)33-15-20(16-33)39-2)14-24(22)34(32-26)28(36)25-21(17-6-7-17)4-3-5-23(25)31/h3-5,8-10,14,17,20H,6-7,11-13,15-16H2,1-2H3,(H,37,38)/t30-/m0/s1	AQIMDWJRLMBKSY-PMERELPUSA-N	256350	US9487490, 2C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 4					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256350	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256350&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118208423	347916152							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446774	COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2c1)C1=CC[C@](C)(CC1)C(O)=O	InChI=1S/C30H30ClN3O5/c1-30(29(37)38)12-10-18(11-13-30)26-22-9-8-19(27(35)33-15-20(16-33)39-2)14-24(22)34(32-26)28(36)25-21(17-6-7-17)4-3-5-23(25)31/h3-5,8-10,14,17,20H,6-7,11-13,15-16H2,1-2H3,(H,37,38)/t30-/m1/s1	AQIMDWJRLMBKSY-SSEXGKCCSA-N	256351	US9487490, 2D	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256351	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256351&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118208424	347916153							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446775	OC(=O)[C@@H]1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12	InChI=1S/C24H20ClFN2O3/c25-17-4-1-3-16(13-7-8-13)20(17)23(29)28-19-6-2-5-18(26)21(19)22(27-28)14-9-11-15(12-10-14)24(30)31/h1-6,9,13,15H,7-8,10-12H2,(H,30,31)/t15-/m0/s1	SEEZLBPQMXZWAU-HNNXBMFYSA-N	256394	US9487490, 3A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256394&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387707	347916196							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446776	OC(=O)[C@H]1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12	InChI=1S/C24H20ClFN2O3/c25-17-4-1-3-16(13-7-8-13)20(17)23(29)28-19-6-2-5-18(26)21(19)22(27-28)14-9-11-15(12-10-14)24(30)31/h1-6,9,13,15H,7-8,10-12H2,(H,30,31)/t15-/m1/s1	SEEZLBPQMXZWAU-OAHLLOKOSA-N	256352	US9487490, 3B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256352&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387824	347916154							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446777	CC(C)(C)OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CC(F)(F)C1	InChI=1S/C30H27ClF5N3O4/c1-28(2,3)43-27(42)17-9-7-16(8-10-17)24-19-12-11-18(25(40)38-14-29(32,33)15-38)13-22(19)39(37-24)26(41)23-20(30(34,35)36)5-4-6-21(23)31/h4-7,11-13,17H,8-10,14-15H2,1-3H3	UEMQXWXIUURCHG-UHFFFAOYSA-N	256353	US9487490, 4A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256353	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256353&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118219044	347916155							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446778	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)NC1CC1	InChI=1S/C26H21ClF3N3O4/c27-19-3-1-2-18(26(28,29)30)21(19)24(35)33-20-12-15(23(34)31-16-9-10-16)8-11-17(20)22(32-33)13-4-6-14(7-5-13)25(36)37/h1-4,8,11-12,14,16H,5-7,9-10H2,(H,31,34)(H,36,37)	GXTKLCIXWCBOHM-UHFFFAOYSA-N	256354	US9487490, 4B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 143					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256354	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256354&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387826	347916156							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446779	CN(C1CC1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C27H23ClF3N3O4/c1-33(17-10-11-17)24(35)16-9-12-18-21(13-16)34(32-23(18)14-5-7-15(8-6-14)26(37)38)25(36)22-19(27(29,30)31)3-2-4-20(22)28/h2-5,9,12-13,15,17H,6-8,10-11H2,1H3,(H,37,38)	ASIUHIHZWLCGSX-UHFFFAOYSA-N	256355	US9487490, 4C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 9					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256355	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256355&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387827	347916157							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446780	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CCC1	InChI=1S/C26H21ClF3N3O4/c27-19-4-1-3-18(26(28,29)30)21(19)24(35)33-20-13-16(23(34)32-11-2-12-32)9-10-17(20)22(31-33)14-5-7-15(8-6-14)25(36)37/h1,3-5,9-10,13,15H,2,6-8,11-12H2,(H,36,37)	MZQZGAYLGDXZIQ-UHFFFAOYSA-N	256356	US9487490, 4D	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 177					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256356	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256356&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387828	347916158							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446781	COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C27H23ClF3N3O5/c1-39-17-12-33(13-17)24(35)16-9-10-18-21(11-16)34(32-23(18)14-5-7-15(8-6-14)26(37)38)25(36)22-19(27(29,30)31)3-2-4-20(22)28/h2-5,9-11,15,17H,6-8,12-13H2,1H3,(H,37,38)	GMWBIQXNRGCABM-UHFFFAOYSA-N	256357	US9487490, 4E	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256357	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256357&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387921	347916159							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446782	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CCCC1	InChI=1S/C27H23ClF3N3O4/c28-20-5-3-4-19(27(29,30)31)22(20)25(36)34-21-14-17(24(35)33-12-1-2-13-33)10-11-18(21)23(32-34)15-6-8-16(9-7-15)26(37)38/h3-6,10-11,14,16H,1-2,7-9,12-13H2,(H,37,38)	VWMRDPIRRQMSDG-UHFFFAOYSA-N	256358	US9487490, 4F	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 30					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256358	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256358&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387922	347916160							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446783	C[C@H]1CCCN1C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O4/c1-15-4-3-13-34(15)25(36)18-11-12-19-22(14-18)35(33-24(19)16-7-9-17(10-8-16)27(38)39)26(37)23-20(28(30,31)32)5-2-6-21(23)29/h2,5-7,11-12,14-15,17H,3-4,8-10,13H2,1H3,(H,38,39)/t15-,17?/m0/s1	WJSVXRQXYZLGEV-MYJWUSKBSA-N	256359	US9487490, 4G	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256359	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256359&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387923	347916161							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446784	C[C@@H]1CCCN1C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O4/c1-15-4-3-13-34(15)25(36)18-11-12-19-22(14-18)35(33-24(19)16-7-9-17(10-8-16)27(38)39)26(37)23-20(28(30,31)32)5-2-6-21(23)29/h2,5-7,11-12,14-15,17H,3-4,8-10,13H2,1H3,(H,38,39)/t15-,17?/m1/s1	WJSVXRQXYZLGEV-LDCVWXEPSA-N	256360	US9487490, 4H	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 115					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256360	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256360&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387924	347916162							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446785	COC1CCN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-40-18-11-12-34(14-18)25(36)17-9-10-19-22(13-17)35(33-24(19)15-5-7-16(8-6-15)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,16,18H,6-8,11-12,14H2,1H3,(H,38,39)	YBBWSYMSKCZLKW-UHFFFAOYSA-N	256361	US9487490, 4I	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256361	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256361&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73387925	347916163							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446786	CC1CN(CCO1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-15-14-34(11-12-40-15)25(36)18-9-10-19-22(13-18)35(33-24(19)16-5-7-17(8-6-16)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,15,17H,6-8,11-12,14H2,1H3,(H,38,39)	DDQRUXMBXOJJAC-UHFFFAOYSA-N	256362	US9487490, 4J	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 24					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256362	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256362&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388023	347916164							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446787	CN(C1CCCCC1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C30H29ClF3N3O4/c1-36(20-6-3-2-4-7-20)27(38)19-14-15-21-24(16-19)37(35-26(21)17-10-12-18(13-11-17)29(40)41)28(39)25-22(30(32,33)34)8-5-9-23(25)31/h5,8-10,14-16,18,20H,2-4,6-7,11-13H2,1H3,(H,40,41)	JGZIIFIESMANPE-UHFFFAOYSA-N	256363	US9487490, 4K	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 94					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256363	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256363&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388024	347916165							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446788	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CCOCC1	InChI=1S/C27H23ClF3N3O5/c28-20-3-1-2-19(27(29,30)31)22(20)25(36)34-21-14-17(24(35)33-10-12-39-13-11-33)8-9-18(21)23(32-34)15-4-6-16(7-5-15)26(37)38/h1-4,8-9,14,16H,5-7,10-13H2,(H,37,38)	DSBPXNGBDIGBRF-UHFFFAOYSA-N	256364	US9487490, 4L	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 36					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256364	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256364&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388025	347916166							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446789	C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C29H27ClF3N3O5/c1-15-13-35(14-16(2)41-15)26(37)19-10-11-20-23(12-19)36(34-25(20)17-6-8-18(9-7-17)28(39)40)27(38)24-21(29(31,32)33)4-3-5-22(24)30/h3-6,10-12,15-16,18H,7-9,13-14H2,1-2H3,(H,39,40)/t15-,16+,18?	KRWYLIPIAGZVDR-BYICEURKSA-N	256365	US9487490, 4M	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 21					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256365	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256365&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388026	347916167							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446790	CN1CCN(CC1=O)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H24ClF3N4O5/c1-34-11-12-35(14-22(34)37)25(38)17-9-10-18-21(13-17)36(33-24(18)15-5-7-16(8-6-15)27(40)41)26(39)23-19(28(30,31)32)3-2-4-20(23)29/h2-5,9-10,13,16H,6-8,11-12,14H2,1H3,(H,40,41)	LQXRTKDPFNHPJT-UHFFFAOYSA-N	256366	US9487490, 4N	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256366	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256366&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388027	347916168							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446791	C[C@H]1COCCN1C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-15-14-40-12-11-34(15)25(36)18-9-10-19-22(13-18)35(33-24(19)16-5-7-17(8-6-16)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,15,17H,6-8,11-12,14H2,1H3,(H,38,39)/t15-,17?/m0/s1	WIWSXCVVUZWXLY-MYJWUSKBSA-N	256367	US9487490, 4O	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 308					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256367	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256367&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90041446	347916169							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446792	CN(C1CCOCC1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C29H27ClF3N3O5/c1-35(19-11-13-41-14-12-19)26(37)18-9-10-20-23(15-18)36(34-25(20)16-5-7-17(8-6-16)28(39)40)27(38)24-21(29(31,32)33)3-2-4-22(24)30/h2-5,9-10,15,17,19H,6-8,11-14H2,1H3,(H,39,40)	OOFHDBBONAVJJF-UHFFFAOYSA-N	256368	US9487490, 4P	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 41					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256368	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256368&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90041818	347916170							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446793	C[C@@H]1COCCN1C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-15-14-40-12-11-34(15)25(36)18-9-10-19-22(13-18)35(33-24(19)16-5-7-17(8-6-16)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,15,17H,6-8,11-12,14H2,1H3,(H,38,39)/t15-,17?/m1/s1	WIWSXCVVUZWXLY-LDCVWXEPSA-N	256369	US9487490, 4Q	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 380					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256369	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256369&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388133	347916171							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446794	C[C@H]1CN(CCO1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-15-14-34(11-12-40-15)25(36)18-9-10-19-22(13-18)35(33-24(19)16-5-7-17(8-6-16)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,15,17H,6-8,11-12,14H2,1H3,(H,38,39)/t15-,17?/m0/s1	DDQRUXMBXOJJAC-MYJWUSKBSA-N	256370	US9487490, 4R	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 21					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256370	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256370&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388134	347916172							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446795	CN(CCO)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C26H23ClF3N3O5/c1-32(11-12-34)23(35)16-9-10-17-20(13-16)33(31-22(17)14-5-7-15(8-6-14)25(37)38)24(36)21-18(26(28,29)30)3-2-4-19(21)27/h2-5,9-10,13,15,34H,6-8,11-12H2,1H3,(H,37,38)	RURBILVXTPQNGT-UHFFFAOYSA-N	256371	US9487490, 4S	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 40					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256371	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256371&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388135	347916173							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446796	CC(C)NC(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C26H23ClF3N3O4/c1-13(2)31-23(34)16-10-11-17-20(12-16)33(32-22(17)14-6-8-15(9-7-14)25(36)37)24(35)21-18(26(28,29)30)4-3-5-19(21)27/h3-6,10-13,15H,7-9H2,1-2H3,(H,31,34)(H,36,37)	GRJJMWMGYUSJAR-UHFFFAOYSA-N	256372	US9487490, 4T	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1116					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256372	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256372&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388136	347916174							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446797	CC(C)N(C)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C27H25ClF3N3O4/c1-14(2)33(3)24(35)17-11-12-18-21(13-17)34(32-23(18)15-7-9-16(10-8-15)26(37)38)25(36)22-19(27(29,30)31)5-4-6-20(22)28/h4-7,11-14,16H,8-10H2,1-3H3,(H,37,38)	MIVJIOPYWAUDFE-UHFFFAOYSA-N	256373	US9487490, 4U	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 164					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256373	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256373&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388137	347916175							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446798	COCCN(C)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C27H25ClF3N3O5/c1-33(12-13-39-2)24(35)17-10-11-18-21(14-17)34(32-23(18)15-6-8-16(9-7-15)26(37)38)25(36)22-19(27(29,30)31)4-3-5-20(22)28/h3-6,10-11,14,16H,7-9,12-13H2,1-2H3,(H,37,38)	PPTPDSALMTVJCV-UHFFFAOYSA-N	256374	US9487490, 4V	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256374	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256374&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388255	347916176							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446799	OC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C26H21ClF3N3O5/c27-19-3-1-2-18(26(28,29)30)21(19)24(36)33-20-10-15(23(35)32-11-16(34)12-32)8-9-17(20)22(31-33)13-4-6-14(7-5-13)25(37)38/h1-4,8-10,14,16,34H,5-7,11-12H2,(H,37,38)	QYKKDMJGDPIYER-UHFFFAOYSA-N	256375	US9487490, 4W	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256375	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256375&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388256	347916177							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446800	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CC(F)C1	InChI=1S/C26H20ClF4N3O4/c27-19-3-1-2-18(26(29,30)31)21(19)24(36)34-20-10-15(23(35)33-11-16(28)12-33)8-9-17(20)22(32-34)13-4-6-14(7-5-13)25(37)38/h1-4,8-10,14,16H,5-7,11-12H2,(H,37,38)	WYFJBTRWRCAZFU-UHFFFAOYSA-N	256376	US9487490, 4X	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256376	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256376&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388257	347916178							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446801	OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CCCCC1	InChI=1S/C28H25ClF3N3O4/c29-21-6-4-5-20(28(30,31)32)23(21)26(37)35-22-15-18(25(36)34-13-2-1-3-14-34)11-12-19(22)24(33-35)16-7-9-17(10-8-16)27(38)39/h4-7,11-12,15,17H,1-3,8-10,13-14H2,(H,38,39)	BOJKDICTPGZHJX-UHFFFAOYSA-N	256377	US9487490, 4Y	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 159					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256377	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256377&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388258	347916179							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446802	CNCC(CO)OC(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C27H25ClF3N3O6/c1-32-12-17(13-35)40-26(39)16-9-10-18-21(11-16)34(33-23(18)14-5-7-15(8-6-14)25(37)38)24(36)22-19(27(29,30)31)3-2-4-20(22)28/h2-5,9-11,15,17,32,35H,6-8,12-13H2,1H3,(H,37,38)	DBVPUALOJKWZOW-UHFFFAOYSA-N	256378	US9487490, 4Z	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 258					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256378	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256378&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388259	347916180							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446803	CO[C@H]1CCN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-40-18-11-12-34(14-18)25(36)17-9-10-19-22(13-17)35(33-24(19)15-5-7-16(8-6-15)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,16,18H,6-8,11-12,14H2,1H3,(H,38,39)/t16?,18-/m0/s1	YBBWSYMSKCZLKW-DAFXYXGESA-N	256379	US9487490, 4AA	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256379	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256379&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388361	347916181							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446804	CO[C@@H]1CCN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)C1=CCC(CC1)C(O)=O	InChI=1S/C28H25ClF3N3O5/c1-40-18-11-12-34(14-18)25(36)17-9-10-19-22(13-17)35(33-24(19)15-5-7-16(8-6-15)27(38)39)26(37)23-20(28(30,31)32)3-2-4-21(23)29/h2-5,9-10,13,16,18H,6-8,11-12,14H2,1H3,(H,38,39)/t16?,18-/m1/s1	YBBWSYMSKCZLKW-UHUGOGIASA-N	256380	US9487490, 4AB	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 8					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256380	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256380&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388362	347916182							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446805	OC(=O)C1CCC(=CC1)c1cn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C23H16ClF4NO3/c24-16-4-1-3-15(23(26,27)28)20(16)21(30)29-11-14(19-17(25)5-2-6-18(19)29)12-7-9-13(10-8-12)22(31)32/h1-7,11,13H,8-10H2,(H,31,32)	PMCCAYCNHYFKOT-UHFFFAOYSA-N	256381	US9487490, 5A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 4					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256381&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388363	347916183							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446806	OC1C=C(CCC1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H15ClF4N2O4/c23-13-4-1-3-12(22(25,26)27)17(13)20(31)29-15-6-2-5-14(24)18(15)19(28-29)10-7-8-11(21(32)33)16(30)9-10/h1-6,9,11,16,30H,7-8H2,(H,32,33)	ULSWXLRBFXSKOO-UHFFFAOYSA-N	256382	US9487490, 6A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256382&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388364	347916184							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446807	OC1CC(=CCC1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H15ClF4N2O4/c23-13-4-1-3-12(22(25,26)27)17(13)20(31)29-15-6-2-5-14(24)18(15)19(28-29)10-7-8-11(21(32)33)16(30)9-10/h1-7,11,16,30H,8-9H2,(H,32,33)	DCEKJNKDTNIZBI-UHFFFAOYSA-N	256395	US9487490, 6B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256395	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256395&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73388365	347916197							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446808	CC1CC(=CC(O)C1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C23H17ClF4N2O4/c1-10-8-11(9-16(31)17(10)22(33)34)20-19-14(25)6-3-7-15(19)30(29-20)21(32)18-12(23(26,27)28)4-2-5-13(18)24/h2-7,9-10,16-17,31H,8H2,1H3,(H,33,34)	DTFLTTVMFQVAJF-UHFFFAOYSA-N	256383	US9487490, 6C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256383	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256383&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386902	347916185							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446809	CC1(CCC(CC1)C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C23H19ClF4N2O3/c1-22(10-8-12(9-11-22)21(32)33)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-7,12H,8-11H2,1H3,(H,32,33)	CHMFHAIDDKZQQX-UHFFFAOYSA-N	256397	US9487490, 7A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1879					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256397	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256397&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386795	347916199							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446810	C[C@@]1(CC[C@@H](CC1)C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C23H19ClF4N2O3/c1-22(10-8-12(9-11-22)21(32)33)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-7,12H,8-11H2,1H3,(H,32,33)/t12-,22-	CHMFHAIDDKZQQX-ZCNVGUKTSA-N	256384	US9487490, 7B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 663					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256384	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256384&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386795	347916186							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446811	C[C@]1(CC[C@@H](CC1)C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C23H19ClF4N2O3/c1-22(10-8-12(9-11-22)21(32)33)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-7,12H,8-11H2,1H3,(H,32,33)/t12-,22+	CHMFHAIDDKZQQX-LMRGUYSOSA-N	256396	US9487490, 7C	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 872					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256396	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256396&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386795	347916198							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446812	OC(=O)[C@H]1CC[C@@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H17ClF4N2O3/c23-14-4-1-3-13(22(25,26)27)17(14)20(30)29-16-6-2-5-15(24)18(16)19(28-29)11-7-9-12(10-8-11)21(31)32/h1-6,11-12H,7-10H2,(H,31,32)/t11-,12-	IJFFCHQCDHHGDN-HAQNSBGRSA-N	256385	US9487490, 8A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 16					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256385	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256385&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386796	347916187							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446813	OC(=O)[C@H]1CC[C@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H17ClF4N2O3/c23-14-4-1-3-13(22(25,26)27)17(14)20(30)29-16-6-2-5-15(24)18(16)19(28-29)11-7-9-12(10-8-11)21(31)32/h1-6,11-12H,7-10H2,(H,31,32)/t11-,12+	IJFFCHQCDHHGDN-TXEJJXNPSA-N	256398	US9487490, 8B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 505					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256398	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256398&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386796	347916200							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446814	C[C@@]1(CC[C@@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O	InChI=1S/C23H19ClF4N2O3/c1-22(21(32)33)10-8-12(9-11-22)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-7,12H,8-11H2,1H3,(H,32,33)/t12-,22-	OJVACVRAWQVAIH-ZCNVGUKTSA-N	256386	US9487490, 9A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256386&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386797	347916188							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446815	C[C@]1(CC[C@@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O	InChI=1S/C23H19ClF4N2O3/c1-22(21(32)33)10-8-12(9-11-22)19-18-15(25)6-3-7-16(18)30(29-19)20(31)17-13(23(26,27)28)4-2-5-14(17)24/h2-7,12H,8-11H2,1H3,(H,32,33)/t12-,22+	OJVACVRAWQVAIH-LMRGUYSOSA-N	256399	US9487490, 9B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5022					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256399	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256399&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386797	347916201							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446816	CC1(C)CC(=CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C24H19ClF4N2O3/c1-23(2)11-12(9-10-14(23)22(33)34)20-19-16(26)7-4-8-17(19)31(30-20)21(32)18-13(24(27,28)29)5-3-6-15(18)25/h3-9,14H,10-11H2,1-2H3,(H,33,34)/t14-/m0/s1	IXHXNWDSLDEFJY-AWEZNQCLSA-N	256387	US9487490, 10A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 343					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256387&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			131709596	347916189							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446817	CC1(C)C=C(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C24H19ClF4N2O3/c1-23(2)11-12(9-10-14(23)22(33)34)20-19-16(26)7-4-8-17(19)31(30-20)21(32)18-13(24(27,28)29)5-3-6-15(18)25/h3-8,11,14H,9-10H2,1-2H3,(H,33,34)/t14-/m1/s1	NLRMPVVVKMFYRF-CQSZACIVSA-N	256392	US9487490, 10B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 96					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256392	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256392&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90041885	347916194							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446818	OC(=O)[C@H]1CC[C@@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12	InChI=1S/C21H17ClF3N3O3/c22-14-4-1-3-13(21(23,24)25)16(14)19(29)28-15-5-2-10-26-18(15)17(27-28)11-6-8-12(9-7-11)20(30)31/h1-5,10-12H,6-9H2,(H,30,31)/t11-,12-	GNTUJCVVEKHONG-HAQNSBGRSA-N	256391	US9487490, 11A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 207					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256391	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256391&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386905	347916193							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446819	OC(=O)[C@H]1CC[C@H](CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12	InChI=1S/C21H17ClF3N3O3/c22-14-4-1-3-13(21(23,24)25)16(14)19(29)28-15-5-2-10-26-18(15)17(27-28)11-6-8-12(9-7-11)20(30)31/h1-5,10-12H,6-9H2,(H,30,31)/t11-,12+	GNTUJCVVEKHONG-TXEJJXNPSA-N	256388	US9487490, 11B	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10000					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256388&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386905	347916190							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446820	CC1CC(CC=C1c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O	InChI=1S/C23H17ClF4N2O3/c1-11-10-12(22(32)33)8-9-13(11)20-19-16(25)6-3-7-17(19)30(29-20)21(31)18-14(23(26,27)28)4-2-5-15(18)24/h2-7,9,11-12H,8,10H2,1H3,(H,32,33)	MZUYAAVZONNWFQ-UHFFFAOYSA-N	256389	US9487490, 12A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 54					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256389&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386998	347916191							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
446821	OC(=O)C1CCC(O)(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12	InChI=1S/C22H17ClF4N2O4/c23-13-4-1-3-12(22(25,26)27)16(13)19(30)29-15-6-2-5-14(24)17(15)18(28-29)21(33)9-7-11(8-10-21)20(31)32/h1-6,11,33H,7-10H2,(H,31,32)	SQOPQHPAVXHAAT-UHFFFAOYSA-N	256390	US9487490, 13A	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2474					7	4.00 C	US Patent		10.7270/Q2GQ6WQN		aid1803597	US9487490	Barr, KJ; Maclean, JK; Zhang, H; Beresis, RT; Zhang, D; Andresen, BM; Anthony, NJ; Lapointe, BT; Sciammetta, N	Merck Sharp & Dohme Corp	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=256390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=256390&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			73386999	347916192							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783544	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)c2noc(=O)[nH]2)c2ccccc12	InChI=1S/C31H39N5O5S2/c1-30(2,3)36-43(39,40)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)33-27(42-25)26(37)32-18-31(4,5)28-34-29(38)41-35-28/h9-10,13-16,19,36H,6-8,11-12,17-18H2,1-5H3,(H,32,37)(H,34,35,38)	IYVGXWZGZUPAGF-UHFFFAOYSA-N	392062	US10301272, Example 6/60	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392062	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392062&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012228	404960402							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783545	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)c1noc(=O)[nH]1)C(F)(F)F			392063	US10301272, Example 6/61	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392063	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392063&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012229	404960403							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783546	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)c1noc(=O)[nH]1)C(F)(F)F			392063	US10301272, Example 6/61	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392063	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392063&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012229	404960403							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783547	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)c1nnn[nH]1)C(F)(F)F			392064	US10301272, Example 6/62	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392064	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392064&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185716	404960404							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783548	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)c1nnn[nH]1)C(F)(F)F			392064	US10301272, Example 6/62	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392064	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392064&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185716	404960404							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783549	Cc1c(Cl)c(c(Cl)cc1-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H37Cl2N3O5S3/c1-16-19(15-20(28)24(22(16)29)40(36,37)32-27(2,3)4)23-21(14-17-8-6-5-7-9-17)31-26(38-23)25(33)30-18-10-12-39(34,35)13-11-18/h15,17-18,32H,5-14H2,1-4H3,(H,30,33)	VZWHYVVKBZIWNW-UHFFFAOYSA-N	392065	US10301272, Example 6/63	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 0.631							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392065	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392065&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185717	404960405							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783550	Cc1c(Cl)c(c(Cl)cc1-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H37Cl2N3O5S3/c1-16-19(15-20(28)24(22(16)29)40(36,37)32-27(2,3)4)23-21(14-17-8-6-5-7-9-17)31-26(38-23)25(33)30-18-10-12-39(34,35)13-11-18/h15,17-18,32H,5-14H2,1-4H3,(H,30,33)	VZWHYVVKBZIWNW-UHFFFAOYSA-N	392065	US10301272, Example 6/63	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392065	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392065&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185717	404960405							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783551	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)C(N)=O)c2ccccc12	InChI=1S/C30H40N4O4S2/c1-29(2,3)34-40(37,38)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)33-27(39-25)26(35)32-18-30(4,5)28(31)36/h9-10,13-16,19,34H,6-8,11-12,17-18H2,1-5H3,(H2,31,36)(H,32,35)	UZGJBTQXRSHORE-UHFFFAOYSA-N	392066	US10301272, Example 6/64	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392066&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185718	404960406							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783552	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)C(N)=O)c2ccccc12	InChI=1S/C30H40N4O4S2/c1-29(2,3)34-40(37,38)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)33-27(39-25)26(35)32-18-30(4,5)28(31)36/h9-10,13-16,19,34H,6-8,11-12,17-18H2,1-5H3,(H2,31,36)(H,32,35)	UZGJBTQXRSHORE-UHFFFAOYSA-N	392066	US10301272, Example 6/64	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392066	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392066&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185718	404960406							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783553	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H44N2O3S/c1-29(2,3)22-17-21(18-23(19-22)31(6)12-13-31)25-24(16-20-10-8-7-9-11-20)33-27(37-25)26(34)32-15-14-30(4,5)28(35)36/h17-20H,7-16H2,1-6H3,(H,32,34)(H,35,36)	JSIWAWWVQCKYAX-UHFFFAOYSA-N	392067	US10301272, Example 7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392067	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392067&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548005	404960407							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783554	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H44N2O3S/c1-29(2,3)22-17-21(18-23(19-22)31(6)12-13-31)25-24(16-20-10-8-7-9-11-20)33-27(37-25)26(34)32-15-14-30(4,5)28(35)36/h17-20H,7-16H2,1-6H3,(H,32,34)(H,35,36)	JSIWAWWVQCKYAX-UHFFFAOYSA-N	392067	US10301272, Example 7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392067	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392067&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548005	404960407							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783555	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H44N2O3S/c1-29(2,3)22-17-21(18-23(19-22)31(6)12-13-31)25-24(16-20-10-8-7-9-11-20)33-27(37-25)26(34)32-15-14-30(4,5)28(35)36/h17-20H,7-16H2,1-6H3,(H,32,34)(H,35,36)	JSIWAWWVQCKYAX-UHFFFAOYSA-N	392067	US10301272, Example 7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392067	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392067&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548005	404960407							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783556	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H47N3O5S2/c1-29(2,3)22-19-21(14-15-24(22)41(38,39)34-30(4,5)6)25-23(18-20-12-10-9-11-13-20)33-27(40-25)26(35)32-17-16-31(7,8)28(36)37/h14-15,19-20,34H,9-13,16-18H2,1-8H3,(H,32,35)(H,36,37)	PSYUVGRQWQIOCW-UHFFFAOYSA-N	392068	US10301272, Example 7/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392068	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392068&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548241	404960408							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783557	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H47N3O5S2/c1-29(2,3)22-19-21(14-15-24(22)41(38,39)34-30(4,5)6)25-23(18-20-12-10-9-11-13-20)33-27(40-25)26(35)32-17-16-31(7,8)28(36)37/h14-15,19-20,34H,9-13,16-18H2,1-8H3,(H,32,35)(H,36,37)	PSYUVGRQWQIOCW-UHFFFAOYSA-N	392068	US10301272, Example 7/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392068	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392068&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548241	404960408							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783558	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C31H47N3O5S2/c1-29(2,3)22-19-21(14-15-24(22)41(38,39)34-30(4,5)6)25-23(18-20-12-10-9-11-13-20)33-27(40-25)26(35)32-17-16-31(7,8)28(36)37/h14-15,19-20,34H,9-13,16-18H2,1-8H3,(H,32,35)(H,36,37)	PSYUVGRQWQIOCW-UHFFFAOYSA-N	392068	US10301272, Example 7/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392068	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392068&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548241	404960408							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783559	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O5S2/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	ABUNLVQVPCSGRD-MEMLXQNLSA-N	392069	US10301272, Example 7/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392069&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548242	404960409							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783560	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O5S2/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	ABUNLVQVPCSGRD-MEMLXQNLSA-N	392069	US10301272, Example 7/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392069&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548242	404960409							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783561	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O5S2/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	ABUNLVQVPCSGRD-MEMLXQNLSA-N	392069	US10301272, Example 7/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392069&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548242	404960409							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783562	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O3S/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	JNHPYHREURDHOD-JKIUYZKVSA-N	392070	US10301272, Example 7/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392070&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548240	404960410							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783563	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O3S/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	JNHPYHREURDHOD-JKIUYZKVSA-N	392070	US10301272, Example 7/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392070&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548240	404960410							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783564	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O3S/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	JNHPYHREURDHOD-JKIUYZKVSA-N	392070	US10301272, Example 7/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392070&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548240	404960410							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783565	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C	InChI=1S/C28H38ClN3O5S2/c1-5-28(3,4)32-39(36,37)22-12-11-20(23(29)16(22)2)24-21(13-17-9-7-6-8-10-17)31-26(38-24)25(33)30-19-14-18(15-19)27(34)35/h11-12,17-19,32H,5-10,13-15H2,1-4H3,(H,30,33)(H,34,35)/t18-,19-	QLKWBZGQDXUAPZ-WGSAOQKQSA-N	50044179	CHEMBL3314002::US10301272, Example 7/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548704	313068130		CHEMBL3314002					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783566	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C	InChI=1S/C28H38ClN3O5S2/c1-5-28(3,4)32-39(36,37)22-12-11-20(23(29)16(22)2)24-21(13-17-9-7-6-8-10-17)31-26(38-24)25(33)30-19-14-18(15-19)27(34)35/h11-12,17-19,32H,5-10,13-15H2,1-4H3,(H,30,33)(H,34,35)/t18-,19-	QLKWBZGQDXUAPZ-WGSAOQKQSA-N	50044179	CHEMBL3314002::US10301272, Example 7/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548704	313068130		CHEMBL3314002					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783567	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C	InChI=1S/C28H38ClN3O5S2/c1-5-28(3,4)32-39(36,37)22-12-11-20(23(29)16(22)2)24-21(13-17-9-7-6-8-10-17)31-26(38-24)25(33)30-19-14-18(15-19)27(34)35/h11-12,17-19,32H,5-10,13-15H2,1-4H3,(H,30,33)(H,34,35)/t18-,19-	QLKWBZGQDXUAPZ-WGSAOQKQSA-N	50044179	CHEMBL3314002::US10301272, Example 7/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548704	313068130		CHEMBL3314002					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783568	CC(C)(C)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)F	InChI=1S/C27H34F2N2O3S/c1-27(2,3)19-11-16(10-17(12-19)23(28)29)22-21(9-15-7-5-4-6-8-15)31-25(35-22)24(32)30-20-13-18(14-20)26(33)34/h10-12,15,18,20,23H,4-9,13-14H2,1-3H3,(H,30,32)(H,33,34)/t18-,20-	OLFNLVXDQKVHBC-KESTWPANSA-N	392072	US10301272, Example 7/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392072&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185719	404960412							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783569	CC(C)(C)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)F	InChI=1S/C27H34F2N2O3S/c1-27(2,3)19-11-16(10-17(12-19)23(28)29)22-21(9-15-7-5-4-6-8-15)31-25(35-22)24(32)30-20-13-18(14-20)26(33)34/h10-12,15,18,20,23H,4-9,13-14H2,1-3H3,(H,30,32)(H,33,34)/t18-,20-	OLFNLVXDQKVHBC-KESTWPANSA-N	392072	US10301272, Example 7/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392072&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185719	404960412							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783570	CC(C)(C)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)F	InChI=1S/C27H34F2N2O3S/c1-27(2,3)19-11-16(10-17(12-19)23(28)29)22-21(9-15-7-5-4-6-8-15)31-25(35-22)24(32)30-20-13-18(14-20)26(33)34/h10-12,15,18,20,23H,4-9,13-14H2,1-3H3,(H,30,32)(H,33,34)/t18-,20-	OLFNLVXDQKVHBC-KESTWPANSA-N	392072	US10301272, Example 7/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392072	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392072&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185719	404960412							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783571	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NCC(F)(F)F	InChI=1S/C29H34F3N3O4S/c1-28(7-8-28)20-11-17(10-18(12-20)24(36)33-15-29(30,31)32)23-22(9-16-5-3-2-4-6-16)35-26(40-23)25(37)34-21-13-19(14-21)27(38)39/h10-12,16,19,21H,2-9,13-15H2,1H3,(H,33,36)(H,34,37)(H,38,39)/t19-,21-	YFVUWRZSDOLCGF-XUTJKUGGSA-N	392073	US10301272, Example 7/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392073&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188702	404960413							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783572	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NCC(F)(F)F	InChI=1S/C29H34F3N3O4S/c1-28(7-8-28)20-11-17(10-18(12-20)24(36)33-15-29(30,31)32)23-22(9-16-5-3-2-4-6-16)35-26(40-23)25(37)34-21-13-19(14-21)27(38)39/h10-12,16,19,21H,2-9,13-15H2,1H3,(H,33,36)(H,34,37)(H,38,39)/t19-,21-	YFVUWRZSDOLCGF-XUTJKUGGSA-N	392073	US10301272, Example 7/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392073&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188702	404960413							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783573	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NCC(F)(F)F	InChI=1S/C29H34F3N3O4S/c1-28(7-8-28)20-11-17(10-18(12-20)24(36)33-15-29(30,31)32)23-22(9-16-5-3-2-4-6-16)35-26(40-23)25(37)34-21-13-19(14-21)27(38)39/h10-12,16,19,21H,2-9,13-15H2,1H3,(H,33,36)(H,34,37)(H,38,39)/t19-,21-	YFVUWRZSDOLCGF-XUTJKUGGSA-N	392073	US10301272, Example 7/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392073	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392073&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188702	404960413							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783574	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S2/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	YYHHVJHYBVCDLG-WKILWMFISA-N	392074	US10301272, Example 7/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392074&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185721	404960414							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783575	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S2/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	YYHHVJHYBVCDLG-WKILWMFISA-N	392074	US10301272, Example 7/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392074&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185721	404960414							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783576	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S2/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	YYHHVJHYBVCDLG-WKILWMFISA-N	392074	US10301272, Example 7/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392074	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392074&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185721	404960414							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783577	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2CCCCc12	InChI=1S/C30H41N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h13-14,18-20,33H,4-12,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	IORGFFCZJYGRQD-MXVIHJGJSA-N	392075	US10301272, Example 7/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392075&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185722	404960415							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783578	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2CCCCc12	InChI=1S/C30H41N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h13-14,18-20,33H,4-12,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	IORGFFCZJYGRQD-MXVIHJGJSA-N	392075	US10301272, Example 7/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392075&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185722	404960415							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783579	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2CCCCc12	InChI=1S/C30H41N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h13-14,18-20,33H,4-12,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	IORGFFCZJYGRQD-MXVIHJGJSA-N	392075	US10301272, Example 7/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392075	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392075&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185722	404960415							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783580	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	KYIGOCCCBXRHNJ-MXVIHJGJSA-N	392076	US10301272, Example 7/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392076&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548703	404960416							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783581	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	KYIGOCCCBXRHNJ-MXVIHJGJSA-N	392076	US10301272, Example 7/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392076&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548703	404960416							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783582	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	KYIGOCCCBXRHNJ-MXVIHJGJSA-N	392076	US10301272, Example 7/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392076	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392076&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548703	404960416							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783583	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12)C(F)(F)F	InChI=1S/C29H32F3N3O5S2/c1-16(29(30,31)32)35-42(39,40)24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)34-27(41-25)26(36)33-19-14-18(15-19)28(37)38/h5-6,9-12,16-19,35H,2-4,7-8,13-15H2,1H3,(H,33,36)(H,37,38)/t16?,18-,19-	ZDBJECNSNPXCFS-YGXOWLSWSA-N	392077	US10301272, Example 7/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392077&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			124001244	404960417							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783584	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12)C(F)(F)F	InChI=1S/C29H32F3N3O5S2/c1-16(29(30,31)32)35-42(39,40)24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)34-27(41-25)26(36)33-19-14-18(15-19)28(37)38/h5-6,9-12,16-19,35H,2-4,7-8,13-15H2,1H3,(H,33,36)(H,37,38)/t16?,18-,19-	ZDBJECNSNPXCFS-YGXOWLSWSA-N	392077	US10301272, Example 7/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392077&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			124001244	404960417							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783585	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12)C(F)(F)F	InChI=1S/C29H32F3N3O5S2/c1-16(29(30,31)32)35-42(39,40)24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)34-27(41-25)26(36)33-19-14-18(15-19)28(37)38/h5-6,9-12,16-19,35H,2-4,7-8,13-15H2,1H3,(H,33,36)(H,37,38)/t16?,18-,19-	ZDBJECNSNPXCFS-YGXOWLSWSA-N	392077	US10301272, Example 7/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392077	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392077&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			124001244	404960417							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783586	CC(C)COc1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O4S/c1-17(2)16-36-24-15-19(14-23(32-24)29(3,4)5)25-22(11-18-9-7-6-8-10-18)31-27(37-25)26(33)30-21-12-20(13-21)28(34)35/h14-15,17-18,20-21H,6-13,16H2,1-5H3,(H,30,33)(H,34,35)/t20-,21-	LNKSNAFFXWHGJC-MEMLXQNLSA-N	392078	US10301272, Example 7/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392078&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185724	404960418							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783587	CC(C)COc1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O4S/c1-17(2)16-36-24-15-19(14-23(32-24)29(3,4)5)25-22(11-18-9-7-6-8-10-18)31-27(37-25)26(33)30-21-12-20(13-21)28(34)35/h14-15,17-18,20-21H,6-13,16H2,1-5H3,(H,30,33)(H,34,35)/t20-,21-	LNKSNAFFXWHGJC-MEMLXQNLSA-N	392078	US10301272, Example 7/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392078&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185724	404960418							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783588	CC(C)COc1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O4S/c1-17(2)16-36-24-15-19(14-23(32-24)29(3,4)5)25-22(11-18-9-7-6-8-10-18)31-27(37-25)26(33)30-21-12-20(13-21)28(34)35/h14-15,17-18,20-21H,6-13,16H2,1-5H3,(H,30,33)(H,34,35)/t20-,21-	LNKSNAFFXWHGJC-MEMLXQNLSA-N	392078	US10301272, Example 7/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392078	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392078&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185724	404960418							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783589	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C(F)(F)F	InChI=1S/C27H33ClF3N3O5S2/c1-26(2,3)34-41(38,39)19-10-9-17(21(28)20(19)27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(40-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	IAWFEFNRFRSAIY-WKILWMFISA-N	392079	US10301272, Example 7/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392079&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185726	404960419							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783590	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C(F)(F)F	InChI=1S/C27H33ClF3N3O5S2/c1-26(2,3)34-41(38,39)19-10-9-17(21(28)20(19)27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(40-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	IAWFEFNRFRSAIY-WKILWMFISA-N	392079	US10301272, Example 7/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392079&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185726	404960419							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783591	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C(F)(F)F	InChI=1S/C27H33ClF3N3O5S2/c1-26(2,3)34-41(38,39)19-10-9-17(21(28)20(19)27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(40-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	IAWFEFNRFRSAIY-WKILWMFISA-N	392079	US10301272, Example 7/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392079	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392079&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185726	404960419							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783592	Cc1c(OC(F)F)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H37F2N3O6S2/c1-15-21(41(37,38)33-28(2,3)4)11-10-19(22(15)39-27(29)30)23-20(12-16-8-6-5-7-9-16)32-25(40-23)24(34)31-18-13-17(14-18)26(35)36/h10-11,16-18,27,33H,5-9,12-14H2,1-4H3,(H,31,34)(H,35,36)/t17-,18-	NSAOHDFDPAPARQ-IYARVYRRSA-N	392080	US10301272, Example 7/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392080&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185723	404960420							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783593	Cc1c(OC(F)F)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H37F2N3O6S2/c1-15-21(41(37,38)33-28(2,3)4)11-10-19(22(15)39-27(29)30)23-20(12-16-8-6-5-7-9-16)32-25(40-23)24(34)31-18-13-17(14-18)26(35)36/h10-11,16-18,27,33H,5-9,12-14H2,1-4H3,(H,31,34)(H,35,36)/t17-,18-	NSAOHDFDPAPARQ-IYARVYRRSA-N	392080	US10301272, Example 7/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392080&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185723	404960420							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783594	Cc1c(OC(F)F)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H37F2N3O6S2/c1-15-21(41(37,38)33-28(2,3)4)11-10-19(22(15)39-27(29)30)23-20(12-16-8-6-5-7-9-16)32-25(40-23)24(34)31-18-13-17(14-18)26(35)36/h10-11,16-18,27,33H,5-9,12-14H2,1-4H3,(H,31,34)(H,35,36)/t17-,18-	NSAOHDFDPAPARQ-IYARVYRRSA-N	392080	US10301272, Example 7/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392080	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392080&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185723	404960420							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783595	Cc1c(ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c1C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C28H36F3N3O5S2/c1-15-21(41(38,39)34-27(2,3)4)11-10-19(22(15)28(29,30)31)23-20(12-16-8-6-5-7-9-16)33-25(40-23)24(35)32-18-13-17(14-18)26(36)37/h10-11,16-18,34H,5-9,12-14H2,1-4H3,(H,32,35)(H,36,37)/t17-,18-	LQDOFOHSWMEENT-IYARVYRRSA-N	392081	US10301272, Example 7/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392081&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188692	404960421							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783596	Cc1c(ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c1C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C28H36F3N3O5S2/c1-15-21(41(38,39)34-27(2,3)4)11-10-19(22(15)28(29,30)31)23-20(12-16-8-6-5-7-9-16)33-25(40-23)24(35)32-18-13-17(14-18)26(36)37/h10-11,16-18,34H,5-9,12-14H2,1-4H3,(H,32,35)(H,36,37)/t17-,18-	LQDOFOHSWMEENT-IYARVYRRSA-N	392081	US10301272, Example 7/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392081&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188692	404960421							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783597	Cc1c(ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c1C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C28H36F3N3O5S2/c1-15-21(41(38,39)34-27(2,3)4)11-10-19(22(15)28(29,30)31)23-20(12-16-8-6-5-7-9-16)33-25(40-23)24(35)32-18-13-17(14-18)26(36)37/h10-11,16-18,34H,5-9,12-14H2,1-4H3,(H,32,35)(H,36,37)/t17-,18-	LQDOFOHSWMEENT-IYARVYRRSA-N	392081	US10301272, Example 7/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392081	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392081&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188692	404960421							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783598	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1C(F)F	InChI=1S/C27H34F3N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(21(28)20(19)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	DIPOXOYHTIKZHF-WKILWMFISA-N	392082	US10301272, Example 7/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392082&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185727	404960422							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783599	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1C(F)F	InChI=1S/C27H34F3N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(21(28)20(19)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	DIPOXOYHTIKZHF-WKILWMFISA-N	392082	US10301272, Example 7/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392082&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185727	404960422							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783600	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1C(F)F	InChI=1S/C27H34F3N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(21(28)20(19)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	DIPOXOYHTIKZHF-WKILWMFISA-N	392082	US10301272, Example 7/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392082	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392082&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185727	404960422							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783601	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(C(F)F)c1Cl	InChI=1S/C27H34ClF2N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(20(21(19)28)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	QFSSUDFXXKGELX-WKILWMFISA-N	392083	US10301272, Example 7/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392083&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548706	404960423							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783602	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(C(F)F)c1Cl	InChI=1S/C27H34ClF2N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(20(21(19)28)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	QFSSUDFXXKGELX-WKILWMFISA-N	392083	US10301272, Example 7/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392083&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548706	404960423							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783603	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(C(F)F)c1Cl	InChI=1S/C27H34ClF2N3O5S2/c1-27(2,3)33-40(37,38)19-10-9-17(20(21(19)28)23(29)30)22-18(11-14-7-5-4-6-8-14)32-25(39-22)24(34)31-16-12-15(13-16)26(35)36/h9-10,14-16,23,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t15-,16-	QFSSUDFXXKGELX-WKILWMFISA-N	392083	US10301272, Example 7/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392083	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392083&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548706	404960423							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783604	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O6S2/c1-28(2,3)32-40(37,38)23-12-11-18(16-21(23)29(4,5)36)24-22(13-17-9-7-6-8-10-17)31-26(39-24)25(33)30-20-14-19(15-20)27(34)35/h11-12,16-17,19-20,32,36H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)/t19-,20-	VOVIZZOAKHUQAS-MXVIHJGJSA-N	392084	US10301272, Example 7/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392084&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185728	404960424							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783605	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O6S2/c1-28(2,3)32-40(37,38)23-12-11-18(16-21(23)29(4,5)36)24-22(13-17-9-7-6-8-10-17)31-26(39-24)25(33)30-20-14-19(15-20)27(34)35/h11-12,16-17,19-20,32,36H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)/t19-,20-	VOVIZZOAKHUQAS-MXVIHJGJSA-N	392084	US10301272, Example 7/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392084&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185728	404960424							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783606	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H41N3O6S2/c1-28(2,3)32-40(37,38)23-12-11-18(16-21(23)29(4,5)36)24-22(13-17-9-7-6-8-10-17)31-26(39-24)25(33)30-20-14-19(15-20)27(34)35/h11-12,16-17,19-20,32,36H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)/t19-,20-	VOVIZZOAKHUQAS-MXVIHJGJSA-N	392084	US10301272, Example 7/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392084	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392084&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185728	404960424							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783607	CC(C)(C)c1cc(cc(c1)C(C)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H36F2N2O3S/c1-27(2,3)19-11-17(12-20(15-19)28(4,29)30)23-22(10-16-8-6-5-7-9-16)32-25(36-23)24(33)31-21-13-18(14-21)26(34)35/h11-12,15-16,18,21H,5-10,13-14H2,1-4H3,(H,31,33)(H,34,35)/t18-,21-	ZCBWGWZHTIWKHS-XGAFWQRZSA-N	392085	US10301272, Example 7/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392085&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185729	404960425							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783608	CC(C)(C)c1cc(cc(c1)C(C)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H36F2N2O3S/c1-27(2,3)19-11-17(12-20(15-19)28(4,29)30)23-22(10-16-8-6-5-7-9-16)32-25(36-23)24(33)31-21-13-18(14-21)26(34)35/h11-12,15-16,18,21H,5-10,13-14H2,1-4H3,(H,31,33)(H,34,35)/t18-,21-	ZCBWGWZHTIWKHS-XGAFWQRZSA-N	392085	US10301272, Example 7/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392085&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185729	404960425							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783609	CC(C)(C)c1cc(cc(c1)C(C)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H36F2N2O3S/c1-27(2,3)19-11-17(12-20(15-19)28(4,29)30)23-22(10-16-8-6-5-7-9-16)32-25(36-23)24(33)31-21-13-18(14-21)26(34)35/h11-12,15-16,18,21H,5-10,13-14H2,1-4H3,(H,31,33)(H,34,35)/t18-,21-	ZCBWGWZHTIWKHS-XGAFWQRZSA-N	392085	US10301272, Example 7/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392085	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392085&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185729	404960425							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783610	CC(NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F	InChI=1S/C30H38F3N3O4S/c1-16(30(31,32)33)34-25(37)19-11-18(12-21(13-19)29(2,3)4)24-23(10-17-8-6-5-7-9-17)36-27(41-24)26(38)35-22-14-20(15-22)28(39)40/h11-13,16-17,20,22H,5-10,14-15H2,1-4H3,(H,34,37)(H,35,38)(H,39,40)/t16?,20-,22-	GZCDNIGGYFEPLV-LKYSKULBSA-N	392086	US10301272, Example 7/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392086&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012230	404960426							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783611	CC(NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F	InChI=1S/C30H38F3N3O4S/c1-16(30(31,32)33)34-25(37)19-11-18(12-21(13-19)29(2,3)4)24-23(10-17-8-6-5-7-9-17)36-27(41-24)26(38)35-22-14-20(15-22)28(39)40/h11-13,16-17,20,22H,5-10,14-15H2,1-4H3,(H,34,37)(H,35,38)(H,39,40)/t16?,20-,22-	GZCDNIGGYFEPLV-LKYSKULBSA-N	392086	US10301272, Example 7/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392086	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392086&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012230	404960426							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783612	COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H30N2O4S/c1-32-24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)29-27(34-25)26(31)28-18-14-19(15-18)33-16-30/h5-6,9-12,16-19H,2-4,7-8,13-15H2,1H3,(H,28,31)/t18-,19-	KLKYGJXHEZXQPG-WGSAOQKQSA-N	392087	US10301272, Example 7/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392087&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185730	404960427							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783613	COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H30N2O4S/c1-32-24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)29-27(34-25)26(31)28-18-14-19(15-18)33-16-30/h5-6,9-12,16-19H,2-4,7-8,13-15H2,1H3,(H,28,31)/t18-,19-	KLKYGJXHEZXQPG-WGSAOQKQSA-N	392087	US10301272, Example 7/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392087&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185730	404960427							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783614	COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H30N2O4S/c1-32-24-12-11-22(20-9-5-6-10-21(20)24)25-23(13-17-7-3-2-4-8-17)29-27(34-25)26(31)28-18-14-19(15-18)33-16-30/h5-6,9-12,16-19H,2-4,7-8,13-15H2,1H3,(H,28,31)/t18-,19-	KLKYGJXHEZXQPG-WGSAOQKQSA-N	392087	US10301272, Example 7/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392087	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392087&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185730	404960427							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783615	FC(F)(F)Oc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H27F3N2O4S/c28-27(29,30)36-23-11-10-21(19-8-4-5-9-20(19)23)24-22(12-16-6-2-1-3-7-16)32-26(37-24)25(34)31-17-13-18(14-17)35-15-33/h4-5,8-11,15-18H,1-3,6-7,12-14H2,(H,31,34)/t17-,18-	KAROPISCKXBLEI-IYARVYRRSA-N	392088	US10301272, Example 7/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1995							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392088&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185731	404960428							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783616	FC(F)(F)Oc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H27F3N2O4S/c28-27(29,30)36-23-11-10-21(19-8-4-5-9-20(19)23)24-22(12-16-6-2-1-3-7-16)32-26(37-24)25(34)31-17-13-18(14-17)35-15-33/h4-5,8-11,15-18H,1-3,6-7,12-14H2,(H,31,34)/t17-,18-	KAROPISCKXBLEI-IYARVYRRSA-N	392088	US10301272, Example 7/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392088&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185731	404960428							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783617	FC(F)(F)Oc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C27H27F3N2O4S/c28-27(29,30)36-23-11-10-21(19-8-4-5-9-20(19)23)24-22(12-16-6-2-1-3-7-16)32-26(37-24)25(34)31-17-13-18(14-17)35-15-33/h4-5,8-11,15-18H,1-3,6-7,12-14H2,(H,31,34)/t17-,18-	KAROPISCKXBLEI-IYARVYRRSA-N	392088	US10301272, Example 7/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392088	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392088&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185731	404960428							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783618	FC(F)(F)COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C28H29F3N2O4S/c29-28(30,31)15-36-24-11-10-22(20-8-4-5-9-21(20)24)25-23(12-17-6-2-1-3-7-17)33-27(38-25)26(35)32-18-13-19(14-18)37-16-34/h4-5,8-11,16-19H,1-3,6-7,12-15H2,(H,32,35)/t18-,19-	ISGXZRGVUXMDPR-WGSAOQKQSA-N	392089	US10301272, Example 7/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392089&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185733	404960429							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783619	FC(F)(F)COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C28H29F3N2O4S/c29-28(30,31)15-36-24-11-10-22(20-8-4-5-9-21(20)24)25-23(12-17-6-2-1-3-7-17)33-27(38-25)26(35)32-18-13-19(14-18)37-16-34/h4-5,8-11,16-19H,1-3,6-7,12-15H2,(H,32,35)/t18-,19-	ISGXZRGVUXMDPR-WGSAOQKQSA-N	392089	US10301272, Example 7/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392089&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185733	404960429							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783620	FC(F)(F)COc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)OC=O)c2ccccc12	InChI=1S/C28H29F3N2O4S/c29-28(30,31)15-36-24-11-10-22(20-8-4-5-9-21(20)24)25-23(12-17-6-2-1-3-7-17)33-27(38-25)26(35)32-18-13-19(14-18)37-16-34/h4-5,8-11,16-19H,1-3,6-7,12-15H2,(H,32,35)/t18-,19-	ISGXZRGVUXMDPR-WGSAOQKQSA-N	392089	US10301272, Example 7/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392089	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392089&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185733	404960429							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783621	CC(C)(O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H36N2O4S2/c1-29(2,33)24-13-12-23(21-10-6-7-11-22(21)24)26-25(18-19-8-4-3-5-9-19)31-28(36-26)27(32)30-20-14-16-37(34,35)17-15-20/h6-7,10-13,19-20,33H,3-5,8-9,14-18H2,1-2H3,(H,30,32)	SUBNBNURHSQFBO-UHFFFAOYSA-N	392090	US10301272, Example 7/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392090&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185734	404960430							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783622	CC(C)(O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H36N2O4S2/c1-29(2,33)24-13-12-23(21-10-6-7-11-22(21)24)26-25(18-19-8-4-3-5-9-19)31-28(36-26)27(32)30-20-14-16-37(34,35)17-15-20/h6-7,10-13,19-20,33H,3-5,8-9,14-18H2,1-2H3,(H,30,32)	SUBNBNURHSQFBO-UHFFFAOYSA-N	392090	US10301272, Example 7/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392090&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185734	404960430							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783623	CC(C)(O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H36N2O4S2/c1-29(2,33)24-13-12-23(21-10-6-7-11-22(21)24)26-25(18-19-8-4-3-5-9-19)31-28(36-26)27(32)30-20-14-16-37(34,35)17-15-20/h6-7,10-13,19-20,33H,3-5,8-9,14-18H2,1-2H3,(H,30,32)	SUBNBNURHSQFBO-UHFFFAOYSA-N	392090	US10301272, Example 7/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392090	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392090&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185734	404960430							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783624	OC1(CCC1)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H36N2O4S2/c33-28(31-21-13-17-38(35,36)18-14-21)29-32-26(19-20-7-2-1-3-8-20)27(37-29)24-11-12-25(30(34)15-6-16-30)23-10-5-4-9-22(23)24/h4-5,9-12,20-21,34H,1-3,6-8,13-19H2,(H,31,33)	SRQJHANWRRXBFO-UHFFFAOYSA-N	392091	US10301272, Example 7/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1995							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392091&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185735	404960431							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783625	OC1(CCC1)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H36N2O4S2/c33-28(31-21-13-17-38(35,36)18-14-21)29-32-26(19-20-7-2-1-3-8-20)27(37-29)24-11-12-25(30(34)15-6-16-30)23-10-5-4-9-22(23)24/h4-5,9-12,20-21,34H,1-3,6-8,13-19H2,(H,31,33)	SRQJHANWRRXBFO-UHFFFAOYSA-N	392091	US10301272, Example 7/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392091&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185735	404960431							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783626	OC1(CCC1)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H36N2O4S2/c33-28(31-21-13-17-38(35,36)18-14-21)29-32-26(19-20-7-2-1-3-8-20)27(37-29)24-11-12-25(30(34)15-6-16-30)23-10-5-4-9-22(23)24/h4-5,9-12,20-21,34H,1-3,6-8,13-19H2,(H,31,33)	SRQJHANWRRXBFO-UHFFFAOYSA-N	392091	US10301272, Example 7/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392091	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392091&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185735	404960431							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783627	CC(C)(C)NC(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H39N3O4S2/c1-31(2,3)34-28(35)25-14-13-24(22-11-7-8-12-23(22)25)27-26(19-20-9-5-4-6-10-20)33-30(39-27)29(36)32-21-15-17-40(37,38)18-16-21/h7-8,11-14,20-21H,4-6,9-10,15-19H2,1-3H3,(H,32,36)(H,34,35)	FXVWIAQJPPVZEJ-UHFFFAOYSA-N	392092	US10301272, Example 7/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392092&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185736	404960432							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783628	CC(C)(C)NC(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H39N3O4S2/c1-31(2,3)34-28(35)25-14-13-24(22-11-7-8-12-23(22)25)27-26(19-20-9-5-4-6-10-20)33-30(39-27)29(36)32-21-15-17-40(37,38)18-16-21/h7-8,11-14,20-21H,4-6,9-10,15-19H2,1-3H3,(H,32,36)(H,34,35)	FXVWIAQJPPVZEJ-UHFFFAOYSA-N	392092	US10301272, Example 7/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392092&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185736	404960432							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783629	CC(C)(C)NC(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H39N3O4S2/c1-31(2,3)34-28(35)25-14-13-24(22-11-7-8-12-23(22)25)27-26(19-20-9-5-4-6-10-20)33-30(39-27)29(36)32-21-15-17-40(37,38)18-16-21/h7-8,11-14,20-21H,4-6,9-10,15-19H2,1-3H3,(H,32,36)(H,34,35)	FXVWIAQJPPVZEJ-UHFFFAOYSA-N	392092	US10301272, Example 7/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392092	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392092&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185736	404960432							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783630	CC1(C)COCCN1Cc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C33H43N3O4S2/c1-33(2)22-40-17-16-36(33)21-24-12-13-28(27-11-7-6-10-26(24)27)30-29(20-23-8-4-3-5-9-23)35-32(41-30)31(37)34-25-14-18-42(38,39)19-15-25/h6-7,10-13,23,25H,3-5,8-9,14-22H2,1-2H3,(H,34,37)	JGANKYZLDWKLMS-UHFFFAOYSA-N	392093	US10301272, Example 7/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392093&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549190	404960433							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783631	CC1(C)COCCN1Cc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C33H43N3O4S2/c1-33(2)22-40-17-16-36(33)21-24-12-13-28(27-11-7-6-10-26(24)27)30-29(20-23-8-4-3-5-9-23)35-32(41-30)31(37)34-25-14-18-42(38,39)19-15-25/h6-7,10-13,23,25H,3-5,8-9,14-22H2,1-2H3,(H,34,37)	JGANKYZLDWKLMS-UHFFFAOYSA-N	392093	US10301272, Example 7/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392093&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549190	404960433							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783632	CC1(C)COCCN1Cc1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C33H43N3O4S2/c1-33(2)22-40-17-16-36(33)21-24-12-13-28(27-11-7-6-10-26(24)27)30-29(20-23-8-4-3-5-9-23)35-32(41-30)31(37)34-25-14-18-42(38,39)19-15-25/h6-7,10-13,23,25H,3-5,8-9,14-22H2,1-2H3,(H,34,37)	JGANKYZLDWKLMS-UHFFFAOYSA-N	392093	US10301272, Example 7/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392093&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549190	404960433							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783633	O=C(NC1CCS(=O)(=O)CC1)c1nc(CC2CCCCC2)c(s1)-c1ccc(N2CCOCC2)c2ccccc12	InChI=1S/C30H37N3O4S2/c34-29(31-22-12-18-39(35,36)19-13-22)30-32-26(20-21-6-2-1-3-7-21)28(38-30)25-10-11-27(33-14-16-37-17-15-33)24-9-5-4-8-23(24)25/h4-5,8-11,21-22H,1-3,6-7,12-20H2,(H,31,34)	ZYYSVXAGRNHONE-UHFFFAOYSA-N	392094	US10301272, Example 7/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392094&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185737	404960434							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783634	O=C(NC1CCS(=O)(=O)CC1)c1nc(CC2CCCCC2)c(s1)-c1ccc(N2CCOCC2)c2ccccc12	InChI=1S/C30H37N3O4S2/c34-29(31-22-12-18-39(35,36)19-13-22)30-32-26(20-21-6-2-1-3-7-21)28(38-30)25-10-11-27(33-14-16-37-17-15-33)24-9-5-4-8-23(24)25/h4-5,8-11,21-22H,1-3,6-7,12-20H2,(H,31,34)	ZYYSVXAGRNHONE-UHFFFAOYSA-N	392094	US10301272, Example 7/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392094&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185737	404960434							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783635	O=C(NC1CCS(=O)(=O)CC1)c1nc(CC2CCCCC2)c(s1)-c1ccc(N2CCOCC2)c2ccccc12	InChI=1S/C30H37N3O4S2/c34-29(31-22-12-18-39(35,36)19-13-22)30-32-26(20-21-6-2-1-3-7-21)28(38-30)25-10-11-27(33-14-16-37-17-15-33)24-9-5-4-8-23(24)25/h4-5,8-11,21-22H,1-3,6-7,12-20H2,(H,31,34)	ZYYSVXAGRNHONE-UHFFFAOYSA-N	392094	US10301272, Example 7/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392094	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392094&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185737	404960434							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783636	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O2S/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	FUZUEQZMCGGQEN-UHFFFAOYSA-N	392095	US10301272, Example 8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392095&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548243	404960435							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783637	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O2S/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	FUZUEQZMCGGQEN-UHFFFAOYSA-N	392095	US10301272, Example 8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392095&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548243	404960435							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783638	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O2S/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	FUZUEQZMCGGQEN-UHFFFAOYSA-N	392095	US10301272, Example 8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392095	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392095&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548243	404960435							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783639	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O4S2/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	ZWTAWYCVVALKKE-UHFFFAOYSA-N	392096	US10301272, Example 8/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392096&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548472	404960436							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783640	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O4S2/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	ZWTAWYCVVALKKE-UHFFFAOYSA-N	392096	US10301272, Example 8/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392096&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548472	404960436							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783641	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O4S2/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	ZWTAWYCVVALKKE-UHFFFAOYSA-N	392096	US10301272, Example 8/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392096	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392096&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548472	404960436							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783642	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(N)=O)c2ccccc12	InChI=1S/C25H31N3O3S2/c1-25(2,3)28-33(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(27-24(32-22)23(26)29)15-16-9-5-4-6-10-16/h7-8,11-14,16,28H,4-6,9-10,15H2,1-3H3,(H2,26,29)	UYKPRQBCYSIDQS-UHFFFAOYSA-N	392097	US10301272, Example 8/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392097&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185740	404960437							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783643	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(N)=O)c2ccccc12	InChI=1S/C25H31N3O3S2/c1-25(2,3)28-33(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(27-24(32-22)23(26)29)15-16-9-5-4-6-10-16/h7-8,11-14,16,28H,4-6,9-10,15H2,1-3H3,(H2,26,29)	UYKPRQBCYSIDQS-UHFFFAOYSA-N	392097	US10301272, Example 8/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392097&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185740	404960437							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783644	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(N)=O)c2ccccc12	InChI=1S/C25H31N3O3S2/c1-25(2,3)28-33(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(27-24(32-22)23(26)29)15-16-9-5-4-6-10-16/h7-8,11-14,16,28H,4-6,9-10,15H2,1-3H3,(H2,26,29)	UYKPRQBCYSIDQS-UHFFFAOYSA-N	392097	US10301272, Example 8/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392097&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185740	404960437							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783645	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C(N)=O	InChI=1S/C29H36N4O5S2/c1-28(2,36)17-31-25(34)26-32-22(16-18-8-4-3-5-9-18)24(39-26)21-12-13-23(20-11-7-6-10-19(20)21)40(37,38)33-29(14-15-29)27(30)35/h6-7,10-13,18,33,36H,3-5,8-9,14-17H2,1-2H3,(H2,30,35)(H,31,34)	JAYVGCFXAOQDHC-UHFFFAOYSA-N	392098	US10301272, Example 8/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392098&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185738	404960438							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783646	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C(N)=O	InChI=1S/C29H36N4O5S2/c1-28(2,36)17-31-25(34)26-32-22(16-18-8-4-3-5-9-18)24(39-26)21-12-13-23(20-11-7-6-10-19(20)21)40(37,38)33-29(14-15-29)27(30)35/h6-7,10-13,18,33,36H,3-5,8-9,14-17H2,1-2H3,(H2,30,35)(H,31,34)	JAYVGCFXAOQDHC-UHFFFAOYSA-N	392098	US10301272, Example 8/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392098&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185738	404960438							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783647	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C(N)=O	InChI=1S/C29H36N4O5S2/c1-28(2,36)17-31-25(34)26-32-22(16-18-8-4-3-5-9-18)24(39-26)21-12-13-23(20-11-7-6-10-19(20)21)40(37,38)33-29(14-15-29)27(30)35/h6-7,10-13,18,33,36H,3-5,8-9,14-17H2,1-2H3,(H2,30,35)(H,31,34)	JAYVGCFXAOQDHC-UHFFFAOYSA-N	392098	US10301272, Example 8/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392098	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392098&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185738	404960438							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783648	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C29H34N4O4S2/c1-28(2,35)18-31-26(34)27-32-23(16-19-8-4-3-5-9-19)25(38-27)22-12-13-24(21-11-7-6-10-20(21)22)39(36,37)33-29(17-30)14-15-29/h6-7,10-13,19,33,35H,3-5,8-9,14-16,18H2,1-2H3,(H,31,34)	ULYHXRTUZSKYEU-UHFFFAOYSA-N	392099	US10301272, Example 8/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392099&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185739	404960439							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783649	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C29H34N4O4S2/c1-28(2,35)18-31-26(34)27-32-23(16-19-8-4-3-5-9-19)25(38-27)22-12-13-24(21-11-7-6-10-20(21)22)39(36,37)33-29(17-30)14-15-29/h6-7,10-13,19,33,35H,3-5,8-9,14-16,18H2,1-2H3,(H,31,34)	ULYHXRTUZSKYEU-UHFFFAOYSA-N	392099	US10301272, Example 8/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392099&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185739	404960439							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783650	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C29H34N4O4S2/c1-28(2,35)18-31-26(34)27-32-23(16-19-8-4-3-5-9-19)25(38-27)22-12-13-24(21-11-7-6-10-20(21)22)39(36,37)33-29(17-30)14-15-29/h6-7,10-13,19,33,35H,3-5,8-9,14-16,18H2,1-2H3,(H,31,34)	ULYHXRTUZSKYEU-UHFFFAOYSA-N	392099	US10301272, Example 8/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392099	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392099&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185739	404960439							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783651	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)COC1	InChI=1S/C29H37N3O5S2/c1-28(2,34)16-30-26(33)27-31-23(15-19-9-5-4-6-10-19)25(38-27)22-13-14-24(21-12-8-7-11-20(21)22)39(35,36)32-29(3)17-37-18-29/h7-8,11-14,19,32,34H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ZGXGRJFUQLOGMK-UHFFFAOYSA-N	392100	US10301272, Example 8/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392100&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185741	404960440							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783652	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)COC1	InChI=1S/C29H37N3O5S2/c1-28(2,34)16-30-26(33)27-31-23(15-19-9-5-4-6-10-19)25(38-27)22-13-14-24(21-12-8-7-11-20(21)22)39(35,36)32-29(3)17-37-18-29/h7-8,11-14,19,32,34H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ZGXGRJFUQLOGMK-UHFFFAOYSA-N	392100	US10301272, Example 8/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392100&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185741	404960440							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783653	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)COC1	InChI=1S/C29H37N3O5S2/c1-28(2,34)16-30-26(33)27-31-23(15-19-9-5-4-6-10-19)25(38-27)22-13-14-24(21-12-8-7-11-20(21)22)39(35,36)32-29(3)17-37-18-29/h7-8,11-14,19,32,34H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ZGXGRJFUQLOGMK-UHFFFAOYSA-N	392100	US10301272, Example 8/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392100	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392100&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185741	404960440							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783654	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O)C(F)(F)F	InChI=1S/C29H38F3N3O3S/c1-17(29(30,31)32)34-24(36)20-13-19(14-21(15-20)28(4)10-11-28)23-22(12-18-8-6-5-7-9-18)35-26(39-23)25(37)33-16-27(2,3)38/h13-15,17-18,38H,5-12,16H2,1-4H3,(H,33,37)(H,34,36)/t17-/m0/s1	NUWGDGWMQLFHAU-KRWDZBQOSA-N	392101	US10301272, Example 8/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392101&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185742	404960441							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783655	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O)C(F)(F)F	InChI=1S/C29H38F3N3O3S/c1-17(29(30,31)32)34-24(36)20-13-19(14-21(15-20)28(4)10-11-28)23-22(12-18-8-6-5-7-9-18)35-26(39-23)25(37)33-16-27(2,3)38/h13-15,17-18,38H,5-12,16H2,1-4H3,(H,33,37)(H,34,36)/t17-/m0/s1	NUWGDGWMQLFHAU-KRWDZBQOSA-N	392101	US10301272, Example 8/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392101&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185742	404960441							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783656	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O)C(F)(F)F	InChI=1S/C29H38F3N3O3S/c1-17(29(30,31)32)34-24(36)20-13-19(14-21(15-20)28(4)10-11-28)23-22(12-18-8-6-5-7-9-18)35-26(39-23)25(37)33-16-27(2,3)38/h13-15,17-18,38H,5-12,16H2,1-4H3,(H,33,37)(H,34,36)/t17-/m0/s1	NUWGDGWMQLFHAU-KRWDZBQOSA-N	392101	US10301272, Example 8/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392101	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392101&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185742	404960441							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783657	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F	InChI=1S/C30H36F3N3O4S/c1-16(30(31,32)33)34-25(37)19-11-18(12-21(13-19)29(2)8-9-29)24-23(10-17-6-4-3-5-7-17)36-27(41-24)26(38)35-22-14-20(15-22)28(39)40/h11-13,16-17,20,22H,3-10,14-15H2,1-2H3,(H,34,37)(H,35,38)(H,39,40)/t16-,20-,22-/m0/s1	PSFPATVFAWGHAJ-BUKVSMQUSA-N	392102	US10301272, Example 8/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392102&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185743	404960442							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783658	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F	InChI=1S/C30H36F3N3O4S/c1-16(30(31,32)33)34-25(37)19-11-18(12-21(13-19)29(2)8-9-29)24-23(10-17-6-4-3-5-7-17)36-27(41-24)26(38)35-22-14-20(15-22)28(39)40/h11-13,16-17,20,22H,3-10,14-15H2,1-2H3,(H,34,37)(H,35,38)(H,39,40)/t16-,20-,22-/m0/s1	PSFPATVFAWGHAJ-BUKVSMQUSA-N	392102	US10301272, Example 8/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392102&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185743	404960442							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783659	C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F	InChI=1S/C30H36F3N3O4S/c1-16(30(31,32)33)34-25(37)19-11-18(12-21(13-19)29(2)8-9-29)24-23(10-17-6-4-3-5-7-17)36-27(41-24)26(38)35-22-14-20(15-22)28(39)40/h11-13,16-17,20,22H,3-10,14-15H2,1-2H3,(H,34,37)(H,35,38)(H,39,40)/t16-,20-,22-/m0/s1	PSFPATVFAWGHAJ-BUKVSMQUSA-N	392102	US10301272, Example 8/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392102	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392102&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185743	404960442							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783660	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3OS/c1-27(2,3)22-16-19(17-23(31-22)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(33-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	MZBIOJSXVQAYSG-UHFFFAOYSA-N	392103	US10301272, Example 8/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392103&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185744	404960443							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783661	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3OS/c1-27(2,3)22-16-19(17-23(31-22)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(33-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	MZBIOJSXVQAYSG-UHFFFAOYSA-N	392103	US10301272, Example 8/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392103&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185744	404960443							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783662	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3OS/c1-27(2,3)22-16-19(17-23(31-22)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(33-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	MZBIOJSXVQAYSG-UHFFFAOYSA-N	392103	US10301272, Example 8/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392103	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392103&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185744	404960443							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783663	CC(C)(C)c1cc(cc([n+]1[O-])C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3O2S/c1-27(2,3)22-16-19(17-23(31(22)33)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(34-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	RMGNKSLXGBISAO-UHFFFAOYSA-N	392104	US10301272, Example 8/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392104&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185745	404960444							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783664	CC(C)(C)c1cc(cc([n+]1[O-])C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3O2S/c1-27(2,3)22-16-19(17-23(31(22)33)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(34-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	RMGNKSLXGBISAO-UHFFFAOYSA-N	392104	US10301272, Example 8/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392104&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185745	404960444							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783665	CC(C)(C)c1cc(cc([n+]1[O-])C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C28H41N3O2S/c1-27(2,3)22-16-19(17-23(31(22)33)28(4,5)6)24-21(15-18-11-8-7-9-12-18)30-26(34-24)25(32)29-20-13-10-14-20/h16-18,20H,7-15H2,1-6H3,(H,29,32)	RMGNKSLXGBISAO-UHFFFAOYSA-N	392104	US10301272, Example 8/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392104	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392104&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185745	404960444							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783666	CC(C)(C)c1cc(cc(n1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C27H39N3O2S/c1-26(2,3)21-15-18(16-22(30-21)27(4,5)32)23-20(14-17-10-7-6-8-11-17)29-25(33-23)24(31)28-19-12-9-13-19/h15-17,19,32H,6-14H2,1-5H3,(H,28,31)	NWKJFXLCOITAKC-UHFFFAOYSA-N	392105	US10301272, Example 8/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392105&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185748	404960445							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783667	CC(C)(C)c1cc(cc(n1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C27H39N3O2S/c1-26(2,3)21-15-18(16-22(30-21)27(4,5)32)23-20(14-17-10-7-6-8-11-17)29-25(33-23)24(31)28-19-12-9-13-19/h15-17,19,32H,6-14H2,1-5H3,(H,28,31)	NWKJFXLCOITAKC-UHFFFAOYSA-N	392105	US10301272, Example 8/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392105&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185748	404960445							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783668	CC(C)(C)c1cc(cc(n1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCC1	InChI=1S/C27H39N3O2S/c1-26(2,3)21-15-18(16-22(30-21)27(4,5)32)23-20(14-17-10-7-6-8-11-17)29-25(33-23)24(31)28-19-12-9-13-19/h15-17,19,32H,6-14H2,1-5H3,(H,28,31)	NWKJFXLCOITAKC-UHFFFAOYSA-N	392105	US10301272, Example 8/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392105	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392105&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185748	404960445							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783669	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12)C(F)(F)F	InChI=1S/C28H32F3N3O5S3/c1-17(28(29,30)31)34-42(38,39)24-11-10-22(20-8-4-5-9-21(20)24)25-23(16-18-6-2-3-7-18)33-27(40-25)26(35)32-19-12-14-41(36,37)15-13-19/h4-5,8-11,17-19,34H,2-3,6-7,12-16H2,1H3,(H,32,35)	BMTBKQOKRUJGCA-UHFFFAOYSA-N	392106	US10301272, Example 8/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392106&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123344921	404960446							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783670	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12)C(F)(F)F	InChI=1S/C28H32F3N3O5S3/c1-17(28(29,30)31)34-42(38,39)24-11-10-22(20-8-4-5-9-21(20)24)25-23(16-18-6-2-3-7-18)33-27(40-25)26(35)32-19-12-14-41(36,37)15-13-19/h4-5,8-11,17-19,34H,2-3,6-7,12-16H2,1H3,(H,32,35)	BMTBKQOKRUJGCA-UHFFFAOYSA-N	392106	US10301272, Example 8/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392106	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392106&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123344921	404960446							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783671	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl)C(F)(F)F	InChI=1S/C24H28Cl2F3N3O5S3/c1-13(24(27,28)29)32-40(36,37)18-7-6-16(19(25)20(18)26)21-17(12-14-4-2-3-5-14)31-23(38-21)22(33)30-15-8-10-39(34,35)11-9-15/h6-7,13-15,32H,2-5,8-12H2,1H3,(H,30,33)	LEWIKIBRQPAJFI-UHFFFAOYSA-N	392107	US10301272, Example 8/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392107&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123676361	404960447							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783672	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl)C(F)(F)F	InChI=1S/C24H28Cl2F3N3O5S3/c1-13(24(27,28)29)32-40(36,37)18-7-6-16(19(25)20(18)26)21-17(12-14-4-2-3-5-14)31-23(38-21)22(33)30-15-8-10-39(34,35)11-9-15/h6-7,13-15,32H,2-5,8-12H2,1H3,(H,30,33)	LEWIKIBRQPAJFI-UHFFFAOYSA-N	392107	US10301272, Example 8/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392107	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392107&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			123676361	404960447							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783673	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C27H36F3N3O4S2/c1-26(2,3)33-39(35,36)22-10-9-18(16-20(22)27(28,29)30)23-21(15-17-7-5-4-6-8-17)32-25(38-23)24(34)31-19-11-13-37-14-12-19/h9-10,16-17,19,33H,4-8,11-15H2,1-3H3,(H,31,34)	JWUWUNHNLFWXMX-UHFFFAOYSA-N	392108	US10301272, Example 9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392108&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160496	404960448							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783674	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C27H36F3N3O4S2/c1-26(2,3)33-39(35,36)22-10-9-18(16-20(22)27(28,29)30)23-21(15-17-7-5-4-6-8-17)32-25(38-23)24(34)31-19-11-13-37-14-12-19/h9-10,16-17,19,33H,4-8,11-15H2,1-3H3,(H,31,34)	JWUWUNHNLFWXMX-UHFFFAOYSA-N	392108	US10301272, Example 9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392108&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160496	404960448							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783675	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C27H36F3N3O4S2/c1-26(2,3)33-39(35,36)22-10-9-18(16-20(22)27(28,29)30)23-21(15-17-7-5-4-6-8-17)32-25(38-23)24(34)31-19-11-13-37-14-12-19/h9-10,16-17,19,33H,4-8,11-15H2,1-3H3,(H,31,34)	JWUWUNHNLFWXMX-UHFFFAOYSA-N	392108	US10301272, Example 9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392108	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392108&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160496	404960448							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783676	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C28H38F3N3O5S2/c1-26(2,3)34-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)33-24(40-22)23(35)32-14-13-27(4,5)25(36)37/h11-12,16-17,34H,6-10,13-15H2,1-5H3,(H,32,35)(H,36,37)	OFKXJNBDQLJIEH-UHFFFAOYSA-N	392109	US10301272, Example 9/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392109&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548474	404960449							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783677	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C28H38F3N3O5S2/c1-26(2,3)34-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)33-24(40-22)23(35)32-14-13-27(4,5)25(36)37/h11-12,16-17,34H,6-10,13-15H2,1-5H3,(H,32,35)(H,36,37)	OFKXJNBDQLJIEH-UHFFFAOYSA-N	392109	US10301272, Example 9/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392109&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548474	404960449							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783678	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(O)=O	InChI=1S/C28H38F3N3O5S2/c1-26(2,3)34-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)33-24(40-22)23(35)32-14-13-27(4,5)25(36)37/h11-12,16-17,34H,6-10,13-15H2,1-5H3,(H,32,35)(H,36,37)	OFKXJNBDQLJIEH-UHFFFAOYSA-N	392109	US10301272, Example 9/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392109	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392109&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548474	404960449							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783679	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H34F3N3O5S2/c1-26(2,3)33-40(37,38)21-10-9-16(14-19(21)27(28,29)30)22-20(11-15-7-5-4-6-8-15)32-24(39-22)23(34)31-18-12-17(13-18)25(35)36/h9-10,14-15,17-18,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t17-,18-	FZWSPVXAVWAUFE-IYARVYRRSA-N	392110	US10301272, Example 9/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392110&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548476	404960450							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783680	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H34F3N3O5S2/c1-26(2,3)33-40(37,38)21-10-9-16(14-19(21)27(28,29)30)22-20(11-15-7-5-4-6-8-15)32-24(39-22)23(34)31-18-12-17(13-18)25(35)36/h9-10,14-15,17-18,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t17-,18-	FZWSPVXAVWAUFE-IYARVYRRSA-N	392110	US10301272, Example 9/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392110&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548476	404960450							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783681	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H34F3N3O5S2/c1-26(2,3)33-40(37,38)21-10-9-16(14-19(21)27(28,29)30)22-20(11-15-7-5-4-6-8-15)32-24(39-22)23(34)31-18-12-17(13-18)25(35)36/h9-10,14-15,17-18,33H,4-8,11-13H2,1-3H3,(H,31,34)(H,35,36)/t17-,18-	FZWSPVXAVWAUFE-IYARVYRRSA-N	392110	US10301272, Example 9/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392110	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392110&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548476	404960450							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783682	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C27H36F3N3O5S2/c1-25(2,3)33-40(37,38)20-12-11-17(14-18(20)27(28,29)30)21-19(13-16-9-7-6-8-10-16)32-23(39-21)22(34)31-15-26(4,5)24(35)36/h11-12,14,16,33H,6-10,13,15H2,1-5H3,(H,31,34)(H,35,36)	FUBAKJMPHVUXBS-UHFFFAOYSA-N	392111	US10301272, Example 9/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392111&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548702	404960451							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783683	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C27H36F3N3O5S2/c1-25(2,3)33-40(37,38)20-12-11-17(14-18(20)27(28,29)30)21-19(13-16-9-7-6-8-10-16)32-23(39-21)22(34)31-15-26(4,5)24(35)36/h11-12,14,16,33H,6-10,13,15H2,1-5H3,(H,31,34)(H,35,36)	FUBAKJMPHVUXBS-UHFFFAOYSA-N	392111	US10301272, Example 9/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392111&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548702	404960451							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783684	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C27H36F3N3O5S2/c1-25(2,3)33-40(37,38)20-12-11-17(14-18(20)27(28,29)30)21-19(13-16-9-7-6-8-10-16)32-23(39-21)22(34)31-15-26(4,5)24(35)36/h11-12,14,16,33H,6-10,13,15H2,1-5H3,(H,31,34)(H,35,36)	FUBAKJMPHVUXBS-UHFFFAOYSA-N	392111	US10301272, Example 9/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392111	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392111&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548702	404960451							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783685	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22-	BTLDXMQHMJIEKL-XYWHTSSQSA-N	392112	US10301272, Example 9/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392112&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960452							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783686	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22-	BTLDXMQHMJIEKL-XYWHTSSQSA-N	392112	US10301272, Example 9/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392112&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960452							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783687	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22-	BTLDXMQHMJIEKL-XYWHTSSQSA-N	392112	US10301272, Example 9/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392112	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392112&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960452							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783688	COC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4S/c1-29(2,36-4)21-13-19(14-22(17-21)30(3)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(37-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	VOXBBILGZNLHCC-JKIUYZKVSA-N	392113	US10301272, Example 9/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392113&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185749	404960453							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783689	COC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4S/c1-29(2,36-4)21-13-19(14-22(17-21)30(3)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(37-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	VOXBBILGZNLHCC-JKIUYZKVSA-N	392113	US10301272, Example 9/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392113&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185749	404960453							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783690	COC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4S/c1-29(2,36-4)21-13-19(14-22(17-21)30(3)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(37-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	VOXBBILGZNLHCC-JKIUYZKVSA-N	392113	US10301272, Example 9/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392113	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392113&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185749	404960453							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783691	CC(C)(C)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H41N3O4S/c1-30(2,3)34-26(35)20-13-19(14-22(15-20)31(4)10-11-31)25-24(12-18-8-6-5-7-9-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,5-12,16-17H2,1-4H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	VTRHQLPYGVWKKI-AFARHQOCSA-N	392114	US10301272, Example 9/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392114&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185750	404960454							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783692	CC(C)(C)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H41N3O4S/c1-30(2,3)34-26(35)20-13-19(14-22(15-20)31(4)10-11-31)25-24(12-18-8-6-5-7-9-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,5-12,16-17H2,1-4H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	VTRHQLPYGVWKKI-AFARHQOCSA-N	392114	US10301272, Example 9/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392114&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185750	404960454							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783693	CC(C)(C)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H41N3O4S/c1-30(2,3)34-26(35)20-13-19(14-22(15-20)31(4)10-11-31)25-24(12-18-8-6-5-7-9-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,5-12,16-17H2,1-4H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	VTRHQLPYGVWKKI-AFARHQOCSA-N	392114	US10301272, Example 9/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392114	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392114&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185750	404960454							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783694	CC(C)(C)NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H43N3O4S/c1-30(2,3)22-14-19(13-20(15-22)26(35)34-31(4,5)6)25-24(12-18-10-8-7-9-11-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,7-12,16-17H2,1-6H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	DDZIKIFYYJUAJN-AFARHQOCSA-N	392115	US10301272, Example 9/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392115&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185751	404960455							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783695	CC(C)(C)NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H43N3O4S/c1-30(2,3)22-14-19(13-20(15-22)26(35)34-31(4,5)6)25-24(12-18-10-8-7-9-11-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,7-12,16-17H2,1-6H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	DDZIKIFYYJUAJN-AFARHQOCSA-N	392115	US10301272, Example 9/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392115&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185751	404960455							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783696	CC(C)(C)NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H43N3O4S/c1-30(2,3)22-14-19(13-20(15-22)26(35)34-31(4,5)6)25-24(12-18-10-8-7-9-11-18)33-28(39-25)27(36)32-23-16-21(17-23)29(37)38/h13-15,18,21,23H,7-12,16-17H2,1-6H3,(H,32,36)(H,34,35)(H,37,38)/t21-,23-	DDZIKIFYYJUAJN-AFARHQOCSA-N	392115	US10301272, Example 9/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392115	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392115&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185751	404960455							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783697	CC1(CC1)c1cc(cc(c1)C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H31F3N2O3S/c1-26(7-8-26)18-10-16(11-19(14-18)27(28,29)30)22-21(9-15-5-3-2-4-6-15)32-24(36-22)23(33)31-20-12-17(13-20)25(34)35/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,31,33)(H,34,35)/t17-,20-	VJGOHHGFZCULJT-IRJFHVNHSA-N	392116	US10301272, Example 9/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392116&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185752	404960456							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783698	CC1(CC1)c1cc(cc(c1)C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H31F3N2O3S/c1-26(7-8-26)18-10-16(11-19(14-18)27(28,29)30)22-21(9-15-5-3-2-4-6-15)32-24(36-22)23(33)31-20-12-17(13-20)25(34)35/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,31,33)(H,34,35)/t17-,20-	VJGOHHGFZCULJT-IRJFHVNHSA-N	392116	US10301272, Example 9/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392116&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185752	404960456							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783699	CC1(CC1)c1cc(cc(c1)C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H31F3N2O3S/c1-26(7-8-26)18-10-16(11-19(14-18)27(28,29)30)22-21(9-15-5-3-2-4-6-15)32-24(36-22)23(33)31-20-12-17(13-20)25(34)35/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,31,33)(H,34,35)/t17-,20-	VJGOHHGFZCULJT-IRJFHVNHSA-N	392116	US10301272, Example 9/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392116	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392116&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185752	404960456							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783700	CC1(CC1)c1cc(Cl)cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C26H31ClN2O3S/c1-26(7-8-26)18-10-16(11-19(27)14-18)22-21(9-15-5-3-2-4-6-15)29-24(33-22)23(30)28-20-12-17(13-20)25(31)32/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,28,30)(H,31,32)/t17-,20-	HZWFAWJNOHBDRP-IRJFHVNHSA-N	392117	US10301272, Example 9/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3981							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392117&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185753	404960457							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783701	CC1(CC1)c1cc(Cl)cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C26H31ClN2O3S/c1-26(7-8-26)18-10-16(11-19(27)14-18)22-21(9-15-5-3-2-4-6-15)29-24(33-22)23(30)28-20-12-17(13-20)25(31)32/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,28,30)(H,31,32)/t17-,20-	HZWFAWJNOHBDRP-IRJFHVNHSA-N	392117	US10301272, Example 9/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392117&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185753	404960457							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783702	CC1(CC1)c1cc(Cl)cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C26H31ClN2O3S/c1-26(7-8-26)18-10-16(11-19(27)14-18)22-21(9-15-5-3-2-4-6-15)29-24(33-22)23(30)28-20-12-17(13-20)25(31)32/h10-11,14-15,17,20H,2-9,12-13H2,1H3,(H,28,30)(H,31,32)/t17-,20-	HZWFAWJNOHBDRP-IRJFHVNHSA-N	392117	US10301272, Example 9/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392117	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392117&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185753	404960457							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783703	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22+	BTLDXMQHMJIEKL-IQGASKDCSA-N	392118	US10301272, Example 9/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392118&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960458							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783704	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22+	BTLDXMQHMJIEKL-IQGASKDCSA-N	392118	US10301272, Example 9/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392118&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960458							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783705	CC(C)(O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@H](C1)C(O)=O	InChI=1S/C29H38N2O4S/c1-28(2,35)20-12-18(13-21(16-20)29(3)9-10-29)24-23(11-17-7-5-4-6-8-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,4-11,14-15H2,1-3H3,(H,30,32)(H,33,34)/t19-,22+	BTLDXMQHMJIEKL-IQGASKDCSA-N	392118	US10301272, Example 9/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392118	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392118&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548475	404960458							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783706	CC(C)(C)NS(=O)(=O)c1ccc(c2CCCc12)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H39N3O5S2/c1-29(2,3)32-39(36,37)24-13-12-22(20-10-7-11-21(20)24)25-23(14-17-8-5-4-6-9-17)31-27(38-25)26(33)30-19-15-18(16-19)28(34)35/h12-13,17-19,32H,4-11,14-16H2,1-3H3,(H,30,33)(H,34,35)/t18-,19-	DZVATTBWRSFOMO-WGSAOQKQSA-N	392119	US10301272, Example 9/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392119&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185754	404960459							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783707	CC(C)(C)NS(=O)(=O)c1ccc(c2CCCc12)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H39N3O5S2/c1-29(2,3)32-39(36,37)24-13-12-22(20-10-7-11-21(20)24)25-23(14-17-8-5-4-6-9-17)31-27(38-25)26(33)30-19-15-18(16-19)28(34)35/h12-13,17-19,32H,4-11,14-16H2,1-3H3,(H,30,33)(H,34,35)/t18-,19-	DZVATTBWRSFOMO-WGSAOQKQSA-N	392119	US10301272, Example 9/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392119&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185754	404960459							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783708	CC(C)(C)NS(=O)(=O)c1ccc(c2CCCc12)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C29H39N3O5S2/c1-29(2,3)32-39(36,37)24-13-12-22(20-10-7-11-21(20)24)25-23(14-17-8-5-4-6-9-17)31-27(38-25)26(33)30-19-15-18(16-19)28(34)35/h12-13,17-19,32H,4-11,14-16H2,1-3H3,(H,30,33)(H,34,35)/t18-,19-	DZVATTBWRSFOMO-WGSAOQKQSA-N	392119	US10301272, Example 9/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392119	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392119&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185754	404960459							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783709	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(N)=O	InChI=1S/C28H39F3N4O4S2/c1-26(2,3)35-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)34-24(40-22)23(36)33-14-13-27(4,5)25(32)37/h11-12,16-17,35H,6-10,13-15H2,1-5H3,(H2,32,37)(H,33,36)	JRDSVVBMAHUIRK-UHFFFAOYSA-N	392120	US10301272, Example 10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392120&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160611	404960460							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783710	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(N)=O	InChI=1S/C28H39F3N4O4S2/c1-26(2,3)35-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)34-24(40-22)23(36)33-14-13-27(4,5)25(32)37/h11-12,16-17,35H,6-10,13-15H2,1-5H3,(H2,32,37)(H,33,36)	JRDSVVBMAHUIRK-UHFFFAOYSA-N	392120	US10301272, Example 10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392120&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160611	404960460							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783711	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NCCC(C)(C)C(N)=O	InChI=1S/C28H39F3N4O4S2/c1-26(2,3)35-41(38,39)21-12-11-18(16-19(21)28(29,30)31)22-20(15-17-9-7-6-8-10-17)34-24(40-22)23(36)33-14-13-27(4,5)25(32)37/h11-12,16-17,35H,6-10,13-15H2,1-5H3,(H2,32,37)(H,33,36)	JRDSVVBMAHUIRK-UHFFFAOYSA-N	392120	US10301272, Example 10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392120	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392120&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160611	404960460							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783712	CNC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C29H41F3N4O4S2/c1-27(2,3)36-42(39,40)22-13-12-19(17-20(22)29(30,31)32)23-21(16-18-10-8-7-9-11-18)35-25(41-23)24(37)34-15-14-28(4,5)26(38)33-6/h12-13,17-18,36H,7-11,14-16H2,1-6H3,(H,33,38)(H,34,37)	KGXUZXYXWMATRZ-UHFFFAOYSA-N	392121	US10301272, Example 10/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392121&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185755	404960461							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783713	CNC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C29H41F3N4O4S2/c1-27(2,3)36-42(39,40)22-13-12-19(17-20(22)29(30,31)32)23-21(16-18-10-8-7-9-11-18)35-25(41-23)24(37)34-15-14-28(4,5)26(38)33-6/h12-13,17-18,36H,7-11,14-16H2,1-6H3,(H,33,38)(H,34,37)	KGXUZXYXWMATRZ-UHFFFAOYSA-N	392121	US10301272, Example 10/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392121&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185755	404960461							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783714	CNC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C29H41F3N4O4S2/c1-27(2,3)36-42(39,40)22-13-12-19(17-20(22)29(30,31)32)23-21(16-18-10-8-7-9-11-18)35-25(41-23)24(37)34-15-14-28(4,5)26(38)33-6/h12-13,17-18,36H,7-11,14-16H2,1-6H3,(H,33,38)(H,34,37)	KGXUZXYXWMATRZ-UHFFFAOYSA-N	392121	US10301272, Example 10/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392121&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185755	404960461							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783715	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)C(=O)NC1(CC1)C#N	InChI=1S/C31H38N4O4S2/c1-30(9-10-30)23-17-21(16-22(18-23)27(36)35-31(19-32)11-12-31)26-25(15-20-5-3-2-4-6-20)34-29(40-26)28(37)33-24-7-13-41(38,39)14-8-24/h16-18,20,24H,2-15H2,1H3,(H,33,37)(H,35,36)	JPHNKXPYJOQEDP-UHFFFAOYSA-N	392122	US10301272, Example 10/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392122&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188670	404960462							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783716	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)C(=O)NC1(CC1)C#N	InChI=1S/C31H38N4O4S2/c1-30(9-10-30)23-17-21(16-22(18-23)27(36)35-31(19-32)11-12-31)26-25(15-20-5-3-2-4-6-20)34-29(40-26)28(37)33-24-7-13-41(38,39)14-8-24/h16-18,20,24H,2-15H2,1H3,(H,33,37)(H,35,36)	JPHNKXPYJOQEDP-UHFFFAOYSA-N	392122	US10301272, Example 10/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392122&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188670	404960462							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783717	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)C(=O)NC1(CC1)C#N	InChI=1S/C31H38N4O4S2/c1-30(9-10-30)23-17-21(16-22(18-23)27(36)35-31(19-32)11-12-31)26-25(15-20-5-3-2-4-6-20)34-29(40-26)28(37)33-24-7-13-41(38,39)14-8-24/h16-18,20,24H,2-15H2,1H3,(H,33,37)(H,35,36)	JPHNKXPYJOQEDP-UHFFFAOYSA-N	392122	US10301272, Example 10/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392122	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392122&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188670	404960462							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783718	CC(C)(CCO)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C32H45N3O5S2/c1-31(2,13-14-36)35-28(37)23-18-22(19-24(20-23)32(3)11-12-32)27-26(17-21-7-5-4-6-8-21)34-30(41-27)29(38)33-25-9-15-42(39,40)16-10-25/h18-21,25,36H,4-17H2,1-3H3,(H,33,38)(H,35,37)	MHMWKIAJTIUBPF-UHFFFAOYSA-N	392123	US10301272, Example 10/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392123&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185756	404960463							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783719	CC(C)(CCO)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C32H45N3O5S2/c1-31(2,13-14-36)35-28(37)23-18-22(19-24(20-23)32(3)11-12-32)27-26(17-21-7-5-4-6-8-21)34-30(41-27)29(38)33-25-9-15-42(39,40)16-10-25/h18-21,25,36H,4-17H2,1-3H3,(H,33,38)(H,35,37)	MHMWKIAJTIUBPF-UHFFFAOYSA-N	392123	US10301272, Example 10/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392123	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392123&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185756	404960463							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783720	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)C(=O)NC1(C)COC1	InChI=1S/C31H41N3O5S2/c1-30(10-11-30)23-16-21(15-22(17-23)27(35)34-31(2)18-39-19-31)26-25(14-20-6-4-3-5-7-20)33-29(40-26)28(36)32-24-8-12-41(37,38)13-9-24/h15-17,20,24H,3-14,18-19H2,1-2H3,(H,32,36)(H,34,35)	JRISJHRKXUDAMA-UHFFFAOYSA-N	392124	US10301272, Example 10/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392124&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185758	404960464							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783721	CC1(CC1)c1cc(cc(c1)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)C(=O)NC1(C)COC1	InChI=1S/C31H41N3O5S2/c1-30(10-11-30)23-16-21(15-22(17-23)27(35)34-31(2)18-39-19-31)26-25(14-20-6-4-3-5-7-20)33-29(40-26)28(36)32-24-8-12-41(37,38)13-9-24/h15-17,20,24H,3-14,18-19H2,1-2H3,(H,32,36)(H,34,35)	JRISJHRKXUDAMA-UHFFFAOYSA-N	392124	US10301272, Example 10/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392124	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392124&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185758	404960464							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783722	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(=O)(=O)NC(=O)OCc1ccccc1	InChI=1S/C32H40N2O4S2/c1-31(2,3)25-18-24(19-26(20-25)32(4)15-16-32)28-27(17-22-11-7-5-8-12-22)33-30(39-28)40(36,37)34-29(35)38-21-23-13-9-6-10-14-23/h6,9-10,13-14,18-20,22H,5,7-8,11-12,15-17,21H2,1-4H3,(H,34,35)	UGQSIGPRQDJPLC-UHFFFAOYSA-N	392125	US10301272, Example 12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3162							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392125&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185757	404960465							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783723	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(=O)(=O)NC(=O)OCc1ccccc1	InChI=1S/C32H40N2O4S2/c1-31(2,3)25-18-24(19-26(20-25)32(4)15-16-32)28-27(17-22-11-7-5-8-12-22)33-30(39-28)40(36,37)34-29(35)38-21-23-13-9-6-10-14-23/h6,9-10,13-14,18-20,22H,5,7-8,11-12,15-17,21H2,1-4H3,(H,34,35)	UGQSIGPRQDJPLC-UHFFFAOYSA-N	392125	US10301272, Example 12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392125&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185757	404960465							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783724	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(=O)(=O)NC(=O)OCc1ccccc1	InChI=1S/C32H40N2O4S2/c1-31(2,3)25-18-24(19-26(20-25)32(4)15-16-32)28-27(17-22-11-7-5-8-12-22)33-30(39-28)40(36,37)34-29(35)38-21-23-13-9-6-10-14-23/h6,9-10,13-14,18-20,22H,5,7-8,11-12,15-17,21H2,1-4H3,(H,34,35)	UGQSIGPRQDJPLC-UHFFFAOYSA-N	392125	US10301272, Example 12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392125	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392125&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185757	404960465							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783725	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H34N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4)10-11-24)21-20(12-16-8-6-5-7-9-16)26-22(29-21)30(25,27)28/h13-16H,5-12H2,1-4H3,(H2,25,27,28)	SCLLYLVVVRMEME-UHFFFAOYSA-N	392126	US10301272, Example 13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392126&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026255	404960466							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783726	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H34N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4)10-11-24)21-20(12-16-8-6-5-7-9-16)26-22(29-21)30(25,27)28/h13-16H,5-12H2,1-4H3,(H2,25,27,28)	SCLLYLVVVRMEME-UHFFFAOYSA-N	392126	US10301272, Example 13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392126&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026255	404960466							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783727	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H34N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4)10-11-24)21-20(12-16-8-6-5-7-9-16)26-22(29-21)30(25,27)28/h13-16H,5-12H2,1-4H3,(H2,25,27,28)	SCLLYLVVVRMEME-UHFFFAOYSA-N	392126	US10301272, Example 13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392126	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392126&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026255	404960466							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783728	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H37N3O4S3/c1-23(2,3)18-15-17(12-13-20(18)34(30,31)27-24(4,5)6)21-19(14-16-10-8-7-9-11-16)26-22(32-21)33(25,28)29/h12-13,15-16,27H,7-11,14H2,1-6H3,(H2,25,28,29)	BFTKANFGFHYDND-UHFFFAOYSA-N	392127	US10301272, Example 13/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392127&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185759	404960467							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783729	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H37N3O4S3/c1-23(2,3)18-15-17(12-13-20(18)34(30,31)27-24(4,5)6)21-19(14-16-10-8-7-9-11-16)26-22(32-21)33(25,28)29/h12-13,15-16,27H,7-11,14H2,1-6H3,(H2,25,28,29)	BFTKANFGFHYDND-UHFFFAOYSA-N	392127	US10301272, Example 13/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392127&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185759	404960467							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783730	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H37N3O4S3/c1-23(2,3)18-15-17(12-13-20(18)34(30,31)27-24(4,5)6)21-19(14-16-10-8-7-9-11-16)26-22(32-21)33(25,28)29/h12-13,15-16,27H,7-11,14H2,1-6H3,(H2,25,28,29)	BFTKANFGFHYDND-UHFFFAOYSA-N	392127	US10301272, Example 13/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392127	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392127&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185759	404960467							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783731	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C21H28F3N3O4S3/c1-20(2,3)27-34(30,31)17-10-9-14(12-15(17)21(22,23)24)18-16(11-13-7-5-4-6-8-13)26-19(32-18)33(25,28)29/h9-10,12-13,27H,4-8,11H2,1-3H3,(H2,25,28,29)	MZHMHJVDYMYWNZ-UHFFFAOYSA-N	392128	US10301272, Example 13/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392128&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185760	404960468							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783732	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C21H28F3N3O4S3/c1-20(2,3)27-34(30,31)17-10-9-14(12-15(17)21(22,23)24)18-16(11-13-7-5-4-6-8-13)26-19(32-18)33(25,28)29/h9-10,12-13,27H,4-8,11H2,1-3H3,(H2,25,28,29)	MZHMHJVDYMYWNZ-UHFFFAOYSA-N	392128	US10301272, Example 13/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392128&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185760	404960468							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783733	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C21H28F3N3O4S3/c1-20(2,3)27-34(30,31)17-10-9-14(12-15(17)21(22,23)24)18-16(11-13-7-5-4-6-8-13)26-19(32-18)33(25,28)29/h9-10,12-13,27H,4-8,11H2,1-3H3,(H2,25,28,29)	MZHMHJVDYMYWNZ-UHFFFAOYSA-N	392128	US10301272, Example 13/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392128	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392128&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185760	404960468							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783734	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)S(N)(=O)=O)c2ccccc12	InChI=1S/C24H31N3O4S3/c1-24(2,3)27-34(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(15-16-9-5-4-6-10-16)26-23(32-22)33(25,28)29/h7-8,11-14,16,27H,4-6,9-10,15H2,1-3H3,(H2,25,28,29)	IKEMCWXULXPXQF-UHFFFAOYSA-N	392129	US10301272, Example 13/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392129&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185761	404960469							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783735	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)S(N)(=O)=O)c2ccccc12	InChI=1S/C24H31N3O4S3/c1-24(2,3)27-34(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(15-16-9-5-4-6-10-16)26-23(32-22)33(25,28)29/h7-8,11-14,16,27H,4-6,9-10,15H2,1-3H3,(H2,25,28,29)	IKEMCWXULXPXQF-UHFFFAOYSA-N	392129	US10301272, Example 13/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392129&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185761	404960469							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783736	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)S(N)(=O)=O)c2ccccc12	InChI=1S/C24H31N3O4S3/c1-24(2,3)27-34(30,31)21-14-13-19(17-11-7-8-12-18(17)21)22-20(15-16-9-5-4-6-10-16)26-23(32-22)33(25,28)29/h7-8,11-14,16,27H,4-6,9-10,15H2,1-3H3,(H2,25,28,29)	IKEMCWXULXPXQF-UHFFFAOYSA-N	392129	US10301272, Example 13/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392129	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392129&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185761	404960469							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783737	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C32H36N4O5S3/c33-19-32(12-13-32)35-44(40,41)27-11-10-25(23-8-4-5-9-24(23)27)28-26(18-22-6-2-1-3-7-22)34-29(42-28)30(37)36-20-31(21-36)14-16-43(38,39)17-15-31/h4-5,8-11,22,35H,1-3,6-7,12-18,20-21H2	AOEHKKQBIXCNHG-UHFFFAOYSA-N	392130	US10301272, Example 14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392130&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160517	404960470							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783738	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C32H36N4O5S3/c33-19-32(12-13-32)35-44(40,41)27-11-10-25(23-8-4-5-9-24(23)27)28-26(18-22-6-2-1-3-7-22)34-29(42-28)30(37)36-20-31(21-36)14-16-43(38,39)17-15-31/h4-5,8-11,22,35H,1-3,6-7,12-18,20-21H2	AOEHKKQBIXCNHG-UHFFFAOYSA-N	392130	US10301272, Example 14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392130&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160517	404960470							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783739	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N	InChI=1S/C32H36N4O5S3/c33-19-32(12-13-32)35-44(40,41)27-11-10-25(23-8-4-5-9-24(23)27)28-26(18-22-6-2-1-3-7-22)34-29(42-28)30(37)36-20-31(21-36)14-16-43(38,39)17-15-31/h4-5,8-11,22,35H,1-3,6-7,12-18,20-21H2	AOEHKKQBIXCNHG-UHFFFAOYSA-N	392130	US10301272, Example 14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392130	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392130&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160517	404960470							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783740	CC(C)(CO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S3/c1-31(2,21-36)34-44(40,41)27-13-12-25(23-10-6-7-11-24(23)27)28-26(18-22-8-4-3-5-9-22)33-29(42-28)30(37)35-19-32(20-35)14-16-43(38,39)17-15-32/h6-7,10-13,22,34,36H,3-5,8-9,14-21H2,1-2H3	XSMXICVDYDSEDP-UHFFFAOYSA-N	392131	US10301272, Example 14/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392131&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185762	404960471							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783741	CC(C)(CO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S3/c1-31(2,21-36)34-44(40,41)27-13-12-25(23-10-6-7-11-24(23)27)28-26(18-22-8-4-3-5-9-22)33-29(42-28)30(37)35-19-32(20-35)14-16-43(38,39)17-15-32/h6-7,10-13,22,34,36H,3-5,8-9,14-21H2,1-2H3	XSMXICVDYDSEDP-UHFFFAOYSA-N	392131	US10301272, Example 14/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392131&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185762	404960471							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783742	CC(C)(CO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S3/c1-31(2,21-36)34-44(40,41)27-13-12-25(23-10-6-7-11-24(23)27)28-26(18-22-8-4-3-5-9-22)33-29(42-28)30(37)35-19-32(20-35)14-16-43(38,39)17-15-32/h6-7,10-13,22,34,36H,3-5,8-9,14-21H2,1-2H3	XSMXICVDYDSEDP-UHFFFAOYSA-N	392131	US10301272, Example 14/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392131	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392131&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185762	404960471							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783743	COCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C33H43N3O6S3/c1-32(2,22-42-3)35-45(40,41)28-14-13-26(24-11-7-8-12-25(24)28)29-27(19-23-9-5-4-6-10-23)34-30(43-29)31(37)36-20-33(21-36)15-17-44(38,39)18-16-33/h7-8,11-14,23,35H,4-6,9-10,15-22H2,1-3H3	NACMOKWDNCZRSL-UHFFFAOYSA-N	392132	US10301272, Example 14/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392132&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185763	404960472							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783744	COCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C33H43N3O6S3/c1-32(2,22-42-3)35-45(40,41)28-14-13-26(24-11-7-8-12-25(24)28)29-27(19-23-9-5-4-6-10-23)34-30(43-29)31(37)36-20-33(21-36)15-17-44(38,39)18-16-33/h7-8,11-14,23,35H,4-6,9-10,15-22H2,1-3H3	NACMOKWDNCZRSL-UHFFFAOYSA-N	392132	US10301272, Example 14/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392132&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185763	404960472							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783745	COCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C33H43N3O6S3/c1-32(2,22-42-3)35-45(40,41)28-14-13-26(24-11-7-8-12-25(24)28)29-27(19-23-9-5-4-6-10-23)34-30(43-29)31(37)36-20-33(21-36)15-17-44(38,39)18-16-33/h7-8,11-14,23,35H,4-6,9-10,15-22H2,1-3H3	NACMOKWDNCZRSL-UHFFFAOYSA-N	392132	US10301272, Example 14/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392132	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392132&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185763	404960472							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783746	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CS(=O)(=O)C1	InChI=1S/C31H37N3O7S4/c35-30(34-19-31(20-34)12-14-43(36,37)15-13-31)29-32-26(16-21-6-2-1-3-7-21)28(42-29)25-10-11-27(24-9-5-4-8-23(24)25)45(40,41)33-22-17-44(38,39)18-22/h4-5,8-11,21-22,33H,1-3,6-7,12-20H2	GZUJRVKHQTXPIB-UHFFFAOYSA-N	392133	US10301272, Example 14/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392133&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185764	404960473							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783747	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CS(=O)(=O)C1	InChI=1S/C31H37N3O7S4/c35-30(34-19-31(20-34)12-14-43(36,37)15-13-31)29-32-26(16-21-6-2-1-3-7-21)28(42-29)25-10-11-27(24-9-5-4-8-23(24)25)45(40,41)33-22-17-44(38,39)18-22/h4-5,8-11,21-22,33H,1-3,6-7,12-20H2	GZUJRVKHQTXPIB-UHFFFAOYSA-N	392133	US10301272, Example 14/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392133&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185764	404960473							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783748	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CS(=O)(=O)C1	InChI=1S/C31H37N3O7S4/c35-30(34-19-31(20-34)12-14-43(36,37)15-13-31)29-32-26(16-21-6-2-1-3-7-21)28(42-29)25-10-11-27(24-9-5-4-8-23(24)25)45(40,41)33-22-17-44(38,39)18-22/h4-5,8-11,21-22,33H,1-3,6-7,12-20H2	GZUJRVKHQTXPIB-UHFFFAOYSA-N	392133	US10301272, Example 14/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392133	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392133&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185764	404960473							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783749	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)N1CCOCC1	InChI=1S/C32H39N3O6S3/c36-31(34-21-32(22-34)12-18-43(37,38)19-13-32)30-33-27(20-23-6-2-1-3-7-23)29(42-30)26-10-11-28(25-9-5-4-8-24(25)26)44(39,40)35-14-16-41-17-15-35/h4-5,8-11,23H,1-3,6-7,12-22H2	RUHQXHHZZAPWBB-UHFFFAOYSA-N	392134	US10301272, Example 14/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392134&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185767	404960474							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783750	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)N1CCOCC1	InChI=1S/C32H39N3O6S3/c36-31(34-21-32(22-34)12-18-43(37,38)19-13-32)30-33-27(20-23-6-2-1-3-7-23)29(42-30)26-10-11-28(25-9-5-4-8-24(25)26)44(39,40)35-14-16-41-17-15-35/h4-5,8-11,23H,1-3,6-7,12-22H2	RUHQXHHZZAPWBB-UHFFFAOYSA-N	392134	US10301272, Example 14/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392134&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185767	404960474							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783751	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)N1CCOCC1	InChI=1S/C32H39N3O6S3/c36-31(34-21-32(22-34)12-18-43(37,38)19-13-32)30-33-27(20-23-6-2-1-3-7-23)29(42-30)26-10-11-28(25-9-5-4-8-24(25)26)44(39,40)35-14-16-41-17-15-35/h4-5,8-11,23H,1-3,6-7,12-22H2	RUHQXHHZZAPWBB-UHFFFAOYSA-N	392134	US10301272, Example 14/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392134&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185767	404960474							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783752	CNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C29H35N3O5S3/c1-30-40(36,37)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-20-7-3-2-4-8-20)31-27(38-26)28(33)32-18-29(19-32)13-15-39(34,35)16-14-29/h5-6,9-12,20,30H,2-4,7-8,13-19H2,1H3	WELNMURBDYFNFX-UHFFFAOYSA-N	392135	US10301272, Example 14/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392135&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185765	404960475							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783753	CNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C29H35N3O5S3/c1-30-40(36,37)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-20-7-3-2-4-8-20)31-27(38-26)28(33)32-18-29(19-32)13-15-39(34,35)16-14-29/h5-6,9-12,20,30H,2-4,7-8,13-19H2,1H3	WELNMURBDYFNFX-UHFFFAOYSA-N	392135	US10301272, Example 14/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392135&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185765	404960475							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783754	CNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C29H35N3O5S3/c1-30-40(36,37)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-20-7-3-2-4-8-20)31-27(38-26)28(33)32-18-29(19-32)13-15-39(34,35)16-14-29/h5-6,9-12,20,30H,2-4,7-8,13-19H2,1H3	WELNMURBDYFNFX-UHFFFAOYSA-N	392135	US10301272, Example 14/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392135	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392135&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185765	404960475							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783755	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-4-31(2,3)34-41(38,39)26-15-14-24(22-12-8-9-13-23(22)26)27-25(16-19-10-6-5-7-11-19)33-29(40-27)28(35)32-21-17-20(18-21)30(36)37/h8-9,12-15,19-21,34H,4-7,10-11,16-18H2,1-3H3,(H,32,35)(H,36,37)/t20-,21-	JFBZAEQCYPRNMQ-MEMLXQNLSA-N	392136	US10301272, Example 14/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392136&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185766	404960476							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783756	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-4-31(2,3)34-41(38,39)26-15-14-24(22-12-8-9-13-23(22)26)27-25(16-19-10-6-5-7-11-19)33-29(40-27)28(35)32-21-17-20(18-21)30(36)37/h8-9,12-15,19-21,34H,4-7,10-11,16-18H2,1-3H3,(H,32,35)(H,36,37)/t20-,21-	JFBZAEQCYPRNMQ-MEMLXQNLSA-N	392136	US10301272, Example 14/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392136	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392136&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185766	404960476							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783757	CC(C)(CCO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O6S2/c1-31(2,14-15-35)34-42(39,40)26-13-12-24(22-10-6-7-11-23(22)26)27-25(16-19-8-4-3-5-9-19)33-29(41-27)28(36)32-21-17-20(18-21)30(37)38/h6-7,10-13,19-21,34-35H,3-5,8-9,14-18H2,1-2H3,(H,32,36)(H,37,38)/t20-,21-	FOIQPNMEMZCIIA-MEMLXQNLSA-N	392137	US10301272, Example 14/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392137&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185768	404960477							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783758	CC(C)(CCO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O6S2/c1-31(2,14-15-35)34-42(39,40)26-13-12-24(22-10-6-7-11-23(22)26)27-25(16-19-8-4-3-5-9-19)33-29(41-27)28(36)32-21-17-20(18-21)30(37)38/h6-7,10-13,19-21,34-35H,3-5,8-9,14-18H2,1-2H3,(H,32,36)(H,37,38)/t20-,21-	FOIQPNMEMZCIIA-MEMLXQNLSA-N	392137	US10301272, Example 14/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392137	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392137&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185768	404960477							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783759	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783760	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783761	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783762	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783763	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783764	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783765	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783766	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783767	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)C1	InChI=1S/C27H39N3O5S3/c1-26(2,3)30-38(34,35)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-37(33)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	NMWCBNAPDBYXPJ-UHFFFAOYSA-N	392139	US10301272, Example 15/1::US10301272, Example 15/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392139	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392139&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185770	404960479							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783768	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)(=O)C1	InChI=1S/C27H39N3O6S3/c1-26(2,3)30-39(35,36)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(37-23)24(31)28-19-15-38(33,34)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	AXGDREKTDUYKAR-UHFFFAOYSA-N	392141	US10301272, Example 15/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392141&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185771	404960480							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783769	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)(=O)C1	InChI=1S/C27H39N3O6S3/c1-26(2,3)30-39(35,36)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(37-23)24(31)28-19-15-38(33,34)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	AXGDREKTDUYKAR-UHFFFAOYSA-N	392141	US10301272, Example 15/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392141&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185771	404960480							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783770	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CS(=O)(=O)C1	InChI=1S/C27H39N3O6S3/c1-26(2,3)30-39(35,36)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(37-23)24(31)28-19-15-38(33,34)16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	AXGDREKTDUYKAR-UHFFFAOYSA-N	392141	US10301272, Example 15/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392141	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392141&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185771	404960480							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783771	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O5S3/c1-24(2,3)29-37(33,34)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(35-21)22(30)27-15-12-36(31,32)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	LPDQEQBZQWIIRO-UHFFFAOYSA-N	392142	US10301272, Example 15/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392142&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185774	404960481							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783772	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O5S3/c1-24(2,3)29-37(33,34)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(35-21)22(30)27-15-12-36(31,32)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	LPDQEQBZQWIIRO-UHFFFAOYSA-N	392142	US10301272, Example 15/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392142&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185774	404960481							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783773	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O5S3/c1-24(2,3)29-37(33,34)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(35-21)22(30)27-15-12-36(31,32)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	LPDQEQBZQWIIRO-UHFFFAOYSA-N	392142	US10301272, Example 15/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392142&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185774	404960481							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783774	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S3/c1-24(2,3)29-36(32,33)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-35(31)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	HEPDNWXPOSGWBG-UHFFFAOYSA-N	392143	US10301272, Example 15/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392143&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185773	404960482							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783775	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S3/c1-24(2,3)29-36(32,33)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-35(31)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	HEPDNWXPOSGWBG-UHFFFAOYSA-N	392143	US10301272, Example 15/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392143&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185773	404960482							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783776	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)C2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S3/c1-24(2,3)29-36(32,33)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-35(31)13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	HEPDNWXPOSGWBG-UHFFFAOYSA-N	392143	US10301272, Example 15/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392143	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392143&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185773	404960482							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783777	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(37-22)24(32)31-12-26(13-31)14-38(33,34)15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	UEXPQLLLMKWEBF-UHFFFAOYSA-N	392144	US10301272, Example 15/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392144	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392144&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185775	404960483							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783778	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(37-22)24(32)31-12-26(13-31)14-38(33,34)15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	UEXPQLLLMKWEBF-UHFFFAOYSA-N	392144	US10301272, Example 15/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392144	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392144&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185775	404960483							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783779	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(37-22)24(32)31-12-26(13-31)14-38(33,34)15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	UEXPQLLLMKWEBF-UHFFFAOYSA-N	392144	US10301272, Example 15/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392144	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392144&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185775	404960483							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783780	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCc2ncc(s2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H32Cl2N4O5S4/c1-26(2,3)32-41(36,37)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(39-23)24(33)30-13-19-29-14-20(38-19)40(4,34)35/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	XXLHZXZWCUQACQ-UHFFFAOYSA-N	392145	US10301272, Example 15/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392145&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185776	404960484							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783781	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCc2ncc(s2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H32Cl2N4O5S4/c1-26(2,3)32-41(36,37)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(39-23)24(33)30-13-19-29-14-20(38-19)40(4,34)35/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	XXLHZXZWCUQACQ-UHFFFAOYSA-N	392145	US10301272, Example 15/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392145&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185776	404960484							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783782	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCc2ncc(s2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H32Cl2N4O5S4/c1-26(2,3)32-41(36,37)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(39-23)24(33)30-13-19-29-14-20(38-19)40(4,34)35/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	XXLHZXZWCUQACQ-UHFFFAOYSA-N	392145	US10301272, Example 15/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392145	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392145&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185776	404960484							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783783	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)32-40(36,37)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-19-9-5-4-6-10-19)31-28(38-26)27(33)30-16-20-17-39(34,35)18-20/h7-8,11-14,19-20,32H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	GCVDJHPKFKRVFR-UHFFFAOYSA-N	392146	US10301272, Example 15/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392146	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392146&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185777	404960485							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783784	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)32-40(36,37)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-19-9-5-4-6-10-19)31-28(38-26)27(33)30-16-20-17-39(34,35)18-20/h7-8,11-14,19-20,32H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	GCVDJHPKFKRVFR-UHFFFAOYSA-N	392146	US10301272, Example 15/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392146	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392146&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185777	404960485							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783785	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O4S3/c1-31(2,3)34-42(38,39)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-41(37)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	HRRIWPVNOCJXPZ-UHFFFAOYSA-N	392147	US10301272, Example 15/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392147&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185778	404960486							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783786	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O4S3/c1-31(2,3)34-42(38,39)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-41(37)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	HRRIWPVNOCJXPZ-UHFFFAOYSA-N	392147	US10301272, Example 15/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392147&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185778	404960486							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783787	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O4S3/c1-31(2,3)34-42(38,39)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-41(37)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	HRRIWPVNOCJXPZ-UHFFFAOYSA-N	392147	US10301272, Example 15/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392147	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392147&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185778	404960486							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783788	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783789	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783790	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(37-25)26(32)29-19-16-38(33,34)17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	KWKFCZMPUXBQEX-UHFFFAOYSA-N	392138	US10301272, Example 15::US10301272, Example 16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392138	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392138&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185769	404960478							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783791	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1Cl)S(N)(=O)=O	InChI=1S/C21H27Cl2N3O4S2/c1-21(2,28)11-25-19(27)20-26-14(10-12-6-4-3-5-7-12)18(31-20)13-8-9-15(32(24,29)30)17(23)16(13)22/h8-9,12,28H,3-7,10-11H2,1-2H3,(H,25,27)(H2,24,29,30)	KVEHQGJPQRRYKL-UHFFFAOYSA-N	392149	US10301272, Example 17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392149	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392149&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026092	404960487							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783792	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1Cl)S(N)(=O)=O	InChI=1S/C21H27Cl2N3O4S2/c1-21(2,28)11-25-19(27)20-26-14(10-12-6-4-3-5-7-12)18(31-20)13-8-9-15(32(24,29)30)17(23)16(13)22/h8-9,12,28H,3-7,10-11H2,1-2H3,(H,25,27)(H2,24,29,30)	KVEHQGJPQRRYKL-UHFFFAOYSA-N	392149	US10301272, Example 17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392149	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392149&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026092	404960487							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783793	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1Cl)S(N)(=O)=O	InChI=1S/C21H27Cl2N3O4S2/c1-21(2,28)11-25-19(27)20-26-14(10-12-6-4-3-5-7-12)18(31-20)13-8-9-15(32(24,29)30)17(23)16(13)22/h8-9,12,28H,3-7,10-11H2,1-2H3,(H,25,27)(H2,24,29,30)	KVEHQGJPQRRYKL-UHFFFAOYSA-N	392149	US10301272, Example 17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392149	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392149&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90026092	404960487							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783794	NS(=O)(=O)c1c(Cl)cc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C23H27ClF3N3O4S2/c24-17-12-14(11-16(23(25,26)27)20(17)36(28,32)33)19-18(10-13-4-2-1-3-5-13)30-22(35-19)21(31)29-15-6-8-34-9-7-15/h11-13,15H,1-10H2,(H,29,31)(H2,28,32,33)	BVODGKALUUEICT-UHFFFAOYSA-N	392150	US10301272, Example 17/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2512							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392150&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185779	404960488							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783795	NS(=O)(=O)c1c(Cl)cc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C23H27ClF3N3O4S2/c24-17-12-14(11-16(23(25,26)27)20(17)36(28,32)33)19-18(10-13-4-2-1-3-5-13)30-22(35-19)21(31)29-15-6-8-34-9-7-15/h11-13,15H,1-10H2,(H,29,31)(H2,28,32,33)	BVODGKALUUEICT-UHFFFAOYSA-N	392150	US10301272, Example 17/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392150&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185779	404960488							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783796	NS(=O)(=O)c1c(Cl)cc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C23H27ClF3N3O4S2/c24-17-12-14(11-16(23(25,26)27)20(17)36(28,32)33)19-18(10-13-4-2-1-3-5-13)30-22(35-19)21(31)29-15-6-8-34-9-7-15/h11-13,15H,1-10H2,(H,29,31)(H2,28,32,33)	BVODGKALUUEICT-UHFFFAOYSA-N	392150	US10301272, Example 17/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392150&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185779	404960488							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783797	Cc1c(Cl)c(c(Cl)cc1-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)S(N)(=O)=O	InChI=1S/C23H29Cl2N3O5S3/c1-13-16(12-17(24)21(19(13)25)36(26,32)33)20-18(11-14-5-3-2-4-6-14)28-23(34-20)22(29)27-15-7-9-35(30,31)10-8-15/h12,14-15H,2-11H2,1H3,(H,27,29)(H2,26,32,33)	FABXPHPYPBGAEI-UHFFFAOYSA-N	392151	US10301272, Example 17/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1995							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392151	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392151&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185780	404960489							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783798	Cc1c(Cl)c(c(Cl)cc1-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1)S(N)(=O)=O	InChI=1S/C23H29Cl2N3O5S3/c1-13-16(12-17(24)21(19(13)25)36(26,32)33)20-18(11-14-5-3-2-4-6-14)28-23(34-20)22(29)27-15-7-9-35(30,31)10-8-15/h12,14-15H,2-11H2,1H3,(H,27,29)(H2,26,32,33)	FABXPHPYPBGAEI-UHFFFAOYSA-N	392151	US10301272, Example 17/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392151	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392151&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185780	404960489							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783799	CCNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-4-27-34(31,32)17-11-10-15(18(24)19(17)25)20-16(12-14-8-6-5-7-9-14)28-22(33-20)21(29)26-13-23(2,3)30/h10-11,14,27,30H,4-9,12-13H2,1-3H3,(H,26,29)	ODXKMZATUCVIIS-UHFFFAOYSA-N	392152	US10301272, Example 18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392152&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160520	404960490							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783800	CCNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-4-27-34(31,32)17-11-10-15(18(24)19(17)25)20-16(12-14-8-6-5-7-9-14)28-22(33-20)21(29)26-13-23(2,3)30/h10-11,14,27,30H,4-9,12-13H2,1-3H3,(H,26,29)	ODXKMZATUCVIIS-UHFFFAOYSA-N	392152	US10301272, Example 18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392152&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160520	404960490							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783801	CCNS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-4-27-34(31,32)17-11-10-15(18(24)19(17)25)20-16(12-14-8-6-5-7-9-14)28-22(33-20)21(29)26-13-23(2,3)30/h10-11,14,27,30H,4-9,12-13H2,1-3H3,(H,26,29)	ODXKMZATUCVIIS-UHFFFAOYSA-N	392152	US10301272, Example 18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392152&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160520	404960490							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783802	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H45N3O6S2/c1-30(2,3)22-17-19(13-14-23(22)42(38,39)34-31(4,5)6)26-24(25(40-7)18-11-9-8-10-12-18)33-28(41-26)27(35)32-21-15-20(16-21)29(36)37/h13-14,17-18,20-21,25,34H,8-12,15-16H2,1-7H3,(H,32,35)(H,36,37)/t20-,21-,25?	CGPVPHWYFNTIGH-FPCUACJBSA-N	392153	US10301272, Example 19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3981							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392153&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160567	404960491							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783803	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H45N3O6S2/c1-30(2,3)22-17-19(13-14-23(22)42(38,39)34-31(4,5)6)26-24(25(40-7)18-11-9-8-10-12-18)33-28(41-26)27(35)32-21-15-20(16-21)29(36)37/h13-14,17-18,20-21,25,34H,8-12,15-16H2,1-7H3,(H,32,35)(H,36,37)/t20-,21-,25?	CGPVPHWYFNTIGH-FPCUACJBSA-N	392153	US10301272, Example 19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392153&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160567	404960491							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783804	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H45N3O6S2/c1-30(2,3)22-17-19(13-14-23(22)42(38,39)34-31(4,5)6)26-24(25(40-7)18-11-9-8-10-12-18)33-28(41-26)27(35)32-21-15-20(16-21)29(36)37/h13-14,17-18,20-21,25,34H,8-12,15-16H2,1-7H3,(H,32,35)(H,36,37)/t20-,21-,25?	CGPVPHWYFNTIGH-FPCUACJBSA-N	392153	US10301272, Example 19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392153&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160567	404960491							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783805	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H47N3O5S2/c1-30(2,3)23-19-21(13-14-24(23)41(36,37)34-31(4,5)6)27-25(26(38-7)20-11-9-8-10-12-20)33-29(40-27)28(35)32-22-15-17-39-18-16-22/h13-14,19-20,22,26,34H,8-12,15-18H2,1-7H3,(H,32,35)	ZBCXVVRLEVDOIQ-UHFFFAOYSA-N	392154	US10301272, Example 19/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392154&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185782	404960492							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783806	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H47N3O5S2/c1-30(2,3)23-19-21(13-14-24(23)41(36,37)34-31(4,5)6)27-25(26(38-7)20-11-9-8-10-12-20)33-29(40-27)28(35)32-22-15-17-39-18-16-22/h13-14,19-20,22,26,34H,8-12,15-18H2,1-7H3,(H,32,35)	ZBCXVVRLEVDOIQ-UHFFFAOYSA-N	392154	US10301272, Example 19/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392154&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185782	404960492							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783807	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(c1)C(C)(C)C)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H47N3O5S2/c1-30(2,3)23-19-21(13-14-24(23)41(36,37)34-31(4,5)6)27-25(26(38-7)20-11-9-8-10-12-20)33-29(40-27)28(35)32-22-15-17-39-18-16-22/h13-14,19-20,22,26,34H,8-12,15-18H2,1-7H3,(H,32,35)	ZBCXVVRLEVDOIQ-UHFFFAOYSA-N	392154	US10301272, Example 19/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392154	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392154&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185782	404960492							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783808	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H42N2O4S/c1-30(2,3)21-13-19(14-22(17-21)31(4)11-12-31)26-24(25(37-5)18-9-7-6-8-10-18)33-28(38-26)27(34)32-23-15-20(16-23)29(35)36/h13-14,17-18,20,23,25H,6-12,15-16H2,1-5H3,(H,32,34)(H,35,36)/t20-,23-,25?	NIYONYQFFZZQFX-HJZAHENMSA-N	392155	US10301272, Example 19/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392155	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392155&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185781	404960493							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783809	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H42N2O4S/c1-30(2,3)21-13-19(14-22(17-21)31(4)11-12-31)26-24(25(37-5)18-9-7-6-8-10-18)33-28(38-26)27(34)32-23-15-20(16-23)29(35)36/h13-14,17-18,20,23,25H,6-12,15-16H2,1-5H3,(H,32,34)(H,35,36)/t20-,23-,25?	NIYONYQFFZZQFX-HJZAHENMSA-N	392155	US10301272, Example 19/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392155	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392155&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185781	404960493							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783810	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C31H42N2O4S/c1-30(2,3)21-13-19(14-22(17-21)31(4)11-12-31)26-24(25(37-5)18-9-7-6-8-10-18)33-28(38-26)27(34)32-23-15-20(16-23)29(35)36/h13-14,17-18,20,23,25H,6-12,15-16H2,1-5H3,(H,32,34)(H,35,36)/t20-,23-,25?	NIYONYQFFZZQFX-HJZAHENMSA-N	392155	US10301272, Example 19/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392155	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392155&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185781	404960493							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783811	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H44N2O3S/c1-30(2,3)22-17-21(18-23(19-22)31(4)13-14-31)27-25(26(35-5)20-9-7-6-8-10-20)33-29(37-27)28(34)32-24-11-15-36-16-12-24/h17-20,24,26H,6-16H2,1-5H3,(H,32,34)	NEXFKLAZJSRAEU-UHFFFAOYSA-N	392156	US10301272, Example 19/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392156	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392156&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185783	404960494							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783812	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H44N2O3S/c1-30(2,3)22-17-21(18-23(19-22)31(4)13-14-31)27-25(26(35-5)20-9-7-6-8-10-20)33-29(37-27)28(34)32-24-11-15-36-16-12-24/h17-20,24,26H,6-16H2,1-5H3,(H,32,34)	NEXFKLAZJSRAEU-UHFFFAOYSA-N	392156	US10301272, Example 19/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392156	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392156&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185783	404960494							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783813	COC(C1CCCCC1)c1nc(sc1-c1cc(cc(c1)C1(C)CC1)C(C)(C)C)C(=O)NC1CCOCC1	InChI=1S/C31H44N2O3S/c1-30(2,3)22-17-21(18-23(19-22)31(4)13-14-31)27-25(26(35-5)20-9-7-6-8-10-20)33-29(37-27)28(34)32-24-11-15-36-16-12-24/h17-20,24,26H,6-16H2,1-5H3,(H,32,34)	NEXFKLAZJSRAEU-UHFFFAOYSA-N	392156	US10301272, Example 19/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392156	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392156&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185783	404960494							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783814	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H35Cl2N3O6S2/c1-27(2,3)32-40(36,37)18-11-10-17(19(28)20(18)29)23-21(22(38-4)14-8-6-5-7-9-14)31-25(39-23)24(33)30-16-12-15(13-16)26(34)35/h10-11,14-16,22,32H,5-9,12-13H2,1-4H3,(H,30,33)(H,34,35)/t15-,16-,22?	MGKFSWKQIATVQR-STFKQGPRSA-N	392157	US10301272, Example 19/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392157&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185784	404960495							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783815	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H35Cl2N3O6S2/c1-27(2,3)32-40(36,37)18-11-10-17(19(28)20(18)29)23-21(22(38-4)14-8-6-5-7-9-14)31-25(39-23)24(33)30-16-12-15(13-16)26(34)35/h10-11,14-16,22,32H,5-9,12-13H2,1-4H3,(H,30,33)(H,34,35)/t15-,16-,22?	MGKFSWKQIATVQR-STFKQGPRSA-N	392157	US10301272, Example 19/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392157&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185784	404960495							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783816	COC(C1CCCCC1)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C27H35Cl2N3O6S2/c1-27(2,3)32-40(36,37)18-11-10-17(19(28)20(18)29)23-21(22(38-4)14-8-6-5-7-9-14)31-25(39-23)24(33)30-16-12-15(13-16)26(34)35/h10-11,14-16,22,32H,5-9,12-13H2,1-4H3,(H,30,33)(H,34,35)/t15-,16-,22?	MGKFSWKQIATVQR-STFKQGPRSA-N	392157	US10301272, Example 19/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392157&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185784	404960495							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783817	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)26-20-14-10-9-13-19(20)21(16-29-26)23-22(15-18-11-7-6-8-12-18)31-25(37-23)24(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	RPKZVBVTIACVGB-UHFFFAOYSA-N	392158	US10301272, Example 19/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392158	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392158&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185785	404960496							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783818	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)26-20-14-10-9-13-19(20)21(16-29-26)23-22(15-18-11-7-6-8-12-18)31-25(37-23)24(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	RPKZVBVTIACVGB-UHFFFAOYSA-N	392158	US10301272, Example 19/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392158	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392158&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185785	404960496							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783819	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)26-20-14-10-9-13-19(20)21(16-29-26)23-22(15-18-11-7-6-8-12-18)31-25(37-23)24(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	RPKZVBVTIACVGB-UHFFFAOYSA-N	392158	US10301272, Example 19/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392158	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392158&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185785	404960496							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783820	CC(C)(C)NS(=O)(=O)c1cnc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)22-16-29-23(20-14-10-9-13-19(20)22)24-21(15-18-11-7-6-8-12-18)31-26(37-24)25(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	YJNAZHIKSBXYOZ-UHFFFAOYSA-N	392159	US10301272, Example 19/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392159&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185786	404960497							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783821	CC(C)(C)NS(=O)(=O)c1cnc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)22-16-29-23(20-14-10-9-13-19(20)22)24-21(15-18-11-7-6-8-12-18)31-26(37-24)25(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	YJNAZHIKSBXYOZ-UHFFFAOYSA-N	392159	US10301272, Example 19/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392159&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185786	404960497							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783822	CC(C)(C)NS(=O)(=O)c1cnc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H38N4O4S2/c1-27(2,3)32-38(35,36)22-16-29-23(20-14-10-9-13-19(20)22)24-21(15-18-11-7-6-8-12-18)31-26(37-24)25(33)30-17-28(4,5)34/h9-10,13-14,16,18,32,34H,6-8,11-12,15,17H2,1-5H3,(H,30,33)	YJNAZHIKSBXYOZ-UHFFFAOYSA-N	392159	US10301272, Example 19/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392159&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185786	404960497							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783823	Cc1c(cc(cc1C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NC(C)(C)C	InChI=1S/C32H43N3O4S/c1-18-23(27(36)35-31(2,3)4)16-20(17-24(18)32(5)11-12-32)26-25(13-19-9-7-6-8-10-19)34-29(40-26)28(37)33-22-14-21(15-22)30(38)39/h16-17,19,21-22H,6-15H2,1-5H3,(H,33,37)(H,35,36)(H,38,39)/t21-,22-	RYAYBMDYXIDMKD-HZCBDIJESA-N	392160	US10301272, Example 19/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392160&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185787	404960498							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783824	Cc1c(cc(cc1C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NC(C)(C)C	InChI=1S/C32H43N3O4S/c1-18-23(27(36)35-31(2,3)4)16-20(17-24(18)32(5)11-12-32)26-25(13-19-9-7-6-8-10-19)34-29(40-26)28(37)33-22-14-21(15-22)30(38)39/h16-17,19,21-22H,6-15H2,1-5H3,(H,33,37)(H,35,36)(H,38,39)/t21-,22-	RYAYBMDYXIDMKD-HZCBDIJESA-N	392160	US10301272, Example 19/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392160&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185787	404960498							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783825	Cc1c(cc(cc1C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(=O)NC(C)(C)C	InChI=1S/C32H43N3O4S/c1-18-23(27(36)35-31(2,3)4)16-20(17-24(18)32(5)11-12-32)26-25(13-19-9-7-6-8-10-19)34-29(40-26)28(37)33-22-14-21(15-22)30(38)39/h16-17,19,21-22H,6-15H2,1-5H3,(H,33,37)(H,35,36)(H,38,39)/t21-,22-	RYAYBMDYXIDMKD-HZCBDIJESA-N	392160	US10301272, Example 19/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392160&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185787	404960498							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783826	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2cccc(F)c12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(19-12-9-13-21(30)24(19)23)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	VOFAAWAGOWNHLE-UHFFFAOYSA-N	392161	US10301272, Example 19/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392161&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185788	404960499							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783827	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2cccc(F)c12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(19-12-9-13-21(30)24(19)23)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	VOFAAWAGOWNHLE-UHFFFAOYSA-N	392161	US10301272, Example 19/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392161&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185788	404960499							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783828	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2cccc(F)c12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(19-12-9-13-21(30)24(19)23)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	VOFAAWAGOWNHLE-UHFFFAOYSA-N	392161	US10301272, Example 19/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392161	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392161&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185788	404960499							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783829	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2c(F)cccc12	InChI=1S/C30H36FN3O5S2/c1-30(2,3)34-41(38,39)24-13-12-21(25-20(24)10-7-11-22(25)31)26-23(14-17-8-5-4-6-9-17)33-28(40-26)27(35)32-19-15-18(16-19)29(36)37/h7,10-13,17-19,34H,4-6,8-9,14-16H2,1-3H3,(H,32,35)(H,36,37)/t18-,19-	YUMGWXKRFFDFPB-WGSAOQKQSA-N	392162	US10301272, Example 19/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392162&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185789	404960500							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783830	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2c(F)cccc12	InChI=1S/C30H36FN3O5S2/c1-30(2,3)34-41(38,39)24-13-12-21(25-20(24)10-7-11-22(25)31)26-23(14-17-8-5-4-6-9-17)33-28(40-26)27(35)32-19-15-18(16-19)29(36)37/h7,10-13,17-19,34H,4-6,8-9,14-16H2,1-3H3,(H,32,35)(H,36,37)/t18-,19-	YUMGWXKRFFDFPB-WGSAOQKQSA-N	392162	US10301272, Example 19/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392162&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185789	404960500							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783831	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2c(F)cccc12	InChI=1S/C30H36FN3O5S2/c1-30(2,3)34-41(38,39)24-13-12-21(25-20(24)10-7-11-22(25)31)26-23(14-17-8-5-4-6-9-17)33-28(40-26)27(35)32-19-15-18(16-19)29(36)37/h7,10-13,17-19,34H,4-6,8-9,14-16H2,1-3H3,(H,32,35)(H,36,37)/t18-,19-	YUMGWXKRFFDFPB-WGSAOQKQSA-N	392162	US10301272, Example 19/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392162	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392162&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185789	404960500							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783832	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1OC(F)(F)F	InChI=1S/C27H33F4N3O6S2/c1-26(2,3)34-42(38,39)19-10-9-17(20(28)21(19)40-27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(41-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	WLGDHJPBHBRUGI-WKILWMFISA-N	392163	US10301272, Example 19/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392163	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392163&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188727	404960501							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783833	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1OC(F)(F)F	InChI=1S/C27H33F4N3O6S2/c1-26(2,3)34-42(38,39)19-10-9-17(20(28)21(19)40-27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(41-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	WLGDHJPBHBRUGI-WKILWMFISA-N	392163	US10301272, Example 19/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392163	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392163&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188727	404960501							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783834	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(F)c1OC(F)(F)F	InChI=1S/C27H33F4N3O6S2/c1-26(2,3)34-42(38,39)19-10-9-17(20(28)21(19)40-27(29,30)31)22-18(11-14-7-5-4-6-8-14)33-24(41-22)23(35)32-16-12-15(13-16)25(36)37/h9-10,14-16,34H,4-8,11-13H2,1-3H3,(H,32,35)(H,36,37)/t15-,16-	WLGDHJPBHBRUGI-WKILWMFISA-N	392163	US10301272, Example 19/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392163	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392163&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188727	404960501							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783835	CC(C)(C)NS(=O)(=O)c1cc(Cl)c(cc1Cl)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C26H33Cl2N3O5S2/c1-26(2,3)31-38(35,36)21-13-18(27)17(12-19(21)28)22-20(9-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-10-15(11-16)25(33)34/h12-16,31H,4-11H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	CRXWBMYQVZBRBZ-WKILWMFISA-N	392164	US10301272, Example 19/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392164&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185791	404960502							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783836	CC(C)(C)NS(=O)(=O)c1cc(Cl)c(cc1Cl)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C26H33Cl2N3O5S2/c1-26(2,3)31-38(35,36)21-13-18(27)17(12-19(21)28)22-20(9-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-10-15(11-16)25(33)34/h12-16,31H,4-11H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	CRXWBMYQVZBRBZ-WKILWMFISA-N	392164	US10301272, Example 19/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392164&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185791	404960502							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783837	CC(C)(C)c1cc(nc(n1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H38N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4)10-11-28)23-20(12-17-8-6-5-7-9-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,5-14H2,1-4H3,(H,29,34)/t18-,19?	QHZANCPXHWSPOT-NZANSXMDSA-N	392165	US10301272, Example 19/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392165&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185792	404960503							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783838	CC(C)(C)c1cc(nc(n1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H38N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4)10-11-28)23-20(12-17-8-6-5-7-9-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,5-14H2,1-4H3,(H,29,34)/t18-,19?	QHZANCPXHWSPOT-NZANSXMDSA-N	392165	US10301272, Example 19/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392165&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185792	404960503							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783839	CC(C)(C)c1cc(nc(n1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H38N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4)10-11-28)23-20(12-17-8-6-5-7-9-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,5-14H2,1-4H3,(H,29,34)/t18-,19?	QHZANCPXHWSPOT-NZANSXMDSA-N	392165	US10301272, Example 19/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392165	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392165&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185792	404960503							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783840	CC(C)(C)c1cc(nc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H40N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4,5)6)23-20(12-17-10-8-7-9-11-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,7-14H2,1-6H3,(H,29,34)/t18-,19?	HANRVFAWFJKDST-NZANSXMDSA-N	392166	US10301272, Example 19/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392166&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185793	404960504							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783841	CC(C)(C)c1cc(nc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H40N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4,5)6)23-20(12-17-10-8-7-9-11-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,7-14H2,1-6H3,(H,29,34)/t18-,19?	HANRVFAWFJKDST-NZANSXMDSA-N	392166	US10301272, Example 19/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392166&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185793	404960504							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783842	CC(C)(C)c1cc(nc(n1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)OC=O	InChI=1S/C28H40N4O3S/c1-27(2,3)22-15-21(31-26(32-22)28(4,5)6)23-20(12-17-10-8-7-9-11-17)30-25(36-23)24(34)29-18-13-19(14-18)35-16-33/h15-19H,7-14H2,1-6H3,(H,29,34)/t18-,19?	HANRVFAWFJKDST-NZANSXMDSA-N	392166	US10301272, Example 19/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392166	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392166&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185793	404960504							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783843	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2c(F)cccc12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(24-19(23)12-9-13-21(24)30)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	DGAVRVFXZASTPB-UHFFFAOYSA-N	392167	US10301272, Example 19/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392167&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185794	404960505							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783844	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2c(F)cccc12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(24-19(23)12-9-13-21(24)30)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	DGAVRVFXZASTPB-UHFFFAOYSA-N	392167	US10301272, Example 19/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392167&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185794	404960505							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783845	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2c(F)cccc12	InChI=1S/C29H38FN3O4S2/c1-28(2,3)33-39(36,37)23-15-14-20(24-19(23)12-9-13-21(24)30)25-22(16-18-10-7-6-8-11-18)32-27(38-25)26(34)31-17-29(4,5)35/h9,12-15,18,33,35H,6-8,10-11,16-17H2,1-5H3,(H,31,34)	DGAVRVFXZASTPB-UHFFFAOYSA-N	392167	US10301272, Example 19/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392167	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392167&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185794	404960505							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783846	CC(C)(CCF)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H38FN3O5S2/c1-31(2,14-15-32)35-42(39,40)26-13-12-24(22-10-6-7-11-23(22)26)27-25(16-19-8-4-3-5-9-19)34-29(41-27)28(36)33-21-17-20(18-21)30(37)38/h6-7,10-13,19-21,35H,3-5,8-9,14-18H2,1-2H3,(H,33,36)(H,37,38)/t20-,21-	FOOFCMISAIJPLF-MEMLXQNLSA-N	392168	US10301272, Example 20::trans-3-(4-(Cyclohexylmethyl-5-(4-(N-(4-fluoro-2-methylbutan-2-yl)sulfamoyl)naphthalen-1-yl)thiazole-2-carboxamido)cyclobutanecarboxylic acid 	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392168	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392168&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188622	404960506							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783847	CC(C)(CCF)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H38FN3O5S2/c1-31(2,14-15-32)35-42(39,40)26-13-12-24(22-10-6-7-11-23(22)26)27-25(16-19-8-4-3-5-9-19)34-29(41-27)28(36)33-21-17-20(18-21)30(37)38/h6-7,10-13,19-21,35H,3-5,8-9,14-18H2,1-2H3,(H,33,36)(H,37,38)/t20-,21-	FOOFCMISAIJPLF-MEMLXQNLSA-N	392168	US10301272, Example 20::trans-3-(4-(Cyclohexylmethyl-5-(4-(N-(4-fluoro-2-methylbutan-2-yl)sulfamoyl)naphthalen-1-yl)thiazole-2-carboxamido)cyclobutanecarboxylic acid 	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392168	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392168&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188622	404960506							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783848	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-22(2,3)28-34(31,32)16-10-9-14(17(24)18(16)25)19-15(11-13-7-6-8-13)27-21(33-19)20(29)26-12-23(4,5)30/h9-10,13,28,30H,6-8,11-12H2,1-5H3,(H,26,29)	UATOMOTUFXJSPU-UHFFFAOYSA-N	392169	US10301272, Example 21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392169&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548956	404960507							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783849	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-22(2,3)28-34(31,32)16-10-9-14(17(24)18(16)25)19-15(11-13-7-6-8-13)27-21(33-19)20(29)26-12-23(4,5)30/h9-10,13,28,30H,6-8,11-12H2,1-5H3,(H,26,29)	UATOMOTUFXJSPU-UHFFFAOYSA-N	392169	US10301272, Example 21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392169&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548956	404960507							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783850	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C23H31Cl2N3O4S2/c1-22(2,3)28-34(31,32)16-10-9-14(17(24)18(16)25)19-15(11-13-7-6-8-13)27-21(33-19)20(29)26-12-23(4,5)30/h9-10,13,28,30H,6-8,11-12H2,1-5H3,(H,26,29)	UATOMOTUFXJSPU-UHFFFAOYSA-N	392169	US10301272, Example 21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392169	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392169&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548956	404960507							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783851	CC(C)(O)CNC(=O)c1nc(CC2CCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C24H32ClF2N3O5S2/c1-23(2,3)30-37(33,34)16-10-9-14(18(17(16)25)35-22(26)27)19-15(11-13-7-6-8-13)29-21(36-19)20(31)28-12-24(4,5)32/h9-10,13,22,30,32H,6-8,11-12H2,1-5H3,(H,28,31)	AFDZQERQBVHMEN-UHFFFAOYSA-N	392170	US10301272, Example 21/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392170&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188679	404960508							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783852	CC(C)(O)CNC(=O)c1nc(CC2CCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C24H32ClF2N3O5S2/c1-23(2,3)30-37(33,34)16-10-9-14(18(17(16)25)35-22(26)27)19-15(11-13-7-6-8-13)29-21(36-19)20(31)28-12-24(4,5)32/h9-10,13,22,30,32H,6-8,11-12H2,1-5H3,(H,28,31)	AFDZQERQBVHMEN-UHFFFAOYSA-N	392170	US10301272, Example 21/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392170&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188679	404960508							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783853	CC(C)(O)CNC(=O)c1nc(CC2CCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C24H32ClF2N3O5S2/c1-23(2,3)30-37(33,34)16-10-9-14(18(17(16)25)35-22(26)27)19-15(11-13-7-6-8-13)29-21(36-19)20(31)28-12-24(4,5)32/h9-10,13,22,30,32H,6-8,11-12H2,1-5H3,(H,28,31)	AFDZQERQBVHMEN-UHFFFAOYSA-N	392170	US10301272, Example 21/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392170	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392170&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188679	404960508							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783854	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C27H35N3O4S2/c1-26(2,3)30-36(33,34)22-14-13-20(18-11-6-7-12-19(18)22)23-21(15-17-9-8-10-17)29-25(35-23)24(31)28-16-27(4,5)32/h6-7,11-14,17,30,32H,8-10,15-16H2,1-5H3,(H,28,31)	ISHVKDWWCNMSLQ-UHFFFAOYSA-N	392171	US10301272, Example 21/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392171&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185796	404960509							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783855	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C27H35N3O4S2/c1-26(2,3)30-36(33,34)22-14-13-20(18-11-6-7-12-19(18)22)23-21(15-17-9-8-10-17)29-25(35-23)24(31)28-16-27(4,5)32/h6-7,11-14,17,30,32H,8-10,15-16H2,1-5H3,(H,28,31)	ISHVKDWWCNMSLQ-UHFFFAOYSA-N	392171	US10301272, Example 21/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392171&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185796	404960509							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783856	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C27H35N3O4S2/c1-26(2,3)30-36(33,34)22-14-13-20(18-11-6-7-12-19(18)22)23-21(15-17-9-8-10-17)29-25(35-23)24(31)28-16-27(4,5)32/h6-7,11-14,17,30,32H,8-10,15-16H2,1-5H3,(H,28,31)	ISHVKDWWCNMSLQ-UHFFFAOYSA-N	392171	US10301272, Example 21/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392171&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185796	404960509							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783857	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(OC(F)F)c1Cl	InChI=1S/C26H34ClF2N3O4S2/c1-26(2,3)32-38(34,35)19-13-12-17(21(20(19)27)36-25(28)29)22-18(14-15-8-5-4-6-9-15)31-24(37-22)23(33)30-16-10-7-11-16/h12-13,15-16,25,32H,4-11,14H2,1-3H3,(H,30,33)	GUOLZVAHLNBJQU-UHFFFAOYSA-N	392172	US10301272, Example 21/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392172	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392172&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012231	404960510							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783858	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(OC(F)F)c1Cl	InChI=1S/C26H34ClF2N3O4S2/c1-26(2,3)32-38(34,35)19-13-12-17(21(20(19)27)36-25(28)29)22-18(14-15-8-5-4-6-9-15)31-24(37-22)23(33)30-16-10-7-11-16/h12-13,15-16,25,32H,4-11,14H2,1-3H3,(H,30,33)	GUOLZVAHLNBJQU-UHFFFAOYSA-N	392172	US10301272, Example 21/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392172	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392172&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012231	404960510							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783859	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(OC(F)F)c1Cl	InChI=1S/C26H34ClF2N3O4S2/c1-26(2,3)32-38(34,35)19-13-12-17(21(20(19)27)36-25(28)29)22-18(14-15-8-5-4-6-9-15)31-24(37-22)23(33)30-16-10-7-11-16/h12-13,15-16,25,32H,4-11,14H2,1-3H3,(H,30,33)	GUOLZVAHLNBJQU-UHFFFAOYSA-N	392172	US10301272, Example 21/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392172	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392172&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012231	404960510							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783860	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O5S2/c1-25(2,3)32-39(35,36)18-12-11-16(20(19(18)27)37-24(28)29)21-17(13-15-9-7-6-8-10-15)31-23(38-21)22(33)30-14-26(4,5)34/h11-12,15,24,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	BQNFYVWDYWWQOW-UHFFFAOYSA-N	392173	US10301272, Example 21/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392173	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392173&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188710	404960511							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783861	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O5S2/c1-25(2,3)32-39(35,36)18-12-11-16(20(19(18)27)37-24(28)29)21-17(13-15-9-7-6-8-10-15)31-23(38-21)22(33)30-14-26(4,5)34/h11-12,15,24,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	BQNFYVWDYWWQOW-UHFFFAOYSA-N	392173	US10301272, Example 21/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392173	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392173&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188710	404960511							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783862	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1OC(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O5S2/c1-25(2,3)32-39(35,36)18-12-11-16(20(19(18)27)37-24(28)29)21-17(13-15-9-7-6-8-10-15)31-23(38-21)22(33)30-14-26(4,5)34/h11-12,15,24,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	BQNFYVWDYWWQOW-UHFFFAOYSA-N	392173	US10301272, Example 21/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392173	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392173&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188710	404960511							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783863	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(c1)C(F)(F)F	InChI=1S/C26H34F3N3O3S2/c1-25(2,3)32-37(34,35)18-12-13-19(20(15-18)26(27,28)29)22-21(14-16-8-5-4-6-9-16)31-24(36-22)23(33)30-17-10-7-11-17/h12-13,15-17,32H,4-11,14H2,1-3H3,(H,30,33)	ROSGQJSBJVQDLH-UHFFFAOYSA-N	392174	US10301272, Example 21/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392174&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012232	404960512							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783864	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(c1)C(F)(F)F	InChI=1S/C26H34F3N3O3S2/c1-25(2,3)32-37(34,35)18-12-13-19(20(15-18)26(27,28)29)22-21(14-16-8-5-4-6-9-16)31-24(36-22)23(33)30-17-10-7-11-17/h12-13,15-17,32H,4-11,14H2,1-3H3,(H,30,33)	ROSGQJSBJVQDLH-UHFFFAOYSA-N	392174	US10301272, Example 21/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392174&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012232	404960512							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783865	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(c1)C(F)(F)F	InChI=1S/C26H34F3N3O3S2/c1-25(2,3)32-37(34,35)18-12-13-19(20(15-18)26(27,28)29)22-21(14-16-8-5-4-6-9-16)31-24(36-22)23(33)30-17-10-7-11-17/h12-13,15-17,32H,4-11,14H2,1-3H3,(H,30,33)	ROSGQJSBJVQDLH-UHFFFAOYSA-N	392174	US10301272, Example 21/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392174&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012232	404960512							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783866	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1	InChI=1S/C25H34ClN3O3S2/c1-25(2,3)29-34(31,32)18-12-13-19(20(26)15-18)22-21(14-16-8-5-4-6-9-16)28-24(33-22)23(30)27-17-10-7-11-17/h12-13,15-17,29H,4-11,14H2,1-3H3,(H,27,30)	XJMBUTPXGMOCEE-UHFFFAOYSA-N	392175	US10301272, Example 21/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392175	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392175&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185800	404960513							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783867	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1	InChI=1S/C25H34ClN3O3S2/c1-25(2,3)29-34(31,32)18-12-13-19(20(26)15-18)22-21(14-16-8-5-4-6-9-16)28-24(33-22)23(30)27-17-10-7-11-17/h12-13,15-17,29H,4-11,14H2,1-3H3,(H,27,30)	XJMBUTPXGMOCEE-UHFFFAOYSA-N	392175	US10301272, Example 21/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392175	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392175&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185800	404960513							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783868	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1	InChI=1S/C25H34ClN3O3S2/c1-25(2,3)29-34(31,32)18-12-13-19(20(26)15-18)22-21(14-16-8-5-4-6-9-16)28-24(33-22)23(30)27-17-10-7-11-17/h12-13,15-17,29H,4-11,14H2,1-3H3,(H,27,30)	XJMBUTPXGMOCEE-UHFFFAOYSA-N	392175	US10301272, Example 21/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392175	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392175&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185800	404960513							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783869	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(OC(F)(F)F)c1	InChI=1S/C26H34F3N3O4S2/c1-25(2,3)32-38(34,35)18-12-13-19(21(15-18)36-26(27,28)29)22-20(14-16-8-5-4-6-9-16)31-24(37-22)23(33)30-17-10-7-11-17/h12-13,15-17,32H,4-11,14H2,1-3H3,(H,30,33)	KLCMTTDFYJUMKX-UHFFFAOYSA-N	392176	US10301272, Example 21/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392176	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392176&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012233	404960514							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783870	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(OC(F)(F)F)c1	InChI=1S/C26H34F3N3O4S2/c1-25(2,3)32-38(34,35)18-12-13-19(21(15-18)36-26(27,28)29)22-20(14-16-8-5-4-6-9-16)31-24(37-22)23(33)30-17-10-7-11-17/h12-13,15-17,32H,4-11,14H2,1-3H3,(H,30,33)	KLCMTTDFYJUMKX-UHFFFAOYSA-N	392176	US10301272, Example 21/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392176	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392176&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012233	404960514							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783871	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C26H36F3N3O5S2/c1-24(2,3)32-39(35,36)17-11-12-18(20(14-17)37-26(27,28)29)21-19(13-16-9-7-6-8-10-16)31-23(38-21)22(33)30-15-25(4,5)34/h11-12,14,16,32,34H,6-10,13,15H2,1-5H3,(H,30,33)	GCSMNPADGYVKSI-UHFFFAOYSA-N	392177	US10301272, Example 21/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392177	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392177&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188682	404960515							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783872	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C26H36F3N3O5S2/c1-24(2,3)32-39(35,36)17-11-12-18(20(14-17)37-26(27,28)29)21-19(13-16-9-7-6-8-10-16)31-23(38-21)22(33)30-15-25(4,5)34/h11-12,14,16,32,34H,6-10,13,15H2,1-5H3,(H,30,33)	GCSMNPADGYVKSI-UHFFFAOYSA-N	392177	US10301272, Example 21/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392177	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392177&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188682	404960515							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783873	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CCOCC1	InChI=1S/C33H41N3O6S3/c37-32(36-21-33(22-36)14-18-44(38,39)19-15-33)31-34-28(20-23-6-2-1-3-7-23)30(43-31)27-10-11-29(26-9-5-4-8-25(26)27)45(40,41)35-24-12-16-42-17-13-24/h4-5,8-11,23-24,35H,1-3,6-7,12-22H2	NQCUBWMDILKGQF-UHFFFAOYSA-N	392178	US10301272, Example 21/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392178	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392178&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188714	404960516							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783874	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CCOCC1	InChI=1S/C33H41N3O6S3/c37-32(36-21-33(22-36)14-18-44(38,39)19-15-33)31-34-28(20-23-6-2-1-3-7-23)30(43-31)27-10-11-29(26-9-5-4-8-25(26)27)45(40,41)35-24-12-16-42-17-13-24/h4-5,8-11,23-24,35H,1-3,6-7,12-22H2	NQCUBWMDILKGQF-UHFFFAOYSA-N	392178	US10301272, Example 21/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392178	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392178&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188714	404960516							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783875	O=C(N1CC2(C1)CCS(=O)(=O)CC2)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1CCOCC1	InChI=1S/C33H41N3O6S3/c37-32(36-21-33(22-36)14-18-44(38,39)19-15-33)31-34-28(20-23-6-2-1-3-7-23)30(43-31)27-10-11-29(26-9-5-4-8-25(26)27)45(40,41)35-24-12-16-42-17-13-24/h4-5,8-11,23-24,35H,1-3,6-7,12-22H2	NQCUBWMDILKGQF-UHFFFAOYSA-N	392178	US10301272, Example 21/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392178	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392178&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188714	404960516							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783876	CC(O)c1c(Cl)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C30H42ClN3O6S3/c1-19(35)24-23(43(39,40)33-29(2,3)4)11-10-21(25(24)31)26-22(16-20-8-6-5-7-9-20)32-27(41-26)28(36)34-17-30(18-34)12-14-42(37,38)15-13-30/h10-11,19-20,33,35H,5-9,12-18H2,1-4H3	SYGXFKWQVPKBRE-UHFFFAOYSA-N	392179	US10301272, Example 21/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188684	404960517							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783877	CC(O)c1c(Cl)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C30H42ClN3O6S3/c1-19(35)24-23(43(39,40)33-29(2,3)4)11-10-21(25(24)31)26-22(16-20-8-6-5-7-9-20)32-27(41-26)28(36)34-17-30(18-34)12-14-42(37,38)15-13-30/h10-11,19-20,33,35H,5-9,12-18H2,1-4H3	SYGXFKWQVPKBRE-UHFFFAOYSA-N	392179	US10301272, Example 21/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188684	404960517							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783878	CC(O)c1c(Cl)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C30H42ClN3O6S3/c1-19(35)24-23(43(39,40)33-29(2,3)4)11-10-21(25(24)31)26-22(16-20-8-6-5-7-9-20)32-27(41-26)28(36)34-17-30(18-34)12-14-42(37,38)15-13-30/h10-11,19-20,33,35H,5-9,12-18H2,1-4H3	SYGXFKWQVPKBRE-UHFFFAOYSA-N	392179	US10301272, Example 21/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392179	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392179&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188684	404960517							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783879	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H37F2N3O4S2/c1-27(2,3)34-40(37,38)23-11-10-21(19-8-6-7-9-20(19)23)24-22(16-18-12-14-29(30,31)15-13-18)33-26(39-24)25(35)32-17-28(4,5)36/h6-11,18,34,36H,12-17H2,1-5H3,(H,32,35)	KIHFMQSGPVESNC-UHFFFAOYSA-N	392180	US10301272, Example 21/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549191	404960518							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783880	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H37F2N3O4S2/c1-27(2,3)34-40(37,38)23-11-10-21(19-8-6-7-9-20(19)23)24-22(16-18-12-14-29(30,31)15-13-18)33-26(39-24)25(35)32-17-28(4,5)36/h6-11,18,34,36H,12-17H2,1-5H3,(H,32,35)	KIHFMQSGPVESNC-UHFFFAOYSA-N	392180	US10301272, Example 21/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549191	404960518							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783881	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H37F2N3O5S3/c1-29(2,3)35-43(39,40)25-9-8-23(21-6-4-5-7-22(21)25)26-24(18-19-10-14-30(31,32)15-11-19)34-28(41-26)27(36)33-20-12-16-42(37,38)17-13-20/h4-9,19-20,35H,10-18H2,1-3H3,(H,33,36)	HLFYKIUEXZPVNL-UHFFFAOYSA-N	392181	US10301272, Example 21/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392181&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549407	404960519							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783882	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H37F2N3O5S3/c1-29(2,3)35-43(39,40)25-9-8-23(21-6-4-5-7-22(21)25)26-24(18-19-10-14-30(31,32)15-11-19)34-28(41-26)27(36)33-20-12-16-42(37,38)17-13-20/h4-9,19-20,35H,10-18H2,1-3H3,(H,33,36)	HLFYKIUEXZPVNL-UHFFFAOYSA-N	392181	US10301272, Example 21/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392181&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549407	404960519							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783883	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccncc12	InChI=1S/C29H38N4O5S3/c1-29(2,3)33-41(37,38)25-10-9-22(21-11-14-30-18-23(21)25)26-24(17-19-7-5-4-6-8-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h9-11,14,18-20,33H,4-8,12-13,15-17H2,1-3H3,(H,31,34)	LWFSZFOEYQVOBE-UHFFFAOYSA-N	392182	US10301272, Example 21/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392182&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188716	404960520							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783884	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccncc12	InChI=1S/C29H38N4O5S3/c1-29(2,3)33-41(37,38)25-10-9-22(21-11-14-30-18-23(21)25)26-24(17-19-7-5-4-6-8-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h9-11,14,18-20,33H,4-8,12-13,15-17H2,1-3H3,(H,31,34)	LWFSZFOEYQVOBE-UHFFFAOYSA-N	392182	US10301272, Example 21/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392182&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188716	404960520							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783885	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccncc12	InChI=1S/C29H38N4O5S3/c1-29(2,3)33-41(37,38)25-10-9-22(21-11-14-30-18-23(21)25)26-24(17-19-7-5-4-6-8-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h9-11,14,18-20,33H,4-8,12-13,15-17H2,1-3H3,(H,31,34)	LWFSZFOEYQVOBE-UHFFFAOYSA-N	392182	US10301272, Example 21/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392182&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188716	404960520							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783886	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O5S3/c1-24(2,3)29-37(33,34)18-8-7-16(19(25)20(18)26)21-17(13-14-5-4-6-14)28-23(35-21)22(30)27-15-9-11-36(31,32)12-10-15/h7-8,14-15,29H,4-6,9-13H2,1-3H3,(H,27,30)	WDWOXUSOFXZJEX-UHFFFAOYSA-N	392183	US10301272, Example 21/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392183	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392183&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188712	404960521							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783887	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O5S3/c1-24(2,3)29-37(33,34)18-8-7-16(19(25)20(18)26)21-17(13-14-5-4-6-14)28-23(35-21)22(30)27-15-9-11-36(31,32)12-10-15/h7-8,14-15,29H,4-6,9-13H2,1-3H3,(H,27,30)	WDWOXUSOFXZJEX-UHFFFAOYSA-N	392183	US10301272, Example 21/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392183	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392183&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188712	404960521							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783888	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCC2)c(Cl)c1Cl	InChI=1S/C23H29Cl2N3O3S2/c1-23(2,3)28-33(30,31)17-11-10-15(18(24)19(17)25)20-16(12-13-6-4-7-13)27-22(32-20)21(29)26-14-8-5-9-14/h10-11,13-14,28H,4-9,12H2,1-3H3,(H,26,29)	CFDRNOFYTVWUQF-UHFFFAOYSA-N	392184	US10301272, Example 21/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392184	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392184&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185807	404960522							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783889	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCC2)c(Cl)c1Cl	InChI=1S/C23H29Cl2N3O3S2/c1-23(2,3)28-33(30,31)17-11-10-15(18(24)19(17)25)20-16(12-13-6-4-7-13)27-22(32-20)21(29)26-14-8-5-9-14/h10-11,13-14,28H,4-9,12H2,1-3H3,(H,26,29)	CFDRNOFYTVWUQF-UHFFFAOYSA-N	392184	US10301272, Example 21/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392184	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392184&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185807	404960522							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783890	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-12-11-22(20-9-4-5-10-21(20)24)25-23(17-18-7-6-8-18)30-27(37-25)26(32)29-19-13-15-38(33,34)16-14-19/h4-5,9-12,18-19,31H,6-8,13-17H2,1-3H3,(H,29,32)	HHEONZPBOLISBI-UHFFFAOYSA-N	392185	US10301272, Example 21/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392185&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188705	404960523							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783891	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H35N3O5S3/c1-28(2,3)31-39(35,36)24-12-11-22(20-9-4-5-10-21(20)24)25-23(17-18-7-6-8-18)30-27(37-25)26(32)29-19-13-15-38(33,34)16-14-19/h4-5,9-12,18-19,31H,6-8,13-17H2,1-3H3,(H,29,32)	HHEONZPBOLISBI-UHFFFAOYSA-N	392185	US10301272, Example 21/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392185	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392185&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188705	404960523							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783892	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCC2)c2ccccc12	InChI=1S/C27H33N3O3S2/c1-27(2,3)30-35(32,33)23-15-14-21(19-12-4-5-13-20(19)23)24-22(16-17-8-6-9-17)29-26(34-24)25(31)28-18-10-7-11-18/h4-5,12-15,17-18,30H,6-11,16H2,1-3H3,(H,28,31)	KTBYQINSRIBHFI-UHFFFAOYSA-N	392186	US10301272, Example 21/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392186&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185809	404960524							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783893	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NC2CCC2)c2ccccc12	InChI=1S/C27H33N3O3S2/c1-27(2,3)30-35(32,33)23-15-14-21(19-12-4-5-13-20(19)23)24-22(16-17-8-6-9-17)29-26(34-24)25(31)28-18-10-7-11-18/h4-5,12-15,17-18,30H,6-11,16H2,1-3H3,(H,28,31)	KTBYQINSRIBHFI-UHFFFAOYSA-N	392186	US10301272, Example 21/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392186	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392186&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185809	404960524							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783894	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1)C(F)(F)F	InChI=1S/C23H27F6N3O5S2/c1-12(22(24,25)26)32-39(35,36)14-7-8-15(17(10-14)37-23(27,28)29)18-16(9-13-5-4-6-13)31-20(38-18)19(33)30-11-21(2,3)34/h7-8,10,12-13,32,34H,4-6,9,11H2,1-3H3,(H,30,33)/t12-/m0/s1	UXOZSACPYDIANF-LBPRGKRZSA-N	392187	US10301272, Example 21/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392187	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392187&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549409	404960525							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783895	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1)C(F)(F)F	InChI=1S/C23H27F6N3O5S2/c1-12(22(24,25)26)32-39(35,36)14-7-8-15(17(10-14)37-23(27,28)29)18-16(9-13-5-4-6-13)31-20(38-18)19(33)30-11-21(2,3)34/h7-8,10,12-13,32,34H,4-6,9,11H2,1-3H3,(H,30,33)/t12-/m0/s1	UXOZSACPYDIANF-LBPRGKRZSA-N	392187	US10301272, Example 21/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392187	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392187&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549409	404960525							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783896	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1)C(F)(F)F	InChI=1S/C22H27ClF3N3O4S2/c1-12(22(24,25)26)29-35(32,33)14-7-8-15(16(23)10-14)18-17(9-13-5-4-6-13)28-20(34-18)19(30)27-11-21(2,3)31/h7-8,10,12-13,29,31H,4-6,9,11H2,1-3H3,(H,27,30)/t12-/m0/s1	UKOJACBVNJLPIO-LBPRGKRZSA-N	392188	US10301272, Example 21/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392188	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392188&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549408	404960526							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783897	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1)C(F)(F)F	InChI=1S/C22H27ClF3N3O4S2/c1-12(22(24,25)26)29-35(32,33)14-7-8-15(16(23)10-14)18-17(9-13-5-4-6-13)28-20(34-18)19(30)27-11-21(2,3)31/h7-8,10,12-13,29,31H,4-6,9,11H2,1-3H3,(H,27,30)/t12-/m0/s1	UKOJACBVNJLPIO-LBPRGKRZSA-N	392188	US10301272, Example 21/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392188	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392188&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549408	404960526							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783898	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(c1)C(F)(F)F)C(F)(F)F	InChI=1S/C23H27F6N3O4S2/c1-12(22(24,25)26)32-38(35,36)14-7-8-15(16(10-14)23(27,28)29)18-17(9-13-5-4-6-13)31-20(37-18)19(33)30-11-21(2,3)34/h7-8,10,12-13,32,34H,4-6,9,11H2,1-3H3,(H,30,33)/t12-/m0/s1	IJCYZVLWRMIOCG-LBPRGKRZSA-N	392189	US10301272, Example 21/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392189	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392189&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188731	404960527							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783899	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(c1)C(F)(F)F)C(F)(F)F	InChI=1S/C23H27F6N3O4S2/c1-12(22(24,25)26)32-38(35,36)14-7-8-15(16(10-14)23(27,28)29)18-17(9-13-5-4-6-13)31-20(37-18)19(33)30-11-21(2,3)34/h7-8,10,12-13,32,34H,4-6,9,11H2,1-3H3,(H,30,33)/t12-/m0/s1	IJCYZVLWRMIOCG-LBPRGKRZSA-N	392189	US10301272, Example 21/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392189	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392189&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188731	404960527							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783900	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)F)c1)C(F)(F)F	InChI=1S/C23H28F5N3O5S2/c1-12(23(26,27)28)31-38(34,35)14-7-8-15(17(10-14)36-21(24)25)18-16(9-13-5-4-6-13)30-20(37-18)19(32)29-11-22(2,3)33/h7-8,10,12-13,21,31,33H,4-6,9,11H2,1-3H3,(H,29,32)/t12-/m0/s1	OZMBUCXLPMWWBK-LBPRGKRZSA-N	392190	US10301272, Example 21/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392190&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188683	404960528							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783901	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)F)c1)C(F)(F)F	InChI=1S/C23H28F5N3O5S2/c1-12(23(26,27)28)31-38(34,35)14-7-8-15(17(10-14)36-21(24)25)18-16(9-13-5-4-6-13)30-20(37-18)19(32)29-11-22(2,3)33/h7-8,10,12-13,21,31,33H,4-6,9,11H2,1-3H3,(H,29,32)/t12-/m0/s1	OZMBUCXLPMWWBK-LBPRGKRZSA-N	392190	US10301272, Example 21/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392190	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392190&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188683	404960528							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783902	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(c1)C(F)F)C(F)(F)F	InChI=1S/C23H28F5N3O4S2/c1-12(23(26,27)28)31-37(34,35)14-7-8-15(16(10-14)19(24)25)18-17(9-13-5-4-6-13)30-21(36-18)20(32)29-11-22(2,3)33/h7-8,10,12-13,19,31,33H,4-6,9,11H2,1-3H3,(H,29,32)/t12-/m0/s1	PNZKBKVBBDIHSC-LBPRGKRZSA-N	392191	US10301272, Example 21/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392191	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392191&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549410	404960529							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783903	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(c1)C(F)F)C(F)(F)F	InChI=1S/C23H28F5N3O4S2/c1-12(23(26,27)28)31-37(34,35)14-7-8-15(16(10-14)19(24)25)18-17(9-13-5-4-6-13)30-21(36-18)20(32)29-11-22(2,3)33/h7-8,10,12-13,19,31,33H,4-6,9,11H2,1-3H3,(H,29,32)/t12-/m0/s1	PNZKBKVBBDIHSC-LBPRGKRZSA-N	392191	US10301272, Example 21/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392191	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392191&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549410	404960529							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783904	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C28H32F5N3O4S2/c1-16(28(31,32)33)36-42(39,40)22-9-8-20(18-6-4-5-7-19(18)22)23-21(14-17-10-12-27(29,30)13-11-17)35-25(41-23)24(37)34-15-26(2,3)38/h4-9,16-17,36,38H,10-15H2,1-3H3,(H,34,37)/t16-/m0/s1	ZKGQGTWOWOVATF-INIZCTEOSA-N	392192	US10301272, Example 21/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392192&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185811	404960530							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783905	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C28H32F5N3O4S2/c1-16(28(31,32)33)36-42(39,40)22-9-8-20(18-6-4-5-7-19(18)22)23-21(14-17-10-12-27(29,30)13-11-17)35-25(41-23)24(37)34-15-26(2,3)38/h4-9,16-17,36,38H,10-15H2,1-3H3,(H,34,37)/t16-/m0/s1	ZKGQGTWOWOVATF-INIZCTEOSA-N	392192	US10301272, Example 21/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.51							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392192	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392192&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185811	404960530							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783906	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C24H32F3N3O5S2/c1-22(2,3)30-37(33,34)15-9-10-16(18(12-15)35-24(25,26)27)19-17(11-14-7-6-8-14)29-21(36-19)20(31)28-13-23(4,5)32/h9-10,12,14,30,32H,6-8,11,13H2,1-5H3,(H,28,31)	HGSZTJBBWZNGKG-UHFFFAOYSA-N	392193	US10301272, Example 21/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392193&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188707	404960531							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783907	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C24H32F3N3O5S2/c1-22(2,3)30-37(33,34)15-9-10-16(18(12-15)35-24(25,26)27)19-17(11-14-7-6-8-14)29-21(36-19)20(31)28-13-23(4,5)32/h9-10,12,14,30,32H,6-8,11,13H2,1-5H3,(H,28,31)	HGSZTJBBWZNGKG-UHFFFAOYSA-N	392193	US10301272, Example 21/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392193	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392193&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188707	404960531							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783908	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C25H34F3N3O5S2/c1-6-23(2,3)31-38(34,35)16-10-11-17(19(13-16)36-25(26,27)28)20-18(12-15-8-7-9-15)30-22(37-20)21(32)29-14-24(4,5)33/h10-11,13,15,31,33H,6-9,12,14H2,1-5H3,(H,29,32)	HHXUILPKYKGAEE-UHFFFAOYSA-N	392194	US10301272, Example 21/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392194&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188623	404960532							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783909	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(OC(F)(F)F)c1	InChI=1S/C25H34F3N3O5S2/c1-6-23(2,3)31-38(34,35)16-10-11-17(19(13-16)36-25(26,27)28)20-18(12-15-8-7-9-15)30-22(37-20)21(32)29-14-24(4,5)33/h10-11,13,15,31,33H,6-9,12,14H2,1-5H3,(H,29,32)	HHXUILPKYKGAEE-UHFFFAOYSA-N	392194	US10301272, Example 21/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392194	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392194&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188623	404960532							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783910	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(C(=O)N[C@H]2CC(C2)C(O)=O)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H41N3O4S/c1-28(2,3)22-15-18(16-23(31-22)29(4,5)6)24-21(12-17-10-8-7-9-11-17)32(36)26(37-24)25(33)30-20-13-19(14-20)27(34)35/h15-17,19-20H,7-14H2,1-6H3,(H,30,33)(H,34,35)/t19?,20-	QSCHTYOTUDVYEK-GUAVBDGJSA-N	392195	US10301272, Example 22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392195&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160583	404960533							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783911	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(C(=O)N[C@H]2CC(C2)C(O)=O)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H41N3O4S/c1-28(2,3)22-15-18(16-23(31-22)29(4,5)6)24-21(12-17-10-8-7-9-11-17)32(36)26(37-24)25(33)30-20-13-19(14-20)27(34)35/h15-17,19-20H,7-14H2,1-6H3,(H,30,33)(H,34,35)/t19?,20-	QSCHTYOTUDVYEK-GUAVBDGJSA-N	392195	US10301272, Example 22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392195&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160583	404960533							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783912	CC(C)(C)c1cc(cc(n1)C(C)(C)C)-c1sc(C(=O)N[C@H]2CC(C2)C(O)=O)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H41N3O4S/c1-28(2,3)22-15-18(16-23(31-22)29(4,5)6)24-21(12-17-10-8-7-9-11-17)32(36)26(37-24)25(33)30-20-13-19(14-20)27(34)35/h15-17,19-20H,7-14H2,1-6H3,(H,30,33)(H,34,35)/t19?,20-	QSCHTYOTUDVYEK-GUAVBDGJSA-N	392195	US10301272, Example 22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392195	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392195&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160583	404960533							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783913	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(C(=O)NC3CCC3)[n+]([O-])c2CC2CCCCC2)c2ccccc12	InChI=1S/C29H37N3O4S2/c1-29(2,3)31-38(35,36)25-17-16-23(21-14-7-8-15-22(21)25)26-24(18-19-10-5-4-6-11-19)32(34)28(37-26)27(33)30-20-12-9-13-20/h7-8,14-17,19-20,31H,4-6,9-13,18H2,1-3H3,(H,30,33)	WKVSFMFIDXGRPH-UHFFFAOYSA-N	392196	US10301272, Example 22/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392196&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012234	404960534							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783914	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(C(=O)NC3CCC3)[n+]([O-])c2CC2CCCCC2)c2ccccc12	InChI=1S/C29H37N3O4S2/c1-29(2,3)31-38(35,36)25-17-16-23(21-14-7-8-15-22(21)25)26-24(18-19-10-5-4-6-11-19)32(34)28(37-26)27(33)30-20-12-9-13-20/h7-8,14-17,19-20,31H,4-6,9-13,18H2,1-3H3,(H,30,33)	WKVSFMFIDXGRPH-UHFFFAOYSA-N	392196	US10301272, Example 22/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392196&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012234	404960534							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783915	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(C(=O)NC3CCC3)[n+]([O-])c2CC2CCCCC2)c2ccccc12	InChI=1S/C29H37N3O4S2/c1-29(2,3)31-38(35,36)25-17-16-23(21-14-7-8-15-22(21)25)26-24(18-19-10-5-4-6-11-19)32(34)28(37-26)27(33)30-20-12-9-13-20/h7-8,14-17,19-20,31H,4-6,9-13,18H2,1-3H3,(H,30,33)	WKVSFMFIDXGRPH-UHFFFAOYSA-N	392196	US10301272, Example 22/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392196	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392196&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012234	404960534							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783916	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(C(=O)NC2CCC2)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H40N2O2S/c1-28(2,3)21-16-20(17-22(18-21)29(4)13-14-29)25-24(15-19-9-6-5-7-10-19)31(33)27(34-25)26(32)30-23-11-8-12-23/h16-19,23H,5-15H2,1-4H3,(H,30,32)	MBGJJRJEEDVEEA-UHFFFAOYSA-N	392197	US10301272, Example 22/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392197&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012235	404960535							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783917	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(C(=O)NC2CCC2)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H40N2O2S/c1-28(2,3)21-16-20(17-22(18-21)29(4)13-14-29)25-24(15-19-9-6-5-7-10-19)31(33)27(34-25)26(32)30-23-11-8-12-23/h16-19,23H,5-15H2,1-4H3,(H,30,32)	MBGJJRJEEDVEEA-UHFFFAOYSA-N	392197	US10301272, Example 22/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392197&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012235	404960535							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783918	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(C(=O)NC2CCC2)[n+]([O-])c1CC1CCCCC1	InChI=1S/C29H40N2O2S/c1-28(2,3)21-16-20(17-22(18-21)29(4)13-14-29)25-24(15-19-9-6-5-7-10-19)31(33)27(34-25)26(32)30-23-11-8-12-23/h16-19,23H,5-15H2,1-4H3,(H,30,32)	MBGJJRJEEDVEEA-UHFFFAOYSA-N	392197	US10301272, Example 22/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392197	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392197&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012235	404960535							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783919	CC(C)(C)c1cc(cc(c1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H40N2O4S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)35)24-23(11-17-9-7-6-8-10-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,6-11,14-15H2,1-5H3,(H,30,32)(H,33,34)/t19?,22-	DJTCUUMWOSSYBE-XVUZFVQRSA-N	392198	US10301272, Example 23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392198&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160547	404960536							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783920	CC(C)(C)c1cc(cc(c1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H40N2O4S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)35)24-23(11-17-9-7-6-8-10-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,6-11,14-15H2,1-5H3,(H,30,32)(H,33,34)/t19?,22-	DJTCUUMWOSSYBE-XVUZFVQRSA-N	392198	US10301272, Example 23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392198&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160547	404960536							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783921	CC(C)(C)c1cc(cc(c1)C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H40N2O4S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)35)24-23(11-17-9-7-6-8-10-17)31-26(36-24)25(32)30-22-14-19(15-22)27(33)34/h12-13,16-17,19,22,35H,6-11,14-15H2,1-5H3,(H,30,32)(H,33,34)/t19?,22-	DJTCUUMWOSSYBE-XVUZFVQRSA-N	392198	US10301272, Example 23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392198	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392198&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160547	404960536							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783922	CC(C)(C)c1cc(cc(c1)C(C)(C)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H39FN2O3S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)30)24-23(11-17-9-7-6-8-10-17)32-26(36-24)25(33)31-22-14-19(15-22)27(34)35/h12-13,16-17,19,22H,6-11,14-15H2,1-5H3,(H,31,33)(H,34,35)/t19?,22-	QLSDOVMAKVXDRG-XVUZFVQRSA-N	392199	US10301272, Example 24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392199&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160528	404960537							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783923	CC(C)(C)c1cc(cc(c1)C(C)(C)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H39FN2O3S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)30)24-23(11-17-9-7-6-8-10-17)32-26(36-24)25(33)31-22-14-19(15-22)27(34)35/h12-13,16-17,19,22H,6-11,14-15H2,1-5H3,(H,31,33)(H,34,35)/t19?,22-	QLSDOVMAKVXDRG-XVUZFVQRSA-N	392199	US10301272, Example 24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392199&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160528	404960537							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783924	CC(C)(C)c1cc(cc(c1)C(C)(C)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C29H39FN2O3S/c1-28(2,3)20-12-18(13-21(16-20)29(4,5)30)24-23(11-17-9-7-6-8-10-17)32-26(36-24)25(33)31-22-14-19(15-22)27(34)35/h12-13,16-17,19,22H,6-11,14-15H2,1-5H3,(H,31,33)(H,34,35)/t19?,22-	QLSDOVMAKVXDRG-XVUZFVQRSA-N	392199	US10301272, Example 24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392199	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392199&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160528	404960537							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783925	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(sc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C30H40N2O3S/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)36-27(32-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20?,23-	UPQMFJFXQYEKTR-TYHZPSRNSA-N	392200	US10301272, Example 25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392200	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392200&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160551	404960538							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783926	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(sc1CC1CCCCC1)C(=O)N[C@H]1CC(C1)C(O)=O	InChI=1S/C30H40N2O3S/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)36-27(32-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20?,23-	UPQMFJFXQYEKTR-TYHZPSRNSA-N	392200	US10301272, Example 25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392200	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392200&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160551	404960538							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783927	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(sc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)39-28(32-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	GQMIUMPESRAULB-MXVIHJGJSA-N	392201	US10301272, Example 25/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.26							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392201	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392201&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185814	404960539							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783928	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(sc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)39-28(32-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	GQMIUMPESRAULB-MXVIHJGJSA-N	392201	US10301272, Example 25/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.58							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392201	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392201&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185814	404960539							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783929	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(sc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)39-29(32-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	DKTDEGPLWZIMFM-UHFFFAOYSA-N	392202	US10301272, Example 25/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392202	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392202&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185815	404960540							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783930	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(sc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)39-29(32-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	DKTDEGPLWZIMFM-UHFFFAOYSA-N	392202	US10301272, Example 25/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392202	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392202&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185815	404960540							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783931	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	KMPMBOMDLPHBHX-UHFFFAOYSA-N	392203	US10301272, Example 100	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392203&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160527	404960541							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783932	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	KMPMBOMDLPHBHX-UHFFFAOYSA-N	392203	US10301272, Example 100	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392203&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160527	404960541							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783933	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	KMPMBOMDLPHBHX-UHFFFAOYSA-N	392203	US10301272, Example 100	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392203	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392203&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160527	404960541							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783934	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O5S/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	PENNQVNUUSBZEI-UHFFFAOYSA-N	392204	US10301272, Example 100/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392204&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72550980	404960542							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783935	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O5S/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	PENNQVNUUSBZEI-UHFFFAOYSA-N	392204	US10301272, Example 100/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392204&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72550980	404960542							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783936	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H45N3O5S/c1-29(2,3)23-19-21(12-13-25(23)39(35,36)33-30(4,5)6)26-24(18-20-10-8-7-9-11-20)32-28(38-26)27(34)31-22-14-16-37-17-15-22/h12-13,19-20,22,33H,7-11,14-18H2,1-6H3,(H,31,34)	PENNQVNUUSBZEI-UHFFFAOYSA-N	392204	US10301272, Example 100/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392204	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392204&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72550980	404960542							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783937	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O6S/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	HHVIPAHRUOSFEE-MEMLXQNLSA-N	392205	US10301272, Example 100/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3162							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392205&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551199	404960543							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783938	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O6S/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	HHVIPAHRUOSFEE-MEMLXQNLSA-N	392205	US10301272, Example 100/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392205&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551199	404960543							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783939	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H43N3O6S/c1-29(2,3)22-17-19(12-13-24(22)40(37,38)33-30(4,5)6)25-23(14-18-10-8-7-9-11-18)32-27(39-25)26(34)31-21-15-20(16-21)28(35)36/h12-13,17-18,20-21,33H,7-11,14-16H2,1-6H3,(H,31,34)(H,35,36)/t20-,21-	HHVIPAHRUOSFEE-MEMLXQNLSA-N	392205	US10301272, Example 100/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392205	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392205&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551199	404960543							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783940	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O5S/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	SAEGZKGDOAFSRY-UHFFFAOYSA-N	392206	US10301272, Example 100/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392206&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551200	404960544							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783941	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O5S/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	SAEGZKGDOAFSRY-UHFFFAOYSA-N	392206	US10301272, Example 100/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392206&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551200	404960544							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783942	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O5S/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	SAEGZKGDOAFSRY-UHFFFAOYSA-N	392206	US10301272, Example 100/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392206	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392206&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551200	404960544							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783943	CN(C1CCOCC1)C(=O)c1nc(CC2CCCCC2)c(o1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C31H41N3O5S/c1-31(2,3)33-40(36,37)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)32-29(39-28)30(35)34(4)22-16-18-38-19-17-22/h8-9,12-15,21-22,33H,5-7,10-11,16-20H2,1-4H3	GVCXWXCTBRAHBX-UHFFFAOYSA-N	392207	US10301272, Example 100/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392207&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186078	404960545							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783944	CN(C1CCOCC1)C(=O)c1nc(CC2CCCCC2)c(o1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C31H41N3O5S/c1-31(2,3)33-40(36,37)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)32-29(39-28)30(35)34(4)22-16-18-38-19-17-22/h8-9,12-15,21-22,33H,5-7,10-11,16-20H2,1-4H3	GVCXWXCTBRAHBX-UHFFFAOYSA-N	392207	US10301272, Example 100/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392207&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186078	404960545							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783945	CN(C1CCOCC1)C(=O)c1nc(CC2CCCCC2)c(o1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C31H41N3O5S/c1-31(2,3)33-40(36,37)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)32-29(39-28)30(35)34(4)22-16-18-38-19-17-22/h8-9,12-15,21-22,33H,5-7,10-11,16-20H2,1-4H3	GVCXWXCTBRAHBX-UHFFFAOYSA-N	392207	US10301272, Example 100/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392207	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392207&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186078	404960545							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783946	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCOCC2)c2ccccc12	InChI=1S/C31H41N3O6S/c1-30(2,3)34-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(40-27)28(35)32-20-31(36)15-17-39-18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RNKINVRKPXKEBW-UHFFFAOYSA-N	392208	US10301272, Example 100/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392208&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551201	404960546							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783947	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCOCC2)c2ccccc12	InChI=1S/C31H41N3O6S/c1-30(2,3)34-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(40-27)28(35)32-20-31(36)15-17-39-18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RNKINVRKPXKEBW-UHFFFAOYSA-N	392208	US10301272, Example 100/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392208&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551201	404960546							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783948	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCOCC2)c2ccccc12	InChI=1S/C31H41N3O6S/c1-30(2,3)34-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(40-27)28(35)32-20-31(36)15-17-39-18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RNKINVRKPXKEBW-UHFFFAOYSA-N	392208	US10301272, Example 100/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392208	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392208&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551201	404960546							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783949	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RYMQDGGJMJDRKS-UHFFFAOYSA-N	392209	US10301272, Example 100/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392209&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551202	404960547							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783950	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RYMQDGGJMJDRKS-UHFFFAOYSA-N	392209	US10301272, Example 100/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392209&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551202	404960547							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783951	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RYMQDGGJMJDRKS-UHFFFAOYSA-N	392209	US10301272, Example 100/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392209	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392209&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551202	404960547							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783952	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O5S/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	SOEFCKZCSLKMCZ-UHFFFAOYSA-N	392210	US10301272, Example 100/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392210&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547764	404960548							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783953	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O5S/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	SOEFCKZCSLKMCZ-UHFFFAOYSA-N	392210	US10301272, Example 100/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392210&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547764	404960548							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783954	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O5S/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	SOEFCKZCSLKMCZ-UHFFFAOYSA-N	392210	US10301272, Example 100/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392210	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392210&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547764	404960548							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783955	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O7S2/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RFAVWFBXMYYLKB-UHFFFAOYSA-N	392211	US10301272, Example 100/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392211	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392211&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547762	404960549							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783956	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O7S2/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RFAVWFBXMYYLKB-UHFFFAOYSA-N	392211	US10301272, Example 100/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392211	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392211&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547762	404960549							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783957	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O7S2/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	RFAVWFBXMYYLKB-UHFFFAOYSA-N	392211	US10301272, Example 100/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392211	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392211&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547762	404960549							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783958	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783959	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783960	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783961	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCOCC3)c2ccccc12	InChI=1S/C32H41N3O5S/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-39-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	VUEICKMKIRYGFL-UHFFFAOYSA-N	392213	US10301272, Example 100/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392213&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186081	404960551							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783962	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCOCC3)c2ccccc12	InChI=1S/C32H41N3O5S/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-39-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	VUEICKMKIRYGFL-UHFFFAOYSA-N	392213	US10301272, Example 100/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392213&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186081	404960551							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783963	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCOCC3)c2ccccc12	InChI=1S/C32H41N3O5S/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(40-28)30(36)35-20-32(21-35)15-17-39-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	VUEICKMKIRYGFL-UHFFFAOYSA-N	392213	US10301272, Example 100/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392213	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392213&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186081	404960551							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783964	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCSCC3)c2ccccc12	InChI=1S/C32H41N3O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(39-28)30(36)35-20-32(21-35)15-17-40-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	RRNYZYULYDRTKJ-UHFFFAOYSA-N	392214	US10301272, Example 100/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392214&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186082	404960552							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783965	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCSCC3)c2ccccc12	InChI=1S/C32H41N3O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(39-28)30(36)35-20-32(21-35)15-17-40-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	RRNYZYULYDRTKJ-UHFFFAOYSA-N	392214	US10301272, Example 100/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392214&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186082	404960552							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783966	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCSCC3)c2ccccc12	InChI=1S/C32H41N3O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(39-28)30(36)35-20-32(21-35)15-17-40-18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	RRNYZYULYDRTKJ-UHFFFAOYSA-N	392214	US10301272, Example 100/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392214	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392214&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186082	404960552							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783967	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15849							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783968	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783969	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O6S2/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JGSCGNUMQKXWTL-UHFFFAOYSA-N	392212	US10301272, Example 100/12::US10301272, Example 100/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392212	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392212&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547763	404960550							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783970	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O6S/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	XCNGDSCXTXNZSP-MXVIHJGJSA-N	392216	US10301272, Example 100/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392216	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392216&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548001	404960553							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783971	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O6S/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	XCNGDSCXTXNZSP-MXVIHJGJSA-N	392216	US10301272, Example 100/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392216	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392216&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548001	404960553							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783972	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H37N3O6S/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h7-8,11-14,18-20,33H,4-6,9-10,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	XCNGDSCXTXNZSP-MXVIHJGJSA-N	392216	US10301272, Example 100/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392216	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392216&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548001	404960553							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783973	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	REXZLGWWWPJQIG-UHFFFAOYSA-N	392217	US10301272, Example 100/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548002	404960554							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783974	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	REXZLGWWWPJQIG-UHFFFAOYSA-N	392217	US10301272, Example 100/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548002	404960554							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783975	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	REXZLGWWWPJQIG-UHFFFAOYSA-N	392217	US10301272, Example 100/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392217	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392217&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548002	404960554							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783976	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783977	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783978	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783979	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783980	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783981	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783982	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O6S/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	VSGFJKOPDFDEDY-WKILWMFISA-N	392220	US10301272, Example 100/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547765	404960557							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783983	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O6S/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	VSGFJKOPDFDEDY-WKILWMFISA-N	392220	US10301272, Example 100/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547765	404960557							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783984	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O6S/c1-26(2,3)31-38(35,36)19-10-9-17(20(27)21(19)28)22-18(11-14-7-5-4-6-8-14)30-24(37-22)23(32)29-16-12-15(13-16)25(33)34/h9-10,14-16,31H,4-8,11-13H2,1-3H3,(H,29,32)(H,33,34)/t15-,16-	VSGFJKOPDFDEDY-WKILWMFISA-N	392220	US10301272, Example 100/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392220	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392220&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547765	404960557							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783985	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O3/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	XDOMKJYYQKINOE-UHFFFAOYSA-N	392221	US10301272, Example 100/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548003	404960558							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783986	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O3/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	XDOMKJYYQKINOE-UHFFFAOYSA-N	392221	US10301272, Example 100/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548003	404960558							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783987	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C30H42N2O3/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)32-28(35-26)27(33)31-24-10-14-34-15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	XDOMKJYYQKINOE-UHFFFAOYSA-N	392221	US10301272, Example 100/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392221	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392221&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548003	404960558							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783988	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C30H42N2O4/c1-28(2,3)21-15-20(16-22(17-21)30(6)12-13-30)24-23(14-19-10-8-7-9-11-19)32-26(36-24)25(33)31-18-29(4,5)27(34)35/h15-17,19H,7-14,18H2,1-6H3,(H,31,33)(H,34,35)	HMPLGOAAXXCXHV-UHFFFAOYSA-N	392222	US10301272, Example 100/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392222	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392222&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548004	404960559							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783989	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C30H42N2O4/c1-28(2,3)21-15-20(16-22(17-21)30(6)12-13-30)24-23(14-19-10-8-7-9-11-19)32-26(36-24)25(33)31-18-29(4,5)27(34)35/h15-17,19H,7-14,18H2,1-6H3,(H,31,33)(H,34,35)	HMPLGOAAXXCXHV-UHFFFAOYSA-N	392222	US10301272, Example 100/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392222	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392222&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548004	404960559							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783990	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)NCC(C)(C)C(O)=O	InChI=1S/C30H42N2O4/c1-28(2,3)21-15-20(16-22(17-21)30(6)12-13-30)24-23(14-19-10-8-7-9-11-19)32-26(36-24)25(33)31-18-29(4,5)27(34)35/h15-17,19H,7-14,18H2,1-6H3,(H,31,33)(H,34,35)	HMPLGOAAXXCXHV-UHFFFAOYSA-N	392222	US10301272, Example 100/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392222	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392222&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548004	404960559							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783991	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	GVBFNUZLZCVBPN-JKIUYZKVSA-N	392223	US10301272, Example 100/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392223	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392223&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72201104	404960560							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783992	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	GVBFNUZLZCVBPN-JKIUYZKVSA-N	392223	US10301272, Example 100/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392223	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392223&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72201104	404960560							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783993	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1oc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C30H40N2O4/c1-29(2,3)21-13-19(14-22(17-21)30(4)10-11-30)25-24(12-18-8-6-5-7-9-18)32-27(36-25)26(33)31-23-15-20(16-23)28(34)35/h13-14,17-18,20,23H,5-12,15-16H2,1-4H3,(H,31,33)(H,34,35)/t20-,23-	GVBFNUZLZCVBPN-JKIUYZKVSA-N	392223	US10301272, Example 100/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392223	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392223&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72201104	404960560							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783994	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCCC(C)(C)C(O)=O)c2ccccc12	InChI=1S/C31H41N3O6S/c1-30(2,3)34-41(38,39)25-16-15-23(21-13-9-10-14-22(21)25)26-24(19-20-11-7-6-8-12-20)33-28(40-26)27(35)32-18-17-31(4,5)29(36)37/h9-10,13-16,20,34H,6-8,11-12,17-19H2,1-5H3,(H,32,35)(H,36,37)	JWHCJHZIURANAH-UHFFFAOYSA-N	392224	US10301272, Example 100/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392224&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186083	404960561							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783995	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCCC(C)(C)C(O)=O)c2ccccc12	InChI=1S/C31H41N3O6S/c1-30(2,3)34-41(38,39)25-16-15-23(21-13-9-10-14-22(21)25)26-24(19-20-11-7-6-8-12-20)33-28(40-26)27(35)32-18-17-31(4,5)29(36)37/h9-10,13-16,20,34H,6-8,11-12,17-19H2,1-5H3,(H,32,35)(H,36,37)	JWHCJHZIURANAH-UHFFFAOYSA-N	392224	US10301272, Example 100/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392224	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392224&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186083	404960561							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783996	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC(C)(CC2)C(O)=O)c2ccccc12	InChI=1S/C33H43N3O6S/c1-32(2,3)36-43(40,41)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)35-30(42-28)29(37)34-22-16-18-33(4,19-17-22)31(38)39/h8-9,12-15,21-22,36H,5-7,10-11,16-20H2,1-4H3,(H,34,37)(H,38,39)	BYEPQRDVQPCSLI-UHFFFAOYSA-N	392225	US10301272, Example 100/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186084	404960562							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783997	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC(C)(CC2)C(O)=O)c2ccccc12	InChI=1S/C33H43N3O6S/c1-32(2,3)36-43(40,41)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)35-30(42-28)29(37)34-22-16-18-33(4,19-17-22)31(38)39/h8-9,12-15,21-22,36H,5-7,10-11,16-20H2,1-4H3,(H,34,37)(H,38,39)	BYEPQRDVQPCSLI-UHFFFAOYSA-N	392225	US10301272, Example 100/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186084	404960562							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783998	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC(C)(CC2)C(O)=O)c2ccccc12	InChI=1S/C33H43N3O6S/c1-32(2,3)36-43(40,41)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)35-30(42-28)29(37)34-22-16-18-33(4,19-17-22)31(38)39/h8-9,12-15,21-22,36H,5-7,10-11,16-20H2,1-4H3,(H,34,37)(H,38,39)	BYEPQRDVQPCSLI-UHFFFAOYSA-N	392225	US10301272, Example 100/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392225	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392225&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186084	404960562							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783999	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(C3)C(O)=O)c2ccccc12	InChI=1S/C33H41N3O6S/c1-31(2,3)36-43(40,41)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)34-29(42-27)28(37)35-33-17-15-32(20-33,16-18-33)30(38)39/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H,35,37)(H,38,39)	BDXRHOJEFBPJTM-UHFFFAOYSA-N	392226	US10301272, Example 100/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392226&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186085	404960563							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784000	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(C3)C(O)=O)c2ccccc12	InChI=1S/C33H41N3O6S/c1-31(2,3)36-43(40,41)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)34-29(42-27)28(37)35-33-17-15-32(20-33,16-18-33)30(38)39/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H,35,37)(H,38,39)	BDXRHOJEFBPJTM-UHFFFAOYSA-N	392226	US10301272, Example 100/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392226&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186085	404960563							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784001	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(C3)C(O)=O)c2ccccc12	InChI=1S/C33H41N3O6S/c1-31(2,3)36-43(40,41)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)34-29(42-27)28(37)35-33-17-15-32(20-33,16-18-33)30(38)39/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H,35,37)(H,38,39)	BDXRHOJEFBPJTM-UHFFFAOYSA-N	392226	US10301272, Example 100/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392226	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392226&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186085	404960563							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784002	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12	InChI=1S/C30H37N3O6S2/c1-29(2,3)32-41(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-20-9-5-4-6-10-20)31-27(39-26)28(34)33-16-30(17-33)18-40(35,36)19-30/h7-8,11-14,20,32H,4-6,9-10,15-19H2,1-3H3	VFSYCKDHKAUECA-UHFFFAOYSA-N	392227	US10301272, Example 100/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392227	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392227&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186087	404960564							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784003	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12	InChI=1S/C30H37N3O6S2/c1-29(2,3)32-41(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-20-9-5-4-6-10-20)31-27(39-26)28(34)33-16-30(17-33)18-40(35,36)19-30/h7-8,11-14,20,32H,4-6,9-10,15-19H2,1-3H3	VFSYCKDHKAUECA-UHFFFAOYSA-N	392227	US10301272, Example 100/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392227	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392227&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186087	404960564							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784004	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784005	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784006	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O6S2/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	IQYDZOOWMUSCMC-UHFFFAOYSA-N	392219	US10301272, Example 100/16::US10301272, Example 100/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392219	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392219&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72551203	404960556							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784007	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784008	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784009	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O5S/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	GRTBNRQFXKQEKY-UHFFFAOYSA-N	392218	US10301272, Example 100/15::US10301272, Example 100/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392218	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392218&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72547766	404960555							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784010	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1Cl	InChI=1S/C25H33Cl2N3O4S/c1-25(2,3)30-35(32,33)19-13-12-17(20(26)21(19)27)22-18(14-15-8-5-4-6-9-15)29-24(34-22)23(31)28-16-10-7-11-16/h12-13,15-16,30H,4-11,14H2,1-3H3,(H,28,31)	LPHABOXKJXVRTH-UHFFFAOYSA-N	392230	US10301272, Example 100/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392230	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392230&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186088	404960565							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784011	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1Cl	InChI=1S/C25H33Cl2N3O4S/c1-25(2,3)30-35(32,33)19-13-12-17(20(26)21(19)27)22-18(14-15-8-5-4-6-9-15)29-24(34-22)23(31)28-16-10-7-11-16/h12-13,15-16,30H,4-11,14H2,1-3H3,(H,28,31)	LPHABOXKJXVRTH-UHFFFAOYSA-N	392230	US10301272, Example 100/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392230	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392230&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186088	404960565							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784012	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCC2)c(Cl)c1Cl	InChI=1S/C25H33Cl2N3O4S/c1-25(2,3)30-35(32,33)19-13-12-17(20(26)21(19)27)22-18(14-15-8-5-4-6-9-15)29-24(34-22)23(31)28-16-10-7-11-16/h12-13,15-16,30H,4-11,14H2,1-3H3,(H,28,31)	LPHABOXKJXVRTH-UHFFFAOYSA-N	392230	US10301272, Example 100/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392230	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392230&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186088	404960565							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784013	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccncc12	InChI=1S/C29H38N4O6S2/c1-29(2,3)33-41(37,38)25-10-9-22(21-11-14-30-18-23(21)25)26-24(17-19-7-5-4-6-8-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h9-11,14,18-20,33H,4-8,12-13,15-17H2,1-3H3,(H,31,34)	AQCCGQDFSLMHEP-UHFFFAOYSA-N	392231	US10301272, Example 100/28	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392231	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392231&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188681	404960566							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784014	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccncc12	InChI=1S/C29H38N4O6S2/c1-29(2,3)33-41(37,38)25-10-9-22(21-11-14-30-18-23(21)25)26-24(17-19-7-5-4-6-8-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h9-11,14,18-20,33H,4-8,12-13,15-17H2,1-3H3,(H,31,34)	AQCCGQDFSLMHEP-UHFFFAOYSA-N	392231	US10301272, Example 100/28	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392231	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392231&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188681	404960566							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784015	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(oc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	CFQCXCVYHPIEOM-UHFFFAOYSA-N	392232	US10301272, Example 101	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392232	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392232&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032716	404960567							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784016	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(oc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	CFQCXCVYHPIEOM-UHFFFAOYSA-N	392232	US10301272, Example 101	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392232	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392232&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032716	404960567							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784017	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(oc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2O2/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	CFQCXCVYHPIEOM-UHFFFAOYSA-N	392232	US10301272, Example 101	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392232	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392232&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032716	404960567							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784018	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C35H46N4O7S2/c1-33(2,3)39-48(44,45)28-15-14-26(24-12-8-9-13-25(24)28)29-27(22-23-10-6-5-7-11-23)36-31(46-29)30(40)37-35-19-16-34(17-20-35,18-21-35)32(41)38-47(4,42)43/h8-9,12-15,23,39H,5-7,10-11,16-22H2,1-4H3,(H,37,40)(H,38,41)	GLIXFZJIJVCUMZ-UHFFFAOYSA-N	392233	US10301272, Example 102	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160569	404960568							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784019	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C35H46N4O7S2/c1-33(2,3)39-48(44,45)28-15-14-26(24-12-8-9-13-25(24)28)29-27(22-23-10-6-5-7-11-23)36-31(46-29)30(40)37-35-19-16-34(17-20-35,18-21-35)32(41)38-47(4,42)43/h8-9,12-15,23,39H,5-7,10-11,16-22H2,1-4H3,(H,37,40)(H,38,41)	GLIXFZJIJVCUMZ-UHFFFAOYSA-N	392233	US10301272, Example 102	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160569	404960568							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784020	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C35H46N4O7S2/c1-33(2,3)39-48(44,45)28-15-14-26(24-12-8-9-13-25(24)28)29-27(22-23-10-6-5-7-11-23)36-31(46-29)30(40)37-35-19-16-34(17-20-35,18-21-35)32(41)38-47(4,42)43/h8-9,12-15,23,39H,5-7,10-11,16-22H2,1-4H3,(H,37,40)(H,38,41)	GLIXFZJIJVCUMZ-UHFFFAOYSA-N	392233	US10301272, Example 102	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392233	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392233&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160569	404960568							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784021	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C31H40N4O7S2/c1-31(2,3)35-44(40,41)26-15-14-24(22-12-8-9-13-23(22)26)27-25(16-19-10-6-5-7-11-19)33-30(42-27)29(37)32-21-17-20(18-21)28(36)34-43(4,38)39/h8-9,12-15,19-21,35H,5-7,10-11,16-18H2,1-4H3,(H,32,37)(H,34,36)/t20-,21-	CAZJDZDXVPUKFP-MEMLXQNLSA-N	392234	US10301272, Example 102/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186089	404960569							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784022	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C31H40N4O7S2/c1-31(2,3)35-44(40,41)26-15-14-24(22-12-8-9-13-23(22)26)27-25(16-19-10-6-5-7-11-19)33-30(42-27)29(37)32-21-17-20(18-21)28(36)34-43(4,38)39/h8-9,12-15,19-21,35H,5-7,10-11,16-18H2,1-4H3,(H,32,37)(H,34,36)/t20-,21-	CAZJDZDXVPUKFP-MEMLXQNLSA-N	392234	US10301272, Example 102/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186089	404960569							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784023	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(=O)NS(C)(=O)=O)c2ccccc12	InChI=1S/C31H40N4O7S2/c1-31(2,3)35-44(40,41)26-15-14-24(22-12-8-9-13-23(22)26)27-25(16-19-10-6-5-7-11-19)33-30(42-27)29(37)32-21-17-20(18-21)28(36)34-43(4,38)39/h8-9,12-15,19-21,35H,5-7,10-11,16-18H2,1-4H3,(H,32,37)(H,34,36)/t20-,21-	CAZJDZDXVPUKFP-MEMLXQNLSA-N	392234	US10301272, Example 102/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392234	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392234&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186089	404960569							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784024	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)39-29(32-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RSTRIEZUQHMPMT-UHFFFAOYSA-N	392235	US10301272, Example 103	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160497	404960570							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784025	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)39-29(32-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RSTRIEZUQHMPMT-UHFFFAOYSA-N	392235	US10301272, Example 103	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160497	404960570							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784026	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O6S2/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)39-29(32-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	RSTRIEZUQHMPMT-UHFFFAOYSA-N	392235	US10301272, Example 103	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392235	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392235&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160497	404960570							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784027	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)43-30(35-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	LDMQAVVRGZTFPR-UHFFFAOYSA-N	392236	US10301272, Example 103/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186092	404960571							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784028	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)43-30(35-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	LDMQAVVRGZTFPR-UHFFFAOYSA-N	392236	US10301272, Example 103/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186092	404960571							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784029	CC(C)(C)NS(=O)(=O)c1ccc(-c2nc(oc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O6S/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)43-30(35-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	LDMQAVVRGZTFPR-UHFFFAOYSA-N	392236	US10301272, Example 103/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392236	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392236&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186092	404960571							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784030	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(oc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)OC=O	InChI=1S/C30H40N2O4/c1-29(2,3)21-13-20(14-22(15-21)30(4)10-11-30)26-25(12-19-8-6-5-7-9-19)36-28(32-26)27(34)31-23-16-24(17-23)35-18-33/h13-15,18-19,23-24H,5-12,16-17H2,1-4H3,(H,31,34)/t23-,24-	LHZXVTHKURLADX-RQNOJGIXSA-N	392237	US10301272, Example 103/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392237&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186091	404960572							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784031	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(oc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)OC=O	InChI=1S/C30H40N2O4/c1-29(2,3)21-13-20(14-22(15-21)30(4)10-11-30)26-25(12-19-8-6-5-7-9-19)36-28(32-26)27(34)31-23-16-24(17-23)35-18-33/h13-15,18-19,23-24H,5-12,16-17H2,1-4H3,(H,31,34)/t23-,24-	LHZXVTHKURLADX-RQNOJGIXSA-N	392237	US10301272, Example 103/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392237	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392237&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186091	404960572							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784032	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(oc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C30H42N2O4S/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)36-28(32-26)27(33)31-24-10-14-37(34,35)15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	SAERRBQYRPWUBN-UHFFFAOYSA-N	392238	US10301272, Example 103/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392238&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186093	404960573							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784033	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1nc(oc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C30H42N2O4S/c1-29(2,3)22-17-21(18-23(19-22)30(4)12-13-30)26-25(16-20-8-6-5-7-9-20)36-28(32-26)27(33)31-24-10-14-37(34,35)15-11-24/h17-20,24H,5-16H2,1-4H3,(H,31,33)	SAERRBQYRPWUBN-UHFFFAOYSA-N	392238	US10301272, Example 103/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392238	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392238&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186093	404960573							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784034	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H35N3O6S2/c1-28(2,3)31-39(35,36)24-12-11-22(20-9-4-5-10-21(20)24)25-23(17-18-7-6-8-18)30-27(37-25)26(32)29-19-13-15-38(33,34)16-14-19/h4-5,9-12,18-19,31H,6-8,13-17H2,1-3H3,(H,29,32)	FMHQBIKDHIHIMD-UHFFFAOYSA-N	392239	US10301272, Example 104	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392239&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160511	404960574							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784035	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H35N3O6S2/c1-28(2,3)31-39(35,36)24-12-11-22(20-9-4-5-10-21(20)24)25-23(17-18-7-6-8-18)30-27(37-25)26(32)29-19-13-15-38(33,34)16-14-19/h4-5,9-12,18-19,31H,6-8,13-17H2,1-3H3,(H,29,32)	FMHQBIKDHIHIMD-UHFFFAOYSA-N	392239	US10301272, Example 104	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392239&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160511	404960574							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784036	CC(C)(C)NS(=O)(=O)c1ccc(-c2oc(nc2CC2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H35N3O6S2/c1-28(2,3)31-39(35,36)24-12-11-22(20-9-4-5-10-21(20)24)25-23(17-18-7-6-8-18)30-27(37-25)26(32)29-19-13-15-38(33,34)16-14-19/h4-5,9-12,18-19,31H,6-8,13-17H2,1-3H3,(H,29,32)	FMHQBIKDHIHIMD-UHFFFAOYSA-N	392239	US10301272, Example 104	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392239	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392239&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160511	404960574							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784037	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NC(=O)CC(C)(C)O)nc1CC1CCCCC1	InChI=1S/C26H36F3N3O4S2/c1-24(2,3)32-38(35,36)20-12-11-17(14-18(20)26(27,28)29)22-19(13-16-9-7-6-8-10-16)30-23(37-22)31-21(33)15-25(4,5)34/h11-12,14,16,32,34H,6-10,13,15H2,1-5H3,(H,30,31,33)	RKHRGJNYGJYPPI-UHFFFAOYSA-N	392240	US10301272, Example 200	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392240&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160549	404960575							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784038	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NC(=O)CC(C)(C)O)nc1CC1CCCCC1	InChI=1S/C26H36F3N3O4S2/c1-24(2,3)32-38(35,36)20-12-11-17(14-18(20)26(27,28)29)22-19(13-16-9-7-6-8-10-16)30-23(37-22)31-21(33)15-25(4,5)34/h11-12,14,16,32,34H,6-10,13,15H2,1-5H3,(H,30,31,33)	RKHRGJNYGJYPPI-UHFFFAOYSA-N	392240	US10301272, Example 200	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392240&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160549	404960575							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784039	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NC(=O)CC(C)(C)O)nc1CC1CCCCC1	InChI=1S/C26H36F3N3O4S2/c1-24(2,3)32-38(35,36)20-12-11-17(14-18(20)26(27,28)29)22-19(13-16-9-7-6-8-10-16)30-23(37-22)31-21(33)15-25(4,5)34/h11-12,14,16,32,34H,6-10,13,15H2,1-5H3,(H,30,31,33)	RKHRGJNYGJYPPI-UHFFFAOYSA-N	392240	US10301272, Example 200	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392240	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392240&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160549	404960575							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784040	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(CC3CCCCC3)c(s2)-c2ccc(c(c2)C(F)(F)F)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C31H38F3N3O5S3/c1-5-44(39,40)23-14-11-21(12-15-23)18-27(38)36-29-35-25(17-20-9-7-6-8-10-20)28(43-29)22-13-16-26(24(19-22)31(32,33)34)45(41,42)37-30(2,3)4/h11-16,19-20,37H,5-10,17-18H2,1-4H3,(H,35,36,38)	VTFSLOIXAMJGJE-UHFFFAOYSA-N	392241	US10301272, Example 200/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392241&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188653	404960576							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784041	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(CC3CCCCC3)c(s2)-c2ccc(c(c2)C(F)(F)F)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C31H38F3N3O5S3/c1-5-44(39,40)23-14-11-21(12-15-23)18-27(38)36-29-35-25(17-20-9-7-6-8-10-20)28(43-29)22-13-16-26(24(19-22)31(32,33)34)45(41,42)37-30(2,3)4/h11-16,19-20,37H,5-10,17-18H2,1-4H3,(H,35,36,38)	VTFSLOIXAMJGJE-UHFFFAOYSA-N	392241	US10301272, Example 200/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392241&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188653	404960576							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784042	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(CC3CCCCC3)c(s2)-c2ccc(c(c2)C(F)(F)F)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C31H38F3N3O5S3/c1-5-44(39,40)23-14-11-21(12-15-23)18-27(38)36-29-35-25(17-20-9-7-6-8-10-20)28(43-29)22-13-16-26(24(19-22)31(32,33)34)45(41,42)37-30(2,3)4/h11-16,19-20,37H,5-10,17-18H2,1-4H3,(H,35,36,38)	VTFSLOIXAMJGJE-UHFFFAOYSA-N	392241	US10301272, Example 200/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392241	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392241&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188653	404960576							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784043	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NS(C)(=O)=O)nc1CC1CCCCC1	InChI=1S/C22H30F3N3O4S3/c1-21(2,3)28-35(31,32)18-11-10-15(13-16(18)22(23,24)25)19-17(12-14-8-6-5-7-9-14)26-20(33-19)27-34(4,29)30/h10-11,13-14,28H,5-9,12H2,1-4H3,(H,26,27)	DLYKMFKSSDEKNW-UHFFFAOYSA-N	392242	US10301272, Example 201	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392242&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160529	404960577							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784044	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NS(C)(=O)=O)nc1CC1CCCCC1	InChI=1S/C22H30F3N3O4S3/c1-21(2,3)28-35(31,32)18-11-10-15(13-16(18)22(23,24)25)19-17(12-14-8-6-5-7-9-14)26-20(33-19)27-34(4,29)30/h10-11,13-14,28H,5-9,12H2,1-4H3,(H,26,27)	DLYKMFKSSDEKNW-UHFFFAOYSA-N	392242	US10301272, Example 201	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392242&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160529	404960577							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784045	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(NS(C)(=O)=O)nc1CC1CCCCC1	InChI=1S/C22H30F3N3O4S3/c1-21(2,3)28-35(31,32)18-11-10-15(13-16(18)22(23,24)25)19-17(12-14-8-6-5-7-9-14)26-20(33-19)27-34(4,29)30/h10-11,13-14,28H,5-9,12H2,1-4H3,(H,26,27)	DLYKMFKSSDEKNW-UHFFFAOYSA-N	392242	US10301272, Example 201	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392242	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392242&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160529	404960577							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784046	CCOC(=O)c1nc(Cc2ccccc2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H28N2O4S2/c1-5-33-26(30)25-28-22(17-18-11-7-6-8-12-18)24(34-25)21-15-16-23(20-14-10-9-13-19(20)21)35(31,32)29-27(2,3)4/h6-16,29H,5,17H2,1-4H3	RLSGORMTMHWNMN-UHFFFAOYSA-N	392243	US10301272, Example 202	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392243	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392243&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032525	404960578							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784047	CCOC(=O)c1nc(Cc2ccccc2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H28N2O4S2/c1-5-33-26(30)25-28-22(17-18-11-7-6-8-12-18)24(34-25)21-15-16-23(20-14-10-9-13-19(20)21)35(31,32)29-27(2,3)4/h6-16,29H,5,17H2,1-4H3	RLSGORMTMHWNMN-UHFFFAOYSA-N	392243	US10301272, Example 202	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392243	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392243&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032525	404960578							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784048	CCOC(=O)c1nc(Cc2ccccc2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H28N2O4S2/c1-5-33-26(30)25-28-22(17-18-11-7-6-8-12-18)24(34-25)21-15-16-23(20-14-10-9-13-19(20)21)35(31,32)29-27(2,3)4/h6-16,29H,5,17H2,1-4H3	RLSGORMTMHWNMN-UHFFFAOYSA-N	392243	US10301272, Example 202	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392243	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392243&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90032525	404960578							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784049	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)[K]O)c2ccccc12	InChI=1S/C25H23N2O3S2.K.H2O/c1-25(2,3)27-32(29,30)22-14-13-20(18-11-7-8-12-19(18)22)24-21(26-23(16-28)31-24)15-17-9-5-4-6-10-17;;/h4-14,27H,15H2,1-3H3;;1H2/q;+1;/p-1	GCVONDIHWVANNJ-UHFFFAOYSA-M	392244	US10301272, Example 203	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392244&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			140677708	404960579							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784050	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)[K]O)c2ccccc12	InChI=1S/C25H23N2O3S2.K.H2O/c1-25(2,3)27-32(29,30)22-14-13-20(18-11-7-8-12-19(18)22)24-21(26-23(16-28)31-24)15-17-9-5-4-6-10-17;;/h4-14,27H,15H2,1-3H3;;1H2/q;+1;/p-1	GCVONDIHWVANNJ-UHFFFAOYSA-M	392244	US10301272, Example 203	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392244&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			140677708	404960579							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784051	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)[K]O)c2ccccc12	InChI=1S/C25H23N2O3S2.K.H2O/c1-25(2,3)27-32(29,30)22-14-13-20(18-11-7-8-12-19(18)22)24-21(26-23(16-28)31-24)15-17-9-5-4-6-10-17;;/h4-14,27H,15H2,1-3H3;;1H2/q;+1;/p-1	GCVONDIHWVANNJ-UHFFFAOYSA-M	392244	US10301272, Example 203	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392244	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392244&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			140677708	404960579							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784052	CCS(=O)(=O)c1ccc(CNC(=O)c2nc(Cc3ccccc3)c(s2)-c2ccc(c3ccccc23)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C34H35N3O5S3/c1-5-44(39,40)25-17-15-24(16-18-25)22-35-32(38)33-36-29(21-23-11-7-6-8-12-23)31(43-33)28-19-20-30(27-14-10-9-13-26(27)28)45(41,42)37-34(2,3)4/h6-20,37H,5,21-22H2,1-4H3,(H,35,38)	AGCBROBSAQQXAU-UHFFFAOYSA-N	392245	US10301272, Example 205	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160572	404960580							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784053	CCS(=O)(=O)c1ccc(CNC(=O)c2nc(Cc3ccccc3)c(s2)-c2ccc(c3ccccc23)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C34H35N3O5S3/c1-5-44(39,40)25-17-15-24(16-18-25)22-35-32(38)33-36-29(21-23-11-7-6-8-12-23)31(43-33)28-19-20-30(27-14-10-9-13-26(27)28)45(41,42)37-34(2,3)4/h6-20,37H,5,21-22H2,1-4H3,(H,35,38)	AGCBROBSAQQXAU-UHFFFAOYSA-N	392245	US10301272, Example 205	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160572	404960580							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784054	CCS(=O)(=O)c1ccc(CNC(=O)c2nc(Cc3ccccc3)c(s2)-c2ccc(c3ccccc23)S(=O)(=O)NC(C)(C)C)cc1	InChI=1S/C34H35N3O5S3/c1-5-44(39,40)25-17-15-24(16-18-25)22-35-32(38)33-36-29(21-23-11-7-6-8-12-23)31(43-33)28-19-20-30(27-14-10-9-13-26(27)28)45(41,42)37-34(2,3)4/h6-20,37H,5,21-22H2,1-4H3,(H,35,38)	AGCBROBSAQQXAU-UHFFFAOYSA-N	392245	US10301272, Example 205	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392245	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392245&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160572	404960580							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784055	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(N)=O	InChI=1S/C26H37N3O/c1-25(2,3)20-13-18(14-21(15-20)26(4,5)6)22-19(12-17-10-8-7-9-11-17)16-28-24(29-22)23(27)30/h13-17H,7-12H2,1-6H3,(H2,27,30)	GVPBUUPFFNYXIF-UHFFFAOYSA-N	392246	US10301272, Example 206	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160542	404960581							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784056	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(N)=O	InChI=1S/C26H37N3O/c1-25(2,3)20-13-18(14-21(15-20)26(4,5)6)22-19(12-17-10-8-7-9-11-17)16-28-24(29-22)23(27)30/h13-17H,7-12H2,1-6H3,(H2,27,30)	GVPBUUPFFNYXIF-UHFFFAOYSA-N	392246	US10301272, Example 206	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160542	404960581							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784057	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(N)=O	InChI=1S/C26H37N3O/c1-25(2,3)20-13-18(14-21(15-20)26(4,5)6)22-19(12-17-10-8-7-9-11-17)16-28-24(29-22)23(27)30/h13-17H,7-12H2,1-6H3,(H2,27,30)	GVPBUUPFFNYXIF-UHFFFAOYSA-N	392246	US10301272, Example 206	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392246&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160542	404960581							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784058	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(=O)NC1COC1	InChI=1S/C29H41N3O2/c1-28(2,3)22-13-20(14-23(15-22)29(4,5)6)25-21(12-19-10-8-7-9-11-19)16-30-26(32-25)27(33)31-24-17-34-18-24/h13-16,19,24H,7-12,17-18H2,1-6H3,(H,31,33)	QXHSLMIJUMDGNK-UHFFFAOYSA-N	392247	US10301272, Example 207	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3981							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90033991	404960582							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784059	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(=O)NC1COC1	InChI=1S/C29H41N3O2/c1-28(2,3)22-13-20(14-23(15-22)29(4,5)6)25-21(12-19-10-8-7-9-11-19)16-30-26(32-25)27(33)31-24-17-34-18-24/h13-16,19,24H,7-12,17-18H2,1-6H3,(H,31,33)	QXHSLMIJUMDGNK-UHFFFAOYSA-N	392247	US10301272, Example 207	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90033991	404960582							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784060	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(ncc1CC1CCCCC1)C(=O)NC1COC1	InChI=1S/C29H41N3O2/c1-28(2,3)22-13-20(14-23(15-22)29(4,5)6)25-21(12-19-10-8-7-9-11-19)16-30-26(32-25)27(33)31-24-17-34-18-24/h13-16,19,24H,7-12,17-18H2,1-6H3,(H,31,33)	QXHSLMIJUMDGNK-UHFFFAOYSA-N	392247	US10301272, Example 207	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392247	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392247&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			90033991	404960582							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784061	CC(C)(O)CNC(=O)c1ncc(CC2CCCCC2)c(n1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C30H45N3O2/c1-28(2,3)23-15-21(16-24(17-23)29(4,5)6)25-22(14-20-12-10-9-11-13-20)18-31-26(33-25)27(34)32-19-30(7,8)35/h15-18,20,35H,9-14,19H2,1-8H3,(H,32,34)	QUGMPTGCIARJIX-UHFFFAOYSA-N	392248	US10301272, Example 207/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392248&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186098	404960583							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784062	CC(C)(O)CNC(=O)c1ncc(CC2CCCCC2)c(n1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C30H45N3O2/c1-28(2,3)23-15-21(16-24(17-23)29(4,5)6)25-22(14-20-12-10-9-11-13-20)18-31-26(33-25)27(34)32-19-30(7,8)35/h15-18,20,35H,9-14,19H2,1-8H3,(H,32,34)	QUGMPTGCIARJIX-UHFFFAOYSA-N	392248	US10301272, Example 207/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392248&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186098	404960583							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784063	CC(C)(O)CNC(=O)c1ncc(CC2CCCCC2)c(n1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C30H45N3O2/c1-28(2,3)23-15-21(16-24(17-23)29(4,5)6)25-22(14-20-12-10-9-11-13-20)18-31-26(33-25)27(34)32-19-30(7,8)35/h15-18,20,35H,9-14,19H2,1-8H3,(H,32,34)	QUGMPTGCIARJIX-UHFFFAOYSA-N	392248	US10301272, Example 207/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392248	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392248&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186098	404960583							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784064	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1cc(ccc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-15-22(16-24(18-23)28(4,5)6)25-17-21(26(29)30)13-12-20(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	PAYMOZXHLCTNFH-UHFFFAOYSA-N	392249	US10301272, Example 208	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160503	404960584							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784065	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1cc(ccc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-15-22(16-24(18-23)28(4,5)6)25-17-21(26(29)30)13-12-20(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	PAYMOZXHLCTNFH-UHFFFAOYSA-N	392249	US10301272, Example 208	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160503	404960584							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784066	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1cc(ccc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-15-22(16-24(18-23)28(4,5)6)25-17-21(26(29)30)13-12-20(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	PAYMOZXHLCTNFH-UHFFFAOYSA-N	392249	US10301272, Example 208	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392249	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392249&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160503	404960584							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784067	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1ccc(cc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-16-22(17-24(18-23)28(4,5)6)25-13-12-20(26(29)30)15-21(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	AZLNWIQPBIQUJP-UHFFFAOYSA-N	392250	US10301272, Example 209	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392250&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186107	404960585							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784068	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1ccc(cc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-16-22(17-24(18-23)28(4,5)6)25-13-12-20(26(29)30)15-21(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	AZLNWIQPBIQUJP-UHFFFAOYSA-N	392250	US10301272, Example 209	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392250&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186107	404960585							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784069	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1ccc(cc1CC1CCCCC1)C(N)=O	InChI=1S/C28H39NO/c1-27(2,3)23-16-22(17-24(18-23)28(4,5)6)25-13-12-20(26(29)30)15-21(25)14-19-10-8-7-9-11-19/h12-13,15-19H,7-11,14H2,1-6H3,(H2,29,30)	AZLNWIQPBIQUJP-UHFFFAOYSA-N	392250	US10301272, Example 209	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392250	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392250&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186107	404960585							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784070	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Cc3ccccc3)s2)-c2ccccc2)cc1	InChI=1S/C26H24N2O3S2/c1-2-33(30,31)22-15-13-20(14-16-22)18-24(29)27-26-28-25(21-11-7-4-8-12-21)23(32-26)17-19-9-5-3-6-10-19/h3-16H,2,17-18H2,1H3,(H,27,28,29)	UVPYBRXTAWOMSZ-UHFFFAOYSA-N	50445901	CHEMBL3105804::US10301272, Example 211	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50445901	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50445901&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			60142607	194943797		CHEMBL3105804					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784071	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Cc3ccccc3)s2)-c2ccccc2)cc1	InChI=1S/C26H24N2O3S2/c1-2-33(30,31)22-15-13-20(14-16-22)18-24(29)27-26-28-25(21-11-7-4-8-12-21)23(32-26)17-19-9-5-3-6-10-19/h3-16H,2,17-18H2,1H3,(H,27,28,29)	UVPYBRXTAWOMSZ-UHFFFAOYSA-N	50445901	CHEMBL3105804::US10301272, Example 211	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50445901	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50445901&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			60142607	194943797		CHEMBL3105804					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784072	CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Cc3ccccc3)s2)-c2ccccc2)cc1	InChI=1S/C26H24N2O3S2/c1-2-33(30,31)22-15-13-20(14-16-22)18-24(29)27-26-28-25(21-11-7-4-8-12-21)23(32-26)17-19-9-5-3-6-10-19/h3-16H,2,17-18H2,1H3,(H,27,28,29)	UVPYBRXTAWOMSZ-UHFFFAOYSA-N	50445901	CHEMBL3105804::US10301272, Example 211	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50445901	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50445901&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			60142607	194943797		CHEMBL3105804					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784073	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H33N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h4-14,21,33H,15-19H2,1-3H3,(H,31,34)	XKPQMCNZIDADTA-UHFFFAOYSA-N	392252	US10301272, Example 300	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160539	404960587							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784074	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H33N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h4-14,21,33H,15-19H2,1-3H3,(H,31,34)	XKPQMCNZIDADTA-UHFFFAOYSA-N	392252	US10301272, Example 300	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160539	404960587							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784075	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H33N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h4-14,21,33H,15-19H2,1-3H3,(H,31,34)	XKPQMCNZIDADTA-UHFFFAOYSA-N	392252	US10301272, Example 300	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392252	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392252&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160539	404960587							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784076	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H31N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h4-14,20,32H,15-18H2,1-3H3,(H,30,33)	DETYWGPTPVJTNT-UHFFFAOYSA-N	392253	US10301272, Example 300/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392253&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186095	404960588							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784077	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H31N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h4-14,20,32H,15-18H2,1-3H3,(H,30,33)	DETYWGPTPVJTNT-UHFFFAOYSA-N	392253	US10301272, Example 300/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392253&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186095	404960588							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784078	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2ccccc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H31N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h4-14,20,32H,15-18H2,1-3H3,(H,30,33)	DETYWGPTPVJTNT-UHFFFAOYSA-N	392253	US10301272, Example 300/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392253	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392253&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186095	404960588							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784079	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h7-8,11-14,19-20,32H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ILZXOVNBYVRZHF-UHFFFAOYSA-N	392254	US10301272, Example 300/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392254&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186100	404960589							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784080	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h7-8,11-14,19-20,32H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ILZXOVNBYVRZHF-UHFFFAOYSA-N	392254	US10301272, Example 300/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392254&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186100	404960589							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784081	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)32-40(36,37)24-14-13-23(21-11-7-8-12-22(21)24)26-25(19-9-5-4-6-10-19)31-28(38-26)27(33)30-20-15-17-39(34,35)18-16-20/h7-8,11-14,19-20,32H,4-6,9-10,15-18H2,1-3H3,(H,30,33)	ILZXOVNBYVRZHF-UHFFFAOYSA-N	392254	US10301272, Example 300/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392254&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186100	404960589							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784082	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C24H31N3O4S2/c1-7-18-20(32-22(26-18)21(28)25-14-24(5,6)29)17-12-13-19(16-11-9-8-10-15(16)17)33(30,31)27-23(2,3)4/h8-13,27,29H,7,14H2,1-6H3,(H,25,28)	HWBLOLKHNRAMBW-UHFFFAOYSA-N	392255	US10301272, Example 300/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392255&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186097	404960590							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784083	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C24H31N3O4S2/c1-7-18-20(32-22(26-18)21(28)25-14-24(5,6)29)17-12-13-19(16-11-9-8-10-15(16)17)33(30,31)27-23(2,3)4/h8-13,27,29H,7,14H2,1-6H3,(H,25,28)	HWBLOLKHNRAMBW-UHFFFAOYSA-N	392255	US10301272, Example 300/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392255&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186097	404960590							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784084	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C24H31N3O4S2/c1-7-18-20(32-22(26-18)21(28)25-14-24(5,6)29)17-12-13-19(16-11-9-8-10-15(16)17)33(30,31)27-23(2,3)4/h8-13,27,29H,7,14H2,1-6H3,(H,25,28)	HWBLOLKHNRAMBW-UHFFFAOYSA-N	392255	US10301272, Example 300/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392255&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186097	404960590							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784085	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)C1CC2(C1)CCOCC2	InChI=1S/C28H34N2O4S2/c1-5-22-25(35-26(29-22)24(31)18-16-28(17-18)12-14-34-15-13-28)21-10-11-23(20-9-7-6-8-19(20)21)36(32,33)30-27(2,3)4/h6-11,18,30H,5,12-17H2,1-4H3	DIKOYTMOYSHXTF-UHFFFAOYSA-N	392256	US10301272, Example 300/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392256&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186109	404960591							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784086	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)C1CC2(C1)CCOCC2	InChI=1S/C28H34N2O4S2/c1-5-22-25(35-26(29-22)24(31)18-16-28(17-18)12-14-34-15-13-28)21-10-11-23(20-9-7-6-8-19(20)21)36(32,33)30-27(2,3)4/h6-11,18,30H,5,12-17H2,1-4H3	DIKOYTMOYSHXTF-UHFFFAOYSA-N	392256	US10301272, Example 300/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392256&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186109	404960591							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784087	CCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)C1CC2(C1)CCOCC2	InChI=1S/C28H34N2O4S2/c1-5-22-25(35-26(29-22)24(31)18-16-28(17-18)12-14-34-15-13-28)21-10-11-23(20-9-7-6-8-19(20)21)36(32,33)30-27(2,3)4/h6-11,18,30H,5,12-17H2,1-4H3	DIKOYTMOYSHXTF-UHFFFAOYSA-N	392256	US10301272, Example 300/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392256	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392256&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186109	404960591							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784088	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C22H29Cl2N3O5S3/c1-5-6-15-19(33-21(26-15)20(28)25-13-9-11-34(29,30)12-10-13)14-7-8-16(18(24)17(14)23)35(31,32)27-22(2,3)4/h7-8,13,27H,5-6,9-12H2,1-4H3,(H,25,28)	DGOHUEQPKSFGKK-UHFFFAOYSA-N	392257	US10301272, Example 300/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392257&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188764	404960592							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784089	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C22H29Cl2N3O5S3/c1-5-6-15-19(33-21(26-15)20(28)25-13-9-11-34(29,30)12-10-13)14-7-8-16(18(24)17(14)23)35(31,32)27-22(2,3)4/h7-8,13,27H,5-6,9-12H2,1-4H3,(H,25,28)	DGOHUEQPKSFGKK-UHFFFAOYSA-N	392257	US10301272, Example 300/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392257&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188764	404960592							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784090	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C22H29Cl2N3O5S3/c1-5-6-15-19(33-21(26-15)20(28)25-13-9-11-34(29,30)12-10-13)14-7-8-16(18(24)17(14)23)35(31,32)27-22(2,3)4/h7-8,13,27H,5-6,9-12H2,1-4H3,(H,25,28)	DGOHUEQPKSFGKK-UHFFFAOYSA-N	392257	US10301272, Example 300/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392257	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392257&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188764	404960592							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784091	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCC1	InChI=1S/C21H27Cl2N3O3S2/c1-5-7-14-18(30-20(25-14)19(27)24-12-8-6-9-12)13-10-11-15(17(23)16(13)22)31(28,29)26-21(2,3)4/h10-12,26H,5-9H2,1-4H3,(H,24,27)	YKQJONURSRTREZ-UHFFFAOYSA-N	392258	US10301272, Example 300/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392258&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186102	404960593							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784092	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCC1	InChI=1S/C21H27Cl2N3O3S2/c1-5-7-14-18(30-20(25-14)19(27)24-12-8-6-9-12)13-10-11-15(17(23)16(13)22)31(28,29)26-21(2,3)4/h10-12,26H,5-9H2,1-4H3,(H,24,27)	YKQJONURSRTREZ-UHFFFAOYSA-N	392258	US10301272, Example 300/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392258&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186102	404960593							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784093	CCCc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCC1	InChI=1S/C21H27Cl2N3O3S2/c1-5-7-14-18(30-20(25-14)19(27)24-12-8-6-9-12)13-10-11-15(17(23)16(13)22)31(28,29)26-21(2,3)4/h10-12,26H,5-9H2,1-4H3,(H,24,27)	YKQJONURSRTREZ-UHFFFAOYSA-N	392258	US10301272, Example 300/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392258	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392258&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186102	404960593							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784094	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C26H33N3O5S3/c1-5-8-21-23(35-25(28-21)24(30)27-17-13-15-36(31,32)16-14-17)20-11-12-22(19-10-7-6-9-18(19)20)37(33,34)29-26(2,3)4/h6-7,9-12,17,29H,5,8,13-16H2,1-4H3,(H,27,30)	GSSDRQRJWHEBTC-UHFFFAOYSA-N	392259	US10301272, Example 300/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392259	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392259&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188724	404960594							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784095	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C26H33N3O5S3/c1-5-8-21-23(35-25(28-21)24(30)27-17-13-15-36(31,32)16-14-17)20-11-12-22(19-10-7-6-9-18(19)20)37(33,34)29-26(2,3)4/h6-7,9-12,17,29H,5,8,13-16H2,1-4H3,(H,27,30)	GSSDRQRJWHEBTC-UHFFFAOYSA-N	392259	US10301272, Example 300/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392259	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392259&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188724	404960594							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784096	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCC1	InChI=1S/C25H31N3O3S2/c1-5-9-20-22(32-24(27-20)23(29)26-16-10-8-11-16)19-14-15-21(18-13-7-6-12-17(18)19)33(30,31)28-25(2,3)4/h6-7,12-16,28H,5,8-11H2,1-4H3,(H,26,29)	MQBWCNWSQNRWGO-UHFFFAOYSA-N	392260	US10301272, Example 300/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392260	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392260&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186096	404960595							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784097	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CCC1	InChI=1S/C25H31N3O3S2/c1-5-9-20-22(32-24(27-20)23(29)26-16-10-8-11-16)19-14-15-21(18-13-7-6-12-17(18)19)33(30,31)28-25(2,3)4/h6-7,12-16,28H,5,8-11H2,1-4H3,(H,26,29)	MQBWCNWSQNRWGO-UHFFFAOYSA-N	392260	US10301272, Example 300/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392260	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392260&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186096	404960595							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784098	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O	InChI=1S/C24H28F3N3O4S2/c1-5-8-18-20(35-22(29-18)21(31)28-13-23(3,4)32)17-11-12-19(16-10-7-6-9-15(16)17)36(33,34)30-14(2)24(25,26)27/h6-7,9-12,14,30,32H,5,8,13H2,1-4H3,(H,28,31)/t14-/m0/s1	YWSPNIWVCRSPOD-AWEZNQCLSA-N	392261	US10301272, Example 300/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392261	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392261&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186104	404960596							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784099	CCCc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O	InChI=1S/C24H28F3N3O4S2/c1-5-8-18-20(35-22(29-18)21(31)28-13-23(3,4)32)17-11-12-19(16-10-7-6-9-15(16)17)36(33,34)30-14(2)24(25,26)27/h6-7,9-12,14,30,32H,5,8,13H2,1-4H3,(H,28,31)/t14-/m0/s1	YWSPNIWVCRSPOD-AWEZNQCLSA-N	392261	US10301272, Example 300/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392261	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392261&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186104	404960596							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784100	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C27H33N3O5S3/c1-27(2,3)30-38(34,35)22-12-11-21(19-9-4-5-10-20(19)22)24-23(17-7-6-8-17)29-26(36-24)25(31)28-18-13-15-37(32,33)16-14-18/h4-5,9-12,17-18,30H,6-8,13-16H2,1-3H3,(H,28,31)	LOPHBQFJYIAKCA-UHFFFAOYSA-N	392262	US10301272, Example 300/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392262&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188669	404960597							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784101	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C27H33N3O5S3/c1-27(2,3)30-38(34,35)22-12-11-21(19-9-4-5-10-20(19)22)24-23(17-7-6-8-17)29-26(36-24)25(31)28-18-13-15-37(32,33)16-14-18/h4-5,9-12,17-18,30H,6-8,13-16H2,1-3H3,(H,28,31)	LOPHBQFJYIAKCA-UHFFFAOYSA-N	392262	US10301272, Example 300/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392262&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188669	404960597							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784102	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(C)(C)C)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C27H35N3O5S3/c1-26(2,3)23-22(36-25(29-23)24(31)28-17-13-15-37(32,33)16-14-17)20-11-12-21(19-10-8-7-9-18(19)20)38(34,35)30-27(4,5)6/h7-12,17,30H,13-16H2,1-6H3,(H,28,31)	IENUAHONTOGODN-UHFFFAOYSA-N	392263	US10301272, Example 300/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392263	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392263&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188765	404960598							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784103	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(C)(C)C)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C27H35N3O5S3/c1-26(2,3)23-22(36-25(29-23)24(31)28-17-13-15-37(32,33)16-14-17)20-11-12-21(19-10-8-7-9-18(19)20)38(34,35)30-27(4,5)6/h7-12,17,30H,13-16H2,1-6H3,(H,28,31)	IENUAHONTOGODN-UHFFFAOYSA-N	392263	US10301272, Example 300/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392263	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392263&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188765	404960598							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784104	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccnc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H30N4O5S3/c1-28(2,3)32-40(36,37)23-11-10-22(20-8-4-5-9-21(20)23)25-24(18-7-6-14-29-17-18)31-27(38-25)26(33)30-19-12-15-39(34,35)16-13-19/h4-11,14,17,19,32H,12-13,15-16H2,1-3H3,(H,30,33)	FLFOORNMPCJMKQ-UHFFFAOYSA-N	392264	US10301272, Example 300/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392264	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392264&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188671	404960599							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784105	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccnc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C28H30N4O5S3/c1-28(2,3)32-40(36,37)23-11-10-22(20-8-4-5-9-21(20)23)25-24(18-7-6-14-29-17-18)31-27(38-25)26(33)30-19-12-15-39(34,35)16-13-19/h4-11,14,17,19,32H,12-13,15-16H2,1-3H3,(H,30,33)	FLFOORNMPCJMKQ-UHFFFAOYSA-N	392264	US10301272, Example 300/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392264	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392264&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188671	404960599							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784106	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2cccnc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H32N4O5S3/c1-29(2,3)33-41(37,38)25-11-10-23(21-8-4-5-9-22(21)25)26-24(17-19-7-6-14-30-18-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h4-11,14,18,20,33H,12-13,15-17H2,1-3H3,(H,31,34)	FKKJUOPEGQBKQM-UHFFFAOYSA-N	392265	US10301272, Example 300/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392265	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392265&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188747	404960600							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784107	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2cccnc2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H32N4O5S3/c1-29(2,3)33-41(37,38)25-11-10-23(21-8-4-5-9-22(21)25)26-24(17-19-7-6-14-30-18-19)32-28(39-26)27(34)31-20-12-15-40(35,36)16-13-20/h4-11,14,18,20,33H,12-13,15-17H2,1-3H3,(H,31,34)	FKKJUOPEGQBKQM-UHFFFAOYSA-N	392265	US10301272, Example 300/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392265	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392265&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188747	404960600							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784108	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(Cl)c2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H30ClN3O5S3/c1-29(2,3)33-41(37,38)24-12-11-23(21-9-4-5-10-22(21)24)26-25(18-7-6-8-19(30)17-18)32-28(39-26)27(34)31-20-13-15-40(35,36)16-14-20/h4-12,17,20,33H,13-16H2,1-3H3,(H,31,34)	JDIMOLKKJSCMPY-UHFFFAOYSA-N	392266	US10301272, Example 300/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392266	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392266&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188726	404960601							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784109	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(Cl)c2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H30ClN3O5S3/c1-29(2,3)33-41(37,38)24-12-11-23(21-9-4-5-10-22(21)24)26-25(18-7-6-8-19(30)17-18)32-28(39-26)27(34)31-20-13-15-40(35,36)16-14-20/h4-12,17,20,33H,13-16H2,1-3H3,(H,31,34)	JDIMOLKKJSCMPY-UHFFFAOYSA-N	392266	US10301272, Example 300/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392266	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392266&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188726	404960601							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784110	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(c2)C#N)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H30N4O5S3/c1-30(2,3)34-42(38,39)25-12-11-24(22-9-4-5-10-23(22)25)27-26(20-8-6-7-19(17-20)18-31)33-29(40-27)28(35)32-21-13-15-41(36,37)16-14-21/h4-12,17,21,34H,13-16H2,1-3H3,(H,32,35)	OPOQHMDDAOUFAE-UHFFFAOYSA-N	392267	US10301272, Example 300/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392267	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392267&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188725	404960602							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784111	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(c2)C#N)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H30N4O5S3/c1-30(2,3)34-42(38,39)25-12-11-24(22-9-4-5-10-23(22)25)27-26(20-8-6-7-19(17-20)18-31)33-29(40-27)28(35)32-21-13-15-41(36,37)16-14-21/h4-12,17,21,34H,13-16H2,1-3H3,(H,32,35)	OPOQHMDDAOUFAE-UHFFFAOYSA-N	392267	US10301272, Example 300/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392267	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392267&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188725	404960602							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784112	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(c2)C(N)=O)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H32N4O6S3/c1-30(2,3)34-43(39,40)24-12-11-23(21-9-4-5-10-22(21)24)26-25(18-7-6-8-19(17-18)27(31)35)33-29(41-26)28(36)32-20-13-15-42(37,38)16-14-20/h4-12,17,20,34H,13-16H2,1-3H3,(H2,31,35)(H,32,36)	CZFUHBGSLLJYRT-UHFFFAOYSA-N	392268	US10301272, Example 300/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392268&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188757	404960603							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784113	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(c2)C(N)=O)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H32N4O6S3/c1-30(2,3)34-43(39,40)24-12-11-23(21-9-4-5-10-22(21)24)26-25(18-7-6-8-19(17-18)27(31)35)33-29(41-26)28(36)32-20-13-15-42(37,38)16-14-20/h4-12,17,20,34H,13-16H2,1-3H3,(H2,31,35)(H,32,36)	CZFUHBGSLLJYRT-UHFFFAOYSA-N	392268	US10301272, Example 300/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392268	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392268&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188757	404960603							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784114	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C29H35N3O5S2/c1-29(2,3)32-39(36,37)23-14-13-22(20-11-7-8-12-21(20)23)25-24(17-9-5-4-6-10-17)31-27(38-25)26(33)30-19-15-18(16-19)28(34)35/h7-8,11-14,17-19,32H,4-6,9-10,15-16H2,1-3H3,(H,30,33)(H,34,35)/t18-,19-	JWWRMAZPNWAWCD-WGSAOQKQSA-N	392269	US10301272, Example 300/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392269	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392269&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186116	404960604							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784115	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C29H35N3O5S2/c1-29(2,3)32-39(36,37)23-14-13-22(20-11-7-8-12-21(20)23)25-24(17-9-5-4-6-10-17)31-27(38-25)26(33)30-19-15-18(16-19)28(34)35/h7-8,11-14,17-19,32H,4-6,9-10,15-16H2,1-3H3,(H,30,33)(H,34,35)/t18-,19-	JWWRMAZPNWAWCD-WGSAOQKQSA-N	392269	US10301272, Example 300/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392269	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392269&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186116	404960604							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784116	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccccc2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C30H31N3O5S2/c1-30(2,3)33-40(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-18-9-5-4-6-10-18)32-28(39-26)27(34)31-20-16-19(17-20)29(35)36/h4-14,19-20,33H,15-17H2,1-3H3,(H,31,34)(H,35,36)/t19-,20-	IGJQQPRGHASVRR-MXVIHJGJSA-N	392270	US10301272, Example 300/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 26.5							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392270	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392270&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186117	404960605							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784117	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1C	InChI=1S/C28H39ClN4O6S3/c1-6-28(4,5)32-42(38,39)21-8-7-20(22(29)18(21)3)24-23(27(35)33-13-9-17(2)10-14-33)31-26(40-24)25(34)30-19-11-15-41(36,37)16-12-19/h7-8,17,19,32H,6,9-16H2,1-5H3,(H,30,34)	UCPALKGPOKCWLE-UHFFFAOYSA-N	392271	US10301272, Example 301	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392271&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160595	404960606							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784118	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1C	InChI=1S/C28H39ClN4O6S3/c1-6-28(4,5)32-42(38,39)21-8-7-20(22(29)18(21)3)24-23(27(35)33-13-9-17(2)10-14-33)31-26(40-24)25(34)30-19-11-15-41(36,37)16-12-19/h7-8,17,19,32H,6,9-16H2,1-5H3,(H,30,34)	UCPALKGPOKCWLE-UHFFFAOYSA-N	392271	US10301272, Example 301	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392271	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392271&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160595	404960606							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784119	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c(Cl)c1C	InChI=1S/C27H39ClN4O5S2/c1-8-26(4,5)31-39(36,37)19-10-9-18(20(28)17(19)3)22-21(25(34)32-13-11-16(2)12-14-32)30-24(38-22)23(33)29-15-27(6,7)35/h9-10,16,31,35H,8,11-15H2,1-7H3,(H,29,33)	WKVRCVRKDBCOON-UHFFFAOYSA-N	392272	US10301272, Example 301/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392272	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392272&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186118	404960607							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784120	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c(Cl)c1C	InChI=1S/C27H39ClN4O5S2/c1-8-26(4,5)31-39(36,37)19-10-9-18(20(28)17(19)3)22-21(25(34)32-13-11-16(2)12-14-32)30-24(38-22)23(33)29-15-27(6,7)35/h9-10,16,31,35H,8,11-15H2,1-7H3,(H,29,33)	WKVRCVRKDBCOON-UHFFFAOYSA-N	392272	US10301272, Example 301/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392272	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392272&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186118	404960607							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784121	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1C	InChI=1S/C28H37ClN4O6S3/c1-6-27(4,5)31-42(38,39)20-8-7-19(21(29)18(20)3)23-22(25(34)32-11-9-17(2)10-12-32)30-24(40-23)26(35)33-13-28(14-33)15-41(36,37)16-28/h7-8,17,31H,6,9-16H2,1-5H3	NTWYLJGBBBYBND-UHFFFAOYSA-N	392273	US10301272, Example 301/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392273	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392273&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186111	404960608							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784122	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1C	InChI=1S/C28H37ClN4O6S3/c1-6-27(4,5)31-42(38,39)20-8-7-19(21(29)18(20)3)23-22(25(34)32-11-9-17(2)10-12-32)30-24(40-23)26(35)33-13-28(14-33)15-41(36,37)16-28/h7-8,17,31H,6,9-16H2,1-5H3	NTWYLJGBBBYBND-UHFFFAOYSA-N	392273	US10301272, Example 301/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392273	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392273&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186111	404960608							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784123	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C	InChI=1S/C28H37ClN4O6S2/c1-6-28(4,5)32-41(38,39)20-8-7-19(21(29)16(20)3)23-22(26(35)33-11-9-15(2)10-12-33)31-25(40-23)24(34)30-18-13-17(14-18)27(36)37/h7-8,15,17-18,32H,6,9-14H2,1-5H3,(H,30,34)(H,36,37)/t17-,18-	NWZDNDKJZPVCCD-IYARVYRRSA-N	392274	US10301272, Example 302	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392274	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392274&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160571	404960609							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784124	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C	InChI=1S/C28H37ClN4O6S2/c1-6-28(4,5)32-41(38,39)20-8-7-19(21(29)16(20)3)23-22(26(35)33-11-9-15(2)10-12-33)31-25(40-23)24(34)30-18-13-17(14-18)27(36)37/h7-8,15,17-18,32H,6,9-14H2,1-5H3,(H,30,34)(H,36,37)/t17-,18-	NWZDNDKJZPVCCD-IYARVYRRSA-N	392274	US10301272, Example 302	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392274	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392274&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160571	404960609							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784125	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCc2ncc(s2)S(C)(=O)=O)c(Cl)c1C	InChI=1S/C28H36ClN5O6S4/c1-7-28(4,5)33-44(39,40)19-9-8-18(22(29)17(19)3)24-23(27(36)34-12-10-16(2)11-13-34)32-26(42-24)25(35)31-14-20-30-15-21(41-20)43(6,37)38/h8-9,15-16,33H,7,10-14H2,1-6H3,(H,31,35)	SAPDWPVKAOFUCN-UHFFFAOYSA-N	392275	US10301272, Example 303	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392275&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160519	404960610							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784126	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCc2ncc(s2)S(C)(=O)=O)c(Cl)c1C	InChI=1S/C28H36ClN5O6S4/c1-7-28(4,5)33-44(39,40)19-9-8-18(22(29)17(19)3)24-23(27(36)34-12-10-16(2)11-13-34)32-26(42-24)25(35)31-14-20-30-15-21(41-20)43(6,37)38/h8-9,15-16,33H,7,10-14H2,1-6H3,(H,31,35)	SAPDWPVKAOFUCN-UHFFFAOYSA-N	392275	US10301272, Example 303	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392275&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160519	404960610							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784127	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H36N4O5S2/c1-27(2,3)31-39(36,37)21-14-13-20(18-11-7-8-12-19(18)21)23-22(26(34)32-15-9-6-10-16-32)30-25(38-23)24(33)29-17-28(4,5)35/h7-8,11-14,31,35H,6,9-10,15-17H2,1-5H3,(H,29,33)	GMZHFKXXDABZPQ-UHFFFAOYSA-N	392276	US10301272, Example 304	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392276&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160505	404960611							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784128	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H36N4O5S2/c1-27(2,3)31-39(36,37)21-14-13-20(18-11-7-8-12-19(18)21)23-22(26(34)32-15-9-6-10-16-32)30-25(38-23)24(33)29-17-28(4,5)35/h7-8,11-14,31,35H,6,9-10,15-17H2,1-5H3,(H,29,33)	GMZHFKXXDABZPQ-UHFFFAOYSA-N	392276	US10301272, Example 304	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392276&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160505	404960611							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784129	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C28H36N4O5S2/c1-27(2,3)31-39(36,37)21-14-13-20(18-11-7-8-12-19(18)21)23-22(26(34)32-15-9-6-10-16-32)30-25(38-23)24(33)29-17-28(4,5)35/h7-8,11-14,31,35H,6,9-10,15-17H2,1-5H3,(H,29,33)	GMZHFKXXDABZPQ-UHFFFAOYSA-N	392276	US10301272, Example 304	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392276&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160505	404960611							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784130	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)NC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H38N4O5S2/c1-28(2,3)33-40(37,38)22-16-15-21(19-13-9-10-14-20(19)22)24-23(25(34)31-18-11-7-6-8-12-18)32-27(39-24)26(35)30-17-29(4,5)36/h9-10,13-16,18,33,36H,6-8,11-12,17H2,1-5H3,(H,30,35)(H,31,34)	RIACUTFRMCZUGY-UHFFFAOYSA-N	392277	US10301272, Example 304/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392277&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186119	404960612							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784131	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)NC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H38N4O5S2/c1-28(2,3)33-40(37,38)22-16-15-21(19-13-9-10-14-20(19)22)24-23(25(34)31-18-11-7-6-8-12-18)32-27(39-24)26(35)30-17-29(4,5)36/h9-10,13-16,18,33,36H,6-8,11-12,17H2,1-5H3,(H,30,35)(H,31,34)	RIACUTFRMCZUGY-UHFFFAOYSA-N	392277	US10301272, Example 304/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392277&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186119	404960612							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784132	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)NC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H38N4O5S2/c1-28(2,3)33-40(37,38)22-16-15-21(19-13-9-10-14-20(19)22)24-23(25(34)31-18-11-7-6-8-12-18)32-27(39-24)26(35)30-17-29(4,5)36/h9-10,13-16,18,33,36H,6-8,11-12,17H2,1-5H3,(H,30,35)(H,31,34)	RIACUTFRMCZUGY-UHFFFAOYSA-N	392277	US10301272, Example 304/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392277&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186119	404960612							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784133	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)C2CCC(C)(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H41N3O5S2/c1-29(2,3)34-41(38,39)23-13-12-22(20-10-8-9-11-21(20)23)26-24(25(35)19-14-16-30(4,5)17-15-19)33-28(40-26)27(36)32-18-31(6,7)37/h8-13,19,34,37H,14-18H2,1-7H3,(H,32,36)	QNAHCNJLYNUFJF-UHFFFAOYSA-N	392278	US10301272, Example 304/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392278&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186120	404960613							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784134	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)C2CCC(C)(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H41N3O5S2/c1-29(2,3)34-41(38,39)23-13-12-22(20-10-8-9-11-21(20)23)26-24(25(35)19-14-16-30(4,5)17-15-19)33-28(40-26)27(36)32-18-31(6,7)37/h8-13,19,34,37H,14-18H2,1-7H3,(H,32,36)	QNAHCNJLYNUFJF-UHFFFAOYSA-N	392278	US10301272, Example 304/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392278&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186120	404960613							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784135	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)C2CCC(C)(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H41N3O5S2/c1-29(2,3)34-41(38,39)23-13-12-22(20-10-8-9-11-21(20)23)26-24(25(35)19-14-16-30(4,5)17-15-19)33-28(40-26)27(36)32-18-31(6,7)37/h8-13,19,34,37H,14-18H2,1-7H3,(H,32,36)	QNAHCNJLYNUFJF-UHFFFAOYSA-N	392278	US10301272, Example 304/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392278	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392278&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186120	404960613							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784136	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-13-15-33(16-14-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-11-12-22(20-10-8-7-9-19(20)21)40(37,38)32-28(2,3)4/h7-12,18,32,36H,13-17H2,1-6H3,(H,30,34)	FUZPBFHPECYRIE-UHFFFAOYSA-N	392279	US10301272, Example 304/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392279&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186121	404960614							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784137	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-13-15-33(16-14-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-11-12-22(20-10-8-7-9-19(20)21)40(37,38)32-28(2,3)4/h7-12,18,32,36H,13-17H2,1-6H3,(H,30,34)	FUZPBFHPECYRIE-UHFFFAOYSA-N	392279	US10301272, Example 304/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392279&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186121	404960614							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784138	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-13-15-33(16-14-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-11-12-22(20-10-8-7-9-19(20)21)40(37,38)32-28(2,3)4/h7-12,18,32,36H,13-17H2,1-6H3,(H,30,34)	FUZPBFHPECYRIE-UHFFFAOYSA-N	392279	US10301272, Example 304/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392279	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392279&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186121	404960614							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784139	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC(C)(C)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-28(2,3)33-41(38,39)22-14-13-21(19-11-8-9-12-20(19)22)24-23(27(36)34-16-10-15-29(4,5)18-34)32-26(40-24)25(35)31-17-30(6,7)37/h8-9,11-14,33,37H,10,15-18H2,1-7H3,(H,31,35)	ICPAZJDAJORAJZ-UHFFFAOYSA-N	392280	US10301272, Example 304/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392280&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186122	404960615							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784140	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC(C)(C)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-28(2,3)33-41(38,39)22-14-13-21(19-11-8-9-12-20(19)22)24-23(27(36)34-16-10-15-29(4,5)18-34)32-26(40-24)25(35)31-17-30(6,7)37/h8-9,11-14,33,37H,10,15-18H2,1-7H3,(H,31,35)	ICPAZJDAJORAJZ-UHFFFAOYSA-N	392280	US10301272, Example 304/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392280&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186122	404960615							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784141	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC(C)(C)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-28(2,3)33-41(38,39)22-14-13-21(19-11-8-9-12-20(19)22)24-23(27(36)34-16-10-15-29(4,5)18-34)32-26(40-24)25(35)31-17-30(6,7)37/h8-9,11-14,33,37H,10,15-18H2,1-7H3,(H,31,35)	ICPAZJDAJORAJZ-UHFFFAOYSA-N	392280	US10301272, Example 304/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392280	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392280&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186122	404960615							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784142	CC1CCCN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-10-9-15-33(16-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-13-14-22(20-12-8-7-11-19(20)21)40(37,38)32-28(2,3)4/h7-8,11-14,18,32,36H,9-10,15-17H2,1-6H3,(H,30,34)	FBKWLQPDCGPROF-UHFFFAOYSA-N	392281	US10301272, Example 304/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392281&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186123	404960616							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784143	CC1CCCN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-10-9-15-33(16-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-13-14-22(20-12-8-7-11-19(20)21)40(37,38)32-28(2,3)4/h7-8,11-14,18,32,36H,9-10,15-17H2,1-6H3,(H,30,34)	FBKWLQPDCGPROF-UHFFFAOYSA-N	392281	US10301272, Example 304/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392281&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186123	404960616							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784144	CC1CCCN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-10-9-15-33(16-18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-13-14-22(20-12-8-7-11-19(20)21)40(37,38)32-28(2,3)4/h7-8,11-14,18,32,36H,9-10,15-17H2,1-6H3,(H,30,34)	FBKWLQPDCGPROF-UHFFFAOYSA-N	392281	US10301272, Example 304/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392281	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392281&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186123	404960616							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784145	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2(C)C)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-28(2,3)33-41(38,39)22-15-14-21(19-12-8-9-13-20(19)22)24-23(27(36)34-17-11-10-16-29(34,4)5)32-26(40-24)25(35)31-18-30(6,7)37/h8-9,12-15,33,37H,10-11,16-18H2,1-7H3,(H,31,35)	WUQSPBZYDFOPHH-UHFFFAOYSA-N	392282	US10301272, Example 304/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392282&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186124	404960617							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784146	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2(C)C)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-28(2,3)33-41(38,39)22-15-14-21(19-12-8-9-13-20(19)22)24-23(27(36)34-17-11-10-16-29(34,4)5)32-26(40-24)25(35)31-18-30(6,7)37/h8-9,12-15,33,37H,10-11,16-18H2,1-7H3,(H,31,35)	WUQSPBZYDFOPHH-UHFFFAOYSA-N	392282	US10301272, Example 304/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392282&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186124	404960617							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784147	CC1CCCCN1C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-11-9-10-16-33(18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-14-15-22(20-13-8-7-12-19(20)21)40(37,38)32-28(2,3)4/h7-8,12-15,18,32,36H,9-11,16-17H2,1-6H3,(H,30,34)	IVQXMUXKJKFABH-UHFFFAOYSA-N	392283	US10301272, Example 304/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392283&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186125	404960618							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784148	CC1CCCCN1C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-11-9-10-16-33(18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-14-15-22(20-13-8-7-12-19(20)21)40(37,38)32-28(2,3)4/h7-8,12-15,18,32,36H,9-11,16-17H2,1-6H3,(H,30,34)	IVQXMUXKJKFABH-UHFFFAOYSA-N	392283	US10301272, Example 304/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392283&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186125	404960618							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784149	CC1CCCCN1C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O5S2/c1-18-11-9-10-16-33(18)27(35)23-24(39-26(31-23)25(34)30-17-29(5,6)36)21-14-15-22(20-13-8-7-12-19(20)21)40(37,38)32-28(2,3)4/h7-8,12-15,18,32,36H,9-11,16-17H2,1-6H3,(H,30,34)	IVQXMUXKJKFABH-UHFFFAOYSA-N	392283	US10301272, Example 304/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392283	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392283&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186125	404960618							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784150	CC1CC(C)CN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-18-14-19(2)16-34(15-18)28(36)24-25(40-27(32-24)26(35)31-17-30(6,7)37)22-12-13-23(21-11-9-8-10-20(21)22)41(38,39)33-29(3,4)5/h8-13,18-19,33,37H,14-17H2,1-7H3,(H,31,35)	AXNNQBSHIFRERU-UHFFFAOYSA-N	392284	US10301272, Example 304/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392284&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186126	404960619							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784151	CC1CC(C)CN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-18-14-19(2)16-34(15-18)28(36)24-25(40-27(32-24)26(35)31-17-30(6,7)37)22-12-13-23(21-11-9-8-10-20(21)22)41(38,39)33-29(3,4)5/h8-13,18-19,33,37H,14-17H2,1-7H3,(H,31,35)	AXNNQBSHIFRERU-UHFFFAOYSA-N	392284	US10301272, Example 304/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392284&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186126	404960619							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784152	CC1CC(C)CN(C1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-18-14-19(2)16-34(15-18)28(36)24-25(40-27(32-24)26(35)31-17-30(6,7)37)22-12-13-23(21-11-9-8-10-20(21)22)41(38,39)33-29(3,4)5/h8-13,18-19,33,37H,14-17H2,1-7H3,(H,31,35)	AXNNQBSHIFRERU-UHFFFAOYSA-N	392284	US10301272, Example 304/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392284	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392284&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186126	404960619							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784153	CC1CCCN(C1C)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-18-11-10-16-34(19(18)2)28(36)24-25(40-27(32-24)26(35)31-17-30(6,7)37)22-14-15-23(21-13-9-8-12-20(21)22)41(38,39)33-29(3,4)5/h8-9,12-15,18-19,33,37H,10-11,16-17H2,1-7H3,(H,31,35)	VSEIRJNWSQNJLY-UHFFFAOYSA-N	392285	US10301272, Example 304/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392285	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392285&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186127	404960620							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784154	CC1CCCN(C1C)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-18-11-10-16-34(19(18)2)28(36)24-25(40-27(32-24)26(35)31-17-30(6,7)37)22-14-15-23(21-13-9-8-12-20(21)22)41(38,39)33-29(3,4)5/h8-9,12-15,18-19,33,37H,10-11,16-17H2,1-7H3,(H,31,35)	VSEIRJNWSQNJLY-UHFFFAOYSA-N	392285	US10301272, Example 304/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392285	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392285&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186127	404960620							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784155	CCC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-7-19-14-16-34(17-15-19)28(36)24-25(40-27(32-24)26(35)31-18-30(5,6)37)22-12-13-23(21-11-9-8-10-20(21)22)41(38,39)33-29(2,3)4/h8-13,19,33,37H,7,14-18H2,1-6H3,(H,31,35)	CKLHEWBUHCHXKW-UHFFFAOYSA-N	392286	US10301272, Example 304/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392286	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392286&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186128	404960621							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784156	CCC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-7-19-14-16-34(17-15-19)28(36)24-25(40-27(32-24)26(35)31-18-30(5,6)37)22-12-13-23(21-11-9-8-10-20(21)22)41(38,39)33-29(2,3)4/h8-13,19,33,37H,7,14-18H2,1-6H3,(H,31,35)	CKLHEWBUHCHXKW-UHFFFAOYSA-N	392286	US10301272, Example 304/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392286	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392286&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186128	404960621							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784157	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC3(CCCC3)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H40N4O5S2/c1-29(2,3)34-42(39,40)23-13-12-22(20-10-6-7-11-21(20)23)25-24(33-27(41-25)26(36)32-18-30(4,5)38)28(37)35-17-16-31(19-35)14-8-9-15-31/h6-7,10-13,34,38H,8-9,14-19H2,1-5H3,(H,32,36)	ODTYQWGJYBGIAF-UHFFFAOYSA-N	392287	US10301272, Example 304/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392287&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186129	404960622							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784158	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC3(CCCC3)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H40N4O5S2/c1-29(2,3)34-42(39,40)23-13-12-22(20-10-6-7-11-21(20)23)25-24(33-27(41-25)26(36)32-18-30(4,5)38)28(37)35-17-16-31(19-35)14-8-9-15-31/h6-7,10-13,34,38H,8-9,14-19H2,1-5H3,(H,32,36)	ODTYQWGJYBGIAF-UHFFFAOYSA-N	392287	US10301272, Example 304/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392287&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186129	404960622							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784159	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC3(CCCC3)C2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H40N4O5S2/c1-29(2,3)34-42(39,40)23-13-12-22(20-10-6-7-11-21(20)23)25-24(33-27(41-25)26(36)32-18-30(4,5)38)28(37)35-17-16-31(19-35)14-8-9-15-31/h6-7,10-13,34,38H,8-9,14-19H2,1-5H3,(H,32,36)	ODTYQWGJYBGIAF-UHFFFAOYSA-N	392287	US10301272, Example 304/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392287	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392287&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186129	404960622							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784160	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C28H33F3N4O5S2/c1-16-11-13-35(14-12-16)26(37)22-23(41-25(33-22)24(36)32-15-27(3,4)38)20-9-10-21(19-8-6-5-7-18(19)20)42(39,40)34-17(2)28(29,30)31/h5-10,16-17,34,38H,11-15H2,1-4H3,(H,32,36)/t17-/m0/s1	JHVZRBBPBMNBCV-KRWDZBQOSA-N	392288	US10301272, Example 304/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392288	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392288&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186130	404960623							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784161	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C28H33F3N4O5S2/c1-16-11-13-35(14-12-16)26(37)22-23(41-25(33-22)24(36)32-15-27(3,4)38)20-9-10-21(19-8-6-5-7-18(19)20)42(39,40)34-17(2)28(29,30)31/h5-10,16-17,34,38H,11-15H2,1-4H3,(H,32,36)/t17-/m0/s1	JHVZRBBPBMNBCV-KRWDZBQOSA-N	392288	US10301272, Example 304/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392288	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392288&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186130	404960623							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784162	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-7-29(3,4)33-41(38,39)23-13-12-22(20-10-8-9-11-21(20)23)25-24(28(36)34-16-14-19(2)15-17-34)32-27(40-25)26(35)31-18-30(5,6)37/h8-13,19,33,37H,7,14-18H2,1-6H3,(H,31,35)	YFKOLSLBNQLFLW-UHFFFAOYSA-N	392289	US10301272, Example 304/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392289	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392289&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186131	404960624							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784163	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C30H40N4O5S2/c1-7-29(3,4)33-41(38,39)23-13-12-22(20-10-8-9-11-21(20)23)25-24(28(36)34-16-14-19(2)15-17-34)32-27(40-25)26(35)31-18-30(5,6)37/h8-13,19,33,37H,7,14-18H2,1-6H3,(H,31,35)	YFKOLSLBNQLFLW-UHFFFAOYSA-N	392289	US10301272, Example 304/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392289	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392289&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186131	404960624							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784164	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H40N4O6S3/c1-5-31(3,4)34-44(40,41)25-11-10-24(22-8-6-7-9-23(22)25)27-26(30(37)35-16-12-20(2)13-17-35)33-29(42-27)28(36)32-21-14-18-43(38,39)19-15-21/h6-11,20-21,34H,5,12-19H2,1-4H3,(H,32,36)	HFFUOJONZMLNPN-UHFFFAOYSA-N	392290	US10301272, Example 304/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392290	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392290&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188738	404960625							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784165	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H40N4O6S3/c1-5-31(3,4)34-44(40,41)25-11-10-24(22-8-6-7-9-23(22)25)27-26(30(37)35-16-12-20(2)13-17-35)33-29(42-27)28(36)32-21-14-18-43(38,39)19-15-21/h6-11,20-21,34H,5,12-19H2,1-4H3,(H,32,36)	HFFUOJONZMLNPN-UHFFFAOYSA-N	392290	US10301272, Example 304/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392290	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392290&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188738	404960625							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784166	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C31H40N4O5S2/c1-5-31(3,4)34-42(38,39)25-11-10-24(22-8-6-7-9-23(22)25)27-26(30(37)35-16-12-20(2)13-17-35)33-29(41-27)28(36)32-21-14-18-40-19-15-21/h6-11,20-21,34H,5,12-19H2,1-4H3,(H,32,36)	AIKCAELVSFTSIR-UHFFFAOYSA-N	392291	US10301272, Example 304/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392291	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392291&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186133	404960626							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784167	CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C31H40N4O5S2/c1-5-31(3,4)34-42(38,39)25-11-10-24(22-8-6-7-9-23(22)25)27-26(30(37)35-16-12-20(2)13-17-35)33-29(41-27)28(36)32-21-14-18-40-19-15-21/h6-11,20-21,34H,5,12-19H2,1-4H3,(H,32,36)	AIKCAELVSFTSIR-UHFFFAOYSA-N	392291	US10301272, Example 304/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392291	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392291&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186133	404960626							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784168	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C32H40N4O6S3/c1-21-11-15-35(16-12-21)29(37)26-27(43-28(33-26)30(38)36-19-32(20-36)13-17-44(39,40)18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)45(41,42)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	NGWSHHFVZFXSTM-UHFFFAOYSA-N	392292	US10301272, Example 304/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392292	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392292&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186153	404960627							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784169	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C32H40N4O6S3/c1-21-11-15-35(16-12-21)29(37)26-27(43-28(33-26)30(38)36-19-32(20-36)13-17-44(39,40)18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)45(41,42)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	NGWSHHFVZFXSTM-UHFFFAOYSA-N	392292	US10301272, Example 304/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392292	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392292&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186153	404960627							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784170	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCOCC2	InChI=1S/C32H40N4O5S2/c1-21-11-15-35(16-12-21)29(37)26-27(42-28(33-26)30(38)36-19-32(20-36)13-17-41-18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)43(39,40)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	BPFUXKAAIAKBBF-UHFFFAOYSA-N	392293	US10301272, Example 304/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392293	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392293&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186135	404960628							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784171	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCOCC2	InChI=1S/C32H40N4O5S2/c1-21-11-15-35(16-12-21)29(37)26-27(42-28(33-26)30(38)36-19-32(20-36)13-17-41-18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)43(39,40)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	BPFUXKAAIAKBBF-UHFFFAOYSA-N	392293	US10301272, Example 304/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392293	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392293&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186135	404960628							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784172	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CC11CCOCC1	InChI=1S/C32H40N4O5S2/c1-20-11-15-36(16-12-20)30(38)26-27(42-29(34-26)28(37)33-25-19-32(25)13-17-41-18-14-32)23-9-10-24(22-8-6-5-7-21(22)23)43(39,40)35-31(2,3)4/h5-10,20,25,35H,11-19H2,1-4H3,(H,33,37)	FLHBPDJMHLVQIG-UHFFFAOYSA-N	392294	US10301272, Example 304/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392294&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186136	404960629							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784173	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)NC1CC11CCOCC1	InChI=1S/C32H40N4O5S2/c1-20-11-15-36(16-12-20)30(38)26-27(42-29(34-26)28(37)33-25-19-32(25)13-17-41-18-14-32)23-9-10-24(22-8-6-5-7-21(22)23)43(39,40)35-31(2,3)4/h5-10,20,25,35H,11-19H2,1-4H3,(H,33,37)	FLHBPDJMHLVQIG-UHFFFAOYSA-N	392294	US10301272, Example 304/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392294&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186136	404960629							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784174	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-19-13-15-34(16-14-19)28(36)24-25(40-27(33-24)26(35)31-18-30(5,6)37)22-11-12-23(21-10-8-7-9-20(21)22)41(38,39)32-17-29(2,3)4/h7-12,19,32,37H,13-18H2,1-6H3,(H,31,35)	RAELYCWHZOTKDM-UHFFFAOYSA-N	392295	US10301272, Example 304/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392295&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186137	404960630							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784175	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C30H40N4O5S2/c1-19-13-15-34(16-14-19)28(36)24-25(40-27(33-24)26(35)31-18-30(5,6)37)22-11-12-23(21-10-8-7-9-20(21)22)41(38,39)32-17-29(2,3)4/h7-12,19,32,37H,13-18H2,1-6H3,(H,31,35)	RAELYCWHZOTKDM-UHFFFAOYSA-N	392295	US10301272, Example 304/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392295&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186137	404960630							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784176	CCN(C(C)(C)C)S(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H42N4O5S2/c1-8-35(30(3,4)5)42(39,40)24-14-13-23(21-11-9-10-12-22(21)24)26-25(29(37)34-17-15-20(2)16-18-34)33-28(41-26)27(36)32-19-31(6,7)38/h9-14,20,38H,8,15-19H2,1-7H3,(H,32,36)	DVTCGFUVCVSVAI-UHFFFAOYSA-N	392296	US10301272, Example 304/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392296&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186138	404960631							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784177	CCN(C(C)(C)C)S(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C31H42N4O5S2/c1-8-35(30(3,4)5)42(39,40)24-14-13-23(21-11-9-10-12-22(21)24)26-25(29(37)34-17-15-20(2)16-18-34)33-28(41-26)27(36)32-19-31(6,7)38/h9-14,20,38H,8,15-19H2,1-7H3,(H,32,36)	DVTCGFUVCVSVAI-UHFFFAOYSA-N	392296	US10301272, Example 304/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392296&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186138	404960631							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783358	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	FJDPZYCZUQHVIE-UHFFFAOYSA-N	391997	US10301272, Example 1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391997	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391997&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160543	404960337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783359	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	FJDPZYCZUQHVIE-UHFFFAOYSA-N	391997	US10301272, Example 1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391997	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391997&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160543	404960337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783360	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(29-23(27-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	FJDPZYCZUQHVIE-UHFFFAOYSA-N	391997	US10301272, Example 1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391997	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391997&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160543	404960337							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783361	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)29-22(26-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	ADURLPIVHIBZBJ-UHFFFAOYSA-N	391998	US10301272, Example 2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391998	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391998&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160559	404960338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783362	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)29-22(26-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	ADURLPIVHIBZBJ-UHFFFAOYSA-N	391998	US10301272, Example 2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391998	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391998&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160559	404960338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783363	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1nc(sc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)29-22(26-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	ADURLPIVHIBZBJ-UHFFFAOYSA-N	391998	US10301272, Example 2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391998	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391998&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160559	404960338							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783364	CC(=O)NS(=O)(=O)c1nc(c(CC2CCCCC2)s1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C26H38N2O3S2/c1-17(29)28-33(30,31)24-27-23(22(32-24)13-18-11-9-8-10-12-18)19-14-20(25(2,3)4)16-21(15-19)26(5,6)7/h14-16,18H,8-13H2,1-7H3,(H,28,29)	OFUJFOTZQUKLDF-UHFFFAOYSA-N	391999	US10301272, Example 3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7943							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391999	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391999&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160568	404960339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783365	CC(=O)NS(=O)(=O)c1nc(c(CC2CCCCC2)s1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C26H38N2O3S2/c1-17(29)28-33(30,31)24-27-23(22(32-24)13-18-11-9-8-10-12-18)19-14-20(25(2,3)4)16-21(15-19)26(5,6)7/h14-16,18H,8-13H2,1-7H3,(H,28,29)	OFUJFOTZQUKLDF-UHFFFAOYSA-N	391999	US10301272, Example 3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391999	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391999&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160568	404960339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783366	CC(=O)NS(=O)(=O)c1nc(c(CC2CCCCC2)s1)-c1cc(cc(c1)C(C)(C)C)C(C)(C)C	InChI=1S/C26H38N2O3S2/c1-17(29)28-33(30,31)24-27-23(22(32-24)13-18-11-9-8-10-12-18)19-14-20(25(2,3)4)16-21(15-19)26(5,6)7/h14-16,18H,8-13H2,1-7H3,(H,28,29)	OFUJFOTZQUKLDF-UHFFFAOYSA-N	391999	US10301272, Example 3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			<19953							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=391999	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=391999&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160568	404960339							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783367	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)26-22(29-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	MMGXJRCFCADXAZ-UHFFFAOYSA-N	392000	US10301272, Example 4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392000	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392000&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160562	404960340							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783368	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)26-22(29-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	MMGXJRCFCADXAZ-UHFFFAOYSA-N	392000	US10301272, Example 4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392000	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392000&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160562	404960340							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783369	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)S(N)(=O)=O	InChI=1S/C24H36N2O2S2/c1-23(2,3)18-13-17(14-19(15-18)24(4,5)6)21-20(12-16-10-8-7-9-11-16)26-22(29-21)30(25,27)28/h13-16H,7-12H2,1-6H3,(H2,25,27,28)	MMGXJRCFCADXAZ-UHFFFAOYSA-N	392000	US10301272, Example 4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392000	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392000&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160562	404960340							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783370	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	QMJBMUBXCCDHPD-UHFFFAOYSA-N	392001	US10301272, Example 5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392001	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392001&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160525	404960341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783371	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	QMJBMUBXCCDHPD-UHFFFAOYSA-N	392001	US10301272, Example 5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392001	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392001&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160525	404960341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783372	CC(C)(C)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(N)=O	InChI=1S/C25H36N2OS/c1-24(2,3)18-13-17(14-19(15-18)25(4,5)6)21-20(27-23(29-21)22(26)28)12-16-10-8-7-9-11-16/h13-16H,7-12H2,1-6H3,(H2,26,28)	QMJBMUBXCCDHPD-UHFFFAOYSA-N	392001	US10301272, Example 5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392001	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392001&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160525	404960341							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783373	COC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1cc(cc(c1)C1(C)CC1)C(C)(C)C	InChI=1S/C32H46N2O3S/c1-30(2,3)23-18-22(19-24(20-23)32(6)13-14-32)26-25(17-21-11-9-8-10-12-21)34-28(38-26)27(35)33-16-15-31(4,5)29(36)37-7/h18-21H,8-17H2,1-7H3,(H,33,35)	VVWIGTHIBADSFK-UHFFFAOYSA-N	392002	US10301272, Example 6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392002	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392002&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160538	404960342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783374	COC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1cc(cc(c1)C1(C)CC1)C(C)(C)C	InChI=1S/C32H46N2O3S/c1-30(2,3)23-18-22(19-24(20-23)32(6)13-14-32)26-25(17-21-11-9-8-10-12-21)34-28(38-26)27(35)33-16-15-31(4,5)29(36)37-7/h18-21H,8-17H2,1-7H3,(H,33,35)	VVWIGTHIBADSFK-UHFFFAOYSA-N	392002	US10301272, Example 6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392002	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392002&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160538	404960342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783375	COC(=O)C(C)(C)CCNC(=O)c1nc(CC2CCCCC2)c(s1)-c1cc(cc(c1)C1(C)CC1)C(C)(C)C	InChI=1S/C32H46N2O3S/c1-30(2,3)23-18-22(19-24(20-23)32(6)13-14-32)26-25(17-21-11-9-8-10-12-21)34-28(38-26)27(35)33-16-15-31(4,5)29(36)37-7/h18-21H,8-17H2,1-7H3,(H,33,35)	VVWIGTHIBADSFK-UHFFFAOYSA-N	392002	US10301272, Example 6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392002	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392002&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160538	404960342							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783376	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H48N4O5S2/c1-30(2,3)23-19-22(12-13-25(23)43(39,40)36-31(4,5)6)26-24(18-21-10-8-7-9-11-21)35-28(42-26)27(37)34-20-32(29(33)38)14-16-41-17-15-32/h12-13,19,21,36H,7-11,14-18,20H2,1-6H3,(H2,33,38)(H,34,37)	WDKKNJMIQKYVKZ-UHFFFAOYSA-N	392003	US10301272, Example 6/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392003	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392003&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548239	404960343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783377	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H48N4O5S2/c1-30(2,3)23-19-22(12-13-25(23)43(39,40)36-31(4,5)6)26-24(18-21-10-8-7-9-11-21)35-28(42-26)27(37)34-20-32(29(33)38)14-16-41-17-15-32/h12-13,19,21,36H,7-11,14-18,20H2,1-6H3,(H2,33,38)(H,34,37)	WDKKNJMIQKYVKZ-UHFFFAOYSA-N	392003	US10301272, Example 6/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392003	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392003&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548239	404960343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783378	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H48N4O5S2/c1-30(2,3)23-19-22(12-13-25(23)43(39,40)36-31(4,5)6)26-24(18-21-10-8-7-9-11-21)35-28(42-26)27(37)34-20-32(29(33)38)14-16-41-17-15-32/h12-13,19,21,36H,7-11,14-18,20H2,1-6H3,(H2,33,38)(H,34,37)	WDKKNJMIQKYVKZ-UHFFFAOYSA-N	392003	US10301272, Example 6/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392003	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392003&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548239	404960343							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783379	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H45N3O3S/c1-30(2,3)23-17-22(18-24(19-23)31(4)10-11-31)26-25(16-21-8-6-5-7-9-21)35-28(39-26)27(36)34-20-32(29(33)37)12-14-38-15-13-32/h17-19,21H,5-16,20H2,1-4H3,(H2,33,37)(H,34,36)	HMCLBVIKHZWRTC-UHFFFAOYSA-N	392004	US10301272, Example 6/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392004	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392004&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185662	404960344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783380	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H45N3O3S/c1-30(2,3)23-17-22(18-24(19-23)31(4)10-11-31)26-25(16-21-8-6-5-7-9-21)35-28(39-26)27(36)34-20-32(29(33)37)12-14-38-15-13-32/h17-19,21H,5-16,20H2,1-4H3,(H2,33,37)(H,34,36)	HMCLBVIKHZWRTC-UHFFFAOYSA-N	392004	US10301272, Example 6/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392004	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392004&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185662	404960344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783381	CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(CCOCC1)C(N)=O	InChI=1S/C32H45N3O3S/c1-30(2,3)23-17-22(18-24(19-23)31(4)10-11-31)26-25(16-21-8-6-5-7-9-21)35-28(39-26)27(36)34-20-32(29(33)37)12-14-38-15-13-32/h17-19,21H,5-16,20H2,1-4H3,(H2,33,37)(H,34,36)	HMCLBVIKHZWRTC-UHFFFAOYSA-N	392004	US10301272, Example 6/2	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392004	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392004&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185662	404960344							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783382	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(N)=O)c2ccccc12	InChI=1S/C32H42N4O5S2/c1-31(2,3)36-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)35-29(42-27)28(37)34-20-32(30(33)38)15-17-41-18-16-32/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H2,33,38)(H,34,37)	LCUPOKVAHBTGTA-UHFFFAOYSA-N	392005	US10301272, Example 6/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392005	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392005&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185663	404960345							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783383	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(N)=O)c2ccccc12	InChI=1S/C32H42N4O5S2/c1-31(2,3)36-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)35-29(42-27)28(37)34-20-32(30(33)38)15-17-41-18-16-32/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H2,33,38)(H,34,37)	LCUPOKVAHBTGTA-UHFFFAOYSA-N	392005	US10301272, Example 6/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392005	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392005&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185663	404960345							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783384	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(N)=O)c2ccccc12	InChI=1S/C32H42N4O5S2/c1-31(2,3)36-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)35-29(42-27)28(37)34-20-32(30(33)38)15-17-41-18-16-32/h7-8,11-14,21,36H,4-6,9-10,15-20H2,1-3H3,(H2,33,38)(H,34,37)	LCUPOKVAHBTGTA-UHFFFAOYSA-N	392005	US10301272, Example 6/3	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392005	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392005&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185663	404960345							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784178	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(F)(F)F)C(=O)NCC(C)(C)O	InChI=1S/C27H31F3N4O5S2/c1-16-10-12-34(13-11-16)25(36)21-22(40-24(33-21)23(35)31-14-26(2,3)37)19-8-9-20(18-7-5-4-6-17(18)19)41(38,39)32-15-27(28,29)30/h4-9,16,32,37H,10-15H2,1-3H3,(H,31,35)	AYFNJCRYFRHBNS-UHFFFAOYSA-N	392297	US10301272, Example 304/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392297&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186139	404960632							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784179	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(F)(F)F)C(=O)NCC(C)(C)O	InChI=1S/C27H31F3N4O5S2/c1-16-10-12-34(13-11-16)25(36)21-22(40-24(33-21)23(35)31-14-26(2,3)37)19-8-9-20(18-7-5-4-6-17(18)19)41(38,39)32-15-27(28,29)30/h4-9,16,32,37H,10-15H2,1-3H3,(H,31,35)	AYFNJCRYFRHBNS-UHFFFAOYSA-N	392297	US10301272, Example 304/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392297&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186139	404960632							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784180	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(C)(C)O)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O6S2/c1-18-12-14-33(15-13-18)27(35)23-24(40-26(32-23)25(34)30-16-28(2,3)36)21-10-11-22(20-9-7-6-8-19(20)21)41(38,39)31-17-29(4,5)37/h6-11,18,31,36-37H,12-17H2,1-5H3,(H,30,34)	ICFPELKNSZLTSL-UHFFFAOYSA-N	392298	US10301272, Example 304/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392298&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186140	404960633							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784181	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NCC(C)(C)O)C(=O)NCC(C)(C)O	InChI=1S/C29H38N4O6S2/c1-18-12-14-33(15-13-18)27(35)23-24(40-26(32-23)25(34)30-16-28(2,3)36)21-10-11-22(20-9-7-6-8-19(20)21)41(38,39)31-17-29(4,5)37/h6-11,18,31,36-37H,12-17H2,1-5H3,(H,30,34)	ICFPELKNSZLTSL-UHFFFAOYSA-N	392298	US10301272, Example 304/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392298&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186140	404960633							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784182	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N(CC(F)(F)F)C(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C31H39F3N4O5S2/c1-19-13-15-37(16-14-19)28(40)24-25(44-27(36-24)26(39)35-17-30(5,6)41)22-11-12-23(21-10-8-7-9-20(21)22)45(42,43)38(29(2,3)4)18-31(32,33)34/h7-12,19,41H,13-18H2,1-6H3,(H,35,39)	NRZRDDUQFXMNRP-UHFFFAOYSA-N	392299	US10301272, Example 304/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392299	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392299&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186141	404960634							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784183	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N(CC(F)(F)F)C(C)(C)C)C(=O)NCC(C)(C)O	InChI=1S/C31H39F3N4O5S2/c1-19-13-15-37(16-14-19)28(40)24-25(44-27(36-24)26(39)35-17-30(5,6)41)22-11-12-23(21-10-8-7-9-20(21)22)45(42,43)38(29(2,3)4)18-31(32,33)34/h7-12,19,41H,13-18H2,1-6H3,(H,35,39)	NRZRDDUQFXMNRP-UHFFFAOYSA-N	392299	US10301272, Example 304/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392299	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392299&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186141	404960634							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784184	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1CCOC1)C(=O)NCC(C)(C)O	InChI=1S/C29H36N4O6S2/c1-18-10-13-33(14-11-18)28(35)24-25(40-27(31-24)26(34)30-17-29(2,3)36)22-8-9-23(21-7-5-4-6-20(21)22)41(37,38)32-19-12-15-39-16-19/h4-9,18-19,32,36H,10-17H2,1-3H3,(H,30,34)	UDFAUISROHNPBT-UHFFFAOYSA-N	392300	US10301272, Example 304/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392300&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186142	404960635							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784185	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1CCOC1)C(=O)NCC(C)(C)O	InChI=1S/C29H36N4O6S2/c1-18-10-13-33(14-11-18)28(35)24-25(40-27(31-24)26(34)30-17-29(2,3)36)22-8-9-23(21-7-5-4-6-20(21)22)41(37,38)32-19-12-15-39-16-19/h4-9,18-19,32,36H,10-17H2,1-3H3,(H,30,34)	UDFAUISROHNPBT-UHFFFAOYSA-N	392300	US10301272, Example 304/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392300&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186142	404960635							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784186	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N1CCCCC1(C)C)C(=O)NCC(C)(C)O	InChI=1S/C32H42N4O5S2/c1-21-14-18-35(19-15-21)30(38)26-27(42-29(34-26)28(37)33-20-32(4,5)39)24-12-13-25(23-11-7-6-10-22(23)24)43(40,41)36-17-9-8-16-31(36,2)3/h6-7,10-13,21,39H,8-9,14-20H2,1-5H3,(H,33,37)	OTJDYJNKOVBYQY-UHFFFAOYSA-N	392301	US10301272, Example 304/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392301&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186143	404960636							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784187	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N1CCCCC1(C)C)C(=O)NCC(C)(C)O	InChI=1S/C32H42N4O5S2/c1-21-14-18-35(19-15-21)30(38)26-27(42-29(34-26)28(37)33-20-32(4,5)39)24-12-13-25(23-11-7-6-10-22(23)24)43(40,41)36-17-9-8-16-31(36,2)3/h6-7,10-13,21,39H,8-9,14-20H2,1-5H3,(H,33,37)	OTJDYJNKOVBYQY-UHFFFAOYSA-N	392301	US10301272, Example 304/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392301&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186143	404960636							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784188	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)CCC1)C(=O)NCC(C)(C)O	InChI=1S/C30H38N4O5S2/c1-19-12-16-34(17-13-19)28(36)24-25(40-27(32-24)26(35)31-18-29(2,3)37)22-10-11-23(21-9-6-5-8-20(21)22)41(38,39)33-30(4)14-7-15-30/h5-6,8-11,19,33,37H,7,12-18H2,1-4H3,(H,31,35)	YQUAPIUFQRKQAC-UHFFFAOYSA-N	392302	US10301272, Example 304/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392302	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392302&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186144	404960637							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784189	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)CCC1)C(=O)NCC(C)(C)O	InChI=1S/C30H38N4O5S2/c1-19-12-16-34(17-13-19)28(36)24-25(40-27(32-24)26(35)31-18-29(2,3)37)22-10-11-23(21-9-6-5-8-20(21)22)41(38,39)33-30(4)14-7-15-30/h5-6,8-11,19,33,37H,7,12-18H2,1-4H3,(H,31,35)	YQUAPIUFQRKQAC-UHFFFAOYSA-N	392302	US10301272, Example 304/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392302	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392302&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186144	404960637							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784190	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)CC1)C(=O)NCC(C)(C)O	InChI=1S/C29H36N4O5S2/c1-18-11-15-33(16-12-18)27(35)23-24(39-26(31-23)25(34)30-17-28(2,3)36)21-9-10-22(20-8-6-5-7-19(20)21)40(37,38)32-29(4)13-14-29/h5-10,18,32,36H,11-17H2,1-4H3,(H,30,34)	SQZXZFFMQLVNBA-UHFFFAOYSA-N	392303	US10301272, Example 304/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392303	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392303&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186145	404960638							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784191	CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)NC1(C)CC1)C(=O)NCC(C)(C)O	InChI=1S/C29H36N4O5S2/c1-18-11-15-33(16-12-18)27(35)23-24(39-26(31-23)25(34)30-17-28(2,3)36)21-9-10-22(20-8-6-5-7-19(20)21)40(37,38)32-29(4)13-14-29/h5-10,18,32,36H,11-17H2,1-4H3,(H,30,34)	SQZXZFFMQLVNBA-UHFFFAOYSA-N	392303	US10301272, Example 304/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392303	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392303&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186145	404960638							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784192	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(F)F)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C23H27F2N3O4S2/c1-22(2,3)28-34(31,32)16-11-10-15(13-8-6-7-9-14(13)16)18-17(19(24)25)27-21(33-18)20(29)26-12-23(4,5)30/h6-11,19,28,30H,12H2,1-5H3,(H,26,29)	YUVFEKYATTYFPC-UHFFFAOYSA-N	392304	US10301272, Example 305	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392304	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392304&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160558	404960639							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784193	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(F)F)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C23H27F2N3O4S2/c1-22(2,3)28-34(31,32)16-11-10-15(13-8-6-7-9-14(13)16)18-17(19(24)25)27-21(33-18)20(29)26-12-23(4,5)30/h6-11,19,28,30H,12H2,1-5H3,(H,26,29)	YUVFEKYATTYFPC-UHFFFAOYSA-N	392304	US10301272, Example 305	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392304	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392304&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160558	404960639							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784194	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)NC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H38N4O5S2/c1-28(2,3)33-40(37,38)22-16-15-21(19-13-9-10-14-20(19)22)24-23(25(34)31-18-11-7-6-8-12-18)32-27(39-24)26(35)30-17-29(4,5)36/h9-10,13-16,18,33,36H,6-8,11-12,17H2,1-5H3,(H,30,35)(H,31,34)	RIACUTFRMCZUGY-UHFFFAOYSA-N	392277	US10301272, Example 304/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392277&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186119	404960612							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784195	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)NC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H38N4O5S2/c1-28(2,3)33-40(37,38)22-16-15-21(19-13-9-10-14-20(19)22)24-23(25(34)31-18-11-7-6-8-12-18)32-27(39-24)26(35)30-17-29(4,5)36/h9-10,13-16,18,33,36H,6-8,11-12,17H2,1-5H3,(H,30,35)(H,31,34)	RIACUTFRMCZUGY-UHFFFAOYSA-N	392277	US10301272, Example 304/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392277&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118186119	404960612							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784196	CC1CCN(CC1)C(=O)c1nc(oc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C32H40N4O7S2/c1-21-11-15-35(16-12-21)29(37)26-27(43-28(33-26)30(38)36-19-32(20-36)13-17-44(39,40)18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)45(41,42)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	OEPIGFXKLYNEHS-UHFFFAOYSA-N	392305	US10301272, Example 306	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2512							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392305&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160606	404960640							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784197	CC1CCN(CC1)C(=O)c1nc(oc1-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C)C(=O)N1CC2(C1)CCS(=O)(=O)CC2	InChI=1S/C32H40N4O7S2/c1-21-11-15-35(16-12-21)29(37)26-27(43-28(33-26)30(38)36-19-32(20-36)13-17-44(39,40)18-14-32)24-9-10-25(23-8-6-5-7-22(23)24)45(41,42)34-31(2,3)4/h5-10,21,34H,11-20H2,1-4H3	OEPIGFXKLYNEHS-UHFFFAOYSA-N	392305	US10301272, Example 306	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2512							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392305&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160606	404960640							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784198	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(cc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H38N2O5S2/c1-31(2,3)33-40(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-20(15-19-9-5-4-6-10-19)18-26(39-28)29(34)32-22-16-21(17-22)30(35)36/h7-8,11-14,18-19,21-22,33H,4-6,9-10,15-17H2,1-3H3,(H,32,34)(H,35,36)/t21-,22-	RPSUNEYWFMEZFB-HZCBDIJESA-N	392306	US10301272, Example 307	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392306	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392306&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160554	404960641							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784199	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(cc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C31H38N2O5S2/c1-31(2,3)33-40(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-20(15-19-9-5-4-6-10-19)18-26(39-28)29(34)32-22-16-21(17-22)30(35)36/h7-8,11-14,18-19,21-22,33H,4-6,9-10,15-17H2,1-3H3,(H,32,34)(H,35,36)/t21-,22-	RPSUNEYWFMEZFB-HZCBDIJESA-N	392306	US10301272, Example 307	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392306	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392306&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118160554	404960641							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784200	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(cc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H40N2O5S3/c1-31(2,3)33-41(37,38)28-14-13-26(24-11-7-8-12-25(24)28)29-22(19-21-9-5-4-6-10-21)20-27(39-29)30(34)32-23-15-17-40(35,36)18-16-23/h7-8,11-14,20-21,23,33H,4-6,9-10,15-19H2,1-3H3,(H,32,34)	PPPLSNSQCJPREY-UHFFFAOYSA-N	392307	US10301272, Example 307/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392307	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392307&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188742	404960642							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
784201	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(cc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H40N2O5S3/c1-31(2,3)33-41(37,38)28-14-13-26(24-11-7-8-12-25(24)28)29-22(19-21-9-5-4-6-10-21)20-27(39-29)30(34)32-23-15-17-40(35,36)18-16-23/h7-8,11-14,20-21,23,33H,4-6,9-10,15-19H2,1-3H3,(H,32,34)	PPPLSNSQCJPREY-UHFFFAOYSA-N	392307	US10301272, Example 307/1	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392307	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392307&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188742	404960642							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783385	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O4S2/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	YBTHMLBUJBBJME-UHFFFAOYSA-N	392006	US10301272, Example 6/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392006	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392006&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548957	404960346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783386	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O4S2/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	YBTHMLBUJBBJME-UHFFFAOYSA-N	392006	US10301272, Example 6/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392006	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392006&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548957	404960346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783387	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12	InChI=1S/C29H39N3O4S2/c1-28(2,3)32-38(35,36)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)31-27(37-25)26(33)30-18-29(4,5)34/h9-10,13-16,19,32,34H,6-8,11-12,17-18H2,1-5H3,(H,30,33)	YBTHMLBUJBBJME-UHFFFAOYSA-N	392006	US10301272, Example 6/4	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392006	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392006&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548957	404960346							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783388	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O6S3/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	APHQPCJAAOPTDM-UHFFFAOYSA-N	392007	US10301272, Example 6/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392007	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392007&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185664	404960347							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783389	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O6S3/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	APHQPCJAAOPTDM-UHFFFAOYSA-N	392007	US10301272, Example 6/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392007	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392007&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185664	404960347							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783390	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(O)CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C31H41N3O6S3/c1-30(2,3)34-43(39,40)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-21-9-5-4-6-10-21)33-29(41-27)28(35)32-20-31(36)15-17-42(37,38)18-16-31/h7-8,11-14,21,34,36H,4-6,9-10,15-20H2,1-3H3,(H,32,35)	APHQPCJAAOPTDM-UHFFFAOYSA-N	392007	US10301272, Example 6/5	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392007	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392007&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185664	404960347							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783391	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	TWURQQLYKYCGLR-UHFFFAOYSA-N	392008	US10301272, Example 6/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392008&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185665	404960348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783392	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	TWURQQLYKYCGLR-UHFFFAOYSA-N	392008	US10301272, Example 6/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392008&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185665	404960348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783393	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C30H39N3O5S3/c1-30(2,3)33-41(37,38)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(39-27)28(34)31-21-15-17-40(35,36)18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	TWURQQLYKYCGLR-UHFFFAOYSA-N	392008	US10301272, Example 6/6	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392008	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392008&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185665	404960348							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783394	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O5S3/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JQFYVJPIAXFVPK-UHFFFAOYSA-N	50044180	CHEMBL3314001::US10301272, Example 6/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185666	313068131		CHEMBL3314001					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783395	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O5S3/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JQFYVJPIAXFVPK-UHFFFAOYSA-N	50044180	CHEMBL3314001::US10301272, Example 6/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185666	313068131		CHEMBL3314001					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783396	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12	InChI=1S/C32H41N3O5S3/c1-31(2,3)34-43(39,40)27-14-13-25(23-11-7-8-12-24(23)27)28-26(19-22-9-5-4-6-10-22)33-29(41-28)30(36)35-20-32(21-35)15-17-42(37,38)18-16-32/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3	JQFYVJPIAXFVPK-UHFFFAOYSA-N	50044180	CHEMBL3314001::US10301272, Example 6/7	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044180	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044180&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185666	313068131		CHEMBL3314001					1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783397	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O5S2/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	XLRXJYWJGFUEPW-UHFFFAOYSA-N	392010	US10301272, Example 6/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392010	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392010&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185667	404960350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783398	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O5S2/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	XLRXJYWJGFUEPW-UHFFFAOYSA-N	392010	US10301272, Example 6/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392010	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392010&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185667	404960350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783399	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CCC(CC2)(CC3)C(O)=O)c2ccccc12	InChI=1S/C34H43N3O5S2/c1-32(2,3)37-44(41,42)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)35-30(43-28)29(38)36-34-18-15-33(16-19-34,17-20-34)31(39)40/h7-8,11-14,22,37H,4-6,9-10,15-21H2,1-3H3,(H,36,38)(H,39,40)	XLRXJYWJGFUEPW-UHFFFAOYSA-N	392010	US10301272, Example 6/8	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392010	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392010&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185667	404960350							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783400	CC(C)(C)NS(=O)(=O)c1cnc(nc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H41N5O5S2/c1-27(2,3)22-20(40(37,38)33-28(4,5)6)15-29-23(32-22)21-19(12-16-10-8-7-9-11-16)31-25(39-21)24(34)30-18-13-17(14-18)26(35)36/h15-18,33H,7-14H2,1-6H3,(H,30,34)(H,35,36)/t17-,18-	GJABJGPNWZAJID-IYARVYRRSA-N	392011	US10301272, Example 6/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392011	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392011&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185668	404960351							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783401	CC(C)(C)NS(=O)(=O)c1cnc(nc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H41N5O5S2/c1-27(2,3)22-20(40(37,38)33-28(4,5)6)15-29-23(32-22)21-19(12-16-10-8-7-9-11-16)31-25(39-21)24(34)30-18-13-17(14-18)26(35)36/h15-18,33H,7-14H2,1-6H3,(H,30,34)(H,35,36)/t17-,18-	GJABJGPNWZAJID-IYARVYRRSA-N	392011	US10301272, Example 6/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392011	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392011&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185668	404960351							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783402	CC(C)(C)NS(=O)(=O)c1cnc(nc1C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O	InChI=1S/C28H41N5O5S2/c1-27(2,3)22-20(40(37,38)33-28(4,5)6)15-29-23(32-22)21-19(12-16-10-8-7-9-11-16)31-25(39-21)24(34)30-18-13-17(14-18)26(35)36/h15-18,33H,7-14H2,1-6H3,(H,30,34)(H,35,36)/t17-,18-	GJABJGPNWZAJID-IYARVYRRSA-N	392011	US10301272, Example 6/9	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392011	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392011&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185668	404960351							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783403	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c2ccccc12	InChI=1S/C32H41N3O5S2/c1-31(2,3)34-42(39,40)26-16-15-24(22-13-9-10-14-23(22)26)27-25(17-20-11-7-6-8-12-20)33-28(41-27)29(36)35-18-21(19-35)32(4,5)30(37)38/h9-10,13-16,20-21,34H,6-8,11-12,17-19H2,1-5H3,(H,37,38)	NKUTUPAMPBDAJJ-UHFFFAOYSA-N	392012	US10301272, Example 6/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392012	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392012&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185669	404960352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783404	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c2ccccc12	InChI=1S/C32H41N3O5S2/c1-31(2,3)34-42(39,40)26-16-15-24(22-13-9-10-14-23(22)26)27-25(17-20-11-7-6-8-12-20)33-28(41-27)29(36)35-18-21(19-35)32(4,5)30(37)38/h9-10,13-16,20-21,34H,6-8,11-12,17-19H2,1-5H3,(H,37,38)	NKUTUPAMPBDAJJ-UHFFFAOYSA-N	392012	US10301272, Example 6/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392012	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392012&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185669	404960352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783405	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c2ccccc12	InChI=1S/C32H41N3O5S2/c1-31(2,3)34-42(39,40)26-16-15-24(22-13-9-10-14-23(22)26)27-25(17-20-11-7-6-8-12-20)33-28(41-27)29(36)35-18-21(19-35)32(4,5)30(37)38/h9-10,13-16,20-21,34H,6-8,11-12,17-19H2,1-5H3,(H,37,38)	NKUTUPAMPBDAJJ-UHFFFAOYSA-N	392012	US10301272, Example 6/10	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392012	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392012&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185669	404960352							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783406	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O4S2/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	XSIGTUMCBGANBN-UHFFFAOYSA-N	392013	US10301272, Example 6/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392013&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185670	404960353							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783407	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O4S2/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	XSIGTUMCBGANBN-UHFFFAOYSA-N	392013	US10301272, Example 6/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392013&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185670	404960353							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783408	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12	InChI=1S/C30H39N3O4S2/c1-30(2,3)33-39(35,36)26-14-13-24(22-11-7-8-12-23(22)26)27-25(19-20-9-5-4-6-10-20)32-29(38-27)28(34)31-21-15-17-37-18-16-21/h7-8,11-14,20-21,33H,4-6,9-10,15-19H2,1-3H3,(H,31,34)	XSIGTUMCBGANBN-UHFFFAOYSA-N	392013	US10301272, Example 6/11	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392013&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185670	404960353							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783409	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12)C(F)(F)F	InChI=1S/C29H34F3N3O4S2/c1-18(29(30,31)32)35-41(37,38)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-19-7-3-2-4-8-19)34-28(40-26)27(36)33-20-13-15-39-16-14-20/h5-6,9-12,18-20,35H,2-4,7-8,13-17H2,1H3,(H,33,36)	TXSZPTCXESKVKJ-UHFFFAOYSA-N	392014	US10301272, Example 6/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392014	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392014&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012227	404960354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783410	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12)C(F)(F)F	InChI=1S/C29H34F3N3O4S2/c1-18(29(30,31)32)35-41(37,38)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-19-7-3-2-4-8-19)34-28(40-26)27(36)33-20-13-15-39-16-14-20/h5-6,9-12,18-20,35H,2-4,7-8,13-17H2,1H3,(H,33,36)	TXSZPTCXESKVKJ-UHFFFAOYSA-N	392014	US10301272, Example 6/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392014	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392014&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012227	404960354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783411	CC(NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12)C(F)(F)F	InChI=1S/C29H34F3N3O4S2/c1-18(29(30,31)32)35-41(37,38)25-12-11-23(21-9-5-6-10-22(21)25)26-24(17-19-7-3-2-4-8-19)34-28(40-26)27(36)33-20-13-15-39-16-14-20/h5-6,9-12,18-20,35H,2-4,7-8,13-17H2,1H3,(H,33,36)	TXSZPTCXESKVKJ-UHFFFAOYSA-N	392014	US10301272, Example 6/12	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392014	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392014&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012227	404960354							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783412	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCOCC2)c2ccccc12	InChI=1S/C31H42N4O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)33-30(40-28)29(36)32-15-16-35-17-19-39-20-18-35/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3,(H,32,36)	GKKPHEJEMPOKNF-UHFFFAOYSA-N	392015	US10301272, Example 6/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 316							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392015	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392015&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185671	404960355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783413	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCOCC2)c2ccccc12	InChI=1S/C31H42N4O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)33-30(40-28)29(36)32-15-16-35-17-19-39-20-18-35/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3,(H,32,36)	GKKPHEJEMPOKNF-UHFFFAOYSA-N	392015	US10301272, Example 6/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392015	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392015&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185671	404960355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783414	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCOCC2)c2ccccc12	InChI=1S/C31H42N4O4S2/c1-31(2,3)34-41(37,38)27-14-13-25(23-11-7-8-12-24(23)27)28-26(21-22-9-5-4-6-10-22)33-30(40-28)29(36)32-15-16-35-17-19-39-20-18-35/h7-8,11-14,22,34H,4-6,9-10,15-21H2,1-3H3,(H,32,36)	GKKPHEJEMPOKNF-UHFFFAOYSA-N	392015	US10301272, Example 6/13	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392015	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392015&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185671	404960355							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783415	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c2ccccc12	InChI=1S/C28H35N3O3S3/c1-28(2,3)31-37(33,34)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(36-25)26(32)29-19-16-35-17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	LGNGYLGTQKSAHX-UHFFFAOYSA-N	392016	US10301272, Example 6/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392016&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185676	404960356							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783416	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c2ccccc12	InChI=1S/C28H35N3O3S3/c1-28(2,3)31-37(33,34)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(36-25)26(32)29-19-16-35-17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	LGNGYLGTQKSAHX-UHFFFAOYSA-N	392016	US10301272, Example 6/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392016&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185676	404960356							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783417	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c2ccccc12	InChI=1S/C28H35N3O3S3/c1-28(2,3)31-37(33,34)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-18-9-5-4-6-10-18)30-27(36-25)26(32)29-19-16-35-17-19/h7-8,11-14,18-19,31H,4-6,9-10,15-17H2,1-3H3,(H,29,32)	LGNGYLGTQKSAHX-UHFFFAOYSA-N	392016	US10301272, Example 6/14	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392016	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392016&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185676	404960356							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783418	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CN3CCC2CC3)c2ccccc12	InChI=1S/C32H42N4O3S2/c1-32(2,3)35-41(38,39)28-14-13-25(23-11-7-8-12-24(23)28)29-26(19-21-9-5-4-6-10-21)34-31(40-29)30(37)33-27-20-36-17-15-22(27)16-18-36/h7-8,11-14,21-22,27,35H,4-6,9-10,15-20H2,1-3H3,(H,33,37)	ZTBKEXCSAPADJV-UHFFFAOYSA-N	392017	US10301272, Example 6/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392017	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392017&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185677	404960357							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783419	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CN3CCC2CC3)c2ccccc12	InChI=1S/C32H42N4O3S2/c1-32(2,3)35-41(38,39)28-14-13-25(23-11-7-8-12-24(23)28)29-26(19-21-9-5-4-6-10-21)34-31(40-29)30(37)33-27-20-36-17-15-22(27)16-18-36/h7-8,11-14,21-22,27,35H,4-6,9-10,15-20H2,1-3H3,(H,33,37)	ZTBKEXCSAPADJV-UHFFFAOYSA-N	392017	US10301272, Example 6/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392017	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392017&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185677	404960357							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783420	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CN3CCC2CC3)c2ccccc12	InChI=1S/C32H42N4O3S2/c1-32(2,3)35-41(38,39)28-14-13-25(23-11-7-8-12-24(23)28)29-26(19-21-9-5-4-6-10-21)34-31(40-29)30(37)33-27-20-36-17-15-22(27)16-18-36/h7-8,11-14,21-22,27,35H,4-6,9-10,15-20H2,1-3H3,(H,33,37)	ZTBKEXCSAPADJV-UHFFFAOYSA-N	392017	US10301272, Example 6/15	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392017	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392017&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185677	404960357							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783421	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCC2)c2ccccc12	InChI=1S/C30H40N4O3S2/c1-30(2,3)33-39(36,37)26-15-14-24(22-12-7-8-13-23(22)26)27-25(20-21-10-5-4-6-11-21)32-29(38-27)28(35)31-16-19-34-17-9-18-34/h7-8,12-15,21,33H,4-6,9-11,16-20H2,1-3H3,(H,31,35)	QTLBLIJVXBTEKN-UHFFFAOYSA-N	392018	US10301272, Example 6/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1259							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392018&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185672	404960358							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783422	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCC2)c2ccccc12	InChI=1S/C30H40N4O3S2/c1-30(2,3)33-39(36,37)26-15-14-24(22-12-7-8-13-23(22)26)27-25(20-21-10-5-4-6-11-21)32-29(38-27)28(35)31-16-19-34-17-9-18-34/h7-8,12-15,21,33H,4-6,9-11,16-20H2,1-3H3,(H,31,35)	QTLBLIJVXBTEKN-UHFFFAOYSA-N	392018	US10301272, Example 6/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392018&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185672	404960358							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783423	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCC2)c2ccccc12	InChI=1S/C30H40N4O3S2/c1-30(2,3)33-39(36,37)26-15-14-24(22-12-7-8-13-23(22)26)27-25(20-21-10-5-4-6-11-21)32-29(38-27)28(35)31-16-19-34-17-9-18-34/h7-8,12-15,21,33H,4-6,9-11,16-20H2,1-3H3,(H,31,35)	QTLBLIJVXBTEKN-UHFFFAOYSA-N	392018	US10301272, Example 6/16	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392018	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392018&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185672	404960358							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783424	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c2ccccc12	InChI=1S/C31H37N3O5S2/c1-29(2,3)34-41(38,39)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-19-9-5-4-6-10-19)32-27(40-25)26(35)33-31-16-30(17-31,18-31)28(36)37/h7-8,11-14,19,34H,4-6,9-10,15-18H2,1-3H3,(H,33,35)(H,36,37)	IXZNFUVIMHGHCV-UHFFFAOYSA-N	392019	US10301272, Example 6/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 631							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392019	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392019&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185679	404960359							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783425	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c2ccccc12	InChI=1S/C31H37N3O5S2/c1-29(2,3)34-41(38,39)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-19-9-5-4-6-10-19)32-27(40-25)26(35)33-31-16-30(17-31,18-31)28(36)37/h7-8,11-14,19,34H,4-6,9-10,15-18H2,1-3H3,(H,33,35)(H,36,37)	IXZNFUVIMHGHCV-UHFFFAOYSA-N	392019	US10301272, Example 6/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392019	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392019&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185679	404960359							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783426	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c2ccccc12	InChI=1S/C31H37N3O5S2/c1-29(2,3)34-41(38,39)24-14-13-22(20-11-7-8-12-21(20)24)25-23(15-19-9-5-4-6-10-19)32-27(40-25)26(35)33-31-16-30(17-31,18-31)28(36)37/h7-8,11-14,19,34H,4-6,9-10,15-18H2,1-3H3,(H,33,35)(H,36,37)	IXZNFUVIMHGHCV-UHFFFAOYSA-N	392019	US10301272, Example 6/17	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392019	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392019&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185679	404960359							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783427	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(F)c1C(F)F	InChI=1S/C26H36F3N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(20(27)19(18)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	AILZNFVZNAMVDG-UHFFFAOYSA-N	392020	US10301272, Example 6/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392020	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392020&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185674	404960360							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783428	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(F)c1C(F)F	InChI=1S/C26H36F3N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(20(27)19(18)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	AILZNFVZNAMVDG-UHFFFAOYSA-N	392020	US10301272, Example 6/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392020	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392020&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185674	404960360							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783429	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(F)c1C(F)F	InChI=1S/C26H36F3N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(20(27)19(18)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	AILZNFVZNAMVDG-UHFFFAOYSA-N	392020	US10301272, Example 6/18	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392020	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392020&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185674	404960360							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783430	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1C(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(19(20(18)27)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	HCDHFTDPQRUZKR-UHFFFAOYSA-N	392021	US10301272, Example 6/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392021&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185675	404960361							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783431	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1C(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(19(20(18)27)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	HCDHFTDPQRUZKR-UHFFFAOYSA-N	392021	US10301272, Example 6/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392021&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185675	404960361							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783432	CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1C(F)F)S(=O)(=O)NC(C)(C)C	InChI=1S/C26H36ClF2N3O4S2/c1-25(2,3)32-38(35,36)18-12-11-16(19(20(18)27)22(28)29)21-17(13-15-9-7-6-8-10-15)31-24(37-21)23(33)30-14-26(4,5)34/h11-12,15,22,32,34H,6-10,13-14H2,1-5H3,(H,30,33)	HCDHFTDPQRUZKR-UHFFFAOYSA-N	392021	US10301272, Example 6/19	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392021	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392021&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185675	404960361							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783433	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCOCC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(36-22)23(32)29-31-11-13-35-14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	RQJVLCZEVWVELI-UHFFFAOYSA-N	392022	US10301272, Example 6/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392022	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392022&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185680	404960362							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783434	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCOCC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(36-22)23(32)29-31-11-13-35-14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	RQJVLCZEVWVELI-UHFFFAOYSA-N	392022	US10301272, Example 6/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392022	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392022&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185680	404960362							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783435	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCOCC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(36-22)23(32)29-31-11-13-35-14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	RQJVLCZEVWVELI-UHFFFAOYSA-N	392022	US10301272, Example 6/20	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392022	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392022&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185680	404960362							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783436	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(37-22)23(32)29-31-11-13-38(33,34)14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	SPDRPVKEOQMNTA-UHFFFAOYSA-N	392023	US10301272, Example 6/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392023&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185684	404960363							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783437	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(37-22)23(32)29-31-11-13-38(33,34)14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	SPDRPVKEOQMNTA-UHFFFAOYSA-N	392023	US10301272, Example 6/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392023&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185684	404960363							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783438	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NN2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C25H34Cl2N4O5S3/c1-25(2,3)30-39(35,36)19-10-9-17(20(26)21(19)27)22-18(15-16-7-5-4-6-8-16)28-24(37-22)23(32)29-31-11-13-38(33,34)14-12-31/h9-10,16,30H,4-8,11-15H2,1-3H3,(H,29,32)	SPDRPVKEOQMNTA-UHFFFAOYSA-N	392023	US10301272, Example 6/21	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392023&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185684	404960363							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783439	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C29H43N3O5S2/c1-28(2,3)32-39(35,36)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(38-25)26(33)30-21-13-15-37-16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	ZVIAXTWXQAIHIL-UHFFFAOYSA-N	392024	US10301272, Example 6/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392024	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392024&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185678	404960364							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783440	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C29H43N3O5S2/c1-28(2,3)32-39(35,36)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(38-25)26(33)30-21-13-15-37-16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	ZVIAXTWXQAIHIL-UHFFFAOYSA-N	392024	US10301272, Example 6/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392024	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392024&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185678	404960364							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783441	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCOCC1	InChI=1S/C29H43N3O5S2/c1-28(2,3)32-39(35,36)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(38-25)26(33)30-21-13-15-37-16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	ZVIAXTWXQAIHIL-UHFFFAOYSA-N	392024	US10301272, Example 6/22	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392024	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392024&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185678	404960364							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783442	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O	InChI=1S/C28H43N3O5S2/c1-26(2,3)31-38(35,36)22-14-13-19(16-20(22)28(6,7)34)23-21(15-18-11-9-8-10-12-18)30-25(37-23)24(32)29-17-27(4,5)33/h13-14,16,18,31,33-34H,8-12,15,17H2,1-7H3,(H,29,32)	YKCVSTKSODSNKW-UHFFFAOYSA-N	392025	US10301272, Example 6/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392025&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185685	404960365							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783443	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O	InChI=1S/C28H43N3O5S2/c1-26(2,3)31-38(35,36)22-14-13-19(16-20(22)28(6,7)34)23-21(15-18-11-9-8-10-12-18)30-25(37-23)24(32)29-17-27(4,5)33/h13-14,16,18,31,33-34H,8-12,15,17H2,1-7H3,(H,29,32)	YKCVSTKSODSNKW-UHFFFAOYSA-N	392025	US10301272, Example 6/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392025&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185685	404960365							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783444	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC(C)(C)O	InChI=1S/C28H43N3O5S2/c1-26(2,3)31-38(35,36)22-14-13-19(16-20(22)28(6,7)34)23-21(15-18-11-9-8-10-12-18)30-25(37-23)24(32)29-17-27(4,5)33/h13-14,16,18,31,33-34H,8-12,15,17H2,1-7H3,(H,29,32)	YKCVSTKSODSNKW-UHFFFAOYSA-N	392025	US10301272, Example 6/23	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392025	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392025&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185685	404960365							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783445	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CSC1	InChI=1S/C27H39N3O4S3/c1-26(2,3)30-37(33,34)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-35-16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	DBMDLBKSOZVQRI-UHFFFAOYSA-N	392026	US10301272, Example 6/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392026	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392026&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185681	404960366							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783446	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CSC1	InChI=1S/C27H39N3O4S3/c1-26(2,3)30-37(33,34)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-35-16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	DBMDLBKSOZVQRI-UHFFFAOYSA-N	392026	US10301272, Example 6/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392026	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392026&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185681	404960366							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783447	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CSC1	InChI=1S/C27H39N3O4S3/c1-26(2,3)30-37(33,34)22-12-11-18(14-20(22)27(4,5)32)23-21(13-17-9-7-6-8-10-17)29-25(36-23)24(31)28-19-15-35-16-19/h11-12,14,17,19,30,32H,6-10,13,15-16H2,1-5H3,(H,28,31)	DBMDLBKSOZVQRI-UHFFFAOYSA-N	392026	US10301272, Example 6/24	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392026	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392026&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185681	404960366							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783448	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCCN1CCOCC1	InChI=1S/C30H46N4O5S2/c1-29(2,3)33-41(37,38)25-12-11-22(20-23(25)30(4,5)36)26-24(19-21-9-7-6-8-10-21)32-28(40-26)27(35)31-13-14-34-15-17-39-18-16-34/h11-12,20-21,33,36H,6-10,13-19H2,1-5H3,(H,31,35)	AGOLNJHNSXNOCB-UHFFFAOYSA-N	392027	US10301272, Example 6/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1585							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392027	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392027&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185683	404960367							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783449	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCCN1CCOCC1	InChI=1S/C30H46N4O5S2/c1-29(2,3)33-41(37,38)25-12-11-22(20-23(25)30(4,5)36)26-24(19-21-9-7-6-8-10-21)32-28(40-26)27(35)31-13-14-34-15-17-39-18-16-34/h11-12,20-21,33,36H,6-10,13-19H2,1-5H3,(H,31,35)	AGOLNJHNSXNOCB-UHFFFAOYSA-N	392027	US10301272, Example 6/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392027	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392027&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185683	404960367							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783450	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCCN1CCOCC1	InChI=1S/C30H46N4O5S2/c1-29(2,3)33-41(37,38)25-12-11-22(20-23(25)30(4,5)36)26-24(19-21-9-7-6-8-10-21)32-28(40-26)27(35)31-13-14-34-15-17-39-18-16-34/h11-12,20-21,33,36H,6-10,13-19H2,1-5H3,(H,31,35)	AGOLNJHNSXNOCB-UHFFFAOYSA-N	392027	US10301272, Example 6/25	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392027	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392027&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185683	404960367							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783451	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C29H43N3O6S3/c1-28(2,3)32-41(37,38)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(39-25)26(33)30-21-13-15-40(35,36)16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	INWXIDWTPUTVFD-UHFFFAOYSA-N	392028	US10301272, Example 6/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392028&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185682	404960368							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783452	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C29H43N3O6S3/c1-28(2,3)32-41(37,38)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(39-25)26(33)30-21-13-15-40(35,36)16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	INWXIDWTPUTVFD-UHFFFAOYSA-N	392028	US10301272, Example 6/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392028&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185682	404960368							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783453	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NC1CCS(=O)(=O)CC1	InChI=1S/C29H43N3O6S3/c1-28(2,3)32-41(37,38)24-12-11-20(18-22(24)29(4,5)34)25-23(17-19-9-7-6-8-10-19)31-27(39-25)26(33)30-21-13-15-40(35,36)16-14-21/h11-12,18-19,21,32,34H,6-10,13-17H2,1-5H3,(H,30,33)	INWXIDWTPUTVFD-UHFFFAOYSA-N	392028	US10301272, Example 6/26	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392028	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392028&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185682	404960368							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783454	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(O)CCOCC1	InChI=1S/C30H45N3O6S2/c1-28(2,3)33-41(37,38)24-12-11-21(18-22(24)29(4,5)35)25-23(17-20-9-7-6-8-10-20)32-27(40-25)26(34)31-19-30(36)13-15-39-16-14-30/h11-12,18,20,33,35-36H,6-10,13-17,19H2,1-5H3,(H,31,34)	YOWNTNMOLBFHJX-UHFFFAOYSA-N	392029	US10301272, Example 6/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 200							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392029	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392029&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185690	404960369							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783455	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(O)CCOCC1	InChI=1S/C30H45N3O6S2/c1-28(2,3)33-41(37,38)24-12-11-21(18-22(24)29(4,5)35)25-23(17-20-9-7-6-8-10-20)32-27(40-25)26(34)31-19-30(36)13-15-39-16-14-30/h11-12,18,20,33,35-36H,6-10,13-17,19H2,1-5H3,(H,31,34)	YOWNTNMOLBFHJX-UHFFFAOYSA-N	392029	US10301272, Example 6/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392029	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392029&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185690	404960369							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783456	CC(C)(C)NS(=O)(=O)c1ccc(cc1C(C)(C)O)-c1sc(nc1CC1CCCCC1)C(=O)NCC1(O)CCOCC1	InChI=1S/C30H45N3O6S2/c1-28(2,3)33-41(37,38)24-12-11-21(18-22(24)29(4,5)35)25-23(17-20-9-7-6-8-10-20)32-27(40-25)26(34)31-19-30(36)13-15-39-16-14-30/h11-12,18,20,33,35-36H,6-10,13-17,19H2,1-5H3,(H,31,34)	YOWNTNMOLBFHJX-UHFFFAOYSA-N	392029	US10301272, Example 6/27	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392029	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392029&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185690	404960369							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783457	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C29H36N4O5S2/c1-29(2,3)33-40(37,38)27-21-12-8-7-11-20(21)22(16-30-27)24-23(13-17-9-5-4-6-10-17)32-26(39-24)25(34)31-19-14-18(15-19)28(35)36/h7-8,11-12,16-19,33H,4-6,9-10,13-15H2,1-3H3,(H,31,34)(H,35,36)/t18-,19-	UOLHOHMCDXPLCY-WGSAOQKQSA-N	392030	US10301272, Example 6/28	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392030&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548705	404960370							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783458	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C29H36N4O5S2/c1-29(2,3)33-40(37,38)27-21-12-8-7-11-20(21)22(16-30-27)24-23(13-17-9-5-4-6-10-17)32-26(39-24)25(34)31-19-14-18(15-19)28(35)36/h7-8,11-12,16-19,33H,4-6,9-10,13-15H2,1-3H3,(H,31,34)(H,35,36)/t18-,19-	UOLHOHMCDXPLCY-WGSAOQKQSA-N	392030	US10301272, Example 6/28	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392030&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548705	404960370							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783459	CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12	InChI=1S/C29H36N4O5S2/c1-29(2,3)33-40(37,38)27-21-12-8-7-11-20(21)22(16-30-27)24-23(13-17-9-5-4-6-10-17)32-26(39-24)25(34)31-19-14-18(15-19)28(35)36/h7-8,11-12,16-19,33H,4-6,9-10,13-15H2,1-3H3,(H,31,34)(H,35,36)/t18-,19-	UOLHOHMCDXPLCY-WGSAOQKQSA-N	392030	US10301272, Example 6/28	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392030	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392030&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72548705	404960370							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783460	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O4S2/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	QNXDBYMJERHWQS-UHFFFAOYSA-N	392031	US10301272, Example 6/29	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392031	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392031&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185688	404960371							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783461	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O4S2/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	QNXDBYMJERHWQS-UHFFFAOYSA-N	392031	US10301272, Example 6/29	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392031	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392031&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185688	404960371							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783462	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl	InChI=1S/C25H35Cl2N3O4S2/c1-24(2,3)30-36(33,34)18-12-11-16(19(26)20(18)27)21-17(13-15-9-7-6-8-10-15)29-23(35-21)22(31)28-14-25(4,5)32/h11-12,15,30,32H,6-10,13-14H2,1-5H3,(H,28,31)	QNXDBYMJERHWQS-UHFFFAOYSA-N	392031	US10301272, Example 6/29	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1.000							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392031	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392031&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185688	404960371							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783463	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S3/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	WDWKSWHEWRKJPR-UHFFFAOYSA-N	392032	US10301272, Example 6/30	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392032&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185687	404960372							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783464	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S3/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	WDWKSWHEWRKJPR-UHFFFAOYSA-N	392032	US10301272, Example 6/30	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392032&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185687	404960372							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783465	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CSC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S3/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	WDWKSWHEWRKJPR-UHFFFAOYSA-N	392032	US10301272, Example 6/30	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392032	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392032&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185687	404960372							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783466	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S2/c1-24(2,3)29-34(31,32)18-12-11-16(19(25)20(18)26)21-17(13-14-7-5-4-6-8-14)28-23(33-21)22(30)27-15-9-10-15/h11-12,14-15,29H,4-10,13H2,1-3H3,(H,27,30)	MFIDUDKMGGBKPL-UHFFFAOYSA-N	392033	US10301272, Example 6/31	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392033	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392033&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185686	404960373							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783467	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S2/c1-24(2,3)29-34(31,32)18-12-11-16(19(25)20(18)26)21-17(13-14-7-5-4-6-8-14)28-23(33-21)22(30)27-15-9-10-15/h11-12,14-15,29H,4-10,13H2,1-3H3,(H,27,30)	MFIDUDKMGGBKPL-UHFFFAOYSA-N	392033	US10301272, Example 6/31	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392033	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392033&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185686	404960373							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783468	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O3S2/c1-24(2,3)29-34(31,32)18-12-11-16(19(25)20(18)26)21-17(13-14-7-5-4-6-8-14)28-23(33-21)22(30)27-15-9-10-15/h11-12,14-15,29H,4-10,13H2,1-3H3,(H,27,30)	MFIDUDKMGGBKPL-UHFFFAOYSA-N	392033	US10301272, Example 6/31	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392033	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392033&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185686	404960373							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783469	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(CSC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O3S3/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	XLMWUZLZXLWOMK-UHFFFAOYSA-N	392034	US10301272, Example 6/32	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392034	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392034&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185689	404960374							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783470	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(CSC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O3S3/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	XLMWUZLZXLWOMK-UHFFFAOYSA-N	392034	US10301272, Example 6/32	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392034	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392034&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185689	404960374							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783471	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(CSC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O3S3/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	XLMWUZLZXLWOMK-UHFFFAOYSA-N	392034	US10301272, Example 6/32	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392034	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392034&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185689	404960374							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783472	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(COC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	FTBAQBAUFGTBQG-UHFFFAOYSA-N	392035	US10301272, Example 6/33	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392035	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392035&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185691	404960375							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783473	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(COC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	FTBAQBAUFGTBQG-UHFFFAOYSA-N	392035	US10301272, Example 6/33	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392035	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392035&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185691	404960375							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783474	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(COC3)C2)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-25(2,3)30-37(33,34)19-10-9-17(20(27)21(19)28)22-18(11-16-7-5-4-6-8-16)29-23(36-22)24(32)31-12-26(13-31)14-35-15-26/h9-10,16,30H,4-8,11-15H2,1-3H3	FTBAQBAUFGTBQG-UHFFFAOYSA-N	392035	US10301272, Example 6/33	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392035	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392035&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185691	404960375							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783475	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2COC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S2/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	PIMGSMBZEJOCRY-UHFFFAOYSA-N	392036	US10301272, Example 6/34	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392036&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185692	404960376							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783476	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2COC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S2/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	PIMGSMBZEJOCRY-UHFFFAOYSA-N	392036	US10301272, Example 6/34	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392036&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185692	404960376							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783477	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2COC2)c(Cl)c1Cl	InChI=1S/C24H31Cl2N3O4S2/c1-24(2,3)29-35(31,32)18-10-9-16(19(25)20(18)26)21-17(11-14-7-5-4-6-8-14)28-23(34-21)22(30)27-15-12-33-13-15/h9-10,14-15,29H,4-8,11-13H2,1-3H3,(H,27,30)	PIMGSMBZEJOCRY-UHFFFAOYSA-N	392036	US10301272, Example 6/34	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392036	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392036&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185692	404960376							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783478	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C23H29Cl2N3O5S3/c1-23(2,3)28-36(32,33)17-7-6-15(18(24)19(17)25)20-16(12-13-4-5-13)27-22(34-20)21(29)26-14-8-10-35(30,31)11-9-14/h6-7,13-14,28H,4-5,8-12H2,1-3H3,(H,26,29)	UPJFBEIADODBQT-UHFFFAOYSA-N	392037	US10301272, Example 6/35	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392037	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392037&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185693	404960377							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783479	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C23H29Cl2N3O5S3/c1-23(2,3)28-36(32,33)17-7-6-15(18(24)19(17)25)20-16(12-13-4-5-13)27-22(34-20)21(29)26-14-8-10-35(30,31)11-9-14/h6-7,13-14,28H,4-5,8-12H2,1-3H3,(H,26,29)	UPJFBEIADODBQT-UHFFFAOYSA-N	392037	US10301272, Example 6/35	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392037	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392037&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185693	404960377							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783480	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C23H29Cl2N3O5S3/c1-23(2,3)28-36(32,33)17-7-6-15(18(24)19(17)25)20-16(12-13-4-5-13)27-22(34-20)21(29)26-14-8-10-35(30,31)11-9-14/h6-7,13-14,28H,4-5,8-12H2,1-3H3,(H,26,29)	UPJFBEIADODBQT-UHFFFAOYSA-N	392037	US10301272, Example 6/35	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 31.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392037	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392037&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185693	404960377							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783481	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O6S2/c1-27(2,3)33-41(37,38)20-10-9-18(21(29)22(20)30)23-19(15-17-7-5-4-6-8-17)32-25(40-23)24(34)31-16-28(26(35)36)11-13-39-14-12-28/h9-10,17,33H,4-8,11-16H2,1-3H3,(H,31,34)(H,35,36)	PWOMHCYFSGEXHS-UHFFFAOYSA-N	392038	US10301272, Example 6/36	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392038	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392038&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185694	404960378							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783482	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O6S2/c1-27(2,3)33-41(37,38)20-10-9-18(21(29)22(20)30)23-19(15-17-7-5-4-6-8-17)32-25(40-23)24(34)31-16-28(26(35)36)11-13-39-14-12-28/h9-10,17,33H,4-8,11-16H2,1-3H3,(H,31,34)(H,35,36)	PWOMHCYFSGEXHS-UHFFFAOYSA-N	392038	US10301272, Example 6/36	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392038	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392038&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185694	404960378							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783483	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2(CCOCC2)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O6S2/c1-27(2,3)33-41(37,38)20-10-9-18(21(29)22(20)30)23-19(15-17-7-5-4-6-8-17)32-25(40-23)24(34)31-16-28(26(35)36)11-13-39-14-12-28/h9-10,17,33H,4-8,11-16H2,1-3H3,(H,31,34)(H,35,36)	PWOMHCYFSGEXHS-UHFFFAOYSA-N	392038	US10301272, Example 6/36	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392038	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392038&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185694	404960378							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783484	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S2/c1-27(2,3)32-40(37,38)20-12-11-18(21(29)22(20)30)23-19(13-16-9-7-6-8-10-16)31-24(39-23)25(34)33-14-17(15-33)28(4,5)26(35)36/h11-12,16-17,32H,6-10,13-15H2,1-5H3,(H,35,36)	FNUUJCQFXVCCGI-UHFFFAOYSA-N	392039	US10301272, Example 6/37	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 794							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392039	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392039&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185695	404960379							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783485	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S2/c1-27(2,3)32-40(37,38)20-12-11-18(21(29)22(20)30)23-19(13-16-9-7-6-8-10-16)31-24(39-23)25(34)33-14-17(15-33)28(4,5)26(35)36/h11-12,16-17,32H,6-10,13-15H2,1-5H3,(H,35,36)	FNUUJCQFXVCCGI-UHFFFAOYSA-N	392039	US10301272, Example 6/37	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392039	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392039&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185695	404960379							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783486	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S2/c1-27(2,3)32-40(37,38)20-12-11-18(21(29)22(20)30)23-19(13-16-9-7-6-8-10-16)31-24(39-23)25(34)33-14-17(15-33)28(4,5)26(35)36/h11-12,16-17,32H,6-10,13-15H2,1-5H3,(H,35,36)	FNUUJCQFXVCCGI-UHFFFAOYSA-N	392039	US10301272, Example 6/37	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392039	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392039&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185695	404960379							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783487	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H33Cl2N3O5S2/c1-25(2,3)32-39(36,37)18-10-9-16(19(28)20(18)29)21-17(11-15-7-5-4-6-8-15)30-23(38-21)22(33)31-27-12-26(13-27,14-27)24(34)35/h9-10,15,32H,4-8,11-14H2,1-3H3,(H,31,33)(H,34,35)	GLQIFPZQCUOUJN-UHFFFAOYSA-N	392040	US10301272, Example 6/38	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392040&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185698	404960380							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783488	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H33Cl2N3O5S2/c1-25(2,3)32-39(36,37)18-10-9-16(19(28)20(18)29)21-17(11-15-7-5-4-6-8-15)30-23(38-21)22(33)31-27-12-26(13-27,14-27)24(34)35/h9-10,15,32H,4-8,11-14H2,1-3H3,(H,31,33)(H,34,35)	GLQIFPZQCUOUJN-UHFFFAOYSA-N	392040	US10301272, Example 6/38	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392040&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185698	404960380							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783489	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H33Cl2N3O5S2/c1-25(2,3)32-39(36,37)18-10-9-16(19(28)20(18)29)21-17(11-15-7-5-4-6-8-15)30-23(38-21)22(33)31-27-12-26(13-27,14-27)24(34)35/h9-10,15,32H,4-8,11-14H2,1-3H3,(H,31,33)(H,34,35)	GLQIFPZQCUOUJN-UHFFFAOYSA-N	392040	US10301272, Example 6/38	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392040&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185698	404960380							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783490	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCC(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H37Cl2N3O5S2/c1-26(2,3)32-39(36,37)19-12-11-17(20(28)21(19)29)22-18(15-16-9-7-6-8-10-16)31-24(38-22)23(33)30-14-13-27(4,5)25(34)35/h11-12,16,32H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)	BWTHTTXTYXYDOH-UHFFFAOYSA-N	392041	US10301272, Example 6/39	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 398							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392041	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392041&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185696	404960381							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783491	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCC(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H37Cl2N3O5S2/c1-26(2,3)32-39(36,37)19-12-11-17(20(28)21(19)29)22-18(15-16-9-7-6-8-10-16)31-24(38-22)23(33)30-14-13-27(4,5)25(34)35/h11-12,16,32H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)	BWTHTTXTYXYDOH-UHFFFAOYSA-N	392041	US10301272, Example 6/39	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392041	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392041&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185696	404960381							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783492	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCC(C)(C)C(O)=O)c(Cl)c1Cl	InChI=1S/C27H37Cl2N3O5S2/c1-26(2,3)32-39(36,37)19-12-11-17(20(28)21(19)29)22-18(15-16-9-7-6-8-10-16)31-24(38-22)23(33)30-14-13-27(4,5)25(34)35/h11-12,16,32H,6-10,13-15H2,1-5H3,(H,30,33)(H,34,35)	BWTHTTXTYXYDOH-UHFFFAOYSA-N	392041	US10301272, Example 6/39	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392041	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392041&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185696	404960381							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783493	CSc1cnc(CNC(=O)c2nc(CC3CCCCC3)c(s2)-c2ccc(c(Cl)c2Cl)S(=O)(=O)NC(C)(C)C)s1	InChI=1S/C26H32Cl2N4O3S4/c1-26(2,3)32-39(34,35)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(38-23)24(33)30-13-19-29-14-20(36-4)37-19/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	HOIWGLVXZBZKHZ-UHFFFAOYSA-N	392042	US10301272, Example 6/40	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392042	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392042&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185697	404960382							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783494	CSc1cnc(CNC(=O)c2nc(CC3CCCCC3)c(s2)-c2ccc(c(Cl)c2Cl)S(=O)(=O)NC(C)(C)C)s1	InChI=1S/C26H32Cl2N4O3S4/c1-26(2,3)32-39(34,35)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(38-23)24(33)30-13-19-29-14-20(36-4)37-19/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	HOIWGLVXZBZKHZ-UHFFFAOYSA-N	392042	US10301272, Example 6/40	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392042	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392042&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185697	404960382							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783495	CSc1cnc(CNC(=O)c2nc(CC3CCCCC3)c(s2)-c2ccc(c(Cl)c2Cl)S(=O)(=O)NC(C)(C)C)s1	InChI=1S/C26H32Cl2N4O3S4/c1-26(2,3)32-39(34,35)18-11-10-16(21(27)22(18)28)23-17(12-15-8-6-5-7-9-15)31-25(38-23)24(33)30-13-19-29-14-20(36-4)37-19/h10-11,14-15,32H,5-9,12-13H2,1-4H3,(H,30,33)	HOIWGLVXZBZKHZ-UHFFFAOYSA-N	392042	US10301272, Example 6/40	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 5.01							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392042	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392042&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185697	404960382							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783496	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17-	JWFDDUGOOFHYGO-QAQDUYKDSA-N	392043	US10301272, Example 6/41	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392043&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960383							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783497	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17-	JWFDDUGOOFHYGO-QAQDUYKDSA-N	392043	US10301272, Example 6/41	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392043&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960383							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783498	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17-	JWFDDUGOOFHYGO-QAQDUYKDSA-N	392043	US10301272, Example 6/41	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392043	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392043&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960383							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783499	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17+	JWFDDUGOOFHYGO-CALCHBBNSA-N	392044	US10301272, Example 6/42	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 63.1							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392044	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392044&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960384							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783500	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17+	JWFDDUGOOFHYGO-CALCHBBNSA-N	392044	US10301272, Example 6/42	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392044	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392044&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960384							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783501	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@H](C2)S(C)(=O)=O)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-11-10-18(21(27)22(20)28)23-19(12-15-8-6-5-7-9-15)30-25(37-23)24(32)29-16-13-17(14-16)38(4,33)34/h10-11,15-17,31H,5-9,12-14H2,1-4H3,(H,29,32)/t16-,17+	JWFDDUGOOFHYGO-CALCHBBNSA-N	392044	US10301272, Example 6/42	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392044	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392044&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185699	404960384							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783502	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	RBANJZJLQVFHEW-UHFFFAOYSA-N	392045	US10301272, Example 6/43	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 100							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392045	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392045&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185700	404960385							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783503	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	RBANJZJLQVFHEW-UHFFFAOYSA-N	392045	US10301272, Example 6/43	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392045	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392045&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185700	404960385							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783504	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl	InChI=1S/C26H35Cl2N3O5S3/c1-26(2,3)31-39(35,36)20-10-9-18(21(27)22(20)28)23-19(15-16-7-5-4-6-8-16)30-25(37-23)24(32)29-17-11-13-38(33,34)14-12-17/h9-10,16-17,31H,4-8,11-15H2,1-3H3,(H,29,32)	RBANJZJLQVFHEW-UHFFFAOYSA-N	392045	US10301272, Example 6/43	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392045	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392045&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185700	404960385							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783505	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3CC(C2)O3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-26(2,3)30-37(33,34)20-10-9-18(21(27)22(20)28)23-19(11-15-7-5-4-6-8-15)29-24(36-23)25(32)31-13-16-12-17(14-31)35-16/h9-10,15-17,30H,4-8,11-14H2,1-3H3	CCMNCDGKGPSCDM-UHFFFAOYSA-N	392046	US10301272, Example 6/44	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392046	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392046&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185701	404960386							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783506	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3CC(C2)O3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-26(2,3)30-37(33,34)20-10-9-18(21(27)22(20)28)23-19(11-15-7-5-4-6-8-15)29-24(36-23)25(32)31-13-16-12-17(14-31)35-16/h9-10,15-17,30H,4-8,11-14H2,1-3H3	CCMNCDGKGPSCDM-UHFFFAOYSA-N	392046	US10301272, Example 6/44	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392046	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392046&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185701	404960386							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783507	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3CC(C2)O3)c(Cl)c1Cl	InChI=1S/C26H33Cl2N3O4S2/c1-26(2,3)30-37(33,34)20-10-9-18(21(27)22(20)28)23-19(11-15-7-5-4-6-8-15)29-24(36-23)25(32)31-13-16-12-17(14-31)35-16/h9-10,15-17,30H,4-8,11-14H2,1-3H3	CCMNCDGKGPSCDM-UHFFFAOYSA-N	392046	US10301272, Example 6/44	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392046	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392046&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185701	404960386							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783508	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S3/c1-27(2,3)32-41(37,38)21-10-9-19(22(29)23(21)30)24-20(15-18-7-5-4-6-8-18)31-25(39-24)26(34)33-16-28(17-33)11-13-40(35,36)14-12-28/h9-10,18,32H,4-8,11-17H2,1-3H3	GGFVCJNGULAGCR-UHFFFAOYSA-N	392047	US10301272, Example 6/45	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392047	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392047&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185702	404960387							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783509	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S3/c1-27(2,3)32-41(37,38)21-10-9-19(22(29)23(21)30)24-20(15-18-7-5-4-6-8-18)31-25(39-24)26(34)33-16-28(17-33)11-13-40(35,36)14-12-28/h9-10,18,32H,4-8,11-17H2,1-3H3	GGFVCJNGULAGCR-UHFFFAOYSA-N	392047	US10301272, Example 6/45	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392047	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392047&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185702	404960387							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783510	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c(Cl)c1Cl	InChI=1S/C28H37Cl2N3O5S3/c1-27(2,3)32-41(37,38)21-10-9-19(22(29)23(21)30)24-20(15-18-7-5-4-6-8-18)31-25(39-24)26(34)33-16-28(17-33)11-13-40(35,36)14-12-28/h9-10,18,32H,4-8,11-17H2,1-3H3	GGFVCJNGULAGCR-UHFFFAOYSA-N	392047	US10301272, Example 6/45	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392047	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392047&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185702	404960387							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783511	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12	InChI=1S/C30H37N3O5S3/c1-29(2,3)32-41(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-20-9-5-4-6-10-20)31-27(39-26)28(34)33-16-30(17-33)18-40(35,36)19-30/h7-8,11-14,20,32H,4-6,9-10,15-19H2,1-3H3	SYEFCMYUCXUVNI-UHFFFAOYSA-N	392048	US10301272, Example 6/46	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392048	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392048&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185703	404960388							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783512	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12	InChI=1S/C30H37N3O5S3/c1-29(2,3)32-41(37,38)25-14-13-23(21-11-7-8-12-22(21)25)26-24(15-20-9-5-4-6-10-20)31-27(39-26)28(34)33-16-30(17-33)18-40(35,36)19-30/h7-8,11-14,20,32H,4-6,9-10,15-19H2,1-3H3	SYEFCMYUCXUVNI-UHFFFAOYSA-N	392048	US10301272, Example 6/46	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392048	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392048&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185703	404960388							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783513	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12)C(F)(F)F	InChI=1S/C26H26F3N3O5S3/c1-15(26(27,28)29)31-40(36,37)21-9-8-19(17-4-2-3-5-18(17)21)22-20(10-16-6-7-16)30-23(38-22)24(33)32-11-25(12-32)13-39(34,35)14-25/h2-5,8-9,15-16,31H,6-7,10-14H2,1H3/t15-/m0/s1	XSWHFQATHCLWSZ-HNNXBMFYSA-N	392049	US10301272, Example 6/47	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392049&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185704	404960389							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783514	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12)C(F)(F)F	InChI=1S/C26H26F3N3O5S3/c1-15(26(27,28)29)31-40(36,37)21-9-8-19(17-4-2-3-5-18(17)21)22-20(10-16-6-7-16)30-23(38-22)24(33)32-11-25(12-32)13-39(34,35)14-25/h2-5,8-9,15-16,31H,6-7,10-14H2,1H3/t15-/m0/s1	XSWHFQATHCLWSZ-HNNXBMFYSA-N	392049	US10301272, Example 6/47	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392049	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392049&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185704	404960389							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783515	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C25H28F3N3O4S2/c1-14(25(26,27)28)31-37(34,35)20-11-10-18(16-6-4-5-7-17(16)20)21-19(12-15-8-9-15)30-23(36-21)22(32)29-13-24(2,3)33/h4-7,10-11,14-15,31,33H,8-9,12-13H2,1-3H3,(H,29,32)/t14-/m0/s1	NAHXYUDPBBTKMC-AWEZNQCLSA-N	392050	US10301272, Example 6/48	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392050	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392050&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185705	404960390							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783516	C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F	InChI=1S/C25H28F3N3O4S2/c1-14(25(26,27)28)31-37(34,35)20-11-10-18(16-6-4-5-7-17(16)20)21-19(12-15-8-9-15)30-23(36-21)22(32)29-13-24(2,3)33/h4-7,10-11,14-15,31,33H,8-9,12-13H2,1-3H3,(H,29,32)/t14-/m0/s1	NAHXYUDPBBTKMC-AWEZNQCLSA-N	392050	US10301272, Example 6/48	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392050	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392050&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185705	404960390							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783517	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C)(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-30(2,3)33-41(38,39)25-15-14-23(21-12-8-9-13-22(21)25)26-24(18-20-10-6-5-7-11-20)32-27(40-26)28(35)34-17-16-31(4,19-34)29(36)37/h8-9,12-15,20,33H,5-7,10-11,16-19H2,1-4H3,(H,36,37)	LQIMYRLGJBRBMG-UHFFFAOYSA-N	392051	US10301272, Example 6/49	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 1995							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392051	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392051&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185706	404960391							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783518	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C)(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-30(2,3)33-41(38,39)25-15-14-23(21-12-8-9-13-22(21)25)26-24(18-20-10-6-5-7-11-20)32-27(40-26)28(35)34-17-16-31(4,19-34)29(36)37/h8-9,12-15,20,33H,5-7,10-11,16-19H2,1-4H3,(H,36,37)	LQIMYRLGJBRBMG-UHFFFAOYSA-N	392051	US10301272, Example 6/49	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 50.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392051	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392051&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185706	404960391							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783519	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C)(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-30(2,3)33-41(38,39)25-15-14-23(21-12-8-9-13-22(21)25)26-24(18-20-10-6-5-7-11-20)32-27(40-26)28(35)34-17-16-31(4,19-34)29(36)37/h8-9,12-15,20,33H,5-7,10-11,16-19H2,1-4H3,(H,36,37)	LQIMYRLGJBRBMG-UHFFFAOYSA-N	392051	US10301272, Example 6/49	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392051	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392051&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185706	404960391							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783520	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C2)C(C)(C)C(O)=O)c2ccccc12	InChI=1S/C33H43N3O5S2/c1-32(2,3)35-43(40,41)27-16-15-25(23-13-9-10-14-24(23)27)28-26(19-21-11-7-6-8-12-21)34-29(42-28)30(37)36-18-17-22(20-36)33(4,5)31(38)39/h9-10,13-16,21-22,35H,6-8,11-12,17-20H2,1-5H3,(H,38,39)	MDFYDUGRDXHQPC-UHFFFAOYSA-N	392052	US10301272, Example 6/50	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392052	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392052&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185707	404960392							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783521	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C2)C(C)(C)C(O)=O)c2ccccc12	InChI=1S/C33H43N3O5S2/c1-32(2,3)35-43(40,41)27-16-15-25(23-13-9-10-14-24(23)27)28-26(19-21-11-7-6-8-12-21)34-29(42-28)30(37)36-18-17-22(20-36)33(4,5)31(38)39/h9-10,13-16,21-22,35H,6-8,11-12,17-20H2,1-5H3,(H,38,39)	MDFYDUGRDXHQPC-UHFFFAOYSA-N	392052	US10301272, Example 6/50	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 20.0							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392052	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392052&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185707	404960392							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783522	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-31(2,3)34-41(38,39)26-16-15-24(22-11-7-8-12-23(22)26)27-25(17-19-9-5-4-6-10-19)33-29(40-27)28(35)32-21-14-13-20(18-21)30(36)37/h7-8,11-12,15-16,19-21,34H,4-6,9-10,13-14,17-18H2,1-3H3,(H,32,35)(H,36,37)	COSPBQHASPZXJY-UHFFFAOYSA-N	392053	US10301272, Example 6/51	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392053&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185708	404960393							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783523	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-31(2,3)34-41(38,39)26-16-15-24(22-11-7-8-12-23(22)26)27-25(17-19-9-5-4-6-10-19)33-29(40-27)28(35)32-21-14-13-20(18-21)30(36)37/h7-8,11-12,15-16,19-21,34H,4-6,9-10,13-14,17-18H2,1-3H3,(H,32,35)(H,36,37)	COSPBQHASPZXJY-UHFFFAOYSA-N	392053	US10301272, Example 6/51	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392053&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185708	404960393							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783524	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCC(C2)C(O)=O)c2ccccc12	InChI=1S/C31H39N3O5S2/c1-31(2,3)34-41(38,39)26-16-15-24(22-11-7-8-12-23(22)26)27-25(17-19-9-5-4-6-10-19)33-29(40-27)28(35)32-21-14-13-20(18-21)30(36)37/h7-8,11-12,15-16,19-21,34H,4-6,9-10,13-14,17-18H2,1-3H3,(H,32,35)(H,36,37)	COSPBQHASPZXJY-UHFFFAOYSA-N	392053	US10301272, Example 6/51	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.98							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392053	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392053&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185708	404960393							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783525	CN(C1CCOCC1)C(=O)c1nc(CC2CCCCC2)c(s1)-c1cc(cc(c1)C1(C)CC1)C(C)(C)C	InChI=1S/C31H44N2O2S/c1-30(2,3)23-18-22(19-24(20-23)31(4)13-14-31)27-26(17-21-9-7-6-8-10-21)32-28(36-27)29(34)33(5)25-11-15-35-16-12-25/h18-21,25H,6-17H2,1-5H3	AIXYUBRRRIHHSZ-UHFFFAOYSA-N	392054	US10301272, Example 6/52	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392054	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392054&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185709	404960394							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783526	CN(C1CCOCC1)C(=O)c1nc(CC2CCCCC2)c(s1)-c1cc(cc(c1)C1(C)CC1)C(C)(C)C	InChI=1S/C31H44N2O2S/c1-30(2,3)23-18-22(19-24(20-23)31(4)13-14-31)27-26(17-21-9-7-6-8-10-21)32-28(36-27)29(34)33(5)25-11-15-35-16-12-25/h18-21,25H,6-17H2,1-5H3	AIXYUBRRRIHHSZ-UHFFFAOYSA-N	392054	US10301272, Example 6/52	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392054	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392054&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185709	404960394							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783527	CN1CCN(CC1)C(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C30H40N4O3S2/c1-30(2,3)32-39(36,37)26-15-14-24(22-12-8-9-13-23(22)26)27-25(20-21-10-6-5-7-11-21)31-28(38-27)29(35)34-18-16-33(4)17-19-34/h8-9,12-15,21,32H,5-7,10-11,16-20H2,1-4H3	SSFKUUBSBMRIIT-UHFFFAOYSA-N	392055	US10301272, Example 6/53	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 251							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392055	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392055&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185710	404960395							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783528	CN1CCN(CC1)C(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C30H40N4O3S2/c1-30(2,3)32-39(36,37)26-15-14-24(22-12-8-9-13-23(22)26)27-25(20-21-10-6-5-7-11-21)31-28(38-27)29(35)34-18-16-33(4)17-19-34/h8-9,12-15,21,32H,5-7,10-11,16-20H2,1-4H3	SSFKUUBSBMRIIT-UHFFFAOYSA-N	392055	US10301272, Example 6/53	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 79.4							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392055	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392055&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185710	404960395							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783529	CN1CCN(CC1)C(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C	InChI=1S/C30H40N4O3S2/c1-30(2,3)32-39(36,37)26-15-14-24(22-12-8-9-13-23(22)26)27-25(20-21-10-6-5-7-11-21)31-28(38-27)29(35)34-18-16-33(4)17-19-34/h8-9,12-15,21,32H,5-7,10-11,16-20H2,1-4H3	SSFKUUBSBMRIIT-UHFFFAOYSA-N	392055	US10301272, Example 6/53	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 39.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392055	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392055&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185710	404960395							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783530	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCN(CC(C)(C)O)CC2)c2ccccc12	InChI=1S/C33H46N4O4S2/c1-32(2,3)35-43(40,41)28-16-15-26(24-13-9-10-14-25(24)28)29-27(21-23-11-7-6-8-12-23)34-30(42-29)31(38)37-19-17-36(18-20-37)22-33(4,5)39/h9-10,13-16,23,35,39H,6-8,11-12,17-22H2,1-5H3	KRJFOZLLWPVOIY-UHFFFAOYSA-N	392056	US10301272, Example 6/54	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 501							US Patent		10.7270/Q2S184TJ		aid1798888	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392056&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185711	404960396							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783531	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCN(CC(C)(C)O)CC2)c2ccccc12	InChI=1S/C33H46N4O4S2/c1-32(2,3)35-43(40,41)28-16-15-26(24-13-9-10-14-25(24)28)29-27(21-23-11-7-6-8-12-23)34-30(42-29)31(38)37-19-17-36(18-20-37)22-33(4,5)39/h9-10,13-16,23,35,39H,6-8,11-12,17-22H2,1-5H3	KRJFOZLLWPVOIY-UHFFFAOYSA-N	392056	US10301272, Example 6/54	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 158							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392056&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185711	404960396							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783532	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCN(CC(C)(C)O)CC2)c2ccccc12	InChI=1S/C33H46N4O4S2/c1-32(2,3)35-43(40,41)28-16-15-26(24-13-9-10-14-25(24)28)29-27(21-23-11-7-6-8-12-23)34-30(42-29)31(38)37-19-17-36(18-20-37)22-33(4,5)39/h9-10,13-16,23,35,39H,6-8,11-12,17-22H2,1-5H3	KRJFOZLLWPVOIY-UHFFFAOYSA-N	392056	US10301272, Example 6/54	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 126							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392056	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392056&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185711	404960396							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783533	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)31-40(36,37)25-14-13-23(21-11-7-8-12-22(21)25)26-24(19-20-9-5-4-6-10-20)30-27(38-26)28(33)32-15-17-39(34,35)18-16-32/h7-8,11-14,20,31H,4-6,9-10,15-19H2,1-3H3	NUOKMVUGNRMHGT-UHFFFAOYSA-N	392057	US10301272, Example 6/55	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 10.0							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392057	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392057&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188708	404960397							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783534	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCS(=O)(=O)CC2)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)31-40(36,37)25-14-13-23(21-11-7-8-12-22(21)25)26-24(19-20-9-5-4-6-10-20)30-27(38-26)28(33)32-15-17-39(34,35)18-16-32/h7-8,11-14,20,31H,4-6,9-10,15-19H2,1-3H3	NUOKMVUGNRMHGT-UHFFFAOYSA-N	392057	US10301272, Example 6/55	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392057	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392057&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118188708	404960397							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783535	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(CC2)S(C)(=O)=O)c2ccccc12	InChI=1S/C31H41N3O5S3/c1-31(2,3)33-42(38,39)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)32-29(40-28)30(35)34-18-16-22(17-19-34)41(4,36)37/h8-9,12-15,21-22,33H,5-7,10-11,16-20H2,1-4H3	MBNLGTPKDOLUJS-UHFFFAOYSA-N	392058	US10301272, Example 6/56	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 7.94							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392058	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392058&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185713	404960398							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783536	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(CC2)S(C)(=O)=O)c2ccccc12	InChI=1S/C31H41N3O5S3/c1-31(2,3)33-42(38,39)27-15-14-25(23-12-8-9-13-24(23)27)28-26(20-21-10-6-5-7-11-21)32-29(40-28)30(35)34-18-16-22(17-19-34)41(4,36)37/h8-9,12-15,21-22,33H,5-7,10-11,16-20H2,1-4H3	MBNLGTPKDOLUJS-UHFFFAOYSA-N	392058	US10301272, Example 6/56	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392058	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392058&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185713	404960398							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783537	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)S(C)(=O)=O)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)31-40(36,37)25-15-14-23(21-12-8-9-13-22(21)25)26-24(16-19-10-6-5-7-11-19)30-27(38-26)28(33)32-17-20(18-32)39(4,34)35/h8-9,12-15,19-20,31H,5-7,10-11,16-18H2,1-4H3	ANPOLCKPTIBCPT-UHFFFAOYSA-N	392059	US10301272, Example 6/57	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 12.6							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392059	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392059&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185714	404960399							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783538	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)S(C)(=O)=O)c2ccccc12	InChI=1S/C29H37N3O5S3/c1-29(2,3)31-40(36,37)25-15-14-23(21-12-8-9-13-22(21)25)26-24(16-19-10-6-5-7-11-19)30-27(38-26)28(33)32-17-20(18-32)39(4,34)35/h8-9,12-15,19-20,31H,5-7,10-11,16-18H2,1-4H3	ANPOLCKPTIBCPT-UHFFFAOYSA-N	392059	US10301272, Example 6/57	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 6.31							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392059	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392059&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			118185714	404960399							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783539	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)C#N)c2ccccc12	InChI=1S/C30H38N4O3S2/c1-29(2,3)34-39(36,37)25-16-15-23(21-13-9-10-14-22(21)25)26-24(17-20-11-7-6-8-12-20)33-28(38-26)27(35)32-19-30(4,5)18-31/h9-10,13-16,20,34H,6-8,11-12,17,19H2,1-5H3,(H,32,35)	IAWSXSVJTHDIPU-UHFFFAOYSA-N	392060	US10301272, Example 6/58	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392060&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549189	404960400							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783540	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)C#N)c2ccccc12	InChI=1S/C30H38N4O3S2/c1-29(2,3)34-39(36,37)25-16-15-23(21-13-9-10-14-22(21)25)26-24(17-20-11-7-6-8-12-20)33-28(38-26)27(35)32-19-30(4,5)18-31/h9-10,13-16,20,34H,6-8,11-12,17,19H2,1-5H3,(H,32,35)	IAWSXSVJTHDIPU-UHFFFAOYSA-N	392060	US10301272, Example 6/58	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 2.00							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392060	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392060&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549189	404960400							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783541	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)c2nn[nH]n2)c2ccccc12	InChI=1S/C30H39N7O3S2/c1-29(2,3)35-42(39,40)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)32-27(41-25)26(38)31-18-30(4,5)28-33-36-37-34-28/h9-10,13-16,19,35H,6-8,11-12,17-18H2,1-5H3,(H,31,38)(H,33,34,36,37)	JPUPUUKSMVXNRM-UHFFFAOYSA-N	392061	US10301272, Example 6/59	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 25.1							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392061	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392061&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549187	404960401							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783542	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)c2nn[nH]n2)c2ccccc12	InChI=1S/C30H39N7O3S2/c1-29(2,3)35-42(39,40)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)32-27(41-25)26(38)31-18-30(4,5)28-33-36-37-34-28/h9-10,13-16,19,35H,6-8,11-12,17-18H2,1-5H3,(H,31,38)(H,33,34,36,37)	JPUPUUKSMVXNRM-UHFFFAOYSA-N	392061	US10301272, Example 6/59	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 15.8							US Patent		10.7270/Q2S184TJ		aid1798890	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392061	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392061&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			72549187	404960401							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
783543	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)c2noc(=O)[nH]2)c2ccccc12	InChI=1S/C31H39N5O5S2/c1-30(2,3)36-43(39,40)24-16-15-22(20-13-9-10-14-21(20)24)25-23(17-19-11-7-6-8-12-19)33-27(42-25)26(37)32-18-31(4,5)28-34-29(38)41-35-28/h9-10,13-16,19,36H,6-8,11-12,17-18H2,1-5H3,(H,32,37)(H,34,35,38)	IYVGXWZGZUPAGF-UHFFFAOYSA-N	392062	US10301272, Example 6/60	Isoform 2 of Nuclear receptor ROR-gamma (RORgT)			 3.16							US Patent		10.7270/Q2S184TJ		aid1798889	US10301272	Gege, C; Steeneck, C; Kinzel, O; Kleymann, G; Hoffmann, T	Phenex Pharmaceuticals AG	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=392062	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=673&target=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=392062&enzyme=Isoform+2+of+Nuclear+receptor+ROR-gamma+%28RORgT%29&column=ki&startPg=0&Increment=50&submit=Search			146012228	404960402							1	MRTQIEVIPCKICGDKSSGIHYGVITCEGCKGFFRRSQRCNAAYSCTRQQNCPIDRTSRNRCQHCRLQKCLALGMSRDAVKFGRMSKKQRDSLHAEVQKQLQQRQQQQQEPVVKTPPAGAQGADTLTYTLGLPDGQLPLGSSPDLPEASACPPGLLKASGSGPSYSNNLAKAGLNGASCHLEYSPERGKAEGRESFYSTGSQLTPDRCGLRFEEHRHPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAAFPPLYKELFSTETESPVGLSK	3B0W,3KYT,3L0J,3L0L,4NB6,4QM0,4S14,4WLB,4WPF,4WQP,4XT9,4YPQ,4ZJR,4ZJW,4ZOM,5APH,5APJ,5APK,5AYG,5EJV,5ETH,5G42,5G43,5G44,5G45,5G46,5K38,5K3L,5K3M,5K3N,5K6E,5K74,5LWP,5NI5,5NI7,5NI8,5NIB,5UFO,5UFR,5UHI,5W4R,5X8S,5X8U,5YP5,5YP6,5ZA1,6B30,6B31,6B33,6BN6,6BR2,6BR3,6CN5,6CVH,6E3E,6E3G,6ESN,6FGQ,6J3N,6NAD,6NWS,6NWT,6NWU,6O98,6P9F,6Q2W,6R7A,6R7J,6R7K,6SAL,6SLZ,6T4G,6T4I,6T4J,6T4K,6T4X,6T4Y,6T50,6TLM,6TLQ,6TLT,6U25,6VQF,6VSW,6W9H,6W9I,6XAE,6XFV,7E3M,7JH2,7JTM,7JYM,7KCO,7KQJ,7KXD,7KXE,7KXF,7LUK,7NEC,7NP5,7NP6,7OFI,7OFK,7QP4,7W3P,7W3Q,8GXP	Nuclear receptor ROR-gamma	RORG_HUMAN	P51449	Q5SZR9 Q8N5V7 Q8NCY8						
