BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID of Ligand	PubChem SID of Ligand	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence	PDB ID(s) of Target Chain	UniProt (SwissProt) Recommended Name of Target Chain	UniProt (SwissProt) Entry Name of Target Chain	UniProt (SwissProt) Primary ID of Target Chain	UniProt (SwissProt) Secondary ID(s) of Target Chain	UniProt (SwissProt) Alternative ID(s) of Target Chain	UniProt (TrEMBL) Submitted Name of Target Chain	UniProt (TrEMBL) Entry Name of Target Chain	UniProt (TrEMBL) Primary ID of Target Chain	UniProt (TrEMBL) Secondary ID(s) of Target Chain	UniProt (TrEMBL) Alternative ID(s) of Target Chain
460919	COc1cc(ccc1Nc1ccc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C32H39N7O3/c1-35-17-19-38(20-18-35)23-13-15-39(16-14-23)31(40)22-9-10-25(28(21-22)42-4)33-29-12-11-27-30(34-29)36(2)26-8-6-5-7-24(26)32(41)37(27)3/h5-12,21,23H,13-20H2,1-4H3,(H,33,34)	SZURENOYVUBGEB-UHFFFAOYSA-N	106150	US9695172, 3	Bromodomain testis-specific protein	Homo sapiens		 3683					7.5	25.00 C	US Patent		10.7270/Q2JD4TX8		aid1794893	US9695172	Bradner, JE; Gray, NS; Qi, J; McKeown, MR; Buckley, D	Dana-Farber Cancer Institute Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=106150	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=106150&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			91826712	174008461						ZINC96177071	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
460922	COc1cc(ccc1Nc1ccc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C28H32N6O3/c1-32-15-13-19(14-16-32)29-27(35)18-9-10-21(24(17-18)37-4)30-25-12-11-23-26(31-25)33(2)22-8-6-5-7-20(22)28(36)34(23)3/h5-12,17,19H,13-16H2,1-4H3,(H,29,35)(H,30,31)	BUWDXYNETOQBNF-UHFFFAOYSA-N	106153	US9695172, 2-227	Bromodomain testis-specific protein	Homo sapiens		 5410					7.5	25.00 C	US Patent		10.7270/Q2JD4TX8		aid1794893	US9695172	Bradner, JE; Gray, NS; Qi, J; McKeown, MR; Buckley, D	Dana-Farber Cancer Institute Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=106153	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=106153&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			118284116	174008464						ZINC96177074	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
460925	CN1c2ccccc2C(=O)N(C)c2ccc(Nc3ccc(cc3)S(N)(=O)=O)nc12	InChI=1S/C20H19N5O3S/c1-24-16-6-4-3-5-15(16)20(26)25(2)17-11-12-18(23-19(17)24)22-13-7-9-14(10-8-13)29(21,27)28/h3-12H,1-2H3,(H,22,23)(H2,21,27,28)	RCVIFGTXCWQDHC-UHFFFAOYSA-N	106152	US9695172, 2-221	Bromodomain testis-specific protein	Homo sapiens		 5660					7.5	25.00 C	US Patent		10.7270/Q2JD4TX8		aid1794893	US9695172	Bradner, JE; Gray, NS; Qi, J; McKeown, MR; Buckley, D	Dana-Farber Cancer Institute Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=106152	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=106152&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			118279322	174008463						ZINC96177073	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
460930	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 147					7.5	25.00 C	US Patent		10.7270/Q2JD4TX8		aid1794893	US9695172	Bradner, JE; Gray, NS; Qi, J; McKeown, MR; Buckley, D	Dana-Farber Cancer Institute Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
460932	C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F	InChI=1S/C27H28F3N5O2S/c1-17(19-5-3-4-6-20(19)27(28,29)30)37-23-14-24(38-25(23)26(31)36)35-16-32-21-8-7-18(13-22(21)35)15-34-11-9-33(2)10-12-34/h3-8,13-14,16-17H,9-12,15H2,1-2H3,(H2,31,36)/t17-/m1/s1	ZHJGWYRLJUCMRT-QGZVFWFLSA-N	50355500	CHEMBL1908394::US9695172, GSK461364	Bromodomain testis-specific protein	Homo sapiens		>50000					7.5	25.00 C	US Patent		10.7270/Q2JD4TX8		aid1794893	US9695172	Bradner, JE; Gray, NS; Qi, J; McKeown, MR; Buckley, D	Dana-Farber Cancer Institute Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50355500	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50355500&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			15983966	136959524		CHEMBL1908394				ZINC43154472	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50238812	C[C@H]1C[C@@H](Nc2ccc(Cl)cc2)c2cc(ccc2N1C(C)=O)-c1ccc(cc1)C(O)=O	InChI=1S/C25H23ClN2O3/c1-15-13-23(27-21-10-8-20(26)9-11-21)22-14-19(7-12-24(22)28(15)16(2)29)17-3-5-18(6-4-17)25(30)31/h3-12,14-15,23,27H,13H2,1-2H3,(H,30,31)/t15-,23+/m0/s1	FAWSUKOIROHXAP-NPMXOYFQSA-N	50028142	CHEMBL2177300	Bromodomain testis-specific protein	Homo sapiens		 31623							ChEMBL	10.1021/jm5010539	10.7270/Q23R0VGR	25249180			Gosmini, R; Nguyen, VL; Toum, J; Simon, C; Brusq, JM; Krysa, G; Mirguet, O; Riou-Eymard, AM; Boursier, EV; Trottet, L; Bamborough, P; Clark, H; Chung, CW; Cutler, L; Demont, EH; Kaur, R; Lewis, AJ; Schilling, MB; Soden, PE; Taylor, S; Walker, AL; Walker, MD; Prinjha, RK; Nicodème, E	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50028142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50028142&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	73B	4BJX,7AMC,4UYF,4UYG	52912222	103937511		CHEMBL2177300				ZINC27554150	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50238813	C[C@H]1C[C@@H](Nc2ccc(Cl)cc2)c2cc(ccc2N1C(C)=O)-c1ccc(cc1)C(O)=O	InChI=1S/C25H23ClN2O3/c1-15-13-23(27-21-10-8-20(26)9-11-21)22-14-19(7-12-24(22)28(15)16(2)29)17-3-5-18(6-4-17)25(30)31/h3-12,14-15,23,27H,13H2,1-2H3,(H,30,31)/t15-,23+/m0/s1	FAWSUKOIROHXAP-NPMXOYFQSA-N	50028142	CHEMBL2177300	Bromodomain testis-specific protein	Homo sapiens		 31623							ChEMBL	10.1021/jm5010539	10.7270/Q23R0VGR	25249180			Gosmini, R; Nguyen, VL; Toum, J; Simon, C; Brusq, JM; Krysa, G; Mirguet, O; Riou-Eymard, AM; Boursier, EV; Trottet, L; Bamborough, P; Clark, H; Chung, CW; Cutler, L; Demont, EH; Kaur, R; Lewis, AJ; Schilling, MB; Soden, PE; Taylor, S; Walker, AL; Walker, MD; Prinjha, RK; Nicodème, E	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50028142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50028142&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	73B	4BJX,7AMC,4UYF,4UYG	52912222	103937511		CHEMBL2177300				ZINC27554150	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50238842	C[C@H]1C[C@@H](Nc2ccc(Cl)cc2)c2cc(ccc2N1C(C)=O)-c1ccc(cc1)C(O)=O	InChI=1S/C25H23ClN2O3/c1-15-13-23(27-21-10-8-20(26)9-11-21)22-14-19(7-12-24(22)28(15)16(2)29)17-3-5-18(6-4-17)25(30)31/h3-12,14-15,23,27H,13H2,1-2H3,(H,30,31)/t15-,23+/m0/s1	FAWSUKOIROHXAP-NPMXOYFQSA-N	50028142	CHEMBL2177300	Bromodomain testis-specific protein	Homo sapiens		 50							ChEMBL	10.1021/jm5010539	10.7270/Q23R0VGR	25249180			Gosmini, R; Nguyen, VL; Toum, J; Simon, C; Brusq, JM; Krysa, G; Mirguet, O; Riou-Eymard, AM; Boursier, EV; Trottet, L; Bamborough, P; Clark, H; Chung, CW; Cutler, L; Demont, EH; Kaur, R; Lewis, AJ; Schilling, MB; Soden, PE; Taylor, S; Walker, AL; Walker, MD; Prinjha, RK; Nicodème, E	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50028142	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50028142&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	73B	4BJX,7AMC,4UYF,4UYG	52912222	103937511		CHEMBL2177300				ZINC27554150	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50323590	CCOC(=O)Nc1cc(nn2c(C)nnc12)-c1ccc(C)c(NS(C)(=O)=O)c1	InChI=1S/C17H20N6O4S/c1-5-27-17(24)18-15-9-14(21-23-11(3)19-20-16(15)23)12-7-6-10(2)13(8-12)22-28(4,25)26/h6-9,22H,5H2,1-4H3,(H,18,24)	UYBRROMMFMPJAN-UHFFFAOYSA-N	50504160	CHEMBL3133807	Bromodomain testis-specific protein	Homo sapiens			 40						ChEMBL		10.7270/Q24J0JPZ	27757418			Picaud, S; Leonards, K; Lambert, JP; Dovey, O; Wells, C; Fedorov, O; Monteiro, O; Fujisawa, T; Wang, CY; Lingard, H; Tallant, C; Nikbin, N; Guetzoyan, L; Ingham, R; Ley, SV; Brennan, P; Muller, S; Samsonova, A; Gingras, AC; Schwaller, J; Vassiliou, G; Knapp, S; Filippakopoulos, P	University of Oxford	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50504160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50504160&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	BMF	7LEL,5IGK,5FEA,5IGM,5IGL,7K1P,7LAH,5C7N,7LB4,5TCK,5U9N,7L6D,6V1H,5C4Q,5CZG,6NIM,6V0U	72943187	440712745							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50323591	CCOC(=O)Nc1cc(nn2c(C)nnc12)-c1ccc(C)c(NS(C)(=O)=O)c1	InChI=1S/C17H20N6O4S/c1-5-27-17(24)18-15-9-14(21-23-11(3)19-20-16(15)23)12-7-6-10(2)13(8-12)22-28(4,25)26/h6-9,22H,5H2,1-4H3,(H,18,24)	UYBRROMMFMPJAN-UHFFFAOYSA-N	50504160	CHEMBL3133807	Bromodomain testis-specific protein	Homo sapiens			 172						ChEMBL		10.7270/Q24J0JPZ	27757418			Picaud, S; Leonards, K; Lambert, JP; Dovey, O; Wells, C; Fedorov, O; Monteiro, O; Fujisawa, T; Wang, CY; Lingard, H; Tallant, C; Nikbin, N; Guetzoyan, L; Ingham, R; Ley, SV; Brennan, P; Muller, S; Samsonova, A; Gingras, AC; Schwaller, J; Vassiliou, G; Knapp, S; Filippakopoulos, P	University of Oxford	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50504160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50504160&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	BMF	7LEL,5IGK,5FEA,5IGM,5IGL,7K1P,7LAH,5C7N,7LB4,5TCK,5U9N,7L6D,6V1H,5C4Q,5CZG,6NIM,6V0U	72943187	440712745							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50358746	Cc1cncc(c1)-c1cnc(NC2CCNCC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C20H23N5O/c1-12-7-14(10-22-9-12)17-11-23-19(24-15-3-5-21-6-4-15)18-16(17)8-13(2)20(26)25-18/h7-11,15,21H,3-6H2,1-2H3,(H,23,24)(H,25,26)	PAGDGWOISBNVEC-UHFFFAOYSA-N	50096300	CHEMBL3585452	Bromodomain testis-specific protein	Homo sapiens		 7943							ChEMBL	10.1021/acs.jmedchem.5b00772	10.7270/Q2PR7XQN	26155854			Demont, EH; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Wellaway, C; Barrett, N; Bridges, AM; Craggs, PD; Diallo, H; Dixon, DP; Douault, C; Emmons, AJ; Jones, EJ; Karamshi, BV; Locke, K; Mitchell, DJ; Mouzon, BH; Prinjha, RK; Roberts, AD; Sheppard, RJ; Watson, RJ; Bamborough, P	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50096300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50096300&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			91827383	103993853		CHEMBL3585452				ZINC96299856	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50358761	COc1cncc(c1)-c1cnc(NC2CCNCC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C15H12N3O6P/c19-12(20)4-7-2-1-3-8-9(7)5-10-13(8)17-15(21)14-16-11(6-18(10)14)25(22,23)24/h1-3,6H,4-5H2,(H,17,21)(H,19,20)(H2,22,23,24)	UGRPUAQGGXFABK-UHFFFAOYSA-N	50096282	CHEMBL3585455	Bromodomain testis-specific protein	Homo sapiens		 6310							ChEMBL	10.1021/acs.jmedchem.5b00772	10.7270/Q2PR7XQN	26155854			Demont, EH; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Wellaway, C; Barrett, N; Bridges, AM; Craggs, PD; Diallo, H; Dixon, DP; Douault, C; Emmons, AJ; Jones, EJ; Karamshi, BV; Locke, K; Mitchell, DJ; Mouzon, BH; Prinjha, RK; Roberts, AD; Sheppard, RJ; Watson, RJ; Bamborough, P	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50096282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50096282&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	NP8	5A5S,5A5R	91820725	103993835		CHEMBL3585455				ZINC01909478	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50351593	Cc1cncc(c1)-c1cnc(NC2CCNCC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C20H23N5O/c1-12-7-14(10-22-9-12)17-11-23-19(24-15-3-5-21-6-4-15)18-16(17)8-13(2)20(26)25-18/h7-11,15,21H,3-6H2,1-2H3,(H,23,24)(H,25,26)	PAGDGWOISBNVEC-UHFFFAOYSA-N	50096300	CHEMBL3585452	Bromodomain testis-specific protein	Homo sapiens		 31623							ChEMBL	10.1021/acs.jmedchem.5b00772	10.7270/Q2PR7XQN	26155854			Demont, EH; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Wellaway, C; Barrett, N; Bridges, AM; Craggs, PD; Diallo, H; Dixon, DP; Douault, C; Emmons, AJ; Jones, EJ; Karamshi, BV; Locke, K; Mitchell, DJ; Mouzon, BH; Prinjha, RK; Roberts, AD; Sheppard, RJ; Watson, RJ; Bamborough, P	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50096300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50096300&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			91827383	103993853		CHEMBL3585452				ZINC96299856	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50351596	COc1cncc(c1)-c1cnc(NC2CCNCC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C15H12N3O6P/c19-12(20)4-7-2-1-3-8-9(7)5-10-13(8)17-15(21)14-16-11(6-18(10)14)25(22,23)24/h1-3,6H,4-5H2,(H,17,21)(H,19,20)(H2,22,23,24)	UGRPUAQGGXFABK-UHFFFAOYSA-N	50096282	CHEMBL3585455	Bromodomain testis-specific protein	Homo sapiens		 25119							ChEMBL	10.1021/acs.jmedchem.5b00772	10.7270/Q2PR7XQN	26155854			Demont, EH; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Wellaway, C; Barrett, N; Bridges, AM; Craggs, PD; Diallo, H; Dixon, DP; Douault, C; Emmons, AJ; Jones, EJ; Karamshi, BV; Locke, K; Mitchell, DJ; Mouzon, BH; Prinjha, RK; Roberts, AD; Sheppard, RJ; Watson, RJ; Bamborough, P	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50096282	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50096282&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	NP8	5A5S,5A5R	91820725	103993835		CHEMBL3585455				ZINC01909478	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50365514	CN1CC[C@@H](Nc2ncc(-c3cncc(C)c3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)OCC1CCS(=O)(=O)CC1			50098311	CHEMBL3590408	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.5b00773	10.7270/Q2FN17Z1	26230603			Bamborough, P; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Sheppard, RJ; Barnett, H; Diallo, H; Dixon, DP; Douault, C; Jones, EJ; Karamshi, B; Mitchell, DJ; Prinjha, RK; Rau, C; Watson, RJ; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50098311	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50098311&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			122363061	318490405		CHEMBL3590408					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50365523	Cc1cncc(c1)-c1cnc(N[C@@H]2CCNC[C@H]2OCC2CCS(=O)(=O)CC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C26H29NO/c1-4-22(19-21-11-7-5-8-12-21)26(23-13-9-6-10-14-23)24-15-17-25(18-16-24)28-20-27(2)3/h5-18H,4,19-20H2,1-3H3/b26-22-	FMHQDBFMJHNCPF-ROMGYVFFSA-N	50098301	CHEMBL3590383	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.5b00773	10.7270/Q2FN17Z1	26230603			Bamborough, P; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Sheppard, RJ; Barnett, H; Diallo, H; Dixon, DP; Douault, C; Jones, EJ; Karamshi, B; Mitchell, DJ; Prinjha, RK; Rau, C; Watson, RJ; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50098301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50098301&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YD4	6VEO	122181550	103995392		CHEMBL3590383				ZINC26017551	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50365524	CN1CC[C@@H](Nc2ncc(-c3cncc(C)c3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)OCC1CCS(=O)(=O)CC1			50098311	CHEMBL3590408	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.5b00773	10.7270/Q2FN17Z1	26230603			Bamborough, P; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Sheppard, RJ; Barnett, H; Diallo, H; Dixon, DP; Douault, C; Jones, EJ; Karamshi, B; Mitchell, DJ; Prinjha, RK; Rau, C; Watson, RJ; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50098311	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50098311&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			122363061	318490405		CHEMBL3590408					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50365491	Cc1cncc(c1)-c1ccc(N[C@@H]2CCNC[C@H]2OCC2CCS(=O)(=O)CC2)c2[nH]c(=O)c(C)cc12			50098305	CHEMBL3590405	Bromodomain testis-specific protein	Homo sapiens			 1995						ChEMBL	10.1021/acs.jmedchem.5b00773	10.7270/Q2FN17Z1	26230603			Bamborough, P; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Sheppard, RJ; Barnett, H; Diallo, H; Dixon, DP; Douault, C; Jones, EJ; Karamshi, B; Mitchell, DJ; Prinjha, RK; Rau, C; Watson, RJ; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50098305	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50098305&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YD3	5A83	122363056	318490400		CHEMBL3590405					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50365513	Cc1cncc(c1)-c1cnc(N[C@@H]2CCNC[C@H]2OCC2CCS(=O)(=O)CC2)c2[nH]c(=O)c(C)cc12	InChI=1S/C26H29NO/c1-4-22(19-21-11-7-5-8-12-21)26(23-13-9-6-10-14-23)24-15-17-25(18-16-24)28-20-27(2)3/h5-18H,4,19-20H2,1-3H3/b26-22-	FMHQDBFMJHNCPF-ROMGYVFFSA-N	50098301	CHEMBL3590383	Bromodomain testis-specific protein	Homo sapiens		 31623							ChEMBL	10.1021/acs.jmedchem.5b00773	10.7270/Q2FN17Z1	26230603			Bamborough, P; Chung, CW; Furze, RC; Grandi, P; Michon, AM; Sheppard, RJ; Barnett, H; Diallo, H; Dixon, DP; Douault, C; Jones, EJ; Karamshi, B; Mitchell, DJ; Prinjha, RK; Rau, C; Watson, RJ; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50098301	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50098301&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YD4	6VEO	122181550	103995392		CHEMBL3590383				ZINC26017551	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50473039	CCn1cnc2n(Cc3ccc(Cl)cc3)c(=O)[nH]c(=O)c12	InChI=1S/C14H13ClN4O2/c1-2-18-8-16-12-11(18)13(20)17-14(21)19(12)7-9-3-5-10(15)6-4-9/h3-6,8H,2,7H2,1H3,(H,17,20,21)	ZUHFEYWVQFKDLX-UHFFFAOYSA-N	50150754	CHEMBL3775058	Bromodomain testis-specific protein	Homo sapiens		 2300							ChEMBL	10.1021/acs.jmedchem.5b01708	10.7270/Q21N830R	26735842			Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X	Centre National de la Recherche Scientifique (CNRS)	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50150754	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50150754&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5OU	5EIS	44396137	104039113		CHEMBL3775058				ZINC34800503	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50473042	CCCCn1c2ncn(CC)c2c(=O)[nH]c1=O	InChI=1S/C11H16N4O2/c1-3-5-6-15-9-8(10(16)13-11(15)17)14(4-2)7-12-9/h7H,3-6H2,1-2H3,(H,13,16,17)	MJFNWOLXWYRXQS-UHFFFAOYSA-N	50150755	CHEMBL3775270	Bromodomain testis-specific protein	Homo sapiens		 7900							ChEMBL	10.1021/acs.jmedchem.5b01708	10.7270/Q21N830R	26735842			Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X	Centre National de la Recherche Scientifique (CNRS)	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50150755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50150755&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			11201422	104039114		CHEMBL3775270					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50473046	CCn1c(CSc2n[nH]c(N)n2)nc2n(Cc3ccc(Cl)cc3)c(=O)[nH]c(=O)c12	InChI=1S/C17H17ClN8O2S/c1-2-25-11(8-29-16-22-15(19)23-24-16)20-13-12(25)14(27)21-17(28)26(13)7-9-3-5-10(18)6-4-9/h3-6H,2,7-8H2,1H3,(H,21,27,28)(H3,19,22,23,24)	HZXIXZPCCYPTDC-UHFFFAOYSA-N	50150752	CHEMBL3774900	Bromodomain testis-specific protein	Homo sapiens		>100000							ChEMBL	10.1021/acs.jmedchem.5b01708	10.7270/Q21N830R	26735842			Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X	Centre National de la Recherche Scientifique (CNRS)	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50150752	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50150752&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44396207	104039111		CHEMBL3774900				ZINC34800501	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50472564	CCCCc1c(C)nc2nc(SCc3nc4n(CCCC)c(=O)[nH]c(=O)c4n3CC)nn2c1C	InChI=1S/C23H32N8O2S/c1-6-9-11-16-14(4)24-21-27-22(28-31(21)15(16)5)34-13-17-25-19-18(29(17)8-3)20(32)26-23(33)30(19)12-10-7-2/h6-13H2,1-5H3,(H,26,32,33)	FTDVJTZJKKOHSY-UHFFFAOYSA-N	50150069	CHEMBL3774931	Bromodomain testis-specific protein	Homo sapiens		 100000							ChEMBL	10.1021/acs.jmedchem.5b01708	10.7270/Q21N830R	26735842			Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X	Centre National de la Recherche Scientifique (CNRS)	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50150069	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50150069&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5NQ	5EGU	44393203	104038602		CHEMBL3774931				ZINC28362738	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50720742	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 190.1						ChEMBL	10.1016/j.bmc.2012.01.018	10.7270/Q2TX3FTN	22316554			Sasaki, K; Ito, A; Yoshida, M	Japan Science and Technology Agency	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552330	Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H36N6O3S/c1-20-19-28-26(30-21-10-12-23(13-11-21)36-17-16-33-14-5-6-15-33)31-25(20)29-22-8-7-9-24(18-22)37(34,35)32-27(2,3)4/h7-13,18-19,32H,5-6,14-17H2,1-4H3,(H2,28,29,30,31)	JOOXLOJCABQBSG-UHFFFAOYSA-N	50332294	CHEMBL1287853::N-tert-butyl-3-(5-methyl-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)pyrimidin-4-ylamino)benzenesulfonamide::US10112907, Example 00018::US10730860, TABLE 1.3::US10766894, Compound TABLE 1.3::US11203595, TABLE 1.3::US11384069, Example T-5	Bromodomain testis-specific protein	Homo sapiens		 340							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50332294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50332294&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2TA	4OGJ,4PS5,6VNE	16722836	123111409		CHEMBL1287853		5716		ZINC19862646	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552348	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(c3)S(=O)(=O)NC(C)(C)C)n2)cc1	InChI=1S/C26H35N7O2S/c1-19-18-27-25(29-20-9-11-22(12-10-20)33-15-13-32(5)14-16-33)30-24(19)28-21-7-6-8-23(17-21)36(34,35)31-26(2,3)4/h6-12,17-18,31H,13-16H2,1-5H3,(H2,27,28,29,30)	JVDOKQYTTYUYDV-UHFFFAOYSA-N	192755	TG101209::US11279703, TABLE 6.171::US11643396, Example TG101209	Bromodomain testis-specific protein	Homo sapiens		 230							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=192755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=192755&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1M3	5HEZ,4O76,4JI9	16722832	317230231							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552353	Cc1nnc2C(CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3	DNVXATUJJDPFDM-UHFFFAOYSA-N	50210164	CHEMBL2132936	Bromodomain testis-specific protein	Homo sapiens		 110							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50210164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50210164&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			49871817	375982585		CHEMBL2132936					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552360	CCc1cnn2c(NCc3ccc[n+]([O-])c3)cc(nc12)N1CCCC[C@H]1CCO	InChI=1S/C21H28N6O2/c1-2-17-14-23-27-19(22-13-16-6-5-9-25(29)15-16)12-20(24-21(17)27)26-10-4-3-7-18(26)8-11-28/h5-6,9,12,14-15,18,22,28H,2-4,7-8,10-11,13H2,1H3/t18-/m0/s1	PIMQWRZWLQKKBJ-SFHVURJKSA-N	50139171	Dinaciclib::MK-7965::SCH-727965::US11643396, Example Dinaciclib	Bromodomain testis-specific protein	Homo sapiens		 37000							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50139171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50139171&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46926350	336952252							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552361	O=c1cc(oc2c(cccc12)-c1cccc2c3ccccc3sc12)N1CCOCC1	InChI=1S/C25H19NO3S/c27-21-15-23(26-11-13-28-14-12-26)29-24-17(6-3-9-20(21)24)19-8-4-7-18-16-5-1-2-10-22(16)30-25(18)19/h1-10,15H,11-14H2	JAMULYFATHSZJM-UHFFFAOYSA-N	50156495	8-(dibenzo[b,d]thiophen-4-yl)-2-morpholino-4H-chromen-4-one::8-Dibenzothiophen-4-yl-2-morpholin-4-yl-chromen-4-one::8-dibenzothiophen-1-yl-2-morpholin-4-yl-chromen-4-one::CHEMBL188678::NU-7432::NU-7441	Bromodomain testis-specific protein	Homo sapiens		 3500							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50156495	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50156495&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2R4	7OTM,4O72	11327430	104043621		CHEMBL188678				ZINC03938693	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552369	Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1	InChI=1S/C20H14FN3O/c21-16-5-1-13(2-6-16)18-19(14-9-11-22-12-10-14)24-20(23-18)15-3-7-17(25)8-4-15/h1-12,25H,(H,23,24)	QHKYPYXTTXKZST-UHFFFAOYSA-N	50044784	CHEBI:79090::SB-202190::US10865384, Compound SB202190	Bromodomain testis-specific protein	Homo sapiens		 20000							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044784	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044784&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RE	4O77	5353940	313068337							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50552512	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m1/s1	XQVVPGYIWAGRNI-JOCHJYFZSA-N	25121	4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide::BI 2536::CHEMBL513909::US10450297, Example 300::US8598172, 5	Bromodomain testis-specific protein	Homo sapiens		 260							ChEMBL	10.1038/nrd.2016.266	10.7270/Q2125VNC	28280261			Munoz, L	The University of Sydney	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=25121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=25121&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	R78	4OGI,6MF9,6BQQ,7K0U,2RKU,6CW0,7LAI,4O74,4PY6,4I5M,5TCM,5C8G,5VBQ,7L9G,7L9L,7N7M	11364421	56374263		CHEMBL513909		5666		ZINC13986815	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50759581	CCS(=O)(=O)Nc1ccc(Oc2ccc(F)cc2F)c(c1)-c1cn(C)c(=O)c2[nH]ccc12	InChI=1S/C22H19F2N3O4S/c1-3-32(29,30)26-14-5-7-19(31-20-6-4-13(23)10-18(20)24)16(11-14)17-12-27(2)22(28)21-15(17)8-9-25-21/h4-12,25-26H,3H2,1-2H3	RDONXGFGWSSFMY-UHFFFAOYSA-N	220447	US10633379, Compound X::US9296741, 36	Bromodomain testis-specific protein	Homo sapiens	 2.2								ChEMBL	10.1021/acs.jmedchem.7b00746	10.7270/Q2251MB8	28949521			McDaniel, KF; Wang, L; Soltwedel, T; Fidanze, SD; Hasvold, LA; Liu, D; Mantei, RA; Pratt, JK; Sheppard, GS; Bui, MH; Faivre, EJ; Huang, X; Li, L; Lin, X; Wang, R; Warder, SE; Wilcox, D; Albert, DH; Magoc, TJ; Rajaraman, G; Park, CH; Hutchins, CW; Shen, JJ; Edalji, RP; Sun, CC; Martin, R; Gao, W; Wong, S; Fang, G; Elmore, SW; Shen, Y; Kati, WM	AbbVie Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=220447	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=220447&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	8NG	5UVW	71600087	329995460							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751197	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H17N3O4/c1-3-21-15-14(16(22)20-18(21)24)12(10-6-4-9(2)5-7-10)13-11(19-15)8-25-17(13)23/h4-7,12,19H,3,8H2,1-2H3,(H,20,22,24)	MUOCQMZJLRQTRD-UHFFFAOYSA-N	50239562	CHEMBL4104179	Bromodomain testis-specific protein	Homo sapiens	 690								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239562&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	6RX	5KDH	44448830	85715051		CHEMBL4104179					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751198	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H17N3O4/c1-3-21-15-14(16(22)20-18(21)24)12(10-6-4-9(2)5-7-10)13-11(19-15)8-25-17(13)23/h4-7,12,19H,3,8H2,1-2H3,(H,20,22,24)	MUOCQMZJLRQTRD-UHFFFAOYSA-N	50239562	CHEMBL4104179	Bromodomain testis-specific protein	Homo sapiens		 5200							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239562&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	6RX	5KDH	44448830	85715051		CHEMBL4104179					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751200	CCn1c(N)cc(=O)[nH]c1=O	InChI=1S/C6H9N3O2/c1-2-9-4(7)3-5(10)8-6(9)11/h3H,2,7H2,1H3,(H,8,10,11)	QHEMDIZENXAVRQ-UHFFFAOYSA-N	50239563	CHEMBL4095390	Bromodomain testis-specific protein	Homo sapiens			 1500000						ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239563	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239563&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448868	85715099		CHEMBL4095390					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751201	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccc(O)cc1)C3	InChI=1S/C26H26N4O4/c1-3-30-23-22(24(32)28-26(30)34)20(17-8-4-15(2)5-9-17)21-19(27-23)14-29(25(21)33)13-12-16-6-10-18(31)11-7-16/h4-11,20,27,31H,3,12-14H2,1-2H3,(H,28,32,34)	VLSYQVCLFAZVNI-UHFFFAOYSA-N	50239567	CHEMBL4085204	Bromodomain testis-specific protein	Homo sapiens	 200								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239567	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239567&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448911	85715159		CHEMBL4085204					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751202	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CC=C)C3	InChI=1S/C21H22N4O3/c1-4-10-24-11-14-16(20(24)27)15(13-8-6-12(3)7-9-13)17-18(22-14)25(5-2)21(28)23-19(17)26/h4,6-9,15,22H,1,5,10-11H2,2-3H3,(H,23,26,28)	SGYUNIXZZZQROD-UHFFFAOYSA-N	50239564	CHEMBL4089152	Bromodomain testis-specific protein	Homo sapiens		 2200							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239564	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239564&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448871	85715102		CHEMBL4089152					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751203	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(Cc1ccccc1)C3	InChI=1S/C25H24N4O3/c1-3-29-22-21(23(30)27-25(29)32)19(17-11-9-15(2)10-12-17)20-18(26-22)14-28(24(20)31)13-16-7-5-4-6-8-16/h4-12,19,26H,3,13-14H2,1-2H3,(H,27,30,32)	ZBRDRGVJFCJFQS-UHFFFAOYSA-N	50239565	CHEMBL4065286	Bromodomain testis-specific protein	Homo sapiens		 550							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239565	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239565&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448870	85715101		CHEMBL4065286					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751205	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccc(O)cc1)C3	InChI=1S/C26H26N4O4/c1-3-30-23-22(24(32)28-26(30)34)20(17-8-4-15(2)5-9-17)21-19(27-23)14-29(25(21)33)13-12-16-6-10-18(31)11-7-16/h4-11,20,27,31H,3,12-14H2,1-2H3,(H,28,32,34)	VLSYQVCLFAZVNI-UHFFFAOYSA-N	50239567	CHEMBL4085204	Bromodomain testis-specific protein	Homo sapiens		 760							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239567	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239567&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448911	85715159		CHEMBL4085204					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751206	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(Cc1ccccc1)C3	InChI=1S/C25H24N4O3/c1-3-29-22-21(23(30)27-25(29)32)19(17-11-9-15(2)10-12-17)20-18(26-22)14-28(24(20)31)13-16-7-5-4-6-8-16/h4-12,19,26H,3,13-14H2,1-2H3,(H,27,30,32)	ZBRDRGVJFCJFQS-UHFFFAOYSA-N	50239565	CHEMBL4065286	Bromodomain testis-specific protein	Homo sapiens	 230								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239565	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239565&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448870	85715101		CHEMBL4065286					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751208	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccc(OC)cc1)C3	InChI=1S/C27H28N4O4/c1-4-31-24-23(25(32)29-27(31)34)21(18-9-5-16(2)6-10-18)22-20(28-24)15-30(26(22)33)14-13-17-7-11-19(35-3)12-8-17/h5-12,21,28H,4,13-15H2,1-3H3,(H,29,32,34)	MWNUDTXWOMXGKW-UHFFFAOYSA-N	50239566	CHEMBL4103140	Bromodomain testis-specific protein	Homo sapiens		 1000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239566	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239566&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448909	85715157		CHEMBL4103140					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751211	CCn1c(N)cc(=O)[nH]c1=O	InChI=1S/C6H9N3O2/c1-2-9-4(7)3-5(10)8-6(9)11/h3H,2,7H2,1H3,(H,8,10,11)	QHEMDIZENXAVRQ-UHFFFAOYSA-N	50239563	CHEMBL4095390	Bromodomain testis-specific protein	Homo sapiens			 1500000						ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239563	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239563&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448868	85715099		CHEMBL4095390					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751212	COc1ccc(cc1)C1C2=C(COC2=O)Nc2c1c(=O)[nH]c(=O)n2C	InChI=1S/C17H15N3O5/c1-20-14-13(15(21)19-17(20)23)11(8-3-5-9(24-2)6-4-8)12-10(18-14)7-25-16(12)22/h3-6,11,18H,7H2,1-2H3,(H,19,21,23)	RDJWSVQIOXAMKF-UHFFFAOYSA-N	50239569	CHEMBL4086263	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239569&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448945	85715214		CHEMBL4086263					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751214	Cn1c2NC3=C(C(c4ccccc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C16H13N3O4/c1-19-13-12(14(20)18-16(19)22)10(8-5-3-2-4-6-8)11-9(17-13)7-23-15(11)21/h2-6,10,17H,7H2,1H3,(H,18,20,22)	LDRPHFMYAJCBFM-UHFFFAOYSA-N	50239570	CHEMBL4066490	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239570	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239570&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448974	85715258		CHEMBL4066490					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751216	CCCn1c2NC3=C(C(c4ccccc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H17N3O4/c1-2-8-21-15-14(16(22)20-18(21)24)12(10-6-4-3-5-7-10)13-11(19-15)9-25-17(13)23/h3-7,12,19H,2,8-9H2,1H3,(H,20,22,24)	JXTZQNJRSYNAJR-UHFFFAOYSA-N	50239571	CHEMBL4088746	Bromodomain testis-specific protein	Homo sapiens	 2400								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239571	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239571&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24959763	85715307		CHEMBL4088746					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751217	Cc1ccc(cc1)C1C2=C(COC2=O)Nc2c1c(=O)n(C)c(=O)n2C	InChI=1S/C18H17N3O4/c1-9-4-6-10(7-5-9)12-13-11(8-25-17(13)23)19-15-14(12)16(22)21(3)18(24)20(15)2/h4-7,12,19H,8H2,1-3H3	AVGOOVXJYOSRNE-UHFFFAOYSA-N	50239572	CHEMBL4060512	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239572	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239572&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24743975	85715309		CHEMBL4060512					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751218	COc1ccc(cc1)C1C2=C(COC2=O)Nc2c1c(=O)n(C)c(=O)n2C	InChI=1S/C18H17N3O5/c1-20-15-14(16(22)21(2)18(20)24)12(9-4-6-10(25-3)7-5-9)13-11(19-15)8-26-17(13)23/h4-7,12,19H,8H2,1-3H3	PWGGLSDTFYJKIA-UHFFFAOYSA-N	50239573	CHEMBL4102160	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239573	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239573&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24960497	85715350		CHEMBL4102160					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751227	CCn1c2NC3=C(C(c4ccc(cc4)C(F)(F)F)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H14F3N3O4/c1-2-24-14-13(15(25)23-17(24)27)11(12-10(22-14)7-28-16(12)26)8-3-5-9(6-4-8)18(19,20)21/h3-6,11,22H,2,7H2,1H3,(H,23,25,27)	GSQMKFKPHLJZSN-UHFFFAOYSA-N	50239574	CHEMBL4094424	Bromodomain testis-specific protein	Homo sapiens	 4700								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239574	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239574&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449026	85715352		CHEMBL4094424					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751230	Cc1ccc(cc1)C1C2=C(COC2=O)Nc2c1c(=O)[nH]c(=O)n2C1CC1	InChI=1S/C19H17N3O4/c1-9-2-4-10(5-3-9)13-14-12(8-26-18(14)24)20-16-15(13)17(23)21-19(25)22(16)11-6-7-11/h2-5,11,13,20H,6-8H2,1H3,(H,21,23,25)	ZEFGFAQVPMQFOV-UHFFFAOYSA-N	50239575	CHEMBL4066935	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239575	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239575&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24959029	85715400		CHEMBL4066935					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751233	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)CC3	InChI=1S/C19H19N3O3/c1-3-22-17-16(18(24)21-19(22)25)14(11-6-4-10(2)5-7-11)15-12(20-17)8-9-13(15)23/h4-7,14,20H,3,8-9H2,1-2H3,(H,21,24,25)	GFYQCHZFSLHBOA-UHFFFAOYSA-N	50239576	CHEMBL4093510	Bromodomain testis-specific protein	Homo sapiens	 23000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239576	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239576&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449075	85715442		CHEMBL4093510					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751235	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(C)C3	InChI=1S/C19H20N4O3/c1-4-23-16-15(17(24)21-19(23)26)13(11-7-5-10(2)6-8-11)14-12(20-16)9-22(3)18(14)25/h5-8,13,20H,4,9H2,1-3H3,(H,21,24,26)	XBNYMTXJOBYHMR-UHFFFAOYSA-N	50239577	CHEMBL4064204	Bromodomain testis-specific protein	Homo sapiens	 5600								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239577	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239577&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449077	85715445		CHEMBL4064204					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751236	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)n(C)c1=O)C(=O)OC3	InChI=1S/C19H19N3O4/c1-4-22-16-15(17(23)21(3)19(22)25)13(11-7-5-10(2)6-8-11)14-12(20-16)9-26-18(14)24/h5-8,13,20H,4,9H2,1-3H3	UVXLCDRWDGHQDE-UHFFFAOYSA-N	50239578	CHEMBL4085767	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239578	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239578&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449104	85715494		CHEMBL4085767					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751238	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccccc1)C3	InChI=1S/C26H26N4O3/c1-3-30-23-22(24(31)28-26(30)33)20(18-11-9-16(2)10-12-18)21-19(27-23)15-29(25(21)32)14-13-17-7-5-4-6-8-17/h4-12,20,27H,3,13-15H2,1-2H3,(H,28,31,33)	DQFBZYXAVHHSEQ-UHFFFAOYSA-N	50239568	CHEMBL4092949	Bromodomain testis-specific protein	Homo sapiens	 220								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239568&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448944	85715212		CHEMBL4092949					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751240	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H17N3O4/c1-3-21-15-14(16(22)20-18(21)24)12(10-6-4-9(2)5-7-10)13-11(19-15)8-25-17(13)23/h4-7,12,19H,3,8H2,1-2H3,(H,20,22,24)	MUOCQMZJLRQTRD-UHFFFAOYSA-N	50239562	CHEMBL4104179	Bromodomain testis-specific protein	Homo sapiens			 1600						ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239562&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	6RX	5KDH	44448830	85715051		CHEMBL4104179					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751241	CON\C=N\c1nc2nccc(-c3cccnc3)n2n1	InChI=1S/C12H11N7O/c1-20-16-8-15-11-17-12-14-6-4-10(19(12)18-11)9-3-2-5-13-7-9/h2-8H,1H3,(H,15,16,18)	OWJDQIQTYCDUAA-UHFFFAOYSA-N	50239579	CHEMBL4059728	Bromodomain testis-specific protein	Homo sapiens		 120000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239579	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239579&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449103	85715493		CHEMBL4059728					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751247	C\N=c1/[nH]c2n(C)c(=O)[nH]c(=O)c2n1Cc1ccc(F)cc1	InChI=1S/C14H14FN5O2/c1-16-13-17-11-10(12(21)18-14(22)19(11)2)20(13)7-8-3-5-9(15)6-4-8/h3-6H,7H2,1-2H3,(H,16,17)(H,18,21,22)	URPANXUHEDIZOO-UHFFFAOYSA-N	50239580	CHEMBL4098168	Bromodomain testis-specific protein	Homo sapiens		 68000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239580	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239580&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449129	85715533		CHEMBL4098168					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751248	O=c1[nH]c(=O)c2c(ccnc2n1CC1CCCO1)-c1ccco1	InChI=1S/C16H15N3O4/c20-15-13-11(12-4-2-8-23-12)5-6-17-14(13)19(16(21)18-15)9-10-3-1-7-22-10/h2,4-6,8,10H,1,3,7,9H2,(H,18,20,21)	OIEHAXQSKYVIJF-UHFFFAOYSA-N	50239581	CHEMBL4080143	Bromodomain testis-specific protein	Homo sapiens		 130000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239581	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239581&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449132	85715536		CHEMBL4080143					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751249	OCC\N=c1\[nH]c2[nH]c(=O)[nH]c(=O)c2n1Cc1cccc2ccccc12	InChI=1S/C18H17N5O3/c24-9-8-19-17-20-15-14(16(25)22-18(26)21-15)23(17)10-12-6-3-5-11-4-1-2-7-13(11)12/h1-7,24H,8-10H2,(H3,19,20,21,22,25,26)	GGBRAEKBAFAXFH-UHFFFAOYSA-N	50239582	CHEMBL4101588	Bromodomain testis-specific protein	Homo sapiens		 87000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239582	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239582&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449164	85715581		CHEMBL4101588					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751250	CCn1c2ccc(C=O)cc2n(CC)c1=O	InChI=1S/C12H14N2O2/c1-3-13-10-6-5-9(8-15)7-11(10)14(4-2)12(13)16/h5-8H,3-4H2,1-2H3	JZPXIWMYTZXPIF-UHFFFAOYSA-N	50239583	CHEMBL4094383	Bromodomain testis-specific protein	Homo sapiens		 140000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239583	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239583&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44449165	85715582		CHEMBL4094383					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751251	CCCN1C(c2c(C)[nH]cc2C1=O)c1cc(OC)ccc1OC	InChI=1S/C18H22N2O3/c1-5-8-20-17(16-11(2)19-10-14(16)18(20)21)13-9-12(22-3)6-7-15(13)23-4/h6-7,9-10,17,19H,5,8H2,1-4H3	CHWGBKSAEUXZHH-UHFFFAOYSA-N	50239584	CHEMBL4066897	Bromodomain testis-specific protein	Homo sapiens		 67000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239584	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239584&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			25099564	85715628		CHEMBL4066897					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751252	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m1/s1	XQVVPGYIWAGRNI-JOCHJYFZSA-N	25121	4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide::BI 2536::CHEMBL513909::US10450297, Example 300::US8598172, 5	Bromodomain testis-specific protein	Homo sapiens		 1400							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=25121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=25121&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	R78	4OGI,6MF9,6BQQ,7K0U,2RKU,6CW0,7LAI,4O74,4PY6,4I5M,5TCM,5C8G,5VBQ,7L9G,7L9L,7N7M	11364421	56374263		CHEMBL513909		5666		ZINC13986815	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751304	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccccc1)C3	InChI=1S/C26H26N4O3/c1-3-30-23-22(24(31)28-26(30)33)20(18-11-9-16(2)10-12-18)21-19(27-23)15-29(25(21)32)14-13-17-7-5-4-6-8-17/h4-12,20,27H,3,13-15H2,1-2H3,(H,28,31,33)	DQFBZYXAVHHSEQ-UHFFFAOYSA-N	50239568	CHEMBL4092949	Bromodomain testis-specific protein	Homo sapiens		 1000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239568	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239568&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448944	85715212		CHEMBL4092949					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751307	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C18H17N3O4/c1-3-21-15-14(16(22)20-18(21)24)12(10-6-4-9(2)5-7-10)13-11(19-15)8-25-17(13)23/h4-7,12,19H,3,8H2,1-2H3,(H,20,22,24)	MUOCQMZJLRQTRD-UHFFFAOYSA-N	50239562	CHEMBL4104179	Bromodomain testis-specific protein	Homo sapiens		 2300							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239562	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239562&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	6RX	5KDH	44448830	85715051		CHEMBL4104179					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751310	CCn1c2NC3=C(C(c4ccccc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C17H15N3O4/c1-2-20-14-13(15(21)19-17(20)23)11(9-6-4-3-5-7-9)12-10(18-14)8-24-16(12)22/h3-7,11,18H,2,8H2,1H3,(H,19,21,23)	WMTVHKOJALQDKD-UHFFFAOYSA-N	50239585	CHEMBL4094028	Bromodomain testis-specific protein	Homo sapiens	 1400								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239585	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239585&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24959031	85715668		CHEMBL4094028					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751311	CCn1c2NC3=C(C(c4ccc(Cl)cc4)c2c(=O)[nH]c1=O)C(=O)OC3	InChI=1S/C17H14ClN3O4/c1-2-21-14-13(15(22)20-17(21)24)11(8-3-5-9(18)6-4-8)12-10(19-14)7-25-16(12)23/h3-6,11,19H,2,7H2,1H3,(H,20,22,24)	SLWPFZUDYLJXOB-UHFFFAOYSA-N	50239588	CHEMBL4077905	Bromodomain testis-specific protein	Homo sapiens	 1100								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239588	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239588&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24958669	85715007		CHEMBL4077905					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751312	Cc1ccc(cc1)C1C2=C(COC2=O)Nc2c1c(=O)[nH]c(=O)n2CC(F)(F)F	InChI=1S/C18H14F3N3O4/c1-8-2-4-9(5-3-8)11-12-10(6-28-16(12)26)22-14-13(11)15(25)23-17(27)24(14)7-18(19,20)21/h2-5,11,22H,6-7H2,1H3,(H,23,25,27)	JNPLKPXUKXLWKV-UHFFFAOYSA-N	50239586	CHEMBL4072799	Bromodomain testis-specific protein	Homo sapiens	 850								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239586	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239586&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24959398	85715671		CHEMBL4072799					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751313	CCn1c2nc3COC(=O)c3c(-c3ccc(C)cc3)c2c(=O)[nH]c1=O	InChI=1S/C18H15N3O4/c1-3-21-15-14(16(22)20-18(21)24)12(10-6-4-9(2)5-7-10)13-11(19-15)8-25-17(13)23/h4-7H,3,8H2,1-2H3,(H,20,22,24)	XQIVSOWGERBFQG-UHFFFAOYSA-N	50239587	CHEMBL4067951	Bromodomain testis-specific protein	Homo sapiens	>40000								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239587	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239587&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			24959030	85714957		CHEMBL4067951					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751314	CCn1c2NC3=C(C(c4ccc(C)cc4)c2c(=O)[nH]c1=O)C(=O)N(CCc1ccc(OC)cc1)C3	InChI=1S/C27H28N4O4/c1-4-31-24-23(25(32)29-27(31)34)21(18-9-5-16(2)6-10-18)22-20(28-24)15-30(26(22)33)14-13-17-7-11-19(35-3)12-8-17/h5-12,21,28H,4,13-15H2,1-3H3,(H,29,32,34)	MWNUDTXWOMXGKW-UHFFFAOYSA-N	50239566	CHEMBL4103140	Bromodomain testis-specific protein	Homo sapiens	 200								ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239566	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239566&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448909	85715157		CHEMBL4103140					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751315	CN1c2ccc(Cl)cc2\C(=N/CCC1=O)c1ccc(Cl)cc1	InChI=1S/C17H14Cl2N2O/c1-21-15-7-6-13(19)10-14(15)17(20-9-8-16(21)22)11-2-4-12(18)5-3-11/h2-7,10H,8-9H2,1H3/b20-17-	RYFVPWCSBPISQS-JZJYNLBNSA-N	50239589	CHEMBL4088018	Bromodomain testis-specific protein	Homo sapiens		 220000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239589	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239589&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448803	85715008		CHEMBL4088018					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50751317	CCC1(C)Cc2ccccc2-c2ncnc(O)c12	InChI=1S/C15H16N2O/c1-3-15(2)8-10-6-4-5-7-11(10)13-12(15)14(18)17-9-16-13/h4-7,9H,3,8H2,1-2H3,(H,16,17,18)	UTJRGNCYPLAFDJ-UHFFFAOYSA-N	50239590	CHEMBL1471174	Bromodomain testis-specific protein	Homo sapiens		 220000							ChEMBL	10.1021/acs.jmedchem.6b01336	10.7270/Q2PC34JK	28535045			Ayoub, AM; Hawk, LML; Herzig, RJ; Jiang, J; Wisniewski, AJ; Gee, CT; Zhao, P; Zhu, JY; Berndt, N; Offei-Addo, NK; Scott, TG; Qi, J; Bradner, JE; Ward, TR; Schönbrunn, E; Georg, GI; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50239590	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50239590&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44448831	85715053		CHEMBL1471174					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50807131	Cc1[nH]c(c2CCNC(=O)c12)-c1cc(ccc1Oc1ccc(F)cc1F)S(C)(=O)=O	InChI=1S/C21H18F2N2O4S/c1-11-19-14(7-8-24-21(19)26)20(25-11)15-10-13(30(2,27)28)4-6-17(15)29-18-5-3-12(22)9-16(18)23/h3-6,9-10,25H,7-8H2,1-2H3,(H,24,26)	QNOJAPBYTXGBLX-UHFFFAOYSA-N	50158624	CHEMBL3786012	Bromodomain testis-specific protein	Homo sapiens	 140								ChEMBL	10.1016/j.bmcl.2017.02.057	10.7270/Q20P12FJ	28268136			Hasvold, LA; Sheppard, GS; Wang, L; Fidanze, SD; Liu, D; Pratt, JK; Mantei, RA; Wada, CK; Hubbard, R; Shen, Y; Lin, X; Huang, X; Warder, SE; Wilcox, D; Li, L; Buchanan, FG; Smithee, L; Albert, DH; Magoc, TJ; Park, CH; Petros, AM; Panchal, SC; Sun, C; Kovar, P; Soni, NB; Elmore, SW; Kati, WM; McDaniel, KF	AbbVie Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50158624	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50158624&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			77843982	104045303		CHEMBL3786012				ZINC13606819	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50807135	Cn1cc(-c2cc(ccc2Oc2ccc(F)cc2F)S(C)(=O)=O)c2cc[nH]c(=O)c12	InChI=1S/C21H16F2N2O4S/c1-25-11-16(14-7-8-24-21(26)20(14)25)15-10-13(30(2,27)28)4-6-18(15)29-19-5-3-12(22)9-17(19)23/h3-11H,1-2H3,(H,24,26)	JGGBFOUTSJEGRT-UHFFFAOYSA-N	50256397	CHEMBL4088466	Bromodomain testis-specific protein	Homo sapiens	 490								ChEMBL	10.1016/j.bmcl.2017.02.057	10.7270/Q20P12FJ	28268136			Hasvold, LA; Sheppard, GS; Wang, L; Fidanze, SD; Liu, D; Pratt, JK; Mantei, RA; Wada, CK; Hubbard, R; Shen, Y; Lin, X; Huang, X; Warder, SE; Wilcox, D; Li, L; Buchanan, FG; Smithee, L; Albert, DH; Magoc, TJ; Park, CH; Petros, AM; Panchal, SC; Sun, C; Kovar, P; Soni, NB; Elmore, SW; Kati, WM; McDaniel, KF	AbbVie Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50256397	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50256397&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			78319129	402360719							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50806892	Cc1[nH]c(c2CCCC(=O)c12)-c1cc(NS(C)(=O)=O)ccc1Oc1ccccc1	InChI=1S/C22H22N2O4S/c1-14-21-17(9-6-10-19(21)25)22(23-14)18-13-15(24-29(2,26)27)11-12-20(18)28-16-7-4-3-5-8-16/h3-5,7-8,11-13,23-24H,6,9-10H2,1-2H3	GZFJPALDEYOFHA-UHFFFAOYSA-N	342597	N-[3-(3-methyl-4-oxo-4,5,6,7-tetrahydro-2H-isoindol-1-yl)-4-phenoxyphenyl]methanesulfonamide::US9776990, Example 40	Bromodomain testis-specific protein	Homo sapiens	 110								ChEMBL	10.1016/j.bmcl.2017.02.057	10.7270/Q20P12FJ	28268136			Hasvold, LA; Sheppard, GS; Wang, L; Fidanze, SD; Liu, D; Pratt, JK; Mantei, RA; Wada, CK; Hubbard, R; Shen, Y; Lin, X; Huang, X; Warder, SE; Wilcox, D; Li, L; Buchanan, FG; Smithee, L; Albert, DH; Magoc, TJ; Park, CH; Petros, AM; Panchal, SC; Sun, C; Kovar, P; Soni, NB; Elmore, SW; Kati, WM; McDaniel, KF	AbbVie Inc	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=342597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=342597&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	87P	5UER	71760902	386048491							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50786848	CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(O)c(C)c1	InChI=1S/C18H19N3O2S/c1-9-6-11(7-10(2)15(9)22)16-19-17(23)14-12-4-5-21(3)8-13(12)24-18(14)20-16/h6-7,22H,4-5,8H2,1-3H3,(H,19,20,23)	PXJZRFLBUBYEPV-UHFFFAOYSA-N	50251045	CHEMBL4077274	Bromodomain testis-specific protein	Homo sapiens		>100000							ChEMBL	10.1021/acs.jmedchem.7b00275	10.7270/Q2M32Z68	29172540			Ouyang, L; Zhang, L; Liu, J; Fu, L; Yao, D; Zhao, Y; Zhang, S; Wang, G; He, G; Liu, B	Sichuan University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50251045	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50251045&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	4V1	4ZW1	135567026	401962583							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50786895	Cc1nnc2C(CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3	DNVXATUJJDPFDM-UHFFFAOYSA-N	50210164	CHEMBL2132936	Bromodomain testis-specific protein	Homo sapiens		 169							ChEMBL	10.1021/acs.jmedchem.7b00275	10.7270/Q2M32Z68	29172540			Ouyang, L; Zhang, L; Liu, J; Fu, L; Yao, D; Zhao, Y; Zhang, S; Wang, G; He, G; Liu, B	Sichuan University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50210164	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50210164&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			49871817	375982585		CHEMBL2132936					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096586	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C28H39N7O3/c1-18-27(37)34(3)23-17-29-28(32-25(23)35(18)21-8-6-5-7-9-21)31-22-11-10-19(16-24(22)38-4)26(36)30-20-12-14-33(2)15-13-20/h10-11,16-18,20-21H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t18-/m1/s1	IRXGEPQYGSUCML-GOSISDBHSA-N	50458967	CHEMBL4202820	Bromodomain testis-specific protein	Homo sapiens		 750							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458967	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458967&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145976012	433926232							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096587	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NC1CCCCC1	InChI=1S/C27H36N6O3/c1-17-26(35)32(2)22-16-28-27(31-24(22)33(17)20-11-7-8-12-20)30-21-14-13-18(15-23(21)36-3)25(34)29-19-9-5-4-6-10-19/h13-17,19-20H,4-12H2,1-3H3,(H,29,34)(H,28,30,31)/t17-/m1/s1	IRCDNPBWELYZBD-QGZVFWFLSA-N	50458961	CHEMBL4210414	Bromodomain testis-specific protein	Homo sapiens		 378							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458961	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458961&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145965219	433926226							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096588	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NC1=CCN(C)C=C1	InChI=1S/C27H33N7O3/c1-17-26(36)33(3)22-16-28-27(31-24(22)34(17)20-7-5-6-8-20)30-21-10-9-18(15-23(21)37-4)25(35)29-19-11-13-32(2)14-12-19/h9-13,15-17,20H,5-8,14H2,1-4H3,(H,29,35)(H,28,30,31)/t17-/m1/s1	LBXYVUXGPFEVSI-QGZVFWFLSA-N	50458968	CHEMBL4216442	Bromodomain testis-specific protein	Homo sapiens		 289							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458968	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458968&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145972360	433926233							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096589	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)N1CCCCC1	InChI=1S/C26H34N6O3/c1-17-24(33)30(2)21-16-27-26(29-23(21)32(17)19-9-5-6-10-19)28-20-12-11-18(15-22(20)35-3)25(34)31-13-7-4-8-14-31/h11-12,15-17,19H,4-10,13-14H2,1-3H3,(H,27,28,29)/t17-/m1/s1	CFTIJALKSHXVNU-QGZVFWFLSA-N	50458956	CHEMBL4202678	Bromodomain testis-specific protein	Homo sapiens		 369							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458956	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458956&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145977980	433926221							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096590	C[C@@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC3CCCC3)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C31H43N7O3/c1-20-30(40)37(3)26-19-32-31(35-28(26)38(20)23-8-4-5-9-23)34-25-13-12-21(18-27(25)41-24-10-6-7-11-24)29(39)33-22-14-16-36(2)17-15-22/h12-13,18-20,22-24H,4-11,14-17H2,1-3H3,(H,33,39)(H,32,34,35)/t20-/m0/s1	HTPNGOWITIWAHM-FQEVSTJZSA-N	50458970	CHEMBL4206381	Bromodomain testis-specific protein	Homo sapiens		 245							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458970	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458970&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145976646	433926235							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096591	COC(=O)c1ccc(Nc2ncc3N(C)C(=O)[C@@H](C)N(C4CCCC4)c3n2)c(OC2CCCC2)c1	InChI=1S/C26H33N5O4/c1-16-24(32)30(2)21-15-27-26(29-23(21)31(16)18-8-4-5-9-18)28-20-13-12-17(25(33)34-3)14-22(20)35-19-10-6-7-11-19/h12-16,18-19H,4-11H2,1-3H3,(H,27,28,29)/t16-/m1/s1	QAXOLKUTJAQVHO-MRXNPFEDSA-N	50458973	CHEMBL4212346	Bromodomain testis-specific protein	Homo sapiens		 933							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458973	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458973&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145964393	433926238							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096592	CCC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC3CCCC3)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C33H47N7O3/c1-4-9-27-32(42)39(3)28-21-34-33(37-30(28)40(27)24-10-5-6-11-24)36-26-15-14-22(20-29(26)43-25-12-7-8-13-25)31(41)35-23-16-18-38(2)19-17-23/h14-15,20-21,23-25,27H,4-13,16-19H2,1-3H3,(H,35,41)(H,34,36,37)/t27-/m1/s1	QIWKCZYPLMKZJX-HHHXNRCGSA-N	50458955	CHEMBL4209192	Bromodomain testis-specific protein	Homo sapiens		 1951							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458955	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458955&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145966579	433926220							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096593	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc3N(C)C(=O)CN(C4CCCC4)c3n2)c(OC2CCCC2)c1	InChI=1S/C30H41N7O3/c1-35-15-13-21(14-16-35)32-29(39)20-11-12-24(26(17-20)40-23-9-5-6-10-23)33-30-31-18-25-28(34-30)37(19-27(38)36(25)2)22-7-3-4-8-22/h11-12,17-18,21-23H,3-10,13-16,19H2,1-2H3,(H,32,39)(H,31,33,34)	OWPIWVDYFAZILM-UHFFFAOYSA-N	50458972	CHEMBL4205459	Bromodomain testis-specific protein	Homo sapiens		 3543							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458972	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458972&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145977109	433926237							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096529	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](CC(C)C)N(C3CCOCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C30H43N7O4/c1-19(2)16-24-29(39)36(4)25-18-31-30(34-27(25)37(24)22-10-14-41-15-11-22)33-23-7-6-20(17-26(23)40-5)28(38)32-21-8-12-35(3)13-9-21/h6-7,17-19,21-22,24H,8-16H2,1-5H3,(H,32,38)(H,31,33,34)/t24-/m1/s1	SDTDGTQRZUJKKU-XMMPIXPASA-N	50458954	CHEMBL4207347	Bromodomain testis-specific protein	Homo sapiens		>50000							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458954	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458954&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145975701	433926219							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096539	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C27H37N7O3/c1-17-26(36)33(3)22-16-28-27(31-24(22)34(17)20-7-5-6-8-20)30-21-10-9-18(15-23(21)37-4)25(35)29-19-11-13-32(2)14-12-19/h9-10,15-17,19-20H,5-8,11-14H2,1-4H3,(H,29,35)(H,28,30,31)/t17-/m1/s1	DYQPKOGFUIEBMS-QGZVFWFLSA-N	50458963	CHEMBL4209902	Bromodomain testis-specific protein	Homo sapiens		 342							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458963	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458963&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			11260691	433926228							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096540	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C(C)C)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C25H35N7O3/c1-15(2)32-16(3)24(34)31(5)20-14-26-25(29-22(20)32)28-19-8-7-17(13-21(19)35-6)23(33)27-18-9-11-30(4)12-10-18/h7-8,13-16,18H,9-12H2,1-6H3,(H,27,33)(H,26,28,29)/t16-/m1/s1	XWNHXTVCPNRSTM-MRXNPFEDSA-N	50458964	CHEMBL4206052	Bromodomain testis-specific protein	Homo sapiens		 978							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458964	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458964&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145967512	433926229							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096541	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NCCN(C)C	InChI=1S/C25H35N7O3/c1-16-24(34)31(4)20-15-27-25(29-22(20)32(16)18-8-6-7-9-18)28-19-11-10-17(14-21(19)35-5)23(33)26-12-13-30(2)3/h10-11,14-16,18H,6-9,12-13H2,1-5H3,(H,26,33)(H,27,28,29)/t16-/m1/s1	VBDIOKSSYUZONA-MRXNPFEDSA-N	50458965	CHEMBL4210571	Bromodomain testis-specific protein	Homo sapiens		 392							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458965	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458965&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145964543	433926230							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096542	C[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC3CCCC3)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C31H43N7O3/c1-20-30(40)37(3)26-19-32-31(35-28(26)38(20)23-8-4-5-9-23)34-25-13-12-21(18-27(25)41-24-10-6-7-11-24)29(39)33-22-14-16-36(2)17-15-22/h12-13,18-20,22-24H,4-11,14-17H2,1-3H3,(H,33,39)(H,32,34,35)/t20-/m1/s1	HTPNGOWITIWAHM-HXUWFJFHSA-N	50458966	CHEMBL4207437	Bromodomain testis-specific protein	Homo sapiens		 102							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458966	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458966&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145975703	433926231							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096544	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 103							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096550	COc1cc(ccc1Nc1ncc2N(C)C(=O)CN(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C26H35N7O3/c1-31-12-10-18(11-13-31)28-25(35)17-8-9-20(22(14-17)36-3)29-26-27-15-21-24(30-26)33(16-23(34)32(21)2)19-6-4-5-7-19/h8-9,14-15,18-19H,4-7,10-13,16H2,1-3H3,(H,28,35)(H,27,29,30)	BWKCRAURLKJCJQ-UHFFFAOYSA-N	50112335	CHEMBL3609304	Bromodomain testis-specific protein	Homo sapiens		 25990							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50112335	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50112335&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			122187519	319493550		CHEMBL3609304					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096551	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NC1CCNCC1	InChI=1S/C26H35N7O3/c1-16-25(35)32(2)21-15-28-26(31-23(21)33(16)19-6-4-5-7-19)30-20-9-8-17(14-22(20)36-3)24(34)29-18-10-12-27-13-11-18/h8-9,14-16,18-19,27H,4-7,10-13H2,1-3H3,(H,29,34)(H,28,30,31)/t16-/m1/s1	YGQSAYAQCWLSAL-MRXNPFEDSA-N	50458962	CHEMBL4213276	Bromodomain testis-specific protein	Homo sapiens		 560							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458962	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458962&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			11283298	433926227							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096556	CCC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C29H41N7O3/c1-5-8-23-28(38)35(3)24-18-30-29(33-26(24)36(23)21-9-6-7-10-21)32-22-12-11-19(17-25(22)39-4)27(37)31-20-13-15-34(2)16-14-20/h11-12,17-18,20-21,23H,5-10,13-16H2,1-4H3,(H,31,37)(H,30,32,33)/t23-/m1/s1	ZUJOXCIHOKDDRE-HSZRJFAPSA-N	50458951	CHEMBL4206171	Bromodomain testis-specific protein	Homo sapiens		 8468							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458951	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458951&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145975649	433926216							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096557	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@@H](C)N(C3CCCC3)c2n1)C(=O)NCCc1ccccc1	InChI=1S/C29H34N6O3/c1-19-28(37)34(2)24-18-31-29(33-26(24)35(19)22-11-7-8-12-22)32-23-14-13-21(17-25(23)38-3)27(36)30-16-15-20-9-5-4-6-10-20/h4-6,9-10,13-14,17-19,22H,7-8,11-12,15-16H2,1-3H3,(H,30,36)(H,31,32,33)/t19-/m1/s1	ITDUQSWFIDASGI-LJQANCHMSA-N	50458952	CHEMBL4203571	Bromodomain testis-specific protein	Homo sapiens		 558							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458952	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458952&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145978238	433926217							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096584	COc1cc(ccc1Nc1ncc2N(C)C(=O)[C@H](C)N(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C27H37N7O3/c1-17-26(36)33(3)22-16-28-27(31-24(22)34(17)20-7-5-6-8-20)30-21-10-9-18(15-23(21)37-4)25(35)29-19-11-13-32(2)14-12-19/h9-10,15-17,19-20H,5-8,11-14H2,1-4H3,(H,29,35)(H,28,30,31)/t17-/m0/s1	DYQPKOGFUIEBMS-KRWDZBQOSA-N	50458960	CHEMBL4216875	Bromodomain testis-specific protein	Homo sapiens		 229							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50458960	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50458960&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145972845	433926225							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51096585	CC[C@@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m0/s1	XQVVPGYIWAGRNI-QFIPXVFZSA-N	50112336	CHEMBL3609305	Bromodomain testis-specific protein	Homo sapiens		 3513							ChEMBL	10.1021/acs.jmedchem.8b00765	10.7270/Q2MP55WQ	30125504			Liu, S; Yosief, HO; Dai, L; Huang, H; Dhawan, G; Zhang, X; Muthengi, AM; Roberts, J; Buckley, DL; Perry, JA; Wu, L; Bradner, JE; Qi, J; Zhang, W	University of Massachusetts-Boston	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50112336	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50112336&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			86295201	319493551		CHEMBL3609305					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111036	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(-c3ccnc4ccccc34)c21	InChI=1S/C26H21N5O2/c1-13-23(14(2)33-31-13)19-11-21-18(12-22(19)32-4)24-25(28-15(3)29-26(24)30-21)17-9-10-27-20-8-6-5-7-16(17)20/h5-12H,1-4H3,(H,28,29,30)	AEANZCXROGPSBY-UHFFFAOYSA-N	179481	US9675697, Cpd. No. 73	Bromodomain testis-specific protein	Homo sapiens			 5.5						ChEMBL	10.1021/acs.jmedchem.7b00193	10.7270/Q28W3GWN	28463487			Zhao, Y; Bai, L; Liu, L; McEachern, D; Stuckey, JA; Meagher, JL; Yang, CY; Ran, X; Zhou, B; Hu, Y; Li, X; Wen, B; Zhao, T; Li, S; Sun, D; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=179481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=179481&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	8FV	5UOO	90395752	363893796							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111087	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(-c3ccnc4ccccc34)c21	InChI=1S/C26H21N5O2/c1-13-23(14(2)33-31-13)19-11-21-18(12-22(19)32-4)24-25(28-15(3)29-26(24)30-21)17-9-10-27-20-8-6-5-7-16(17)20/h5-12H,1-4H3,(H,28,29,30)	AEANZCXROGPSBY-UHFFFAOYSA-N	179481	US9675697, Cpd. No. 73	Bromodomain testis-specific protein	Homo sapiens			 15						ChEMBL	10.1021/acs.jmedchem.7b00193	10.7270/Q28W3GWN	28463487			Zhao, Y; Bai, L; Liu, L; McEachern, D; Stuckey, JA; Meagher, JL; Yang, CY; Ran, X; Zhou, B; Hu, Y; Li, X; Wen, B; Zhao, T; Li, S; Sun, D; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=179481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=179481&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	8FV	5UOO	90395752	363893796							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111088	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(-c3ccnc4ccccc34)c21	InChI=1S/C26H21N5O2/c1-13-23(14(2)33-31-13)19-11-21-18(12-22(19)32-4)24-25(28-15(3)29-26(24)30-21)17-9-10-27-20-8-6-5-7-16(17)20/h5-12H,1-4H3,(H,28,29,30)	AEANZCXROGPSBY-UHFFFAOYSA-N	179481	US9675697, Cpd. No. 73	Bromodomain testis-specific protein	Homo sapiens			 9.7						ChEMBL	10.1021/acs.jmedchem.7b00193	10.7270/Q28W3GWN	28463487			Zhao, Y; Bai, L; Liu, L; McEachern, D; Stuckey, JA; Meagher, JL; Yang, CY; Ran, X; Zhou, B; Hu, Y; Li, X; Wen, B; Zhao, T; Li, S; Sun, D; Wang, S	University of Michigan	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=179481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=179481&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	8FV	5UOO	90395752	363893796							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114762	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)-c1cnc(nc1)C(N)=O)C1CC1	InChI=1S/C26H27N5O3/c1-16(33)31-22-9-8-18(21-11-28-26(25(27)34)29-12-21)10-23(22)30(14-24(31)17-6-7-17)13-19-4-2-3-5-20(19)15-32/h2-5,8-12,17,24,32H,6-7,13-15H2,1H3,(H2,27,34)/t24-/m1/s1	JVAKWUYUZCOCKR-XMMPIXPASA-N	50455493	CHEMBL4213809	Bromodomain testis-specific protein	Homo sapiens		 100							ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455493	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455493&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7H	6FFF	137321203	433923585							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114764	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)C1=CCNCC1)C1CC1	InChI=1S/C26H31N3O2/c1-18(31)29-24-9-8-21(19-10-12-27-13-11-19)14-25(24)28(16-26(29)20-6-7-20)15-22-4-2-3-5-23(22)17-30/h2-5,8-10,14,20,26-27,30H,6-7,11-13,15-17H2,1H3/t26-/m1/s1	ARWMKZDWGIOCEU-AREMUKBSSA-N	50455480	CHEMBL4218735	Bromodomain testis-specific protein	Homo sapiens		 1585							ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455480&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7B	6FFG	137321204	433923572							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114783	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)C1=CCNCC1)C1CC1	InChI=1S/C26H31N3O2/c1-18(31)29-24-9-8-21(19-10-12-27-13-11-19)14-25(24)28(16-26(29)20-6-7-20)15-22-4-2-3-5-23(22)17-30/h2-5,8-10,14,20,26-27,30H,6-7,11-13,15-17H2,1H3/t26-/m1/s1	ARWMKZDWGIOCEU-AREMUKBSSA-N	50455480	CHEMBL4218735	Bromodomain testis-specific protein	Homo sapiens			 21						ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455480&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7B	6FFG	137321204	433923572							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51119049	Cn1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(c23)c1=O)c1ccc(F)cc1F	InChI=1S/C23H19F2N3O3S/c1-27-11-17-16-7-13(12-32(2,30)31)3-5-19(16)28(20-6-4-15(24)8-18(20)25)10-14-9-26-22(21(14)17)23(27)29/h3-9,11,26H,10,12H2,1-2H3	UNODBAFOZVBZBF-UHFFFAOYSA-N	50457496	CHEMBL4217457	Bromodomain testis-specific protein	Homo sapiens	 4.2								ChEMBL	10.1016/j.bmcl.2018.04.020	10.7270/Q2542R63	29678460			Fidanze, SD; Liu, D; Mantei, RA; Hasvold, LA; Pratt, JK; Sheppard, GS; Wang, L; Holms, JH; Dai, Y; Aguirre, A; Bogdan, A; Dietrich, JD; Marjanovic, J; Park, CH; Hutchins, CW; Lin, X; Bui, MH; Huang, X; Wilcox, D; Li, L; Wang, R; Kovar, P; Magoc, TJ; Rajaraman, G; Albert, DH; Shen, Y; Kati, WM; McDaniel, KF	AbbVie Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50457496	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50457496&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			86270928	433924763							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114816	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)-c1cnc(nc1)C(N)=O)C1CC1	InChI=1S/C26H27N5O3/c1-16(33)31-22-9-8-18(21-11-28-26(25(27)34)29-12-21)10-23(22)30(14-24(31)17-6-7-17)13-19-4-2-3-5-20(19)15-32/h2-5,8-12,17,24,32H,6-7,13-15H2,1H3,(H2,27,34)/t24-/m1/s1	JVAKWUYUZCOCKR-XMMPIXPASA-N	50455493	CHEMBL4213809	Bromodomain testis-specific protein	Homo sapiens		 501							ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455493	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455493&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7H	6FFF	137321203	433923585							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114819	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)C1=CCNCC1)C1CC1	InChI=1S/C26H31N3O2/c1-18(31)29-24-9-8-21(19-10-12-27-13-11-19)14-25(24)28(16-26(29)20-6-7-20)15-22-4-2-3-5-23(22)17-30/h2-5,8-10,14,20,26-27,30H,6-7,11-13,15-17H2,1H3/t26-/m1/s1	ARWMKZDWGIOCEU-AREMUKBSSA-N	50455480	CHEMBL4218735	Bromodomain testis-specific protein	Homo sapiens		 200							ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455480&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7B	6FFG	137321204	433923572							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51119092	Cn1cc2CN(c3ccc(F)cc3)c3ccc(CS(C)(=O)=O)cc3-c3c[nH]c(=O)c1c23	InChI=1S/C23H20FN3O3S/c1-26-11-15-12-27(17-6-4-16(24)5-7-17)20-8-3-14(13-31(2,29)30)9-18(20)19-10-25-23(28)22(26)21(15)19/h3-11H,12-13H2,1-2H3,(H,25,28)	QGTJNNMFLDHNQH-UHFFFAOYSA-N	50457495	CHEMBL4215988	Bromodomain testis-specific protein	Homo sapiens	 5.9								ChEMBL	10.1016/j.bmcl.2018.04.020	10.7270/Q2542R63	29678460			Fidanze, SD; Liu, D; Mantei, RA; Hasvold, LA; Pratt, JK; Sheppard, GS; Wang, L; Holms, JH; Dai, Y; Aguirre, A; Bogdan, A; Dietrich, JD; Marjanovic, J; Park, CH; Hutchins, CW; Lin, X; Bui, MH; Huang, X; Wilcox, D; Li, L; Wang, R; Kovar, P; Magoc, TJ; Rajaraman, G; Albert, DH; Shen, Y; Kati, WM; McDaniel, KF	AbbVie Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50457495	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50457495&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145972103	433924762							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51119093	Cn1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(c23)c1=O)c1ccccn1	InChI=1S/C22H20N4O3S/c1-25-12-17-16-9-14(13-30(2,28)29)6-7-18(16)26(19-5-3-4-8-23-19)11-15-10-24-21(20(15)17)22(25)27/h3-10,12,24H,11,13H2,1-2H3	LJLJARSDBHJRGG-UHFFFAOYSA-N	50457489	CHEMBL4208129	Bromodomain testis-specific protein	Homo sapiens	 0.690000								ChEMBL	10.1016/j.bmcl.2018.04.020	10.7270/Q2542R63	29678460			Fidanze, SD; Liu, D; Mantei, RA; Hasvold, LA; Pratt, JK; Sheppard, GS; Wang, L; Holms, JH; Dai, Y; Aguirre, A; Bogdan, A; Dietrich, JD; Marjanovic, J; Park, CH; Hutchins, CW; Lin, X; Bui, MH; Huang, X; Wilcox, D; Li, L; Wang, R; Kovar, P; Magoc, TJ; Rajaraman, G; Albert, DH; Shen, Y; Kati, WM; McDaniel, KF	AbbVie Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50457489	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50457489&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			78425807	433924756							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51114877	CC(=O)N1[C@H](CN(Cc2ccccc2CO)c2cc(ccc12)C1=CCNCC1)C1CC1	InChI=1S/C26H31N3O2/c1-18(31)29-24-9-8-21(19-10-12-27-13-11-19)14-25(24)28(16-26(29)20-6-7-20)15-22-4-2-3-5-23(22)17-30/h2-5,8-10,14,20,26-27,30H,6-7,11-13,15-17H2,1H3/t26-/m1/s1	ARWMKZDWGIOCEU-AREMUKBSSA-N	50455480	CHEMBL4218735	Bromodomain testis-specific protein	Homo sapiens			 1862						ChEMBL	10.1021/acs.jmedchem.7b01666	10.7270/Q27H1N6W	29656650			Law, RP; Atkinson, SJ; Bamborough, P; Chung, CW; Demont, EH; Gordon, LJ; Lindon, M; Prinjha, RK; Watson, AJB; Hirst, DJ	University of Strathclyde	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50455480	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50455480&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	D7B	6FFG	137321204	433923572							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111618	CNC(=O)c1ccc(cn1)-c1cc2cccc(-c3nn(C4CCOCC4)c4CCN(Cc34)C(C)=O)c2cn1	InChI=1S/C29H30N6O3/c1-18(36)34-11-8-27-24(17-34)28(33-35(27)21-9-12-38-13-10-21)22-5-3-4-19-14-26(32-16-23(19)22)20-6-7-25(31-15-20)29(37)30-2/h3-7,14-16,21H,8-13,17H2,1-2H3,(H,30,37)	MUJXZEDIWKGKQD-UHFFFAOYSA-N	50453949	CHEMBL4208820::US11247989, Example 87	Bromodomain testis-specific protein	Homo sapiens			 1200						ChEMBL	10.1016/j.bmcl.2017.11.025	10.7270/Q2ZG6VVZ	29169673			Lai, KW; Romero, FA; Tsui, V; Beresini, MH; de Leon Boenig, G; Bronner, SM; Chen, K; Chen, Z; Choo, EF; Crawford, TD; Cyr, P; Kaufman, S; Li, Y; Liao, J; Liu, W; Ly, J; Murray, J; Shen, W; Wai, J; Wang, F; Zhu, C; Zhu, X; Magnuson, S	WuXi AppTec Co., Ltd.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50453949	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50453949&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186469	433922358							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111619	CNC(=O)c1ccc(cn1)-c1cc2cccc(-c3nn(C4CCOCC4)c4CCN(Cc34)C(C)=O)c2cn1	InChI=1S/C29H30N6O3/c1-18(36)34-11-8-27-24(17-34)28(33-35(27)21-9-12-38-13-10-21)22-5-3-4-19-14-26(32-16-23(19)22)20-6-7-25(31-15-20)29(37)30-2/h3-7,14-16,21H,8-13,17H2,1-2H3,(H,30,37)	MUJXZEDIWKGKQD-UHFFFAOYSA-N	50453949	CHEMBL4208820::US11247989, Example 87	Bromodomain testis-specific protein	Homo sapiens			>10000						ChEMBL	10.1016/j.bmcl.2017.11.025	10.7270/Q2ZG6VVZ	29169673			Lai, KW; Romero, FA; Tsui, V; Beresini, MH; de Leon Boenig, G; Bronner, SM; Chen, K; Chen, Z; Choo, EF; Crawford, TD; Cyr, P; Kaufman, S; Li, Y; Liao, J; Liu, W; Ly, J; Murray, J; Shen, W; Wai, J; Wang, F; Zhu, C; Zhu, X; Magnuson, S	WuXi AppTec Co., Ltd.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50453949	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50453949&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186469	433922358							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51111659	CNC(=O)c1ccc(cn1)-c1cc2cccc(-c3nn(C4CCOCC4)c4CCN(Cc34)C(C)=O)c2cn1	InChI=1S/C29H30N6O3/c1-18(36)34-11-8-27-24(17-34)28(33-35(27)21-9-12-38-13-10-21)22-5-3-4-19-14-26(32-16-23(19)22)20-6-7-25(31-15-20)29(37)30-2/h3-7,14-16,21H,8-13,17H2,1-2H3,(H,30,37)	MUJXZEDIWKGKQD-UHFFFAOYSA-N	50453949	CHEMBL4208820::US11247989, Example 87	Bromodomain testis-specific protein	Homo sapiens			 3600						ChEMBL	10.1016/j.bmcl.2017.11.025	10.7270/Q2ZG6VVZ	29169673			Lai, KW; Romero, FA; Tsui, V; Beresini, MH; de Leon Boenig, G; Bronner, SM; Chen, K; Chen, Z; Choo, EF; Crawford, TD; Cyr, P; Kaufman, S; Li, Y; Liao, J; Liu, W; Ly, J; Murray, J; Shen, W; Wai, J; Wang, F; Zhu, C; Zhu, X; Magnuson, S	WuXi AppTec Co., Ltd.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50453949	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50453949&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186469	433922358							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51098429	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(Nc3cc(nn3C)C3CC3)c21	InChI=1S/C24H25N7O2/c1-11-21(12(2)33-30-11)16-8-18-15(9-19(16)32-5)22-23(27-18)25-13(3)26-24(22)28-20-10-17(14-6-7-14)29-31(20)4/h8-10,14H,6-7H2,1-5H3,(H2,25,26,27,28)	JIYPVUCBRQNICX-UHFFFAOYSA-N	50366670	CHEMBL4173488	Bromodomain testis-specific protein	Homo sapiens			 2.0						ChEMBL	10.1021/acs.jmedchem.8b00483	10.7270/Q26M39B1	30015487			Zhao, Y; Zhou, B; Bai, L; Liu, L; Yang, CY; Meagher, JL; Stuckey, JA; McEachern, D; Przybranowski, S; Wang, M; Ran, X; Aguilar, A; Hu, Y; Kampf, JW; Li, X; Zhao, T; Li, S; Wen, B; Sun, D; Wang, S	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50366670	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50366670&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	EO4	6C7R	118340554	160845772						ZINC49785250	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100015	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 217							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100022	Cc1cc(\N=N\c2ccc(cc2)S(=O)(=O)NC2CCCC2)c(N)cc1O	InChI=1S/C18H22N4O3S/c1-12-10-17(16(19)11-18(12)23)21-20-13-6-8-15(9-7-13)26(24,25)22-14-4-2-3-5-14/h6-11,14,22-23H,2-5,19H2,1H3/b21-20+	IRKMSULWLDLTIK-QZQOTICOSA-N	50370181	CHEMBL4159382::US11117865, Compound ZL0454	Bromodomain testis-specific protein	Homo sapiens		 3292							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50370181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50370181&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			137285009	160849283							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100027	Cc1cc(\N=N\c2ccc3NC(=O)CCc3c2)c(N)cc1O	InChI=1S/C16H16N4O2/c1-9-6-14(12(17)8-15(9)21)20-19-11-3-4-13-10(7-11)2-5-16(22)18-13/h3-4,6-8,21H,2,5,17H2,1H3,(H,18,22)/b20-19+	ANMQADUROYWADA-FMQUCBEESA-N	50370182	CHEMBL4176038::US11117865, Compound ZL0420	Bromodomain testis-specific protein	Homo sapiens		 2781							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50370182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50370182&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			137285011	160849284							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100056	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 183							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100057	Cc1cc(\N=N\c2ccc3NC(=O)CCc3c2)c(N)cc1O	InChI=1S/C16H16N4O2/c1-9-6-14(12(17)8-15(9)21)20-19-11-3-4-13-10(7-11)2-5-16(22)18-13/h3-4,6-8,21H,2,5,17H2,1H3,(H,18,22)/b20-19+	ANMQADUROYWADA-FMQUCBEESA-N	50370182	CHEMBL4176038::US11117865, Compound ZL0420	Bromodomain testis-specific protein	Homo sapiens		 3183							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50370182	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50370182&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			137285011	160849284							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100058	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens		 4836							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100059	Cc1cc(\N=N\c2ccc(cc2)S(=O)(=O)NC2CCCC2)c(N)cc1O	InChI=1S/C18H22N4O3S/c1-12-10-17(16(19)11-18(12)23)21-20-13-6-8-15(9-7-13)26(24,25)22-14-4-2-3-5-14/h6-11,14,22-23H,2-5,19H2,1H3/b21-20+	IRKMSULWLDLTIK-QZQOTICOSA-N	50370181	CHEMBL4159382::US11117865, Compound ZL0454	Bromodomain testis-specific protein	Homo sapiens		 3082							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50370181	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50370181&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			137285009	160849283							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51100060	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens		 708							ChEMBL	10.1016/j.ejmech.2018.04.006	10.7270/Q2X069KM	29649741			Liu, Z; Tian, B; Chen, H; Wang, P; Brasier, AR; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51098415	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(Nc3cc(nn3C)C3CC3)c21	InChI=1S/C24H25N7O2/c1-11-21(12(2)33-30-11)16-8-18-15(9-19(16)32-5)22-23(27-18)25-13(3)26-24(22)28-20-10-17(14-6-7-14)29-31(20)4/h8-10,14H,6-7H2,1-5H3,(H2,25,26,27,28)	JIYPVUCBRQNICX-UHFFFAOYSA-N	50366670	CHEMBL4173488	Bromodomain testis-specific protein	Homo sapiens			 2.1						ChEMBL	10.1021/acs.jmedchem.8b00483	10.7270/Q26M39B1	30015487			Zhao, Y; Zhou, B; Bai, L; Liu, L; Yang, CY; Meagher, JL; Stuckey, JA; McEachern, D; Przybranowski, S; Wang, M; Ran, X; Aguilar, A; Hu, Y; Kampf, JW; Li, X; Zhao, T; Li, S; Wen, B; Sun, D; Wang, S	TBA	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50366670	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50366670&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	EO4	6C7R	118340554	160845772						ZINC49785250	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51137095	CN(C)CCN1CCN(CC1)c1nc(NCc2cccc(Cl)c2)c2cc(ccc2n1)-c1ccc(=O)n(C)c1	InChI=1S/C29H34ClN7O/c1-34(2)11-12-36-13-15-37(16-14-36)29-32-26-9-7-22(23-8-10-27(38)35(3)20-23)18-25(26)28(33-29)31-19-21-5-4-6-24(30)17-21/h4-10,17-18,20H,11-16,19H2,1-3H3,(H,31,32,33)	POKZINYHLOHGEB-UHFFFAOYSA-N	50466254	CHEMBL4288569	Bromodomain testis-specific protein	Homo sapiens			 67						ChEMBL	10.1016/j.bmcl.2018.08.039	10.7270/Q28S4SKP	30268702			Yang, SM; Urban, DJ; Yoshioka, M; Strovel, JW; Fletcher, S; Wang, AQ; Xu, X; Shah, P; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50466254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50466254&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HRY	6E4A	129182189	433933519							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51137096	CN(C)CCN1CCN(CC1)c1nc(NCc2cccc(Cl)c2)c2cc(ccc2n1)-c1ccc(=O)n(C)c1	InChI=1S/C29H34ClN7O/c1-34(2)11-12-36-13-15-37(16-14-36)29-32-26-9-7-22(23-8-10-27(38)35(3)20-23)18-25(26)28(33-29)31-19-21-5-4-6-24(30)17-21/h4-10,17-18,20H,11-16,19H2,1-3H3,(H,31,32,33)	POKZINYHLOHGEB-UHFFFAOYSA-N	50466254	CHEMBL4288569	Bromodomain testis-specific protein	Homo sapiens			 160						ChEMBL	10.1016/j.bmcl.2018.08.039	10.7270/Q28S4SKP	30268702			Yang, SM; Urban, DJ; Yoshioka, M; Strovel, JW; Fletcher, S; Wang, AQ; Xu, X; Shah, P; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50466254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50466254&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HRY	6E4A	129182189	433933519							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51137144	CN(C)CCN1CCN(CC1)c1nc(NCc2cccc(Cl)c2)c2cc(ccc2n1)-c1ccc(=O)n(C)c1	InChI=1S/C29H34ClN7O/c1-34(2)11-12-36-13-15-37(16-14-36)29-32-26-9-7-22(23-8-10-27(38)35(3)20-23)18-25(26)28(33-29)31-19-21-5-4-6-24(30)17-21/h4-10,17-18,20H,11-16,19H2,1-3H3,(H,31,32,33)	POKZINYHLOHGEB-UHFFFAOYSA-N	50466254	CHEMBL4288569	Bromodomain testis-specific protein	Homo sapiens			 20						ChEMBL	10.1016/j.bmcl.2018.08.039	10.7270/Q28S4SKP	30268702			Yang, SM; Urban, DJ; Yoshioka, M; Strovel, JW; Fletcher, S; Wang, AQ; Xu, X; Shah, P; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50466254	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50466254&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HRY	6E4A	129182189	433933519							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51251642	CCNC(=O)c1cc2c(cn(C)c(=O)c2[nH]1)-c1cc(ccc1Oc1c(C)cc(F)cc1C)C(C)(C)O	InChI=1S/C28H30FN3O4/c1-7-30-26(33)22-13-20-21(14-32(6)27(34)24(20)31-22)19-12-17(28(4,5)35)8-9-23(19)36-25-15(2)10-18(29)11-16(25)3/h8-14,31,35H,7H2,1-6H3,(H,30,33)	OEDSFMUSNZDJFD-UHFFFAOYSA-N	439497	US10633379, Example 35::US10633379, Example 82	Bromodomain testis-specific protein	Homo sapiens	 1.000000								ChEMBL	10.1021/acs.jmedchem.0c00628	10.7270/Q2057K8M	32324999			Sheppard, GS; Wang, L; Fidanze, SD; Hasvold, LA; Liu, D; Pratt, JK; Park, CH; Longenecker, K; Qiu, W; Torrent, M; Kovar, PJ; Bui, M; Faivre, E; Huang, X; Lin, X; Wilcox, D; Zhang, L; Shen, Y; Albert, DH; Magoc, TJ; Rajaraman, G; Kati, WM; McDaniel, KF	AbbVie Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=439497	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=439497&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HWV	6E6J,6ONY	132010322	439661049							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51251708	CCNC(=O)c1cc2c(cn(C)c(=O)c2[nH]1)-c1cc(ccc1Oc1c(C)cc(F)cc1C)C(C)(C)O	InChI=1S/C28H30FN3O4/c1-7-30-26(33)22-13-20-21(14-32(6)27(34)24(20)31-22)19-12-17(28(4,5)35)8-9-23(19)36-25-15(2)10-18(29)11-16(25)3/h8-14,31,35H,7H2,1-6H3,(H,30,33)	OEDSFMUSNZDJFD-UHFFFAOYSA-N	439497	US10633379, Example 35::US10633379, Example 82	Bromodomain testis-specific protein	Homo sapiens	 917								ChEMBL	10.1021/acs.jmedchem.0c00628	10.7270/Q2057K8M	32324999			Sheppard, GS; Wang, L; Fidanze, SD; Hasvold, LA; Liu, D; Pratt, JK; Park, CH; Longenecker, K; Qiu, W; Torrent, M; Kovar, PJ; Bui, M; Faivre, E; Huang, X; Lin, X; Wilcox, D; Zhang, L; Shen, Y; Albert, DH; Magoc, TJ; Rajaraman, G; Kati, WM; McDaniel, KF	AbbVie Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=439497	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=439497&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HWV	6E6J,6ONY	132010322	439661049							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51228575	CC1(NC(=O)N(CC(=O)Nc2ccc(Br)c(c2)S(=O)(=O)N2CCCCC2)C1=O)C1CC1	InChI=1S/C20H25BrN4O5S/c1-20(13-5-6-13)18(27)25(19(28)23-20)12-17(26)22-14-7-8-15(21)16(11-14)31(29,30)24-9-3-2-4-10-24/h7-8,11,13H,2-6,9-10,12H2,1H3,(H,22,26)(H,23,28)	CDJMQOCUCVPNIU-UHFFFAOYSA-N	50504159	CHEMBL4583297	Bromodomain testis-specific protein	Homo sapiens		 15849							ChEMBL	10.1021/acs.jmedchem.9b00673	10.7270/Q22R3VZV	31398032			Bamborough, P; Chung, CW; Demont, EH; Bridges, AM; Craggs, PD; Dixon, DP; Francis, P; Furze, RC; Grandi, P; Jones, EJ; Karamshi, B; Locke, K; Lucas, SCC; Michon, AM; Mitchell, DJ; Pogány, P; Prinjha, RK; Rau, C; Roa, AM; Roberts, AD; Sheppard, RJ; Watson, RJ	Cellzome	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50504159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50504159&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			139030526	440712744							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51228593	CC1(NC(=O)N(CC(=O)Nc2ccc(Br)c(c2)S(=O)(=O)N2CCCCC2)C1=O)C1CC1	InChI=1S/C20H25BrN4O5S/c1-20(13-5-6-13)18(27)25(19(28)23-20)12-17(26)22-14-7-8-15(21)16(11-14)31(29,30)24-9-3-2-4-10-24/h7-8,11,13H,2-6,9-10,12H2,1H3,(H,22,26)(H,23,28)	CDJMQOCUCVPNIU-UHFFFAOYSA-N	50504159	CHEMBL4583297	Bromodomain testis-specific protein	Homo sapiens		 25119							ChEMBL	10.1021/acs.jmedchem.9b00673	10.7270/Q22R3VZV	31398032			Bamborough, P; Chung, CW; Demont, EH; Bridges, AM; Craggs, PD; Dixon, DP; Francis, P; Furze, RC; Grandi, P; Jones, EJ; Karamshi, B; Locke, K; Lucas, SCC; Michon, AM; Mitchell, DJ; Pogány, P; Prinjha, RK; Rau, C; Roa, AM; Roberts, AD; Sheppard, RJ; Watson, RJ	Cellzome	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50504159	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50504159&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			139030526	440712744							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51242088	Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1	InChI=1S/C25H22N4O/c1-13-6-9-20-18(5-4-10-26-20)22(13)19-11-17(23-14(2)29-30-15(23)3)12-21-24(19)28-25(27-21)16-7-8-16/h4-6,9-12,16H,7-8H2,1-3H3,(H,27,28)	KHQQNXFBTALTQF-UHFFFAOYSA-N	249277	US10017501, Compound 1020-18::US9458145, 1020-18	Bromodomain testis-specific protein	Homo sapiens			 19						ChEMBL	10.1016/j.bmc.2018.11.020	10.7270/Q2HD7ZZ6	30606676			Sperandio, D; Aktoudianakis, V; Babaoglu, K; Chen, X; Elbel, K; Chin, G; Corkey, B; Du, J; Jiang, B; Kobayashi, T; Mackman, R; Martinez, R; Yang, H; Zablocki, J; Kusam, S; Jordan, K; Webb, H; Bates, JG; Lad, L; Mish, M; Niedziela-Majka, A; Metobo, S; Sapre, A; Hung, M; Jin, D; Fung, W; Kan, E; Eisenberg, G; Larson, N; Newby, ZER; Lansdon, E; Tay, C; Neve, RM; Shevick, SL; Breckenridge, DG	Gilead Sciences, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=249277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=249277&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			86301666	346543778							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51242089	Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1	InChI=1S/C25H22N4O/c1-13-6-9-20-18(5-4-10-26-20)22(13)19-11-17(23-14(2)29-30-15(23)3)12-21-24(19)28-25(27-21)16-7-8-16/h4-6,9-12,16H,7-8H2,1-3H3,(H,27,28)	KHQQNXFBTALTQF-UHFFFAOYSA-N	249277	US10017501, Compound 1020-18::US9458145, 1020-18	Bromodomain testis-specific protein	Homo sapiens			 5.0						ChEMBL	10.1016/j.bmc.2018.11.020	10.7270/Q2HD7ZZ6	30606676			Sperandio, D; Aktoudianakis, V; Babaoglu, K; Chen, X; Elbel, K; Chin, G; Corkey, B; Du, J; Jiang, B; Kobayashi, T; Mackman, R; Martinez, R; Yang, H; Zablocki, J; Kusam, S; Jordan, K; Webb, H; Bates, JG; Lad, L; Mish, M; Niedziela-Majka, A; Metobo, S; Sapre, A; Hung, M; Jin, D; Fung, W; Kan, E; Eisenberg, G; Larson, N; Newby, ZER; Lansdon, E; Tay, C; Neve, RM; Shevick, SL; Breckenridge, DG	Gilead Sciences, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=249277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=249277&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			86301666	346543778							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51242109	Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1	InChI=1S/C25H22N4O/c1-13-6-9-20-18(5-4-10-26-20)22(13)19-11-17(23-14(2)29-30-15(23)3)12-21-24(19)28-25(27-21)16-7-8-16/h4-6,9-12,16H,7-8H2,1-3H3,(H,27,28)	KHQQNXFBTALTQF-UHFFFAOYSA-N	249277	US10017501, Compound 1020-18::US9458145, 1020-18	Bromodomain testis-specific protein	Homo sapiens			 4.9						ChEMBL	10.1016/j.bmc.2018.11.020	10.7270/Q2HD7ZZ6	30606676			Sperandio, D; Aktoudianakis, V; Babaoglu, K; Chen, X; Elbel, K; Chin, G; Corkey, B; Du, J; Jiang, B; Kobayashi, T; Mackman, R; Martinez, R; Yang, H; Zablocki, J; Kusam, S; Jordan, K; Webb, H; Bates, JG; Lad, L; Mish, M; Niedziela-Majka, A; Metobo, S; Sapre, A; Hung, M; Jin, D; Fung, W; Kan, E; Eisenberg, G; Larson, N; Newby, ZER; Lansdon, E; Tay, C; Neve, RM; Shevick, SL; Breckenridge, DG	Gilead Sciences, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=249277	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=249277&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			86301666	346543778							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51249932	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 134							ChEMBL	10.1021/acs.jmedchem.9b02178	10.7270/Q27W6GHJ	32153186			Pan, Z; Li, X; Wang, Y; Jiang, Q; Jiang, L; Zhang, M; Zhang, N; Wu, F; Liu, B; He, G	Sichuan University and Collaborative Innovation Center of Biotherapy	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51249935	CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1	InChI=1S/C24H30N4O4S/c1-14-11-16(12-15(2)21(14)32-10-6-4-5-7-19(29)27-31)22-25-23(30)20-17-8-9-28(3)13-18(17)33-24(20)26-22/h11-12,31H,4-10,13H2,1-3H3,(H,27,29)(H,25,26,30)	BBFKONWWIAFKEJ-UHFFFAOYSA-N	50511231	CHEMBL4514808	Bromodomain testis-specific protein	Homo sapiens		>20000							ChEMBL	10.1021/acs.jmedchem.9b02178	10.7270/Q27W6GHJ	32153186			Pan, Z; Li, X; Wang, Y; Jiang, Q; Jiang, L; Zhang, M; Zhang, N; Wu, F; Liu, B; He, G	Sichuan University and Collaborative Innovation Center of Biotherapy	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50511231	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50511231&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			153534005	440719813							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51262552	Cc1nnc2CC[C@@H](Nc3ccc(Cl)cc3)c3cc(ccc3-n12)-c1cnn(C)c1	InChI=1S/C22H21ClN6/c1-14-26-27-22-10-8-20(25-18-6-4-17(23)5-7-18)19-11-15(3-9-21(19)29(14)22)16-12-24-28(2)13-16/h3-7,9,11-13,20,25H,8,10H2,1-2H3/t20-/m1/s1	MDRXOFSNECSECW-HXUWFJFHSA-N	50515771	CHEMBL4528047	Bromodomain testis-specific protein	Homo sapiens			 3.0						ChEMBL	10.1016/j.ejmech.2019.111633	10.7270/Q2MK6H84	31461688			Chen, D; Lu, T; Yan, Z; Lu, W; Zhou, F; Lyu, X; Xu, B; Jiang, H; Chen, K; Luo, C; Zhao, Y	University of Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50515771	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50515771&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	CQF	6K05,6K04	139035062	440724353							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51262561	Cc1nnc2CC[C@@H](Nc3ccc(Cl)cc3)c3cc(ccc3-n12)-c1cnn(C)c1	InChI=1S/C22H21ClN6/c1-14-26-27-22-10-8-20(25-18-6-4-17(23)5-7-18)19-11-15(3-9-21(19)29(14)22)16-12-24-28(2)13-16/h3-7,9,11-13,20,25H,8,10H2,1-2H3/t20-/m1/s1	MDRXOFSNECSECW-HXUWFJFHSA-N	50515771	CHEMBL4528047	Bromodomain testis-specific protein	Homo sapiens			 64						ChEMBL	10.1016/j.ejmech.2019.111633	10.7270/Q2MK6H84	31461688			Chen, D; Lu, T; Yan, Z; Lu, W; Zhou, F; Lyu, X; Xu, B; Jiang, H; Chen, K; Luo, C; Zhao, Y	University of Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50515771	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50515771&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	CQF	6K05,6K04	139035062	440724353							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225780	Fc1ccc(cc1)-c1ncn(C2CCNCC2)c1-c1ccnc(Oc2cc(F)cc(F)c2)n1	InChI=1S/C24H20F3N5O/c25-16-3-1-15(2-4-16)22-23(32(14-30-22)19-5-8-28-9-6-19)21-7-10-29-24(31-21)33-20-12-17(26)11-18(27)13-20/h1-4,7,10-14,19,28H,5-6,8-9H2	IXQGHOZDNBWZOU-UHFFFAOYSA-N	50099339	2-(3,5-Difluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL14339	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099339&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44269241	103996255		CHEMBL14339				ZINC36127104	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225781	Cc1nnn(C2CCNCC2)c1-c1ccnc(Nc2cc(C)cc(C)c2)n1	InChI=1S/C20H25N7/c1-13-10-14(2)12-16(11-13)23-20-22-9-6-18(24-20)19-15(3)25-26-27(19)17-4-7-21-8-5-17/h6,9-12,17,21H,4-5,7-8H2,1-3H3,(H,22,23,24)	CIBHWLGHOAYWGR-UHFFFAOYSA-N	50503386	CHEMBL4441390	Bromodomain testis-specific protein	Homo sapiens		 1600							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503386	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503386&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155514936	440711971							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225787	Cc1ccc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1	InChI=1S/C25H24FN5O/c1-17-2-8-21(9-3-17)32-25-28-15-12-22(30-25)24-23(18-4-6-19(26)7-5-18)29-16-31(24)20-10-13-27-14-11-20/h2-9,12,15-16,20,27H,10-11,13-14H2,1H3	MYXXRVIYUKHKPI-UHFFFAOYSA-N	50099352	4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-2-p-tolyloxy-pyrimidine::CHEMBL14682	Bromodomain testis-specific protein	Homo sapiens		 88000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099352&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536647	103996268		CHEMBL14682				ZINC36127110	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225788	Cc1ccc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1C	InChI=1S/C26H26FN5O/c1-17-3-8-22(15-18(17)2)33-26-29-14-11-23(31-26)25-24(19-4-6-20(27)7-5-19)30-16-32(25)21-9-12-28-13-10-21/h3-8,11,14-16,21,28H,9-10,12-13H2,1-2H3	ZPVIXTLWEIXXCD-UHFFFAOYSA-N	50099347	2-(3,4-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL13880	Bromodomain testis-specific protein	Homo sapiens		 13000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099347&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536615	103996263		CHEMBL13880				ZINC36127072	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225789	Cc1cc(C)cc(Nc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C26H27FN6/c1-17-13-18(2)15-21(14-17)31-26-29-12-9-23(32-26)25-24(19-3-5-20(27)6-4-19)30-16-33(25)22-7-10-28-11-8-22/h3-6,9,12-16,22,28H,7-8,10-11H2,1-2H3,(H,29,31,32)	DGOVBHLIYNOJOQ-UHFFFAOYSA-N	50503388	CHEMBL4521096	Bromodomain testis-specific protein	Homo sapiens		 3500							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503388&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JQP	6MH1	137701509	440711973							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225794	Cc1ccc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1C	InChI=1S/C26H26FN5O/c1-17-3-8-22(15-18(17)2)33-26-29-14-11-23(31-26)25-24(19-4-6-20(27)7-5-19)30-16-32(25)21-9-12-28-13-10-21/h3-8,11,14-16,21,28H,9-10,12-13H2,1-2H3	ZPVIXTLWEIXXCD-UHFFFAOYSA-N	50099347	2-(3,4-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL13880	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099347	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099347&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536615	103996263		CHEMBL13880				ZINC36127072	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225795	Cc1ccc(Nc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1C	InChI=1S/C26H27FN6/c1-17-3-8-21(15-18(17)2)31-26-29-14-11-23(32-26)25-24(19-4-6-20(27)7-5-19)30-16-33(25)22-9-12-28-13-10-22/h3-8,11,14-16,22,28H,9-10,12-13H2,1-2H3,(H,29,31,32)	OGDBBVMMKPWVLG-UHFFFAOYSA-N	50503389	CHEMBL4452281	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503389&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JQY	6MH7	138756791	440711974							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225796	Cc1cc(C)cc(Nc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C26H27FN6/c1-17-13-18(2)15-21(14-17)31-26-29-12-9-23(32-26)25-24(19-3-5-20(27)6-4-19)30-16-33(25)22-7-10-28-11-8-22/h3-6,9,12-16,22,28H,7-8,10-11H2,1-2H3,(H,29,31,32)	DGOVBHLIYNOJOQ-UHFFFAOYSA-N	50503388	CHEMBL4521096	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503388&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JQP	6MH1	137701509	440711973							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225812	Cc1cc(C)cc(Nc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C26H27FN6/c1-17-13-18(2)15-21(14-17)31-26-29-12-9-23(32-26)25-24(19-3-5-20(27)6-4-19)30-16-33(25)22-7-10-28-11-8-22/h3-6,9,12-16,22,28H,7-8,10-11H2,1-2H3,(H,29,31,32)	DGOVBHLIYNOJOQ-UHFFFAOYSA-N	50503388	CHEMBL4521096	Bromodomain testis-specific protein	Homo sapiens		 5300							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503388	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503388&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JQP	6MH1	137701509	440711973							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225813	Cc1cc(C)cc(Nc2nccc(n2)-c2c(nnn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C25H26FN7/c1-16-13-17(2)15-20(14-16)29-25-28-12-9-22(30-25)24-23(18-3-5-19(26)6-4-18)31-32-33(24)21-7-10-27-11-8-21/h3-6,9,12-15,21,27H,7-8,10-11H2,1-2H3,(H,28,29,30)	KNBRONAEQNUZRY-UHFFFAOYSA-N	50503387	CHEMBL4475135	Bromodomain testis-specific protein	Homo sapiens		 36000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503387	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503387&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155352361	440711972							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225830	Cc1ccc(Nc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1C	InChI=1S/C26H27FN6/c1-17-3-8-21(15-18(17)2)31-26-29-14-11-23(32-26)25-24(19-4-6-20(27)7-5-19)30-16-33(25)22-9-12-28-13-10-22/h3-8,11,14-16,22,28H,9-10,12-13H2,1-2H3,(H,29,31,32)	OGDBBVMMKPWVLG-UHFFFAOYSA-N	50503389	CHEMBL4452281	Bromodomain testis-specific protein	Homo sapiens		 4700							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503389	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503389&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JQY	6MH7	138756791	440711974							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225839	Cc1ccc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)cc1	InChI=1S/C25H24FN5O/c1-17-2-8-21(9-3-17)32-25-28-15-12-22(30-25)24-23(18-4-6-19(26)7-5-18)29-16-31(24)20-10-13-27-14-11-20/h2-9,12,15-16,20,27H,10-11,13-14H2,1H3	MYXXRVIYUKHKPI-UHFFFAOYSA-N	50099352	4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-2-p-tolyloxy-pyrimidine::CHEMBL14682	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099352	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099352&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536647	103996268		CHEMBL14682				ZINC36127110	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225848	Cc1cc(C)cc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C26H26FN5O/c1-17-13-18(2)15-22(14-17)33-26-29-12-9-23(31-26)25-24(19-3-5-20(27)6-4-19)30-16-32(25)21-7-10-28-11-8-21/h3-6,9,12-16,21,28H,7-8,10-11H2,1-2H3	UVLWMBRFRAMDOW-UHFFFAOYSA-N	50099333	2-(3,5-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL417255::D3RKN_55	Bromodomain testis-specific protein	Homo sapiens		 18000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099333	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099333&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536633	103996249		CHEMBL417255				ZINC36127094	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225851	Cc1cc(C)cc(Oc2nccc(n2)-c2c(ncn2C2CCNCC2)-c2ccc(F)cc2)c1	InChI=1S/C26H26FN5O/c1-17-13-18(2)15-22(14-17)33-26-29-12-9-23(31-26)25-24(19-3-5-20(27)6-4-19)30-16-32(25)21-7-10-28-11-8-21/h3-6,9,12-16,21,28H,7-8,10-11H2,1-2H3	UVLWMBRFRAMDOW-UHFFFAOYSA-N	50099333	2-(3,5-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL417255::D3RKN_55	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099333	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099333&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			18536633	103996249		CHEMBL417255				ZINC36127094	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225852	Fc1ccc(cc1)-c1ncn(C2CCNCC2)c1-c1ccnc(Oc2cc(F)cc(F)c2)n1	InChI=1S/C24H20F3N5O/c25-16-3-1-15(2-4-16)22-23(32(14-30-22)19-5-8-28-9-6-19)21-7-10-29-24(31-21)33-20-12-17(26)11-18(27)13-20/h1-4,7,10-14,19,28H,5-6,8-9H2	IXQGHOZDNBWZOU-UHFFFAOYSA-N	50099339	2-(3,5-Difluoro-phenoxy)-4-[5-(4-fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-pyrimidine::CHEMBL14339	Bromodomain testis-specific protein	Homo sapiens		>250000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099339&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			44269241	103996255		CHEMBL14339				ZINC36127104	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51225854	Cc1cc(C)cc(Nc2nccc(n2)-c2c(CO)nnn2C2CCNCC2)c1	InChI=1S/C20H25N7O/c1-13-9-14(2)11-15(10-13)23-20-22-8-5-17(24-20)19-18(12-28)25-26-27(19)16-3-6-21-7-4-16/h5,8-11,16,21,28H,3-4,6-7,12H2,1-2H3,(H,22,23,24)	PYRVHRPHHLORKP-UHFFFAOYSA-N	50503390	CHEMBL4533090	Bromodomain testis-specific protein	Homo sapiens		 110000							ChEMBL	10.1021/acs.jmedchem.8b01248	10.7270/Q25T3PRQ	30253095			Divakaran, A; Talluri, SK; Ayoub, AM; Mishra, NK; Cui, H; Widen, JC; Berndt, N; Zhu, JY; Carlson, AS; Topczewski, JJ; Schonbrunn, EK; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50503390	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50503390&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155352401	440711975							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51258461	COc1ccccc1S(=O)(=O)Nc1ccc2N(C)C(=O)c3cc(nc1c23)-n1cnc(C)c1	InChI=1S/C22H19N5O4S/c1-13-11-27(12-23-13)19-10-14-20-16(26(2)22(14)28)9-8-15(21(20)24-19)25-32(29,30)18-7-5-4-6-17(18)31-3/h4-12,25H,1-3H3	FSMTUHGXWGJNKK-UHFFFAOYSA-N	50514312	CHEMBL4446421	Bromodomain testis-specific protein	Homo sapiens		 357							ChEMBL	10.1021/acs.jmedchem.9b01010	10.7270/Q2280BZP	31789032			Jiang, F; Hu, Q; Zhang, Z; Li, H; Li, H; Zhang, D; Li, H; Ma, Y; Xu, J; Chen, H; Cui, Y; Zhi, Y; Zhang, Y; Xu, J; Zhu, J; Lu, T; Chen, Y	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50514312	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50514312&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			145925666	440722894							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51321770	COc1nnc2ccc(nn12)N1CCC(CC1)c1ccc(OCCN2CCN(C)C(=O)[C@H]2C)cc1	InChI=1S/C25H33N7O3/c1-18-24(33)29(2)14-15-30(18)16-17-35-21-6-4-19(5-7-21)20-10-12-31(13-11-20)23-9-8-22-26-27-25(34-3)32(22)28-23/h4-9,18,20H,10-17H2,1-3H3/t18-/m1/s1	RSMYFSPOTCDHHJ-GOSISDBHSA-N	50260093	CHEMBL4078100	Bromodomain testis-specific protein	Homo sapiens	 100								ChEMBL	10.1021/acs.jmedchem.6b00070	10.7270/Q2697721	27528113			Bradbury, RH; Callis, R; Carr, GR; Chen, H; Clark, E; Feron, L; Glossop, S; Graham, MA; Hattersley, M; Jones, C; Lamont, SG; Ouvry, G; Patel, A; Patel, J; Rabow, AA; Roberts, CA; Stokes, S; Stratton, N; Walker, GE; Ward, L; Whalley, D; Whittaker, D; Wrigley, G; Waring, MJ	AstraZeneca	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50260093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50260093&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XNH	5KHM	118693659	404339980							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51321771	COc1nnc2ccc(nn12)N1CCC(CC1)c1ccc(OCCN2CCN(C)C(=O)[C@H]2C)cc1	InChI=1S/C25H33N7O3/c1-18-24(33)29(2)14-15-30(18)16-17-35-21-6-4-19(5-7-21)20-10-12-31(13-11-20)23-9-8-22-26-27-25(34-3)32(22)28-23/h4-9,18,20H,10-17H2,1-3H3/t18-/m1/s1	RSMYFSPOTCDHHJ-GOSISDBHSA-N	50260093	CHEMBL4078100	Bromodomain testis-specific protein	Homo sapiens	 501								ChEMBL	10.1021/acs.jmedchem.6b00070	10.7270/Q2697721	27528113			Bradbury, RH; Callis, R; Carr, GR; Chen, H; Clark, E; Feron, L; Glossop, S; Graham, MA; Hattersley, M; Jones, C; Lamont, SG; Ouvry, G; Patel, A; Patel, J; Rabow, AA; Roberts, CA; Stokes, S; Stratton, N; Walker, GE; Ward, L; Whalley, D; Whittaker, D; Wrigley, G; Waring, MJ	AstraZeneca	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50260093	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50260093&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XNH	5KHM	118693659	404339980							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294607	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@@H](O)CN2CCN(C)CC2)c(C)c1	InChI=1S/C27H34N2O6/c1-17-10-19(23-14-22(31)26-24(33-5)12-21(32-4)13-25(26)35-23)11-18(2)27(17)34-16-20(30)15-29-8-6-28(3)7-9-29/h10-14,20,30H,6-9,15-16H2,1-5H3/t20-/m0/s1	UDPXIEUTIPNLKC-FQEVSTJZSA-N	50527823	CHEMBL4517875	Bromodomain testis-specific protein	Homo sapiens			 2545						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527823	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527823&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155541119	440736405							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294608	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@H](O)CN2CCN(C)CC2)c(C)c1	InChI=1S/C27H34N2O6/c1-17-10-19(23-14-22(31)26-24(33-5)12-21(32-4)13-25(26)35-23)11-18(2)27(17)34-16-20(30)15-29-8-6-28(3)7-9-29/h10-14,20,30H,6-9,15-16H2,1-5H3/t20-/m1/s1	UDPXIEUTIPNLKC-HXUWFJFHSA-N	50527819	CHEMBL4557050::US11117865, Compound ZL0516	Bromodomain testis-specific protein	Homo sapiens			 3176						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527819	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527819&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QKP	6UWU	135126189	440736401							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294622	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens			 4836						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294623	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@H](O)CN2CCN(C)CC2)c(C)c1	InChI=1S/C27H34N2O6/c1-17-10-19(23-14-22(31)26-24(33-5)12-21(32-4)13-25(26)35-23)11-18(2)27(17)34-16-20(30)15-29-8-6-28(3)7-9-29/h10-14,20,30H,6-9,15-16H2,1-5H3/t20-/m1/s1	UDPXIEUTIPNLKC-HXUWFJFHSA-N	50527819	CHEMBL4557050::US11117865, Compound ZL0516	Bromodomain testis-specific protein	Homo sapiens			 3592						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527819	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527819&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QKP	6UWU	135126189	440736401							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294624	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@H](O)CN2CCCCC2)c(C)c1	InChI=1S/C27H33NO6/c1-17-10-19(11-18(2)27(17)33-16-20(29)15-28-8-6-5-7-9-28)23-14-22(30)26-24(32-4)12-21(31-3)13-25(26)34-23/h10-14,20,29H,5-9,15-16H2,1-4H3/t20-/m1/s1	CSTRBRUZBLYKBT-HXUWFJFHSA-N	50527821	CHEMBL4455209	Bromodomain testis-specific protein	Homo sapiens			 2317						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527821	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527821&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			135126546	440736403							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294632	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@H](O)CN2CCCCC2)c(C)c1	InChI=1S/C27H33NO6/c1-17-10-19(11-18(2)27(17)33-16-20(29)15-28-8-6-5-7-9-28)23-14-22(30)26-24(32-4)12-21(31-3)13-25(26)34-23/h10-14,20,29H,5-9,15-16H2,1-4H3/t20-/m1/s1	CSTRBRUZBLYKBT-HXUWFJFHSA-N	50527821	CHEMBL4455209	Bromodomain testis-specific protein	Homo sapiens			 2869						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527821	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527821&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			135126546	440736403							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294638	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 217						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51299391	COC(=O)N1CCSC(CC1)c1cccs1	InChI=1S/C11H15NO2S2/c1-14-11(13)12-5-4-10(16-8-6-12)9-3-2-7-15-9/h2-3,7,10H,4-6,8H2,1H3	GTUMUZDXWXZZSA-UHFFFAOYSA-N	50529527	CHEMBL4435656	Bromodomain testis-specific protein	Homo sapiens			 270000						ChEMBL	10.1021/acsmedchemlett.9b00414	10.7270/Q2WM1HVP	31857841			Johnson, JA; Nicolaou, CA; Kirberger, SE; Pandey, AK; Hu, H; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50529527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50529527&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QJ1	6UVJ,7UU0	155511200	440738109							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51299392	COC(=O)N1CCSC(CC1)c1cccs1	InChI=1S/C11H15NO2S2/c1-14-11(13)12-5-4-10(16-8-6-12)9-3-2-7-15-9/h2-3,7,10H,4-6,8H2,1H3	GTUMUZDXWXZZSA-UHFFFAOYSA-N	50529527	CHEMBL4435656	Bromodomain testis-specific protein	Homo sapiens			 270000						ChEMBL	10.1021/acsmedchemlett.9b00414	10.7270/Q2WM1HVP	31857841			Johnson, JA; Nicolaou, CA; Kirberger, SE; Pandey, AK; Hu, H; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50529527	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50529527&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QJ1	6UVJ,7UU0	155511200	440738109							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294077	CCS(=O)(=O)Cc1cnc(Oc2ccc(F)cc2F)c(c1)-c1cc(C)c2n1cc[nH]c2=O	InChI=1S/C22H19F2N3O4S/c1-3-32(29,30)12-14-9-16(18-8-13(2)20-21(28)25-6-7-27(18)20)22(26-11-14)31-19-5-4-15(23)10-17(19)24/h4-11H,3,12H2,1-2H3,(H,25,28)	UETQFSCWDMJWMM-UHFFFAOYSA-N	50527569	CHEMBL4440098::US11427593, Compound ZB-BD-216	Bromodomain testis-specific protein	Homo sapiens			 2.1						ChEMBL	10.1021/acs.jmedchem.9b01784	10.7270/Q2V98CHS	32208600			Li, Z; Xiao, S; Yang, Y; Chen, C; Lu, T; Chen, Z; Jiang, H; Chen, S; Luo, C; Zhou, B	Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527569	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527569&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			146047136	440736151							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294574	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@@H](O)CN2CCCCC2)c(C)c1	InChI=1S/C27H33NO6/c1-17-10-19(11-18(2)27(17)33-16-20(29)15-28-8-6-5-7-9-28)23-14-22(30)26-24(32-4)12-21(31-3)13-25(26)34-23/h10-14,20,29H,5-9,15-16H2,1-4H3/t20-/m0/s1	CSTRBRUZBLYKBT-FQEVSTJZSA-N	50527820	CHEMBL4549898	Bromodomain testis-specific protein	Homo sapiens			 2411						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527820	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527820&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155550409	440736402							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294603	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@@H](O)CN2CCCCC2)c(C)c1	InChI=1S/C27H33NO6/c1-17-10-19(11-18(2)27(17)33-16-20(29)15-28-8-6-5-7-9-28)23-14-22(30)26-24(32-4)12-21(31-3)13-25(26)34-23/h10-14,20,29H,5-9,15-16H2,1-4H3/t20-/m0/s1	CSTRBRUZBLYKBT-FQEVSTJZSA-N	50527820	CHEMBL4549898	Bromodomain testis-specific protein	Homo sapiens			 2502						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527820	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527820&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155550409	440736402							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294604	COc1cc(OC)c2c(c1)oc(cc2=O)-c1cc(C)c(OC[C@@H](O)CN2CCN(C)CC2)c(C)c1	InChI=1S/C27H34N2O6/c1-17-10-19(23-14-22(31)26-24(33-5)12-21(32-4)13-25(26)35-23)11-18(2)27(17)34-16-20(30)15-29-8-6-28(3)7-9-29/h10-14,20,30H,6-9,15-16H2,1-5H3/t20-/m0/s1	UDPXIEUTIPNLKC-FQEVSTJZSA-N	50527823	CHEMBL4517875	Bromodomain testis-specific protein	Homo sapiens			 2765						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50527823	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50527823&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			155541119	440736405							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294605	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 183						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51294606	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens			 708						ChEMBL	10.1021/acs.jmedchem.0c00035	10.7270/Q2PK0KMS	32255647			Liu, Z; Chen, H; Wang, P; Li, Y; Wold, EA; Leonard, PG; Joseph, S; Brasier, AR; Tian, B; Zhou, J	University of Texas Medical Branch	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51333375	CCS(=O)(=O)Nc1cc(cc2n(ccc12)C(C)(c1ccccn1)c1ccccn1)-c1cn(C)c2c1cc[nH]c2=O	InChI=1S/C30H28N6O3S/c1-4-40(38,39)34-24-17-20(23-19-35(3)28-21(23)11-15-33-29(28)37)18-25-22(24)12-16-36(25)30(2,26-9-5-7-13-31-26)27-10-6-8-14-32-27/h5-19,34H,4H2,1-3H3,(H,33,37)	LMLIBNUOIWAJFC-UHFFFAOYSA-N	50539801	CHEMBL4648912	Bromodomain testis-specific protein	Homo sapiens			<1.000000						ChEMBL	10.1021/acs.jmedchem.0c00456	10.7270/Q2PK0KPP	32453591			Li, Y; Zhao, J; Gutgesell, LM; Shen, Z; Ratia, K; Dye, K; Dubrovskyi, O; Zhao, H; Huang, F; Tonetti, DA; Thatcher, GRJ; Xiong, R	University of Illinois at Chicago	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50539801	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50539801&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YF2	6P05,7JUO	146036007	442141364							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51333376	CCS(=O)(=O)Nc1cc(cc2n(ccc12)C(C)(c1ccccn1)c1ccccn1)-c1cn(C)c2c1cc[nH]c2=O	InChI=1S/C30H28N6O3S/c1-4-40(38,39)34-24-17-20(23-19-35(3)28-21(23)11-15-33-29(28)37)18-25-22(24)12-16-36(25)30(2,26-9-5-7-13-31-26)27-10-6-8-14-32-27/h5-19,34H,4H2,1-3H3,(H,33,37)	LMLIBNUOIWAJFC-UHFFFAOYSA-N	50539801	CHEMBL4648912	Bromodomain testis-specific protein	Homo sapiens			<1.000000						ChEMBL	10.1021/acs.jmedchem.0c00456	10.7270/Q2PK0KPP	32453591			Li, Y; Zhao, J; Gutgesell, LM; Shen, Z; Ratia, K; Dye, K; Dubrovskyi, O; Zhao, H; Huang, F; Tonetti, DA; Thatcher, GRJ; Xiong, R	University of Illinois at Chicago	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50539801	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50539801&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YF2	6P05,7JUO	146036007	442141364							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51333377	CCS(=O)(=O)Nc1cc(cc2n(ccc12)C(C)(c1ccccn1)c1ccccn1)-c1cn(C)c2c1cc[nH]c2=O	InChI=1S/C30H28N6O3S/c1-4-40(38,39)34-24-17-20(23-19-35(3)28-21(23)11-15-33-29(28)37)18-25-22(24)12-16-36(25)30(2,26-9-5-7-13-31-26)27-10-6-8-14-32-27/h5-19,34H,4H2,1-3H3,(H,33,37)	LMLIBNUOIWAJFC-UHFFFAOYSA-N	50539801	CHEMBL4648912	Bromodomain testis-specific protein	Homo sapiens			<1.000000						ChEMBL	10.1021/acs.jmedchem.0c00456	10.7270/Q2PK0KPP	32453591			Li, Y; Zhao, J; Gutgesell, LM; Shen, Z; Ratia, K; Dye, K; Dubrovskyi, O; Zhao, H; Huang, F; Tonetti, DA; Thatcher, GRJ; Xiong, R	University of Illinois at Chicago	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50539801	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50539801&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	YF2	6P05,7JUO	146036007	442141364							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991938	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 77.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991940	C[C@H](O)CNC(=O)C[C@H]1N=C(c2c(C)c(C)sc2-n2c(C)nnc12)c1ccc(Cl)cc1	InChI=1S/C22H24ClN5O2S/c1-11(29)10-24-18(30)9-17-21-27-26-14(4)28(21)22-19(12(2)13(3)31-22)20(25-17)15-5-7-16(23)8-6-15/h5-8,11,17,29H,9-10H2,1-4H3,(H,24,30)/t11-,17+/m0/s1	ZXGRKOXAZLNTEL-APPDUMDISA-N	474457	US10881668, Compound 501	Bromodomain testis-specific protein	Homo sapiens		 82.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=474457	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=474457&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156027022	442136550							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991942	C[C@@H](O)CNC(=O)C[C@H]1N=C(c2c(C)c(C)sc2-n2c(C)nnc12)c1ccc(Cl)cc1	InChI=1S/C22H24ClN5O2S/c1-11(29)10-24-18(30)9-17-21-27-26-14(4)28(21)22-19(12(2)13(3)31-22)20(25-17)15-5-7-16(23)8-6-15/h5-8,11,17,29H,9-10H2,1-4H3,(H,24,30)/t11-,17-/m1/s1	ZXGRKOXAZLNTEL-PIGZYNQJSA-N	474458	US10881668, Compound 502	Bromodomain testis-specific protein	Homo sapiens		 61.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=474458	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=474458&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156027023	442136551							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991944	Cc1nnc2[C@@H](CC(=O)NCC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C24H28ClN5OS/c1-13-14(2)32-23-20(13)21(16-7-9-17(25)10-8-16)27-18(22-29-28-15(3)30(22)23)11-19(31)26-12-24(4,5)6/h7-10,18H,11-12H2,1-6H3,(H,26,31)/t18-/m1/s1	QXWJFGXUZLPVCL-GOSISDBHSA-N	474459	US10881668, Compound 503	Bromodomain testis-specific protein	Homo sapiens		 89.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=474459	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=474459&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			126544231	442136552							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991946	Cc1sc-2c(c1C)C(=N[C@H](CC(=O)NCC(F)F)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C21H20ClF2N5OS/c1-10-11(2)31-21-18(10)19(13-4-6-14(22)7-5-13)26-15(8-17(30)25-9-16(23)24)20-28-27-12(3)29(20)21/h4-7,15-16H,8-9H2,1-3H3,(H,25,30)/t15-/m1/s1	SKANTSCEPLCAJH-OAHLLOKOSA-N	474460	US10881668, Compound 504	Bromodomain testis-specific protein	Homo sapiens		 69.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=474460	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=474460&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156027024	442136553							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
991948	Cc1sc-2c(c1C)C(=N[C@H](CC(=O)NCCC(F)F)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C22H22ClF2N5OS/c1-11-12(2)32-22-19(11)20(14-4-6-15(23)7-5-14)27-16(21-29-28-13(3)30(21)22)10-18(31)26-9-8-17(24)25/h4-7,16-17H,8-10H2,1-3H3,(H,26,31)/t16-/m1/s1	NHMJYXDPZTZGQX-MRXNPFEDSA-N	474461	US10881668, Compound 505	Bromodomain testis-specific protein	Homo sapiens		 75.0							US Patent		10.7270/Q2TQ64NR		aid1805148	US10881668	Bradner, JE; Qi, J; Tanaka, M	Dana-Farber Cancer Institute, Inc.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=474461	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=474461&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156027025	442136554							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345913	COCc1nc2cnc3cc(-c4c(C)noc4C)c(OC[C@H]4CCNC4)cc3c2n1[C@H](C)c1ccccc1	InChI=1S/C30H33N5O3/c1-18-29(20(3)38-34-18)24-12-25-23(13-27(24)37-16-21-10-11-31-14-21)30-26(15-32-25)33-28(17-36-4)35(30)19(2)22-8-6-5-7-9-22/h5-9,12-13,15,19,21,31H,10-11,14,16-17H2,1-4H3/t19-,21+/m1/s1	ZORLJXWXFABTPZ-CTNGQTDRSA-N	50544597	GSK778	Bromodomain testis-specific protein	Homo sapiens		 158							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544597&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	LWB	6SWN,6SWO	146018691	442146160							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345917	COCc1nc2cnc3cc(-c4c(C)noc4C)c(OC[C@H]4CCNC4)cc3c2n1[C@H](C)c1ccccc1	InChI=1S/C30H33N5O3/c1-18-29(20(3)38-34-18)24-12-25-23(13-27(24)37-16-21-10-11-31-14-21)30-26(15-32-25)33-28(17-36-4)35(30)19(2)22-8-6-5-7-9-22/h5-9,12-13,15,19,21,31H,10-11,14,16-17H2,1-4H3/t19-,21+/m1/s1	ZORLJXWXFABTPZ-CTNGQTDRSA-N	50544597	GSK778	Bromodomain testis-specific protein	Homo sapiens		 15849							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544597	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544597&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	LWB	6SWN,6SWO	146018691	442146160							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345924	COc1cc2c3n([C@H](C)c4ccccn4)c(=O)[nH]c3cnc2cc1-c1c(C)noc1C	InChI=1S/C23H21N5O3/c1-12-21(14(3)31-27-12)16-9-18-15(10-20(16)30-4)22-19(11-25-18)26-23(29)28(22)13(2)17-7-5-6-8-24-17/h5-11,13H,1-4H3,(H,26,29)/t13-/m1/s1	VUVUVNZRUGEAHB-CYBMUJFWSA-N	50380682	CHEMBL2017291::I-BET151 (16)	Bromodomain testis-specific protein	Homo sapiens		 126							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50380682	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50380682&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1GH	3ZYU,4PKL,4ALG	52912189	160859765		CHEMBL2017291				ZINC73069302	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345928	COc1cc2c3n([C@H](C)c4ccccn4)c(=O)[nH]c3cnc2cc1-c1c(C)noc1C	InChI=1S/C23H21N5O3/c1-12-21(14(3)31-27-12)16-9-18-15(10-20(16)30-4)22-19(11-25-18)26-23(29)28(22)13(2)17-7-5-6-8-24-17/h5-11,13H,1-4H3,(H,26,29)/t13-/m1/s1	VUVUVNZRUGEAHB-CYBMUJFWSA-N	50380682	CHEMBL2017291::I-BET151 (16)	Bromodomain testis-specific protein	Homo sapiens		 1585							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50380682	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50380682&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1GH	3ZYU,4PKL,4ALG	52912189	160859765		CHEMBL2017291				ZINC73069302	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345932	COCc1nc2cnc3cc(-c4c(C)noc4C)c(OC)cc3c2n1[C@H](C)c1ccccc1	InChI=1S/C26H26N4O3/c1-15-25(17(3)33-29-15)20-11-21-19(12-23(20)32-5)26-22(13-27-21)28-24(14-31-4)30(26)16(2)18-9-7-6-8-10-18/h6-13,16H,14H2,1-5H3/t16-/m1/s1	ZYJNOYAZLFPWBD-MRXNPFEDSA-N	50544616	CHEMBL4635329	Bromodomain testis-specific protein	Homo sapiens		 25							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544616	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544616&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156014722	442146179							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51345936	COCc1nc2cnc3cc(-c4c(C)noc4C)c(OC)cc3c2n1[C@H](C)c1ccccc1	InChI=1S/C26H26N4O3/c1-15-25(17(3)33-29-15)20-11-21-19(12-23(20)32-5)26-22(13-27-21)28-24(14-31-4)30(26)16(2)18-9-7-6-8-10-18/h6-13,16H,14H2,1-5H3/t16-/m1/s1	ZYJNOYAZLFPWBD-MRXNPFEDSA-N	50544616	CHEMBL4635329	Bromodomain testis-specific protein	Homo sapiens		 316							ChEMBL	10.1021/acs.jmedchem.0c00566	10.7270/Q2348Q0N	32787145			Wellaway, CR; Bamborough, P; Bernard, SG; Chung, CW; Craggs, PD; Cutler, L; Demont, EH; Evans, JP; Gordon, L; Karamshi, B; Lewis, AJ; Lindon, MJ; Mitchell, DJ; Rioja, I; Soden, PE; Taylor, S; Watson, RJ; Willis, R; Woolven, JM; Wyspiańska, BS; Kerr, WJ; Prinjha, RK	GSK	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544616	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544616&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			156014722	442146179							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51346958	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCNC(=O)COc1cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c13)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C38H37ClN8O7S/c1-19-20(2)55-38-31(19)33(22-9-11-23(39)12-10-22)42-25(34-45-44-21(3)46(34)38)17-29(49)40-15-4-5-16-41-30(50)18-54-27-8-6-7-24-32(27)37(53)47(36(24)52)26-13-14-28(48)43-35(26)51/h6-12,25-26H,4-5,13-18H2,1-3H3,(H,40,49)(H,41,50)(H,43,48,51)/t25-,26?/m0/s1	LKEGXJXRNBALBV-PMCHYTPCSA-N	50544938	CHEMBL4094346::US11059801, Compound dBET1	Bromodomain testis-specific protein	Homo sapiens			 6.0						ChEMBL	10.1016/j.bmcl.2020.126958	10.7270/Q2M0491W	32019712			Wisniewski, A; Georg, GI	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544938	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544938&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			91799313	442146501							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51344902	CNC(=O)c1ccc(=O)n(Cc2cc(Br)ccc2F)c1	InChI=1S/C14H12BrFN2O2/c1-17-14(20)9-2-5-13(19)18(7-9)8-10-6-11(15)3-4-12(10)16/h2-7H,8H2,1H3,(H,17,20)	GWUMCWHPIGGSQS-UHFFFAOYSA-N	50544297	CHEMBL4637442	Bromodomain testis-specific protein	Homo sapiens		 39811							ChEMBL	10.1021/acs.jmedchem.0c00796	10.7270/Q27W6GS4	32702236			Seal, JT; Atkinson, SJ; Aylott, H; Bamborough, P; Chung, CW; Copley, RCB; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Lindon, M; Messenger, C; Michon, AM; Mitchell, D; Preston, A; Prinjha, RK; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544297	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544297&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			47449090	442145860							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51344903	CNC(=O)c1ccc(=O)n(Cc2ccccc2)c1	InChI=1S/C14H14N2O2/c1-15-14(18)12-7-8-13(17)16(10-12)9-11-5-3-2-4-6-11/h2-8,10H,9H2,1H3,(H,15,18)	HKTUSCZNSARQMH-UHFFFAOYSA-N	50544298	CHEMBL4639878	Bromodomain testis-specific protein	Homo sapiens		 31623							ChEMBL	10.1021/acs.jmedchem.0c00796	10.7270/Q27W6GS4	32702236			Seal, JT; Atkinson, SJ; Aylott, H; Bamborough, P; Chung, CW; Copley, RCB; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Lindon, M; Messenger, C; Michon, AM; Mitchell, D; Preston, A; Prinjha, RK; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544298	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544298&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			47394458	442145861							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51344904	CNC(=O)c1cccn(Cc2ccccc2)c1=O	InChI=1S/C14H14N2O2/c1-15-13(17)12-8-5-9-16(14(12)18)10-11-6-3-2-4-7-11/h2-9H,10H2,1H3,(H,15,17)	FPNFBPWMDHIOEK-UHFFFAOYSA-N	50543339	CHEMBL4633353	Bromodomain testis-specific protein	Homo sapiens		 10000							ChEMBL	10.1021/acs.jmedchem.0c00796	10.7270/Q27W6GS4	32702236			Seal, JT; Atkinson, SJ; Aylott, H; Bamborough, P; Chung, CW; Copley, RCB; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Lindon, M; Messenger, C; Michon, AM; Mitchell, D; Preston, A; Prinjha, RK; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50543339	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50543339&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QCW	6ZB0	48157449	442144902							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51344905	CNC(=O)c1cc(cn(Cc2ccccc2)c1=O)C(=O)NC1CC1	InChI=1S/C18H19N3O3/c1-19-17(23)15-9-13(16(22)20-14-7-8-14)11-21(18(15)24)10-12-5-3-2-4-6-12/h2-6,9,11,14H,7-8,10H2,1H3,(H,19,23)(H,20,22)	QZZCUOVXHPAQRQ-UHFFFAOYSA-N	50543359	GSK620	Bromodomain testis-specific protein	Homo sapiens		 25119							ChEMBL	10.1021/acs.jmedchem.0c00796	10.7270/Q27W6GS4	32702236			Seal, JT; Atkinson, SJ; Aylott, H; Bamborough, P; Chung, CW; Copley, RCB; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Lindon, M; Messenger, C; Michon, AM; Mitchell, D; Preston, A; Prinjha, RK; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50543359	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50543359&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QCZ	6ZB3,6ZB1	126648559	442144922							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51344906	CNC(=O)c1cc(cn(Cc2cccc3[nH]ccc23)c1=O)C(=O)NC1CC1	InChI=1S/C20H20N4O3/c1-21-19(26)16-9-13(18(25)23-14-5-6-14)11-24(20(16)27)10-12-3-2-4-17-15(12)7-8-22-17/h2-4,7-9,11,14,22H,5-6,10H2,1H3,(H,21,26)(H,23,25)	PDCBJZVPIGAEBL-UHFFFAOYSA-N	50544335	CHEMBL4648431	Bromodomain testis-specific protein	Homo sapiens		 19953							ChEMBL	10.1021/acs.jmedchem.0c00796	10.7270/Q27W6GS4	32702236			Seal, JT; Atkinson, SJ; Aylott, H; Bamborough, P; Chung, CW; Copley, RCB; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Lindon, M; Messenger, C; Michon, AM; Mitchell, D; Preston, A; Prinjha, RK; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544335	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544335&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QD5	6ZB2	126648444	442145898							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51380544	C[C@@H]1CN(c2ccc(Cl)cc2)c2cc(ccc2-n2c(C)nnc12)-c1ccc(N)nc1	InChI=1S/C23H21ClN6/c1-14-13-29(19-7-5-18(24)6-8-19)21-11-16(17-4-10-22(25)26-12-17)3-9-20(21)30-15(2)27-28-23(14)30/h3-12,14H,13H2,1-2H3,(H2,25,26)/t14-/m1/s1	SBRJLPKKZHHGCO-CQSZACIVSA-N	50558065	CHEMBL4780530	Bromodomain testis-specific protein	Homo sapiens		 3.0							ChEMBL	10.1021/ml500411h	10.7270/Q2DV1PK7	26985289			Taylor, AM; Vaswani, RG; Gehling, VS; Hewitt, MC; Leblanc, Y; Audia, JE; Bellon, S; Cummings, RT; Côté, A; Harmange, JC; Jayaram, H; Joshi, S; Lora, JM; Mertz, JA; Neiss, A; Pardo, E; Nasveschuk, CG; Poy, F; Sandy, P; Setser, JW; Sims, RJ; Tang, Y; Albrecht, BK	Constellation Pharmaceuticals	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50558065	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50558065&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	558	4Z1Q	71466419	461828457							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51380545	C[C@@H]1CN(c2ccc(Cl)cc2)c2cc(ccc2-n2c(C)nnc12)-c1ccc(N)nc1	InChI=1S/C23H21ClN6/c1-14-13-29(19-7-5-18(24)6-8-19)21-11-16(17-4-10-22(25)26-12-17)3-9-20(21)30-15(2)27-28-23(14)30/h3-12,14H,13H2,1-2H3,(H2,25,26)/t14-/m1/s1	SBRJLPKKZHHGCO-CQSZACIVSA-N	50558065	CHEMBL4780530	Bromodomain testis-specific protein	Homo sapiens		 3.0							ChEMBL	10.1021/ml500411h	10.7270/Q2DV1PK7	26985289			Taylor, AM; Vaswani, RG; Gehling, VS; Hewitt, MC; Leblanc, Y; Audia, JE; Bellon, S; Cummings, RT; Côté, A; Harmange, JC; Jayaram, H; Joshi, S; Lora, JM; Mertz, JA; Neiss, A; Pardo, E; Nasveschuk, CG; Poy, F; Sandy, P; Setser, JW; Sims, RJ; Tang, Y; Albrecht, BK	Constellation Pharmaceuticals	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50558065	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50558065&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	558	4Z1Q	71466419	461828457							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51384900	CN1c2cnc(N[C@H]3CC[C@H](O)CC3)cc2Oc2cccc(F)c2C1=O	InChI=1S/C19H20FN3O3/c1-23-14-10-21-17(22-11-5-7-12(24)8-6-11)9-16(14)26-15-4-2-3-13(20)18(15)19(23)25/h2-4,9-12,24H,5-8H2,1H3,(H,21,22)/t11-,12-	GFDDTDKCZCGJLM-HAQNSBGRSA-N	50559467	CHEMBL4763016	Bromodomain testis-specific protein	Homo sapiens			 170						ChEMBL	10.1016/j.bmc.2021.116015	10.7270/Q2TF021T	33549905			Sato, M; Kondo, T; Kohno, Y; Seto, S	Kyorin Pharmaceutical Co., Ltd	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50559467	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50559467&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			124182258	461829859							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51384901	CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12	InChI=1S/C22H22ClN5O2/c1-4-24-20(29)12-18-22-27-26-13(2)28(22)19-10-9-16(30-3)11-17(19)21(25-18)14-5-7-15(23)8-6-14/h5-11,18H,4,12H2,1-3H3,(H,24,29)/t18-/m0/s1	AAAQFGUYHFJNHI-SFHVURJKSA-N	50365463	CHEMBL1232461	Bromodomain testis-specific protein	Homo sapiens			 112						ChEMBL	10.1016/j.bmc.2021.116015	10.7270/Q2TF021T	33549905			Sato, M; Kondo, T; Kohno, Y; Seto, S	Kyorin Pharmaceutical Co., Ltd	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365463	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365463&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	EAM	5DFC,3P5O,2YEK,7AQT	46943432	136969525		CHEMBL1232461				ZINC58655571	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51384902	CN1c2cnc(N[C@H]3CC[C@H](O)CC3)cc2Oc2cccc(F)c2C1=O	InChI=1S/C19H20FN3O3/c1-23-14-10-21-17(22-11-5-7-12(24)8-6-11)9-16(14)26-15-4-2-3-13(20)18(15)19(23)25/h2-4,9-12,24H,5-8H2,1H3,(H,21,22)/t11-,12-	GFDDTDKCZCGJLM-HAQNSBGRSA-N	50559467	CHEMBL4763016	Bromodomain testis-specific protein	Homo sapiens			 220						ChEMBL	10.1016/j.bmc.2021.116015	10.7270/Q2TF021T	33549905			Sato, M; Kondo, T; Kohno, Y; Seto, S	Kyorin Pharmaceutical Co., Ltd	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50559467	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50559467&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			124182258	461829859							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51384903	CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12	InChI=1S/C22H22ClN5O2/c1-4-24-20(29)12-18-22-27-26-13(2)28(22)19-10-9-16(30-3)11-17(19)21(25-18)14-5-7-15(23)8-6-14/h5-11,18H,4,12H2,1-3H3,(H,24,29)/t18-/m0/s1	AAAQFGUYHFJNHI-SFHVURJKSA-N	50365463	CHEMBL1232461	Bromodomain testis-specific protein	Homo sapiens			 60						ChEMBL	10.1016/j.bmc.2021.116015	10.7270/Q2TF021T	33549905			Sato, M; Kondo, T; Kohno, Y; Seto, S	Kyorin Pharmaceutical Co., Ltd	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365463	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365463&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	EAM	5DFC,3P5O,2YEK,7AQT	46943432	136969525		CHEMBL1232461				ZINC58655571	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51386430	CN1CC[C@@H](Nc2ncc(-c3ccco3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)C(=O)NC1CCCCC1	InChI=1S/C26H33N5O3/c1-16-13-18-19(22-9-6-12-34-22)14-27-24(23(18)30-25(16)32)29-21-10-11-31(2)15-20(21)26(33)28-17-7-4-3-5-8-17/h6,9,12-14,17,20-21H,3-5,7-8,10-11,15H2,1-2H3,(H,27,29)(H,28,33)(H,30,32)/t20-,21-/m1/s1	NDEORODKVUYMFQ-NHCUHLMSSA-N	50560174	GSK789	Bromodomain testis-specific protein	Homo sapiens			 20						ChEMBL	10.1021/acs.jmedchem.0c00614	10.7270/Q27D2ZVG	32691589			Watson, RJ; Bamborough, P; Barnett, H; Chung, CW; Davis, R; Gordon, L; Grandi, P; Petretich, M; Phillipou, A; Prinjha, RK; Rioja, I; Soden, P; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50560174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50560174&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QAN	6Z7L	146681130	461830566							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51386434	CN1CC[C@@H](Nc2ncc(-c3ccco3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)C(=O)NC1CCCCC1	InChI=1S/C26H33N5O3/c1-16-13-18-19(22-9-6-12-34-22)14-27-24(23(18)30-25(16)32)29-21-10-11-31(2)15-20(21)26(33)28-17-7-4-3-5-8-17/h6,9,12-14,17,20-21H,3-5,7-8,10-11,15H2,1-2H3,(H,27,29)(H,28,33)(H,30,32)/t20-,21-/m1/s1	NDEORODKVUYMFQ-NHCUHLMSSA-N	50560174	GSK789	Bromodomain testis-specific protein	Homo sapiens			 19953						ChEMBL	10.1021/acs.jmedchem.0c00614	10.7270/Q27D2ZVG	32691589			Watson, RJ; Bamborough, P; Barnett, H; Chung, CW; Davis, R; Gordon, L; Grandi, P; Petretich, M; Phillipou, A; Prinjha, RK; Rioja, I; Soden, P; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50560174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50560174&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QAN	6Z7L	146681130	461830566							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51386440	CN1CC[C@@H](Nc2ncc(-c3ccco3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)C(=O)NC1CCCCC1	InChI=1S/C26H33N5O3/c1-16-13-18-19(22-9-6-12-34-22)14-27-24(23(18)30-25(16)32)29-21-10-11-31(2)15-20(21)26(33)28-17-7-4-3-5-8-17/h6,9,12-14,17,20-21H,3-5,7-8,10-11,15H2,1-2H3,(H,27,29)(H,28,33)(H,30,32)/t20-,21-/m1/s1	NDEORODKVUYMFQ-NHCUHLMSSA-N	50560174	GSK789	Bromodomain testis-specific protein	Homo sapiens			 10.0						ChEMBL	10.1021/acs.jmedchem.0c00614	10.7270/Q27D2ZVG	32691589			Watson, RJ; Bamborough, P; Barnett, H; Chung, CW; Davis, R; Gordon, L; Grandi, P; Petretich, M; Phillipou, A; Prinjha, RK; Rioja, I; Soden, P; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50560174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50560174&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QAN	6Z7L	146681130	461830566							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51386442	CN1CC[C@@H](Nc2ncc(-c3ccco3)c3cc(C)c(=O)[nH]c23)[C@@H](C1)C(=O)NC1CCCCC1	InChI=1S/C26H33N5O3/c1-16-13-18-19(22-9-6-12-34-22)14-27-24(23(18)30-25(16)32)29-21-10-11-31(2)15-20(21)26(33)28-17-7-4-3-5-8-17/h6,9,12-14,17,20-21H,3-5,7-8,10-11,15H2,1-2H3,(H,27,29)(H,28,33)(H,30,32)/t20-,21-/m1/s1	NDEORODKVUYMFQ-NHCUHLMSSA-N	50560174	GSK789	Bromodomain testis-specific protein	Homo sapiens			<31623						ChEMBL	10.1021/acs.jmedchem.0c00614	10.7270/Q27D2ZVG	32691589			Watson, RJ; Bamborough, P; Barnett, H; Chung, CW; Davis, R; Gordon, L; Grandi, P; Petretich, M; Phillipou, A; Prinjha, RK; Rioja, I; Soden, P; Werner, T; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50560174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50560174&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	QAN	6Z7L	146681130	461830566							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51350670	C[C@H](Oc1cc(cc(F)c1NC(C)=O)C(=O)N[C@H]1CC[C@H](O)CC1)c1ccccc1	InChI=1S/C23H27FN2O4/c1-14(16-6-4-3-5-7-16)30-21-13-17(12-20(24)22(21)25-15(2)27)23(29)26-18-8-10-19(28)11-9-18/h3-7,12-14,18-19,28H,8-11H2,1-2H3,(H,25,27)(H,26,29)/t14-,18-,19-/m0/s1	FRBRZGLUFOZRGD-JVPBZIDWSA-N	50544300	GSK046	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.0c00605	10.7270/Q2XP78HK	32691591			Preston, A; Atkinson, S; Bamborough, P; Chung, CW; Craggs, PD; Gordon, L; Grandi, P; Gray, JRJ; Jones, EJ; Lindon, M; Michon, AM; Mitchell, DJ; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, J; Taylor, S; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544300&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	LW5	6SWP,6SWQ	146018690	442145863							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51350671	C[C@H](Oc1cc(cc(F)c1NC(C)=O)C(=O)N[C@H]1CC[C@H](O)CC1)c1ccccc1	InChI=1S/C23H27FN2O4/c1-14(16-6-4-3-5-7-16)30-21-13-17(12-20(24)22(21)25-15(2)27)23(29)26-18-8-10-19(28)11-9-18/h3-7,12-14,18-19,28H,8-11H2,1-2H3,(H,25,27)(H,26,29)/t14-,18-,19-/m0/s1	FRBRZGLUFOZRGD-JVPBZIDWSA-N	50544300	GSK046	Bromodomain testis-specific protein	Homo sapiens		 200							ChEMBL	10.1021/acs.jmedchem.0c00605	10.7270/Q2XP78HK	32691591			Preston, A; Atkinson, S; Bamborough, P; Chung, CW; Craggs, PD; Gordon, L; Grandi, P; Gray, JRJ; Jones, EJ; Lindon, M; Michon, AM; Mitchell, DJ; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, J; Taylor, S; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50544300	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50544300&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	LW5	6SWP,6SWQ	146018690	442145863							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50886309	Cc1noc(C)c1-c1ccc2nc(nc(N3CCOC[C@@H]3c3ccccc3)c2c1)-c1cnn(CC(C)(C)O)c1	InChI=1S/C30H32N6O3/c1-19-27(20(2)39-34-19)22-10-11-25-24(14-22)29(36-12-13-38-17-26(36)21-8-6-5-7-9-21)33-28(32-25)23-15-31-35(16-23)18-30(3,4)37/h5-11,14-16,26,37H,12-13,17-18H2,1-4H3/t26-/m1/s1	SUFVOUWYHJXPBW-AREMUKBSSA-N	50545912	CHEMBL4749664	Bromodomain testis-specific protein	Homo sapiens			 76						ChEMBL	10.1016/j.bmcl.2019.03.014	10.7270/Q2FT8QMQ	30905542			Yang, SM; Yoshioka, M; Strovel, JW; Urban, DJ; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50545912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50545912&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JBS	6MAU	129166067	461689675							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50886310	Cc1noc(C)c1-c1ccc2nc(nc(N3CCOC[C@@H]3c3ccccc3)c2c1)-c1cnn(CC(C)(C)O)c1	InChI=1S/C30H32N6O3/c1-19-27(20(2)39-34-19)22-10-11-25-24(14-22)29(36-12-13-38-17-26(36)21-8-6-5-7-9-21)33-28(32-25)23-15-31-35(16-23)18-30(3,4)37/h5-11,14-16,26,37H,12-13,17-18H2,1-4H3/t26-/m1/s1	SUFVOUWYHJXPBW-AREMUKBSSA-N	50545912	CHEMBL4749664	Bromodomain testis-specific protein	Homo sapiens			 160						ChEMBL	10.1016/j.bmcl.2019.03.014	10.7270/Q2FT8QMQ	30905542			Yang, SM; Yoshioka, M; Strovel, JW; Urban, DJ; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50545912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50545912&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JBS	6MAU	129166067	461689675							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
50886311	Cc1noc(C)c1-c1ccc2nc(nc(N3CCOC[C@@H]3c3ccccc3)c2c1)-c1cnn(CC(C)(C)O)c1	InChI=1S/C30H32N6O3/c1-19-27(20(2)39-34-19)22-10-11-25-24(14-22)29(36-12-13-38-17-26(36)21-8-6-5-7-9-21)33-28(32-25)23-15-31-35(16-23)18-30(3,4)37/h5-11,14-16,26,37H,12-13,17-18H2,1-4H3/t26-/m1/s1	SUFVOUWYHJXPBW-AREMUKBSSA-N	50545912	CHEMBL4749664	Bromodomain testis-specific protein	Homo sapiens			 170						ChEMBL	10.1016/j.bmcl.2019.03.014	10.7270/Q2FT8QMQ	30905542			Yang, SM; Yoshioka, M; Strovel, JW; Urban, DJ; Hu, X; Hall, MD; Jadhav, A; Maloney, DJ	National Institutes of Health	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50545912	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50545912&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JBS	6MAU	129166067	461689675							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51402742	CNC(=O)c1cc(cc(n1)C(O)c1ccccc1)C(=O)N[C@H]1C[C@@H]1C	InChI=1S/C19H21N3O3/c1-11-8-14(11)22-18(24)13-9-15(21-16(10-13)19(25)20-2)17(23)12-6-4-3-5-7-12/h3-7,9-11,14,17,23H,8H2,1-2H3,(H,20,25)(H,22,24)/t11-,14-,17?/m0/s1	OJSKWCXPUVTNCF-UKOIWPHMSA-N	50566697	CHEMBL4862372	Bromodomain testis-specific protein	Homo sapiens		 25119							ChEMBL	10.1021/acs.jmedchem.0c02155	10.7270/Q2JH3QXP	34232650			Harrison, LA; Atkinson, SJ; Bassil, A; Chung, CW; Grandi, P; Gray, JRJ; Levernier, E; Lewis, A; Lugo, D; Messenger, C; Michon, AM; Mitchell, DJ; Preston, A; Prinjha, RK; Rioja, I; Seal, JT; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50566697	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50566697&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186095	471056842							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51402743	CNC(=O)c1cc(cc(n1)C(O)c1ccccc1)C(=O)N[C@H]1C[C@@H]1C	InChI=1S/C19H21N3O3/c1-11-8-14(11)22-18(24)13-9-15(21-16(10-13)19(25)20-2)17(23)12-6-4-3-5-7-12/h3-7,9-11,14,17,23H,8H2,1-2H3,(H,20,25)(H,22,24)/t11-,14-,17?/m0/s1	OJSKWCXPUVTNCF-UKOIWPHMSA-N	50566697	CHEMBL4862372	Bromodomain testis-specific protein	Homo sapiens		 25							ChEMBL	10.1021/acs.jmedchem.0c02155	10.7270/Q2JH3QXP	34232650			Harrison, LA; Atkinson, SJ; Bassil, A; Chung, CW; Grandi, P; Gray, JRJ; Levernier, E; Lewis, A; Lugo, D; Messenger, C; Michon, AM; Mitchell, DJ; Preston, A; Prinjha, RK; Rioja, I; Seal, JT; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50566697	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50566697&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186095	471056842							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51402750	CNC(=O)c1cc(cc(n1)C(O)c1ccccc1)C(=O)N[C@H]1C[C@@H]1C	InChI=1S/C19H21N3O3/c1-11-8-14(11)22-18(24)13-9-15(21-16(10-13)19(25)20-2)17(23)12-6-4-3-5-7-12/h3-7,9-11,14,17,23H,8H2,1-2H3,(H,20,25)(H,22,24)/t11-,14-,17?/m0/s1	OJSKWCXPUVTNCF-UKOIWPHMSA-N	50566697	CHEMBL4862372	Bromodomain testis-specific protein	Homo sapiens			 25119						ChEMBL	10.1021/acs.jmedchem.0c02155	10.7270/Q2JH3QXP	34232650			Harrison, LA; Atkinson, SJ; Bassil, A; Chung, CW; Grandi, P; Gray, JRJ; Levernier, E; Lewis, A; Lugo, D; Messenger, C; Michon, AM; Mitchell, DJ; Preston, A; Prinjha, RK; Rioja, I; Seal, JT; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50566697	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50566697&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186095	471056842							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51402751	CNC(=O)c1cc(cc(n1)C(O)c1ccccc1)C(=O)N[C@H]1C[C@@H]1C	InChI=1S/C19H21N3O3/c1-11-8-14(11)22-18(24)13-9-15(21-16(10-13)19(25)20-2)17(23)12-6-4-3-5-7-12/h3-7,9-11,14,17,23H,8H2,1-2H3,(H,20,25)(H,22,24)/t11-,14-,17?/m0/s1	OJSKWCXPUVTNCF-UKOIWPHMSA-N	50566697	CHEMBL4862372	Bromodomain testis-specific protein	Homo sapiens			 2.0						ChEMBL	10.1021/acs.jmedchem.0c02155	10.7270/Q2JH3QXP	34232650			Harrison, LA; Atkinson, SJ; Bassil, A; Chung, CW; Grandi, P; Gray, JRJ; Levernier, E; Lewis, A; Lugo, D; Messenger, C; Michon, AM; Mitchell, DJ; Preston, A; Prinjha, RK; Rioja, I; Seal, JT; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50566697	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50566697&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			132186095	471056842							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51424999	CCNC(=O)c1ccc(OCc2cccc(C)n2)c(c1)-c1cn(C)nn1	InChI=1S/C19H21N5O2/c1-4-20-19(25)14-8-9-18(16(10-14)17-11-24(3)23-22-17)26-12-15-7-5-6-13(2)21-15/h5-11H,4,12H2,1-3H3,(H,20,25)	BHUOTMULUBCHII-UHFFFAOYSA-N	50575643	CHEMBL4856289	Bromodomain testis-specific protein	Homo sapiens		 398							ChEMBL	10.1021/acs.jmedchem.0c02156	10.7270/Q2F193JT	33662213			Aylott, HE; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, JT; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50575643	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50575643&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164613009	471051766							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51425000	CCNC(=O)c1cc(Cc2cccc3[nH]ccc23)nc(c1)-c1cn(C)nn1	InChI=1S/C20H20N6O/c1-3-21-20(27)14-10-15(23-18(11-14)19-12-26(2)25-24-19)9-13-5-4-6-17-16(13)7-8-22-17/h4-8,10-12,22H,3,9H2,1-2H3,(H,21,27)	MMMRGZLSUKMQOD-UHFFFAOYSA-N	50575644	CHEMBL4856853	Bromodomain testis-specific protein	Homo sapiens		 50							ChEMBL	10.1021/acs.jmedchem.0c02156	10.7270/Q2F193JT	33662213			Aylott, HE; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, JT; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50575644	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50575644&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164614664	471051767							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51425001	CCNC(=O)c1ccc(OCc2cccc(C)n2)c(c1)-c1cn(C)nn1	InChI=1S/C19H21N5O2/c1-4-20-19(25)14-8-9-18(16(10-14)17-11-24(3)23-22-17)26-12-15-7-5-6-13(2)21-15/h5-11H,4,12H2,1-3H3,(H,20,25)	BHUOTMULUBCHII-UHFFFAOYSA-N	50575643	CHEMBL4856289	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.0c02156	10.7270/Q2F193JT	33662213			Aylott, HE; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, JT; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50575643	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50575643&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164613009	471051766							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51425002	CCNC(=O)c1cc(Cc2cccc3[nH]ccc23)nc(c1)-c1cn(C)nn1	InChI=1S/C20H20N6O/c1-3-21-20(27)14-10-15(23-18(11-14)19-12-26(2)25-24-19)9-13-5-4-6-17-16(13)7-8-22-17/h4-8,10-12,22H,3,9H2,1-2H3,(H,21,27)	MMMRGZLSUKMQOD-UHFFFAOYSA-N	50575644	CHEMBL4856853	Bromodomain testis-specific protein	Homo sapiens		 25119							ChEMBL	10.1021/acs.jmedchem.0c02156	10.7270/Q2F193JT	33662213			Aylott, HE; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Hayhow, TG; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Seal, JT; Wall, ID; Watson, RJ; Woolven, JM; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50575644	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50575644&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164614664	471051767							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426944	CNC(=O)c1cc(C(=O)N[C@H]2CC[C@H](O)CC2)n(n1)[C@@H](C)c1ccccc1	InChI=1S/C20H26N4O3/c1-13(14-6-4-3-5-7-14)24-18(12-17(23-24)19(26)21-2)20(27)22-15-8-10-16(25)11-9-15/h3-7,12-13,15-16,25H,8-11H2,1-2H3,(H,21,26)(H,22,27)/t13-,15-,16-/m0/s1	LEXSRVMWXAFLMV-BPUTZDHNSA-N	50576426	CHEMBL4854042	Bromodomain testis-specific protein	Homo sapiens		 79							ChEMBL	10.1021/acs.jmedchem.1c00365	10.7270/Q21N84ZQ	34255512			Seal, JT; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Foley, J; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Kruger, RG; Matteo, JJ; McCabe, MT; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Wyce, A; Zhang, XP; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576426	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576426&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	V9H	7OE5	142417949	471052549							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426945	CNC(=O)c1cc(C(=O)N[C@H]2CC[C@H](O)CC2)c(o1)[C@@H](C)c1ccccc1	InChI=1S/C21H26N2O4/c1-13(14-6-4-3-5-7-14)19-17(12-18(27-19)21(26)22-2)20(25)23-15-8-10-16(24)11-9-15/h3-7,12-13,15-16,24H,8-11H2,1-2H3,(H,22,26)(H,23,25)/t13-,15-,16-/m0/s1	BRAMSTZRKUJRKS-BPUTZDHNSA-N	50576427	CHEMBL4865767	Bromodomain testis-specific protein	Homo sapiens		 25							ChEMBL	10.1021/acs.jmedchem.1c00365	10.7270/Q21N84ZQ	34255512			Seal, JT; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Foley, J; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Kruger, RG; Matteo, JJ; McCabe, MT; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Wyce, A; Zhang, XP; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576427	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576427&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	V9K	7OE6	146434124	471052550							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426946	CNC(=O)c1cc(C(=O)N[C@H]2CC[C@H](O)CC2)n(n1)[C@@H](C)c1ccccc1	InChI=1S/C20H26N4O3/c1-13(14-6-4-3-5-7-14)24-18(12-17(23-24)19(26)21-2)20(27)22-15-8-10-16(25)11-9-15/h3-7,12-13,15-16,25H,8-11H2,1-2H3,(H,21,26)(H,22,27)/t13-,15-,16-/m0/s1	LEXSRVMWXAFLMV-BPUTZDHNSA-N	50576426	CHEMBL4854042	Bromodomain testis-specific protein	Homo sapiens		<50119							ChEMBL	10.1021/acs.jmedchem.1c00365	10.7270/Q21N84ZQ	34255512			Seal, JT; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Foley, J; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Kruger, RG; Matteo, JJ; McCabe, MT; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Wyce, A; Zhang, XP; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576426	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576426&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	V9H	7OE5	142417949	471052549							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426947	CNC(=O)c1cc(C(=O)N[C@H]2CC[C@H](O)CC2)c(o1)[C@@H](C)c1ccccc1	InChI=1S/C21H26N2O4/c1-13(14-6-4-3-5-7-14)19-17(12-18(27-19)21(26)22-2)20(25)23-15-8-10-16(24)11-9-15/h3-7,12-13,15-16,24H,8-11H2,1-2H3,(H,22,26)(H,23,25)/t13-,15-,16-/m0/s1	BRAMSTZRKUJRKS-BPUTZDHNSA-N	50576427	CHEMBL4865767	Bromodomain testis-specific protein	Homo sapiens		 39811							ChEMBL	10.1021/acs.jmedchem.1c00365	10.7270/Q21N84ZQ	34255512			Seal, JT; Atkinson, SJ; Bamborough, P; Bassil, A; Chung, CW; Foley, J; Gordon, L; Grandi, P; Gray, JRJ; Harrison, LA; Kruger, RG; Matteo, JJ; McCabe, MT; Messenger, C; Mitchell, D; Phillipou, A; Preston, A; Prinjha, RK; Rianjongdee, F; Rioja, I; Taylor, S; Wall, ID; Watson, RJ; Woolven, JM; Wyce, A; Zhang, XP; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576427	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576427&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	V9K	7OE6	146434124	471052550							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426966	CNC(=O)c1cc(cc2c1OC[C@@]2(C)c1ccccc1)C(=O)N[C@@H]1[C@H]2C[C@H](O)C[C@@H]12	InChI=1S/C24H26N2O4/c1-24(14-6-4-3-5-7-14)12-30-21-18(23(29)25-2)8-13(9-19(21)24)22(28)26-20-16-10-15(27)11-17(16)20/h3-9,15-17,20,27H,10-12H2,1-2H3,(H,25,29)(H,26,28)/t15-,16-,17+,20+,24-/m0/s1	FNHHVPPSBFQMEL-HURDOVMISA-N	50576438	CHEMBL4869149	Bromodomain testis-specific protein	Homo sapiens		 1.6							ChEMBL	10.1021/acs.jmedchem.1c00344	10.7270/Q2S46WSG	34260229			Lucas, SCC; Atkinson, SJ; Chung, CW; Davis, R; Gordon, L; Grandi, P; Gray, JJR; Grimes, T; Phillipou, A; Preston, AG; Prinjha, RK; Rioja, I; Taylor, S; Tomkinson, NCO; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138533986	471052561							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426967	CNC(=O)c1cc(cc2c1OC[C@@]2(C)c1ccccc1)C(=O)N[C@@H]1[C@H]2C[C@H](O)C[C@@H]12	InChI=1S/C24H26N2O4/c1-24(14-6-4-3-5-7-14)12-30-21-18(23(29)25-2)8-13(9-19(21)24)22(28)26-20-16-10-15(27)11-17(16)20/h3-9,15-17,20,27H,10-12H2,1-2H3,(H,25,29)(H,26,28)/t15-,16-,17+,20+,24-/m0/s1	FNHHVPPSBFQMEL-HURDOVMISA-N	50576438	CHEMBL4869149	Bromodomain testis-specific protein	Homo sapiens		 15849							ChEMBL	10.1021/acs.jmedchem.1c00344	10.7270/Q2S46WSG	34260229			Lucas, SCC; Atkinson, SJ; Chung, CW; Davis, R; Gordon, L; Grandi, P; Gray, JJR; Grimes, T; Phillipou, A; Preston, AG; Prinjha, RK; Rioja, I; Taylor, S; Tomkinson, NCO; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138533986	471052561							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426974	CNC(=O)c1cc(cc2c1OC[C@@]2(C)c1ccccc1)C(=O)N[C@@H]1[C@H]2C[C@H](O)C[C@@H]12	InChI=1S/C24H26N2O4/c1-24(14-6-4-3-5-7-14)12-30-21-18(23(29)25-2)8-13(9-19(21)24)22(28)26-20-16-10-15(27)11-17(16)20/h3-9,15-17,20,27H,10-12H2,1-2H3,(H,25,29)(H,26,28)/t15-,16-,17+,20+,24-/m0/s1	FNHHVPPSBFQMEL-HURDOVMISA-N	50576438	CHEMBL4869149	Bromodomain testis-specific protein	Homo sapiens		 19953							ChEMBL	10.1021/acs.jmedchem.1c00344	10.7270/Q2S46WSG	34260229			Lucas, SCC; Atkinson, SJ; Chung, CW; Davis, R; Gordon, L; Grandi, P; Gray, JJR; Grimes, T; Phillipou, A; Preston, AG; Prinjha, RK; Rioja, I; Taylor, S; Tomkinson, NCO; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138533986	471052561							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51426975	CNC(=O)c1cc(cc2c1OC[C@@]2(C)c1ccccc1)C(=O)N[C@@H]1[C@H]2C[C@H](O)C[C@@H]12	InChI=1S/C24H26N2O4/c1-24(14-6-4-3-5-7-14)12-30-21-18(23(29)25-2)8-13(9-19(21)24)22(28)26-20-16-10-15(27)11-17(16)20/h3-9,15-17,20,27H,10-12H2,1-2H3,(H,25,29)(H,26,28)/t15-,16-,17+,20+,24-/m0/s1	FNHHVPPSBFQMEL-HURDOVMISA-N	50576438	CHEMBL4869149	Bromodomain testis-specific protein	Homo sapiens		 7.9							ChEMBL	10.1021/acs.jmedchem.1c00344	10.7270/Q2S46WSG	34260229			Lucas, SCC; Atkinson, SJ; Chung, CW; Davis, R; Gordon, L; Grandi, P; Gray, JJR; Grimes, T; Phillipou, A; Preston, AG; Prinjha, RK; Rioja, I; Taylor, S; Tomkinson, NCO; Wall, I; Watson, RJ; Woolven, J; Demont, EH	GlaxoSmithKline	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50576438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50576438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138533986	471052561							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453813	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1ccc(OCC(=O)Nc2ccc(N3CCN(C)CC3)c(Cl)c2)cc1	InChI=1S/C29H30ClN5O5/c1-34-10-12-35(13-11-34)24-9-6-19(14-22(24)30)31-26(36)17-40-20-7-4-18(5-8-20)28-32-23-15-21(38-2)16-25(39-3)27(23)29(37)33-28/h4-9,14-16H,10-13,17H2,1-3H3,(H,31,36)(H,32,33,37)	UZWCUBDJHDWTFV-UHFFFAOYSA-N	50587013	CHEMBL5091216	Bromodomain testis-specific protein	Homo sapiens		>10000							ChEMBL	10.1021/acs.jmedchem.1c01382	10.7270/Q25D8WRZ	34908415			Zhang, J; Tang, P; Zou, L; Zhang, J; Chen, J; Yang, C; He, G; Liu, B; Liu, J; Chiang, CM; Wang, G; Ye, T; Ouyang, L	Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50587013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50587013&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			162641712	476023100							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453814	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 207							ChEMBL	10.1021/acs.jmedchem.1c01382	10.7270/Q25D8WRZ	34908415			Zhang, J; Tang, P; Zou, L; Zhang, J; Chen, J; Yang, C; He, G; Liu, B; Liu, J; Chiang, CM; Wang, G; Ye, T; Ouyang, L	Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453815	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1ccc(OCC(=O)Nc2ccc(N3CCN(C)CC3)c(Cl)c2)cc1	InChI=1S/C29H30ClN5O5/c1-34-10-12-35(13-11-34)24-9-6-19(14-22(24)30)31-26(36)17-40-20-7-4-18(5-8-20)28-32-23-15-21(38-2)16-25(39-3)27(23)29(37)33-28/h4-9,14-16H,10-13,17H2,1-3H3,(H,31,36)(H,32,33,37)	UZWCUBDJHDWTFV-UHFFFAOYSA-N	50587013	CHEMBL5091216	Bromodomain testis-specific protein	Homo sapiens		>10000							ChEMBL	10.1021/acs.jmedchem.1c01382	10.7270/Q25D8WRZ	34908415			Zhang, J; Tang, P; Zou, L; Zhang, J; Chen, J; Yang, C; He, G; Liu, B; Liu, J; Chiang, CM; Wang, G; Ye, T; Ouyang, L	Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50587013	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50587013&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			162641712	476023100							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453816	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 185							ChEMBL	10.1021/acs.jmedchem.1c01382	10.7270/Q25D8WRZ	34908415			Zhang, J; Tang, P; Zou, L; Zhang, J; Chen, J; Yang, C; He, G; Liu, B; Liu, J; Chiang, CM; Wang, G; Ye, T; Ouyang, L	Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446453	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 178							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446454	FC(F)(F)c1ccc(NC(=O)Nc2ccc(cc2)S(=O)(=O)N2CCC[C@H]2CN2CCOCC2)cc1	InChI=1S/C23H27F3N4O4S/c24-23(25,26)17-3-5-18(6-4-17)27-22(31)28-19-7-9-21(10-8-19)35(32,33)30-11-1-2-20(30)16-29-12-14-34-15-13-29/h3-10,20H,1-2,11-16H2,(H2,27,28,31)/t20-/m0/s1	ZPMULUKHFNMJPF-FQEVSTJZSA-N	50584382	CHEMBL5090401	Bromodomain testis-specific protein	Homo sapiens		 2416							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50584382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50584382&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	POJ	6U0D	135144027	476020469							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446455	OC1CCN(C[C@@H]2CCCN2S(=O)(=O)c2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2)CC1	InChI=1S/C24H29F3N4O4S/c25-24(26,27)17-3-5-18(6-4-17)28-23(33)29-19-7-9-22(10-8-19)36(34,35)31-13-1-2-20(31)16-30-14-11-21(32)12-15-30/h3-10,20-21,32H,1-2,11-16H2,(H2,28,29,33)/t20-/m0/s1	CFXFHVGCTLQYSO-FQEVSTJZSA-N	518799	US11117865, Compound ZL0591	Bromodomain testis-specific protein	Homo sapiens		 2217							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=518799	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=518799&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			135126198	461604814							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446456	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens		 5027							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446457	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 224							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446458	FC(F)(F)c1ccc(NC(=O)Nc2ccc(cc2)S(=O)(=O)N2CCC[C@H]2CN2CCOCC2)cc1	InChI=1S/C23H27F3N4O4S/c24-23(25,26)17-3-5-18(6-4-17)27-22(31)28-19-7-9-21(10-8-19)35(32,33)30-11-1-2-20(30)16-29-12-14-34-15-13-29/h3-10,20H,1-2,11-16H2,(H2,27,28,31)/t20-/m0/s1	ZPMULUKHFNMJPF-FQEVSTJZSA-N	50584382	CHEMBL5090401	Bromodomain testis-specific protein	Homo sapiens		 1902							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50584382	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50584382&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	POJ	6U0D	135144027	476020469							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446459	OC1CCN(C[C@@H]2CCCN2S(=O)(=O)c2ccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)cc2)CC1	InChI=1S/C24H29F3N4O4S/c25-24(26,27)17-3-5-18(6-4-17)28-23(33)29-19-7-9-22(10-8-19)36(34,35)31-13-1-2-20(31)16-30-14-11-21(32)12-15-30/h3-10,20-21,32H,1-2,11-16H2,(H2,28,29,33)/t20-/m0/s1	CFXFHVGCTLQYSO-FQEVSTJZSA-N	518799	US11117865, Compound ZL0591	Bromodomain testis-specific protein	Homo sapiens		 1987							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=518799	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=518799&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			135126198	461604814							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446460	COc1cc(OC)c2c(c1)nc([nH]c2=O)-c1cc(C)c(OCCO)c(C)c1	InChI=1S/C20H22N2O5/c1-11-7-13(8-12(2)18(11)27-6-5-23)19-21-15-9-14(25-3)10-16(26-4)17(15)20(24)22-19/h7-10,23H,5-6H2,1-4H3,(H,21,22,24)	NETXMUIMUZJUTB-UHFFFAOYSA-N	50103503	CHEMBL2393130::US11117865, Compound RVX-208	Bromodomain testis-specific protein	Homo sapiens		 696							ChEMBL	10.1021/acs.jmedchem.1c01851	10.7270/Q2HD80K2	34982556			Liu, Z; Li, Y; Chen, H; Lai, HT; Wang, P; Wu, SY; Wold, EA; Leonard, PG; Joseph, S; Hu, H; Chiang, CM; Brasier, AR; Tian, B; Zhou, J	MD Anderson Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50103503	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50103503&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1K0	4MR6,4MR5,4MR4,4MR3,4J1P,4J3I	122362584	318491278		CHEMBL2393130					1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51446527	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 120							ChEMBL	10.1021/acs.jmedchem.1c01779	10.7270/Q28056H6	35007061			Cui, H; Divakaran, A; Hoell, ZJ; Ellingson, MO; Scholtz, CR; Zahid, H; Johnson, JA; Griffith, EC; Gee, CT; Lee, AL; Khanal, S; Shi, K; Aihara, H; Shah, VH; Lee, RE; Harki, DA; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435487	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m1/s1	XQVVPGYIWAGRNI-JOCHJYFZSA-N	25121	4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide::BI 2536::CHEMBL513909::US10450297, Example 300::US8598172, 5	Bromodomain testis-specific protein	Homo sapiens			 240						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=25121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=25121&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	R78	4OGI,6MF9,6BQQ,7K0U,2RKU,6CW0,7LAI,4O74,4PY6,4I5M,5TCM,5C8G,5VBQ,7L9G,7L9L,7N7M	11364421	56374263		CHEMBL513909		5666		ZINC13986815	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435488	CC[C@H]1N(C(C)C)c2nc(Nc3ccc(cc3OC)C(=O)N[C@H]3CC[C@@H](CC3)N3CCN(CC4CC4)CC3)ncc2N(C)C1=O	InChI=1S/C34H50N8O3/c1-6-28-33(44)39(4)29-20-35-34(38-31(29)42(28)22(2)3)37-27-14-9-24(19-30(27)45-5)32(43)36-25-10-12-26(13-11-25)41-17-15-40(16-18-41)21-23-7-8-23/h9,14,19-20,22-23,25-26,28H,6-8,10-13,15-18,21H2,1-5H3,(H,36,43)(H,35,37,38)/t25-,26-,28-/m1/s1	SXNJFOWDRLKDSF-STROYTFGSA-N	50402023	BI 6727::VOLASERTIB	Bromodomain testis-specific protein	Homo sapiens			 1030						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50402023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50402023&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	IBI	7LEJ,7N7N,7LAK,3FC2,5VBR,5V67	10461508	163351047						ZINC39716290	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435489	COc1cc(ccc1Nc1ncc2N(C)C(=O)C(F)(F)CN(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C27H35F2N7O3/c1-34-12-10-18(11-13-34)31-24(37)17-8-9-20(22(14-17)39-3)32-26-30-15-21-23(33-26)36(19-6-4-5-7-19)16-27(28,29)25(38)35(21)2/h8-9,14-15,18-19H,4-7,10-13,16H2,1-3H3,(H,31,37)(H,30,32,33)	DJNZZLZKAXGMMC-UHFFFAOYSA-N	50435735	CHEMBL2392553	Bromodomain testis-specific protein	Homo sapiens			 1900						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50435735	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50435735&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	79C	7BJY,7LAJ,5VBP,7L9J,5TA8,7L72	25015677	175448052		CHEMBL2392553				ZINC96271651	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435490	COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C31H38N8O3/c1-35-15-17-38(18-16-35)22-11-13-39(14-12-22)29(40)21-9-10-24(27(19-21)42-4)33-31-32-20-26-28(34-31)36(2)25-8-6-5-7-23(25)30(41)37(26)3/h5-10,19-20,22H,11-18H2,1-4H3,(H,32,33,34)	IWMCPJZTADUIFX-UHFFFAOYSA-N	482157	BDBM50379529::LRRK2-IN-1::US11370796, Compound LRRK2-IN-1	Bromodomain testis-specific protein	Homo sapiens			 700						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=482157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=482157&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46843906	443551320							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435491	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C3CCCC3)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C36H46N8O3/c1-4-47-32-23-25(34(45)43-17-15-26(16-18-43)42-21-19-40(2)20-22-42)13-14-29(32)38-36-37-24-31-33(39-36)44(27-9-5-6-10-27)30-12-8-7-11-28(30)35(46)41(31)3/h7-8,11-14,23-24,26-27H,4-6,9-10,15-22H2,1-3H3,(H,37,38,39)	XVBGRTMNFNMINE-UHFFFAOYSA-N	50434070	CHEMBL2381340	Bromodomain testis-specific protein	Homo sapiens			 1600						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50434070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50434070&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	VYJ	7LEK,7LAU,7LAZ,7LBT,7L73,7K6G	71604307	175446387		CHEMBL2381340				ZINC96270216	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435492	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCC(O)CC1	InChI=1S/C26H30N6O3/c1-4-35-23-15-17(32-13-11-18(33)12-14-32)9-10-20(23)28-26-27-16-22-24(29-26)30(2)21-8-6-5-7-19(21)25(34)31(22)3/h5-10,15-16,18,33H,4,11-14H2,1-3H3,(H,27,28,29)	QAPAJIZPZGWAND-UHFFFAOYSA-N	50337134	2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5,11-dimethyl-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one::CHEMBL1673046::Scaffold, B46::US9266890, IV-6	Bromodomain testis-specific protein	Homo sapiens			 3500						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50337134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50337134&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	4WG	7K6H,5LRQ,5BYY	46843772	125087236	60325	CHEMBL1673046				ZINC64633932	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435493	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 260						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435494	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m1/s1	XQVVPGYIWAGRNI-JOCHJYFZSA-N	25121	4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide::BI 2536::CHEMBL513909::US10450297, Example 300::US8598172, 5	Bromodomain testis-specific protein	Homo sapiens			 105						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=25121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=25121&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	R78	4OGI,6MF9,6BQQ,7K0U,2RKU,6CW0,7LAI,4O74,4PY6,4I5M,5TCM,5C8G,5VBQ,7L9G,7L9L,7N7M	11364421	56374263		CHEMBL513909		5666		ZINC13986815	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435495	CC[C@H]1N(C(C)C)c2nc(Nc3ccc(cc3OC)C(=O)N[C@H]3CC[C@@H](CC3)N3CCN(CC4CC4)CC3)ncc2N(C)C1=O	InChI=1S/C34H50N8O3/c1-6-28-33(44)39(4)29-20-35-34(38-31(29)42(28)22(2)3)37-27-14-9-24(19-30(27)45-5)32(43)36-25-10-12-26(13-11-25)41-17-15-40(16-18-41)21-23-7-8-23/h9,14,19-20,22-23,25-26,28H,6-8,10-13,15-18,21H2,1-5H3,(H,36,43)(H,35,37,38)/t25-,26-,28-/m1/s1	SXNJFOWDRLKDSF-STROYTFGSA-N	50402023	BI 6727::VOLASERTIB	Bromodomain testis-specific protein	Homo sapiens			 113						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50402023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50402023&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	IBI	7LEJ,7N7N,7LAK,3FC2,5VBR,5V67	10461508	163351047						ZINC39716290	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435496	COc1cc(ccc1Nc1ncc2N(C)C(=O)C(F)(F)CN(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C27H35F2N7O3/c1-34-12-10-18(11-13-34)31-24(37)17-8-9-20(22(14-17)39-3)32-26-30-15-21-23(33-26)36(19-6-4-5-7-19)16-27(28,29)25(38)35(21)2/h8-9,14-15,18-19H,4-7,10-13,16H2,1-3H3,(H,31,37)(H,30,32,33)	DJNZZLZKAXGMMC-UHFFFAOYSA-N	50435735	CHEMBL2392553	Bromodomain testis-specific protein	Homo sapiens			 390						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50435735	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50435735&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	79C	7BJY,7LAJ,5VBP,7L9J,5TA8,7L72	25015677	175448052		CHEMBL2392553				ZINC96271651	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435497	COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C31H38N8O3/c1-35-15-17-38(18-16-35)22-11-13-39(14-12-22)29(40)21-9-10-24(27(19-21)42-4)33-31-32-20-26-28(34-31)36(2)25-8-6-5-7-23(25)30(41)37(26)3/h5-10,19-20,22H,11-18H2,1-4H3,(H,32,33,34)	IWMCPJZTADUIFX-UHFFFAOYSA-N	482157	BDBM50379529::LRRK2-IN-1::US11370796, Compound LRRK2-IN-1	Bromodomain testis-specific protein	Homo sapiens			 390						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=482157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=482157&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46843906	443551320							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435498	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C3CCCC3)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C36H46N8O3/c1-4-47-32-23-25(34(45)43-17-15-26(16-18-43)42-21-19-40(2)20-22-42)13-14-29(32)38-36-37-24-31-33(39-36)44(27-9-5-6-10-27)30-12-8-7-11-28(30)35(46)41(31)3/h7-8,11-14,23-24,26-27H,4-6,9-10,15-22H2,1-3H3,(H,37,38,39)	XVBGRTMNFNMINE-UHFFFAOYSA-N	50434070	CHEMBL2381340	Bromodomain testis-specific protein	Homo sapiens			 500						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50434070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50434070&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	VYJ	7LEK,7LAU,7LAZ,7LBT,7L73,7K6G	71604307	175446387		CHEMBL2381340				ZINC96270216	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435499	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCC(O)CC1	InChI=1S/C26H30N6O3/c1-4-35-23-15-17(32-13-11-18(33)12-14-32)9-10-20(23)28-26-27-16-22-24(29-26)30(2)21-8-6-5-7-19(21)25(34)31(22)3/h5-10,15-16,18,33H,4,11-14H2,1-3H3,(H,27,28,29)	QAPAJIZPZGWAND-UHFFFAOYSA-N	50337134	2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5,11-dimethyl-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one::CHEMBL1673046::Scaffold, B46::US9266890, IV-6	Bromodomain testis-specific protein	Homo sapiens			 675						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50337134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50337134&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	4WG	7K6H,5LRQ,5BYY	46843772	125087236	60325	CHEMBL1673046				ZINC64633932	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435500	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 22						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435501	CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O	InChI=1S/C28H39N7O3/c1-5-22-27(37)34(3)23-17-29-28(32-25(23)35(22)20-8-6-7-9-20)31-21-11-10-18(16-24(21)38-4)26(36)30-19-12-14-33(2)15-13-19/h10-11,16-17,19-20,22H,5-9,12-15H2,1-4H3,(H,30,36)(H,29,31,32)/t22-/m1/s1	XQVVPGYIWAGRNI-JOCHJYFZSA-N	25121	4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide::BI 2536::CHEMBL513909::US10450297, Example 300::US8598172, 5	Bromodomain testis-specific protein	Homo sapiens			 806						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=25121	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=25121&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	R78	4OGI,6MF9,6BQQ,7K0U,2RKU,6CW0,7LAI,4O74,4PY6,4I5M,5TCM,5C8G,5VBQ,7L9G,7L9L,7N7M	11364421	56374263		CHEMBL513909		5666		ZINC13986815	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435502	CC[C@H]1N(C(C)C)c2nc(Nc3ccc(cc3OC)C(=O)N[C@H]3CC[C@@H](CC3)N3CCN(CC4CC4)CC3)ncc2N(C)C1=O	InChI=1S/C34H50N8O3/c1-6-28-33(44)39(4)29-20-35-34(38-31(29)42(28)22(2)3)37-27-14-9-24(19-30(27)45-5)32(43)36-25-10-12-26(13-11-25)41-17-15-40(16-18-41)21-23-7-8-23/h9,14,19-20,22-23,25-26,28H,6-8,10-13,15-18,21H2,1-5H3,(H,36,43)(H,35,37,38)/t25-,26-,28-/m1/s1	SXNJFOWDRLKDSF-STROYTFGSA-N	50402023	BI 6727::VOLASERTIB	Bromodomain testis-specific protein	Homo sapiens			 1700						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50402023	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50402023&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	IBI	7LEJ,7N7N,7LAK,3FC2,5VBR,5V67	10461508	163351047						ZINC39716290	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435503	COc1cc(ccc1Nc1ncc2N(C)C(=O)C(F)(F)CN(C3CCCC3)c2n1)C(=O)NC1CCN(C)CC1	InChI=1S/C27H35F2N7O3/c1-34-12-10-18(11-13-34)31-24(37)17-8-9-20(22(14-17)39-3)32-26-30-15-21-23(33-26)36(19-6-4-5-7-19)16-27(28,29)25(38)35(21)2/h8-9,14-15,18-19H,4-7,10-13,16H2,1-3H3,(H,31,37)(H,30,32,33)	DJNZZLZKAXGMMC-UHFFFAOYSA-N	50435735	CHEMBL2392553	Bromodomain testis-specific protein	Homo sapiens			 1800						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50435735	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50435735&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	79C	7BJY,7LAJ,5VBP,7L9J,5TA8,7L72	25015677	175448052		CHEMBL2392553				ZINC96271651	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435504	COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C31H38N8O3/c1-35-15-17-38(18-16-35)22-11-13-39(14-12-22)29(40)21-9-10-24(27(19-21)42-4)33-31-32-20-26-28(34-31)36(2)25-8-6-5-7-23(25)30(41)37(26)3/h5-10,19-20,22H,11-18H2,1-4H3,(H,32,33,34)	IWMCPJZTADUIFX-UHFFFAOYSA-N	482157	BDBM50379529::LRRK2-IN-1::US11370796, Compound LRRK2-IN-1	Bromodomain testis-specific protein	Homo sapiens			 1700						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=482157	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=482157&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46843906	443551320							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435505	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C3CCCC3)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1	InChI=1S/C36H46N8O3/c1-4-47-32-23-25(34(45)43-17-15-26(16-18-43)42-21-19-40(2)20-22-42)13-14-29(32)38-36-37-24-31-33(39-36)44(27-9-5-6-10-27)30-12-8-7-11-28(30)35(46)41(31)3/h7-8,11-14,23-24,26-27H,4-6,9-10,15-22H2,1-3H3,(H,37,38,39)	XVBGRTMNFNMINE-UHFFFAOYSA-N	50434070	CHEMBL2381340	Bromodomain testis-specific protein	Homo sapiens			 2100						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50434070	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50434070&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	VYJ	7LEK,7LAU,7LAZ,7LBT,7L73,7K6G	71604307	175446387		CHEMBL2381340				ZINC96270216	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435506	CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCC(O)CC1	InChI=1S/C26H30N6O3/c1-4-35-23-15-17(32-13-11-18(33)12-14-32)9-10-20(23)28-26-27-16-22-24(29-26)30(2)21-8-6-5-7-19(21)25(34)31(22)3/h5-10,15-16,18,33H,4,11-14H2,1-3H3,(H,27,28,29)	QAPAJIZPZGWAND-UHFFFAOYSA-N	50337134	2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5,11-dimethyl-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6(11H)-one::CHEMBL1673046::Scaffold, B46::US9266890, IV-6	Bromodomain testis-specific protein	Homo sapiens			 4200						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50337134	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50337134&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	4WG	7K6H,5LRQ,5BYY	46843772	125087236	60325	CHEMBL1673046				ZINC64633932	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435507	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C28H35ClFN7O3S/c1-17-16-31-27(34-19-6-8-21(23(30)14-19)26(38)33-18-10-12-37(5)13-11-18)35-25(17)32-20-7-9-22(29)24(15-20)36-41(39,40)28(2,3)4/h6-9,14-16,18,36H,10-13H2,1-5H3,(H,33,38)(H2,31,32,34,35)	RBZRCEPYYVFROZ-UHFFFAOYSA-N	50557394	CHEMBL4760892::US11643396, Example SG3-179	Bromodomain testis-specific protein	Homo sapiens			 59						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50557394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50557394&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W2	5F63,7KO0,7LAY,6VNL	118889467	461696162							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51435508	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 188						ChEMBL	10.1021/acs.jmedchem.1c01096	10.7270/Q26H4N8M	34710325			Karim, RM; Bikowitz, MJ; Chan, A; Zhu, JY; Grassie, D; Becker, A; Berndt, N; Gunawan, S; Lawrence, NJ; Schönbrunn, E	Moffitt Cancer Center	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51448005	CC(C)[C@H]1NC(=O)[C@@H]2Cc3ccccc3[C@H]1N2C(=O)c1cc(NC2CCN(CC(C)(C)F)CC2)c2nnc(C)n2n1	InChI=1S/C30H39FN8O2/c1-17(2)25-26-21-9-7-6-8-19(21)14-24(28(40)33-25)38(26)29(41)23-15-22(27-35-34-18(3)39(27)36-23)32-20-10-12-37(13-11-20)16-30(4,5)31/h6-9,15,17,20,24-26,32H,10-14,16H2,1-5H3,(H,33,40)/t24-,25+,26+/m0/s1	NGXAMXNWIHBLBN-JIMJEQGWSA-N	50584925	CHEMBL5079885	Bromodomain testis-specific protein	Homo sapiens			 200						ChEMBL	10.1021/acs.jmedchem.1c01871	10.7270/Q2280CH8	35133824			Winter-Holt, JJ; Bardelle, C; Chiarparin, E; Dale, IL; Davey, PRJ; Davies, NL; Denz, C; Fillery, SM; Guérot, CM; Han, F; Hughes, SJ; Kulkarni, M; Liu, Z; Milbradt, A; Moss, TA; Niu, H; Patel, J; Rabow, AA; Schimpl, M; Shi, J; Sun, D; Yang, D; Guichard, S	AstraZeneca	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50584925	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50584925&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	96L	7Q6T	162422438	476021012							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1257009	Cc1nnc2C(Cc3nnc(o3)C3CC3)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H21ClN6OS/c1-11-12(2)32-23-19(11)20(14-6-8-16(24)9-7-14)25-17(21-28-26-13(3)30(21)23)10-18-27-29-22(31-18)15-4-5-15/h6-9,15,17H,4-5,10H2,1-3H3	JKLFTZFZNNCDAE-UHFFFAOYSA-N	592405	US11572371, Compound 20	Bromodomain testis-specific protein	Homo sapiens		 49.0							US Patent		10.7270/Q2SQ94BJ			US11572371	Fan, L; Xu, K; Chen, K; Wang, F; Wu, X; Luo, T; Zhang, S; Li, X; Chen, Y	HINOVA PHARMACEUTICALS INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=592405	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=592405&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			167844896	479270589							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1257013	CCOCc1nnc(CC2N=C(c3c(C)c(C)sc3-n3c(C)nnc23)c2ccc(Cl)cc2)o1	InChI=1S/C23H23ClN6O2S/c1-5-31-11-19-28-27-18(32-19)10-17-22-29-26-14(4)30(22)23-20(12(2)13(3)33-23)21(25-17)15-6-8-16(24)9-7-15/h6-9,17H,5,10-11H2,1-4H3	USNVRJYSAUJTNT-UHFFFAOYSA-N	592506	US11572371, Compound 6	Bromodomain testis-specific protein	Homo sapiens		 46.0							US Patent		10.7270/Q2SQ94BJ			US11572371	Fan, L; Xu, K; Chen, K; Wang, F; Wu, X; Luo, T; Zhang, S; Li, X; Chen, Y	HINOVA PHARMACEUTICALS INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=592506	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=592506&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			167844897	479270690							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1257017	CC(C)c1nnc(CC2N=C(c3c(C)c(C)sc3-n3c(C)nnc23)c2ccc(Cl)cc2)o1	InChI=1S/C23H23ClN6OS/c1-11(2)22-29-27-18(31-22)10-17-21-28-26-14(5)30(21)23-19(12(3)13(4)32-23)20(25-17)15-6-8-16(24)9-7-15/h6-9,11,17H,10H2,1-5H3	NHQWTZLQTWSZGU-UHFFFAOYSA-N	592507	US11572371, Compound 19	Bromodomain testis-specific protein	Homo sapiens		 51.0							US Patent		10.7270/Q2SQ94BJ			US11572371	Fan, L; Xu, K; Chen, K; Wang, F; Wu, X; Luo, T; Zhang, S; Li, X; Chen, Y	HINOVA PHARMACEUTICALS INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=592507	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=592507&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			167844898	479270691							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1257021	Cc1nnc2C(Cc3nnc(o3)C(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C24H25ClN6OS/c1-12-13(2)33-22-19(12)20(15-7-9-16(25)10-8-15)26-17(21-29-27-14(3)31(21)22)11-18-28-30-23(32-18)24(4,5)6/h7-10,17H,11H2,1-6H3	LLRPIXCDTAUFLE-UHFFFAOYSA-N	592508	US11572371, Compound 22	Bromodomain testis-specific protein	Homo sapiens		 46.0							US Patent		10.7270/Q2SQ94BJ			US11572371	Fan, L; Xu, K; Chen, K; Wang, F; Wu, X; Luo, T; Zhang, S; Li, X; Chen, Y	HINOVA PHARMACEUTICALS INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=592508	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=592508&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			167844899	479270692							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453569	CC[C@H]1N(C2CCCC2)c2nc(ncc2N(C)C1=O)N(C)c1ccc(cc1OC)-c1nc2c(cccc2[nH]1)C(N)=O			50586865	CHEMBL5084388	Bromodomain testis-specific protein	Homo sapiens		 1198							ChEMBL	10.1021/acs.jmedchem.1c01535	10.7270/Q22N566V	34813314			Wang, SP; Li, Y; Huang, SH; Wu, SQ; Gao, LL; Sun, Q; Lin, QW; Huang, L; Meng, LQ; Zou, Y; Zhu, QH; Xu, YG	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50586865	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50586865&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			166633451	476022952							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453570	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 588							ChEMBL	10.1021/acs.jmedchem.1c01535	10.7270/Q22N566V	34813314			Wang, SP; Li, Y; Huang, SH; Wu, SQ; Gao, LL; Sun, Q; Lin, QW; Huang, L; Meng, LQ; Zou, Y; Zhu, QH; Xu, YG	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453571	CC[C@H]1N(C2CCCC2)c2nc(ncc2N(C)C1=O)N(C)c1ccc(cc1OC)-c1nc2c(cccc2[nH]1)C(N)=O			50586865	CHEMBL5084388	Bromodomain testis-specific protein	Homo sapiens		 1401							ChEMBL	10.1021/acs.jmedchem.1c01535	10.7270/Q22N566V	34813314			Wang, SP; Li, Y; Huang, SH; Wu, SQ; Gao, LL; Sun, Q; Lin, QW; Huang, L; Meng, LQ; Zou, Y; Zhu, QH; Xu, YG	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50586865	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50586865&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			166633451	476022952							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51453572	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 325							ChEMBL	10.1021/acs.jmedchem.1c01535	10.7270/Q22N566V	34813314			Wang, SP; Li, Y; Huang, SH; Wu, SQ; Gao, LL; Sun, Q; Lin, QW; Huang, L; Meng, LQ; Zou, Y; Zhu, QH; Xu, YG	China Pharmaceutical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51440811	CN(C)CCN1CCC(CC1)n1nnc(C)c1-c1cccc(Oc2cc(C)cc(C)c2)n1	InChI=1S/C25H34N6O/c1-18-15-19(2)17-22(16-18)32-24-8-6-7-23(26-24)25-20(3)27-28-31(25)21-9-11-30(12-10-21)14-13-29(4)5/h6-8,15-17,21H,9-14H2,1-5H3	PIKWYDHWUKSWAQ-UHFFFAOYSA-N	50582040	CHEMBL5083660	Bromodomain testis-specific protein	Homo sapiens			 15						ChEMBL	10.1021/acs.jmedchem.1c00933	10.7270/Q2PR80VN	34236185			Cui, H; Carlson, AS; Schleiff, MA; Divakaran, A; Johnson, JA; Buchholz, CR; Zahid, H; Vail, NR; Shi, K; Aihara, H; Harki, DA; Miller, GP; Topczewski, JJ; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50582040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50582040&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZHS	7MLR	156022514	476027045							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51440819	CN(C)CCN1CCC(CC1)n1nnc(C)c1-c1cccc(Oc2cc(C)cc(C)c2)n1	InChI=1S/C25H34N6O/c1-18-15-19(2)17-22(16-18)32-24-8-6-7-23(26-24)25-20(3)27-28-31(25)21-9-11-30(12-10-21)14-13-29(4)5/h6-8,15-17,21H,9-14H2,1-5H3	PIKWYDHWUKSWAQ-UHFFFAOYSA-N	50582040	CHEMBL5083660	Bromodomain testis-specific protein	Homo sapiens			 250						ChEMBL	10.1021/acs.jmedchem.1c00933	10.7270/Q2PR80VN	34236185			Cui, H; Carlson, AS; Schleiff, MA; Divakaran, A; Johnson, JA; Buchholz, CR; Zahid, H; Vail, NR; Shi, K; Aihara, H; Harki, DA; Miller, GP; Topczewski, JJ; Pomerantz, WCK	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50582040	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50582040&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZHS	7MLR	156022514	476027045							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274624	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C28H35ClFN7O3S/c1-17-16-31-27(34-19-6-8-21(23(30)14-19)26(38)33-18-10-12-37(5)13-11-18)35-25(17)32-20-7-9-22(29)24(15-20)36-41(39,40)28(2,3)4/h6-9,14-16,18,36H,10-13H2,1-5H3,(H,33,38)(H2,31,32,34,35)	RBZRCEPYYVFROZ-UHFFFAOYSA-N	50557394	CHEMBL4760892::US11643396, Example SG3-179	Bromodomain testis-specific protein	Homo sapiens		 22.5							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50557394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50557394&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W2	5F63,7KO0,7LAY,6VNL	118889467	461696162							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274630	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C26H33ClFN7O2S/c1-17-16-29-25(31-18-7-9-23(21(28)14-18)35-12-10-34(5)11-13-35)32-24(17)30-19-6-8-20(27)22(15-19)33-38(36,37)26(2,3)4/h6-9,14-16,33H,10-13H2,1-5H3,(H2,29,30,31,32)	QHSBHADJYBAJTJ-UHFFFAOYSA-N	601877	US11643396, Example MA4-022-2	Bromodomain testis-specific protein	Homo sapiens		 19.0							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=601877	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=601877&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W1		124081171	482092963							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274636	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C26H34FN7O2S/c1-18-17-28-25(30-20-9-10-23(22(27)16-20)34-13-11-33(5)12-14-34)31-24(18)29-19-7-6-8-21(15-19)32-37(35,36)26(2,3)4/h6-10,15-17,32H,11-14H2,1-5H3,(H2,28,29,30,31)	OGJFKWUOCYNWAB-UHFFFAOYSA-N	601876	US11643396, Example MA4-022-1	Bromodomain testis-specific protein	Homo sapiens		 41.3							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=601876	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=601876&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W0		124081170	482092962							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274644	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1	InChI=1S/C26H34ClN7O2S/c1-18-17-28-25(30-19-6-9-21(10-7-19)34-14-12-33(5)13-15-34)31-24(18)29-20-8-11-22(27)23(16-20)32-37(35,36)26(2,3)4/h6-11,16-17,32H,12-15H2,1-5H3,(H2,28,29,30,31)	OKUXIUAKYDKHDY-UHFFFAOYSA-N	601857	US11643396, Example SG3-014	Bromodomain testis-specific protein	Homo sapiens		 27.8							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=601857	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=601857&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5VZ		124081169	482092943							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274652	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(NS(=O)(=O)C(C)(C)C)c3)n2)cc1	InChI=1S/C26H35N7O2S/c1-19-18-27-25(29-20-9-11-23(12-10-20)33-15-13-32(5)14-16-33)30-24(19)28-21-7-6-8-22(17-21)31-36(34,35)26(2,3)4/h6-12,17-18,31H,13-16H2,1-5H3,(H2,27,28,29,30)	ZFVWPEWZIRRFOU-UHFFFAOYSA-N	543516	US11279703, TABLE 6.119::US11279703, TABLE 6.128::US11279703, TABLE 6.149::US11279703, TABLE 6.154::US11279703, TABLE 6.168::US11279703, TABLE 6.181::US11279703, TABLE 6.194::US11279703, TABLE 6.199::US11279703, TABLE 6.204::US11279703, TABLE 6.215::US11279703, TABLE 6.244::US11279703, TABLE 6.262::US11279703, TABLE 6.276::US11279703, TABLE 6.298::US11279703, TABLE 6.307::US11279703, TABLE 6.314::US11279703, TABLE 6.319::US11279703, TABLE 6.328::US11279703, TABLE 6.37::US11643396, Example MA2-014	Bromodomain testis-specific protein	Homo sapiens		 29.1							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=543516	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=543516&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5VY	5F5Z	118889482	469686131							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
1274662	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(c3)S(=O)(=O)NC(C)(C)C)n2)cc1	InChI=1S/C26H35N7O2S/c1-19-18-27-25(29-20-9-11-22(12-10-20)33-15-13-32(5)14-16-33)30-24(19)28-21-7-6-8-23(17-21)36(34,35)31-26(2,3)4/h6-12,17-18,31H,13-16H2,1-5H3,(H2,27,28,29,30)	JVDOKQYTTYUYDV-UHFFFAOYSA-N	192755	TG101209::US11279703, TABLE 6.171::US11643396, Example TG101209	Bromodomain testis-specific protein	Homo sapiens		 290							US Patent		10.7270/Q2833WX4			US11643396	Schonbrunn, E; Lawrence, NJ; Lawrence, HR	H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC.	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=192755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=192755&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1M3	5HEZ,4O76,4JI9	16722832	317230231							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51455537	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C26H23ClN6O3S/c1-13-14(2)37-26-22(13)23(16-4-8-18(27)9-5-16)29-20(24-31-30-15(3)33(24)26)12-21(34)28-19-10-6-17(7-11-19)25(35)32-36/h4-11,20,36H,12H2,1-3H3,(H,28,34)(H,32,35)/t20-/m0/s1	JBPWXWQIGDWQHR-FQEVSTJZSA-N	50569836	CHEMBL4850926	Bromodomain testis-specific protein	Homo sapiens		 11							ChEMBL		10.7270/Q2RN3CS0	33229136			Ren, Q; Gao, W	The First Affiliated Hospital of Zhengzhou University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50569836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50569836&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			154716332	471059981							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51455538	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C26H23ClN6O3S/c1-13-14(2)37-26-22(13)23(16-4-8-18(27)9-5-16)29-20(24-31-30-15(3)33(24)26)12-21(34)28-19-10-6-17(7-11-19)25(35)32-36/h4-11,20,36H,12H2,1-3H3,(H,28,34)(H,32,35)/t20-/m0/s1	JBPWXWQIGDWQHR-FQEVSTJZSA-N	50569836	CHEMBL4850926	Bromodomain testis-specific protein	Homo sapiens		 11							ChEMBL		10.7270/Q2RN3CS0	33229136			Ren, Q; Gao, W	The First Affiliated Hospital of Zhengzhou University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50569836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50569836&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			154716332	471059981							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51456100	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C26H23ClN6O3S/c1-13-14(2)37-26-22(13)23(16-4-8-18(27)9-5-16)29-20(24-31-30-15(3)33(24)26)12-21(34)28-19-10-6-17(7-11-19)25(35)32-36/h4-11,20,36H,12H2,1-3H3,(H,28,34)(H,32,35)/t20-/m0/s1	JBPWXWQIGDWQHR-FQEVSTJZSA-N	50569836	CHEMBL4850926	Bromodomain testis-specific protein	Homo sapiens		 11							ChEMBL		10.7270/Q2K07870	33685790			Ren, Q; Gao, W	the First Affiliated Hospital of Zhengzhou University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50569836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50569836&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			154716332	471059981							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51456101	Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1	InChI=1S/C26H23ClN6O3S/c1-13-14(2)37-26-22(13)23(16-4-8-18(27)9-5-16)29-20(24-31-30-15(3)33(24)26)12-21(34)28-19-10-6-17(7-11-19)25(35)32-36/h4-11,20,36H,12H2,1-3H3,(H,28,34)(H,32,35)/t20-/m0/s1	JBPWXWQIGDWQHR-FQEVSTJZSA-N	50569836	CHEMBL4850926	Bromodomain testis-specific protein	Homo sapiens		 11							ChEMBL		10.7270/Q2K07870	33685790			Ren, Q; Gao, W	the First Affiliated Hospital of Zhengzhou University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50569836	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50569836&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			154716332	471059981							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473370	Cn1cc(-c2cccc(c2)N2CCCC2=O)c2ccccc2c1=O	InChI=1S/C20H18N2O2/c1-21-13-18(16-8-2-3-9-17(16)20(21)24)14-6-4-7-15(12-14)22-11-5-10-19(22)23/h2-4,6-9,12-13H,5,10-11H2,1H3	IQHRPUHKLPCOKF-UHFFFAOYSA-N	50594434	CHEMBL5170344	Bromodomain testis-specific protein	Homo sapiens			 875						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594434	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594434&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMM		164607239	482605286							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473371	CCS(=O)(=O)Nc1cccc(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C18H18N2O3S/c1-3-24(22,23)19-14-8-6-7-13(11-14)17-12-20(2)18(21)16-10-5-4-9-15(16)17/h4-12,19H,3H2,1-2H3	QIEVBHRUPLMWFP-UHFFFAOYSA-N	284968	N-[3-(2-methyl-1-oxoisoquinolin-4-yl) phenyl]ethanesulfonamide::US10023592, Example 13::US10941160, Example 13	Bromodomain testis-specific protein	Homo sapiens			 77						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=284968	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=284968&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMJ	7MRH,7MRA	118021879	378168616							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473372	CCS(=O)(=O)Nc1ccc(Oc2ccc(Cl)cc2)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C24H21ClN2O4S/c1-3-32(29,30)26-17-10-13-23(31-18-11-8-16(25)9-12-18)21(14-17)22-15-27(2)24(28)20-7-5-4-6-19(20)22/h4-15,26H,3H2,1-2H3	LMYMWXJBPLXESU-UHFFFAOYSA-N	50594435	CHEMBL5184876	Bromodomain testis-specific protein	Homo sapiens			 5.0						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594435	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594435&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	N49		164607223	482605287							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473373	CCS(=O)(=O)Nc1ccc(OCCOCCOCCOCCOc2ccc(NS(=O)(=O)CC)cc2-c2cn(C)c(=O)c3ccccc23)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C44H50N4O11S2/c1-5-60(51,52)45-31-15-17-41(37(27-31)39-29-47(3)43(49)35-13-9-7-11-33(35)39)58-25-23-56-21-19-55-20-22-57-24-26-59-42-18-16-32(46-61(53,54)6-2)28-38(42)40-30-48(4)44(50)36-14-10-8-12-34(36)40/h7-18,27-30,45-46H,5-6,19-26H2,1-4H3	VGOFJMULWAVDMV-UHFFFAOYSA-N	50594436	CHEMBL5170488	Bromodomain testis-specific protein	Homo sapiens			 0.089000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594436	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594436&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR7		162394475	482605288							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473374	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C28H35ClFN7O3S/c1-17-16-31-27(34-19-6-8-21(23(30)14-19)26(38)33-18-10-12-37(5)13-11-18)35-25(17)32-20-7-9-22(29)24(15-20)36-41(39,40)28(2,3)4/h6-9,14-16,18,36H,10-13H2,1-5H3,(H,33,38)(H2,31,32,34,35)	RBZRCEPYYVFROZ-UHFFFAOYSA-N	50557394	CHEMBL4760892::US11643396, Example SG3-179	Bromodomain testis-specific protein	Homo sapiens			 9.5						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50557394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50557394&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W2	5F63,7KO0,7LAY,6VNL	118889467	461696162							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473375	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C62H76Cl2F2N14O11S2/c1-37-33-67-59(75-55(37)69-43-11-15-47(63)51(31-43)77-92(85,86)61(3,4)5)73-41-9-13-45(49(65)29-41)57(83)71-39-17-21-79(22-18-39)53(81)35-90-27-25-89-26-28-91-36-54(82)80-23-19-40(20-24-80)72-58(84)46-14-10-42(30-50(46)66)74-60-68-34-38(2)56(76-60)70-44-12-16-48(64)52(32-44)78-93(87,88)62(6,7)8/h9-16,29-34,39-40,77-78H,17-28,35-36H2,1-8H3,(H,71,83)(H,72,84)(H2,67,69,73,75)(H2,68,70,74,76)	QKJZSKDMERAPEK-UHFFFAOYSA-N	50594437	CHEMBL5204093	Bromodomain testis-specific protein	Homo sapiens			 0.600000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMS		163321846	482605289							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473376	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C60H72Cl2F2N14O10S2/c1-35-31-65-57(73-53(35)67-41-11-15-45(61)49(29-41)75-89(83,84)59(3,4)5)71-39-9-13-43(47(63)27-39)55(81)69-37-17-21-77(22-18-37)51(79)33-87-25-26-88-34-52(80)78-23-19-38(20-24-78)70-56(82)44-14-10-40(28-48(44)64)72-58-66-32-36(2)54(74-58)68-42-12-16-46(62)50(30-42)76-90(85,86)60(6,7)8/h9-16,27-32,37-38,75-76H,17-26,33-34H2,1-8H3,(H,69,81)(H,70,82)(H2,65,67,71,73)(H2,66,68,72,74)	YTJRGAPMTDBXIK-UHFFFAOYSA-N	50594438	CHEMBL5201173	Bromodomain testis-specific protein	Homo sapiens			 0.840000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164946925	482605290							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473377	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C66H84Cl2F2N14O12S2/c1-41-39-71-63(79-59(41)73-47-11-15-51(67)55(37-47)81-97(89,90)65(3,4)5)77-45-9-13-49(53(69)35-45)61(87)75-43-17-23-83(24-18-43)57(85)21-27-93-29-31-95-33-34-96-32-30-94-28-22-58(86)84-25-19-44(20-26-84)76-62(88)50-14-10-46(36-54(50)70)78-64-72-40-42(2)60(80-64)74-48-12-16-52(68)56(38-48)82-98(91,92)66(6,7)8/h9-16,35-40,43-44,81-82H,17-34H2,1-8H3,(H,75,87)(H,76,88)(H2,71,73,77,79)(H2,72,74,78,80)	AMHWRJBEKUEFFO-UHFFFAOYSA-N	50594439	CHEMBL5178175	Bromodomain testis-specific protein	Homo sapiens			 0.920000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594439	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594439&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMV		163321847	482605291							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473378	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C68H88Cl2F2N14O13S2/c1-43-41-73-65(81-61(43)75-49-11-15-53(69)57(39-49)83-100(91,92)67(3,4)5)79-47-9-13-51(55(71)37-47)63(89)77-45-17-23-85(24-18-45)59(87)21-27-95-29-31-97-33-35-99-36-34-98-32-30-96-28-22-60(88)86-25-19-46(20-26-86)78-64(90)52-14-10-48(38-56(52)72)80-66-74-42-44(2)62(82-66)76-50-12-16-54(70)58(40-50)84-101(93,94)68(6,7)8/h9-16,37-42,45-46,83-84H,17-36H2,1-8H3,(H,77,89)(H,78,90)(H2,73,75,79,81)(H2,74,76,80,82)	VLYMRIROHVATMC-UHFFFAOYSA-N	50594440	CHEMBL5206426	Bromodomain testis-specific protein	Homo sapiens			 0.600000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594440	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594440&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR4		162394473	482605292							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473379	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCNC(=O)c3cc(Nc4nc(Nc5ccc(C(=O)NC6CCNCC6)c(F)c5)ncc4C)cc(NS(=O)(=O)C(C)(C)C)c3)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C64H82ClF2N15O11S2/c1-39-37-70-61(78-56(39)72-46-11-14-51(65)54(36-46)81-95(89,90)64(6,7)8)76-44-10-13-50(53(67)35-44)60(86)75-43-17-23-82(24-18-43)55(83)19-25-91-27-29-93-30-28-92-26-22-69-58(84)41-31-47(33-48(32-41)80-94(87,88)63(3,4)5)73-57-40(2)38-71-62(79-57)77-45-9-12-49(52(66)34-45)59(85)74-42-15-20-68-21-16-42/h9-14,31-38,42-43,68,80-81H,15-30H2,1-8H3,(H,69,84)(H,74,85)(H,75,86)(H2,70,72,76,78)(H2,71,73,77,79)	DPQKUYBPPCXREN-UHFFFAOYSA-N	50594441	CHEMBL5188470	Bromodomain testis-specific protein	Homo sapiens			 0.160000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594441	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594441&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZN1		163321848	482605293							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473380	CCS(=O)(=O)Nc1ccc(Oc2ccc(Cl)cc2)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C24H21ClN2O4S/c1-3-32(29,30)26-17-10-13-23(31-18-11-8-16(25)9-12-18)21(14-17)22-15-27(2)24(28)20-7-5-4-6-19(20)22/h4-15,26H,3H2,1-2H3	LMYMWXJBPLXESU-UHFFFAOYSA-N	50594435	CHEMBL5184876	Bromodomain testis-specific protein	Homo sapiens			 12						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594435	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594435&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	N49		164607223	482605287							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473381	CCS(=O)(=O)Nc1ccc(OCCOCCOCCOCCOc2ccc(NS(=O)(=O)CC)cc2-c2cn(C)c(=O)c3ccccc23)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C44H50N4O11S2/c1-5-60(51,52)45-31-15-17-41(37(27-31)39-29-47(3)43(49)35-13-9-7-11-33(35)39)58-25-23-56-21-19-55-20-22-57-24-26-59-42-18-16-32(46-61(53,54)6-2)28-38(42)40-30-48(4)44(50)36-14-10-8-12-34(36)40/h7-18,27-30,45-46H,5-6,19-26H2,1-4H3	VGOFJMULWAVDMV-UHFFFAOYSA-N	50594436	CHEMBL5170488	Bromodomain testis-specific protein	Homo sapiens			 5.5						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594436	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594436&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR7		162394475	482605288							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473382	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C28H35ClFN7O3S/c1-17-16-31-27(34-19-6-8-21(23(30)14-19)26(38)33-18-10-12-37(5)13-11-18)35-25(17)32-20-7-9-22(29)24(15-20)36-41(39,40)28(2,3)4/h6-9,14-16,18,36H,10-13H2,1-5H3,(H,33,38)(H2,31,32,34,35)	RBZRCEPYYVFROZ-UHFFFAOYSA-N	50557394	CHEMBL4760892::US11643396, Example SG3-179	Bromodomain testis-specific protein	Homo sapiens			 25						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50557394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50557394&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W2	5F63,7KO0,7LAY,6VNL	118889467	461696162							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473383	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C62H76Cl2F2N14O11S2/c1-37-33-67-59(75-55(37)69-43-11-15-47(63)51(31-43)77-92(85,86)61(3,4)5)73-41-9-13-45(49(65)29-41)57(83)71-39-17-21-79(22-18-39)53(81)35-90-27-25-89-26-28-91-36-54(82)80-23-19-40(20-24-80)72-58(84)46-14-10-42(30-50(46)66)74-60-68-34-38(2)56(76-60)70-44-12-16-48(64)52(32-44)78-93(87,88)62(6,7)8/h9-16,29-34,39-40,77-78H,17-28,35-36H2,1-8H3,(H,71,83)(H,72,84)(H2,67,69,73,75)(H2,68,70,74,76)	QKJZSKDMERAPEK-UHFFFAOYSA-N	50594437	CHEMBL5204093	Bromodomain testis-specific protein	Homo sapiens			 8.4						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMS		163321846	482605289							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473384	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C60H72Cl2F2N14O10S2/c1-35-31-65-57(73-53(35)67-41-11-15-45(61)49(29-41)75-89(83,84)59(3,4)5)71-39-9-13-43(47(63)27-39)55(81)69-37-17-21-77(22-18-37)51(79)33-87-25-26-88-34-52(80)78-23-19-38(20-24-78)70-56(82)44-14-10-40(28-48(44)64)72-58-66-32-36(2)54(74-58)68-42-12-16-46(62)50(30-42)76-90(85,86)60(6,7)8/h9-16,27-32,37-38,75-76H,17-26,33-34H2,1-8H3,(H,69,81)(H,70,82)(H2,65,67,71,73)(H2,66,68,72,74)	YTJRGAPMTDBXIK-UHFFFAOYSA-N	50594438	CHEMBL5201173	Bromodomain testis-specific protein	Homo sapiens			 3.5						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164946925	482605290							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473385	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C66H84Cl2F2N14O12S2/c1-41-39-71-63(79-59(41)73-47-11-15-51(67)55(37-47)81-97(89,90)65(3,4)5)77-45-9-13-49(53(69)35-45)61(87)75-43-17-23-83(24-18-43)57(85)21-27-93-29-31-95-33-34-96-32-30-94-28-22-58(86)84-25-19-44(20-26-84)76-62(88)50-14-10-46(36-54(50)70)78-64-72-40-42(2)60(80-64)74-48-12-16-52(68)56(38-48)82-98(91,92)66(6,7)8/h9-16,35-40,43-44,81-82H,17-34H2,1-8H3,(H,75,87)(H,76,88)(H2,71,73,77,79)(H2,72,74,78,80)	AMHWRJBEKUEFFO-UHFFFAOYSA-N	50594439	CHEMBL5178175	Bromodomain testis-specific protein	Homo sapiens			 1.7						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594439	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594439&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMV		163321847	482605291							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473386	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C68H88Cl2F2N14O13S2/c1-43-41-73-65(81-61(43)75-49-11-15-53(69)57(39-49)83-100(91,92)67(3,4)5)79-47-9-13-51(55(71)37-47)63(89)77-45-17-23-85(24-18-45)59(87)21-27-95-29-31-97-33-35-99-36-34-98-32-30-96-28-22-60(88)86-25-19-46(20-26-86)78-64(90)52-14-10-48(38-56(52)72)80-66-74-42-44(2)62(82-66)76-50-12-16-54(70)58(40-50)84-101(93,94)68(6,7)8/h9-16,37-42,45-46,83-84H,17-36H2,1-8H3,(H,77,89)(H,78,90)(H2,73,75,79,81)(H2,74,76,80,82)	VLYMRIROHVATMC-UHFFFAOYSA-N	50594440	CHEMBL5206426	Bromodomain testis-specific protein	Homo sapiens			 2.2						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594440	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594440&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR4		162394473	482605292							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473387	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCNC(=O)c3cc(Nc4nc(Nc5ccc(C(=O)NC6CCNCC6)c(F)c5)ncc4C)cc(NS(=O)(=O)C(C)(C)C)c3)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C64H82ClF2N15O11S2/c1-39-37-70-61(78-56(39)72-46-11-14-51(65)54(36-46)81-95(89,90)64(6,7)8)76-44-10-13-50(53(67)35-44)60(86)75-43-17-23-82(24-18-43)55(83)19-25-91-27-29-93-30-28-92-26-22-69-58(84)41-31-47(33-48(32-41)80-94(87,88)63(3,4)5)73-57-40(2)38-71-62(79-57)77-45-9-12-49(52(66)34-45)59(85)74-42-15-20-68-21-16-42/h9-14,31-38,42-43,68,80-81H,15-30H2,1-8H3,(H,69,84)(H,74,85)(H,75,86)(H2,70,72,76,78)(H2,71,73,77,79)	DPQKUYBPPCXREN-UHFFFAOYSA-N	50594441	CHEMBL5188470	Bromodomain testis-specific protein	Homo sapiens			 3.1						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594441	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594441&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZN1		163321848	482605293							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473388	CCS(=O)(=O)Nc1ccc(Oc2ccc(Cl)cc2)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C24H21ClN2O4S/c1-3-32(29,30)26-17-10-13-23(31-18-11-8-16(25)9-12-18)21(14-17)22-15-27(2)24(28)20-7-5-4-6-19(20)22/h4-15,26H,3H2,1-2H3	LMYMWXJBPLXESU-UHFFFAOYSA-N	50594435	CHEMBL5184876	Bromodomain testis-specific protein	Homo sapiens			 6.0						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594435	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594435&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	N49		164607223	482605287							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473389	CCS(=O)(=O)Nc1ccc(OCCOCCOCCOCCOc2ccc(NS(=O)(=O)CC)cc2-c2cn(C)c(=O)c3ccccc23)c(c1)-c1cn(C)c(=O)c2ccccc12	InChI=1S/C44H50N4O11S2/c1-5-60(51,52)45-31-15-17-41(37(27-31)39-29-47(3)43(49)35-13-9-7-11-33(35)39)58-25-23-56-21-19-55-20-22-57-24-26-59-42-18-16-32(46-61(53,54)6-2)28-38(42)40-30-48(4)44(50)36-14-10-8-12-34(36)40/h7-18,27-30,45-46H,5-6,19-26H2,1-4H3	VGOFJMULWAVDMV-UHFFFAOYSA-N	50594436	CHEMBL5170488	Bromodomain testis-specific protein	Homo sapiens			 0.058000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594436	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594436&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR7		162394475	482605288							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473390	CN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(C)c(Nc3ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c3)n2)cc1F	InChI=1S/C28H35ClFN7O3S/c1-17-16-31-27(34-19-6-8-21(23(30)14-19)26(38)33-18-10-12-37(5)13-11-18)35-25(17)32-20-7-9-22(29)24(15-20)36-41(39,40)28(2,3)4/h6-9,14-16,18,36H,10-13H2,1-5H3,(H,33,38)(H2,31,32,34,35)	RBZRCEPYYVFROZ-UHFFFAOYSA-N	50557394	CHEMBL4760892::US11643396, Example SG3-179	Bromodomain testis-specific protein	Homo sapiens			 18						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50557394	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50557394&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	5W2	5F63,7KO0,7LAY,6VNL	118889467	461696162							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473391	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C62H76Cl2F2N14O11S2/c1-37-33-67-59(75-55(37)69-43-11-15-47(63)51(31-43)77-92(85,86)61(3,4)5)73-41-9-13-45(49(65)29-41)57(83)71-39-17-21-79(22-18-39)53(81)35-90-27-25-89-26-28-91-36-54(82)80-23-19-40(20-24-80)72-58(84)46-14-10-42(30-50(46)66)74-60-68-34-38(2)56(76-60)70-44-12-16-48(64)52(32-44)78-93(87,88)62(6,7)8/h9-16,29-34,39-40,77-78H,17-28,35-36H2,1-8H3,(H,71,83)(H,72,84)(H2,67,69,73,75)(H2,68,70,74,76)	QKJZSKDMERAPEK-UHFFFAOYSA-N	50594437	CHEMBL5204093	Bromodomain testis-specific protein	Homo sapiens			 2.6						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMS		163321846	482605289							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473392	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)COCCOCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C60H72Cl2F2N14O10S2/c1-35-31-65-57(73-53(35)67-41-11-15-45(61)49(29-41)75-89(83,84)59(3,4)5)71-39-9-13-43(47(63)27-39)55(81)69-37-17-21-77(22-18-37)51(79)33-87-25-26-88-34-52(80)78-23-19-38(20-24-78)70-56(82)44-14-10-40(28-48(44)64)72-58-66-32-36(2)54(74-58)68-42-12-16-46(62)50(30-42)76-90(85,86)60(6,7)8/h9-16,27-32,37-38,75-76H,17-26,33-34H2,1-8H3,(H,69,81)(H,70,82)(H2,65,67,71,73)(H2,66,68,72,74)	YTJRGAPMTDBXIK-UHFFFAOYSA-N	50594438	CHEMBL5201173	Bromodomain testis-specific protein	Homo sapiens			 0.590000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594438	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594438&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			164946925	482605290							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473393	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C66H84Cl2F2N14O12S2/c1-41-39-71-63(79-59(41)73-47-11-15-51(67)55(37-47)81-97(89,90)65(3,4)5)77-45-9-13-49(53(69)35-45)61(87)75-43-17-23-83(24-18-43)57(85)21-27-93-29-31-95-33-34-96-32-30-94-28-22-58(86)84-25-19-44(20-26-84)76-62(88)50-14-10-46(36-54(50)70)78-64-72-40-42(2)60(80-64)74-48-12-16-52(68)56(38-48)82-98(91,92)66(6,7)8/h9-16,35-40,43-44,81-82H,17-34H2,1-8H3,(H,75,87)(H,76,88)(H2,71,73,77,79)(H2,72,74,78,80)	AMHWRJBEKUEFFO-UHFFFAOYSA-N	50594439	CHEMBL5178175	Bromodomain testis-specific protein	Homo sapiens			 1.6						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594439	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594439&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZMV		163321847	482605291							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473394	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCOCCOCCC(=O)N3CCC(CC3)NC(=O)c3ccc(Nc4ncc(C)c(Nc5ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c5)n4)cc3F)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C68H88Cl2F2N14O13S2/c1-43-41-73-65(81-61(43)75-49-11-15-53(69)57(39-49)83-100(91,92)67(3,4)5)79-47-9-13-51(55(71)37-47)63(89)77-45-17-23-85(24-18-45)59(87)21-27-95-29-31-97-33-35-99-36-34-98-32-30-96-28-22-60(88)86-25-19-46(20-26-86)78-64(90)52-14-10-48(38-56(52)72)80-66-74-42-44(2)62(82-66)76-50-12-16-54(70)58(40-50)84-101(93,94)68(6,7)8/h9-16,37-42,45-46,83-84H,17-36H2,1-8H3,(H,77,89)(H,78,90)(H2,73,75,79,81)(H2,74,76,80,82)	VLYMRIROHVATMC-UHFFFAOYSA-N	50594440	CHEMBL5206426	Bromodomain testis-specific protein	Homo sapiens			 0.800000						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594440	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594440&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	XR4		162394473	482605292							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51473395	Cc1cnc(Nc2ccc(C(=O)NC3CCN(CC3)C(=O)CCOCCOCCOCCNC(=O)c3cc(Nc4nc(Nc5ccc(C(=O)NC6CCNCC6)c(F)c5)ncc4C)cc(NS(=O)(=O)C(C)(C)C)c3)c(F)c2)nc1Nc1ccc(Cl)c(NS(=O)(=O)C(C)(C)C)c1	InChI=1S/C64H82ClF2N15O11S2/c1-39-37-70-61(78-56(39)72-46-11-14-51(65)54(36-46)81-95(89,90)64(6,7)8)76-44-10-13-50(53(67)35-44)60(86)75-43-17-23-82(24-18-43)55(83)19-25-91-27-29-93-30-28-92-26-22-69-58(84)41-31-47(33-48(32-41)80-94(87,88)63(3,4)5)73-57-40(2)38-71-62(79-57)77-45-9-12-49(52(66)34-45)59(85)74-42-15-20-68-21-16-42/h9-14,31-38,42-43,68,80-81H,15-30H2,1-8H3,(H,69,84)(H,74,85)(H,75,86)(H2,70,72,76,78)(H2,71,73,77,79)	DPQKUYBPPCXREN-UHFFFAOYSA-N	50594441	CHEMBL5188470	Bromodomain testis-specific protein	Homo sapiens			 1.3						ChEMBL		10.7270/Q2MG7THB	35867655			Guan, X; Cheryala, N; Karim, RM; Chan, A; Berndt, N; Qi, J; Georg, GI; Schönbrunn, E	University of Minnesota	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50594441	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50594441&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	ZN1		163321848	482605293							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51497102	C[C@H]1C[C@@H](Nc2ncc(Cl)cn2)c2cc(ccc2N1C(C)=O)C(N)=O	InChI=1S/C17H18ClN5O2/c1-9-5-14(22-17-20-7-12(18)8-21-17)13-6-11(16(19)25)3-4-15(13)23(9)10(2)24/h3-4,6-9,14H,5H2,1-2H3,(H2,19,25)(H,20,21,22)/t9-,14+/m0/s1	KNBYFXZNSOENGW-LKFCYVNXSA-N	50603097	CHEMBL5195288	Bromodomain testis-specific protein	Homo sapiens			 25						ChEMBL		10.7270/Q23B646M	34995458			Humphreys, PG; Atkinson, SJ; Bamborough, P; Bit, RA; Chung, CW; Craggs, PD; Cutler, L; Davis, R; Ferrie, A; Gong, G; Gordon, LJ; Gray, M; Harrison, LA; Hayhow, TG; Haynes, A; Henley, N; Hirst, DJ; Holyer, ID; Lindon, MJ; Lovatt, C; Lugo, D; McCleary, S; Molnar, J; Osmani, Q; Patten, C; Preston, A; Rioja, I; Seal, JT; Smithers, N; Sun, F; Tang, D; Taylor, S; Theodoulou, NH; Thomas, C; Watson, RJ; Wellaway, CR; Zhu, L; Tomkinson, NCO; Prinjha, RK	GlaxoSmithKline R&D	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50603097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50603097&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	AKQ		118948181	482613948							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51497103	C[C@H]1C[C@@H](Nc2ncc(Cl)cn2)c2cc(ccc2N1C(C)=O)C(N)=O	InChI=1S/C17H18ClN5O2/c1-9-5-14(22-17-20-7-12(18)8-21-17)13-6-11(16(19)25)3-4-15(13)23(9)10(2)24/h3-4,6-9,14H,5H2,1-2H3,(H2,19,25)(H,20,21,22)/t9-,14+/m0/s1	KNBYFXZNSOENGW-LKFCYVNXSA-N	50603097	CHEMBL5195288	Bromodomain testis-specific protein	Homo sapiens			 25						ChEMBL		10.7270/Q23B646M	34995458			Humphreys, PG; Atkinson, SJ; Bamborough, P; Bit, RA; Chung, CW; Craggs, PD; Cutler, L; Davis, R; Ferrie, A; Gong, G; Gordon, LJ; Gray, M; Harrison, LA; Hayhow, TG; Haynes, A; Henley, N; Hirst, DJ; Holyer, ID; Lindon, MJ; Lovatt, C; Lugo, D; McCleary, S; Molnar, J; Osmani, Q; Patten, C; Preston, A; Rioja, I; Seal, JT; Smithers, N; Sun, F; Tang, D; Taylor, S; Theodoulou, NH; Thomas, C; Watson, RJ; Wellaway, CR; Zhu, L; Tomkinson, NCO; Prinjha, RK	GlaxoSmithKline R&D	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50603097	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50603097&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	AKQ		118948181	482613948							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51498211	CN1C=C(C2C=CNC2C1=O)c1ccc2ccn(Cc3ccccn3)c2c1	InChI=1S/C22H20N4O/c1-25-14-19(18-7-10-24-21(18)22(25)27)16-6-5-15-8-11-26(20(15)12-16)13-17-4-2-3-9-23-17/h2-12,14,18,21,24H,13H2,1H3	RUUNUTOBMVHUHT-UHFFFAOYSA-N	50603594	CHEMBL5205457	Bromodomain testis-specific protein	Homo sapiens		>1000							ChEMBL		10.7270/Q2ZC86Z5	35149305			Tao, S; Tao, S; Guo, F; Zhang, L; Zhao, L; Fu, P; Ma, L	West China Hospital of Sichuan University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50603594	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50603594&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			168295363	482614445							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51500671	Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2cc(oc12)-c1cnc([nH]1)C1CCCC1)C(C)(C)O	InChI=1S/C33H34FN3O4/c1-18-12-22(34)13-19(2)29(18)40-27-11-10-21(33(3,4)39)14-23(27)25-17-37(5)32(38)24-15-28(41-30(24)25)26-16-35-31(36-26)20-8-6-7-9-20/h10-17,20,39H,6-9H2,1-5H3,(H,35,36)	QSRRNUBIKNVQHO-UHFFFAOYSA-N	50604624	CHEMBL5206088	Bromodomain testis-specific protein	Homo sapiens			 3668						ChEMBL		10.7270/Q2QJ7NBN	35333526			Li, J; Zhang, C; Xu, H; Wang, C; Dong, R; Shen, H; Zhuang, X; Chen, X; Li, Q; Lu, J; Zhang, M; Wu, X; Loomes, KM; Zhou, Y; Zhang, Y; Liu, J; Xu, Y	Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50604624	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50604624&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JFR		164607215	482615475							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51500672	Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2cc(oc12)-c1cnc([nH]1)C1CCCCC1)C(C)(C)O	InChI=1S/C34H36FN3O4/c1-19-13-23(35)14-20(2)30(19)41-28-12-11-22(34(3,4)40)15-24(28)26-18-38(5)33(39)25-16-29(42-31(25)26)27-17-36-32(37-27)21-9-7-6-8-10-21/h11-18,21,40H,6-10H2,1-5H3,(H,36,37)	UCJMBWXOKLINTN-UHFFFAOYSA-N	50604625	CHEMBL5204783	Bromodomain testis-specific protein	Homo sapiens			 3308						ChEMBL		10.7270/Q2QJ7NBN	35333526			Li, J; Zhang, C; Xu, H; Wang, C; Dong, R; Shen, H; Zhuang, X; Chen, X; Li, Q; Lu, J; Zhang, M; Wu, X; Loomes, KM; Zhou, Y; Zhang, Y; Liu, J; Xu, Y	Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50604625	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50604625&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			168295310	482615476							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51500673	Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2cc(oc12)-c1cnc([nH]1)C1CCCC1)C(C)(C)O	InChI=1S/C33H34FN3O4/c1-18-12-22(34)13-19(2)29(18)40-27-11-10-21(33(3,4)39)14-23(27)25-17-37(5)32(38)24-15-28(41-30(24)25)26-16-35-31(36-26)20-8-6-7-9-20/h10-17,20,39H,6-9H2,1-5H3,(H,35,36)	QSRRNUBIKNVQHO-UHFFFAOYSA-N	50604624	CHEMBL5206088	Bromodomain testis-specific protein	Homo sapiens			 39						ChEMBL		10.7270/Q2QJ7NBN	35333526			Li, J; Zhang, C; Xu, H; Wang, C; Dong, R; Shen, H; Zhuang, X; Chen, X; Li, Q; Lu, J; Zhang, M; Wu, X; Loomes, KM; Zhou, Y; Zhang, Y; Liu, J; Xu, Y	Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50604624	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50604624&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JFR		164607215	482615475							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51500674	Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2cc(oc12)-c1cnc([nH]1)C1CCCCC1)C(C)(C)O	InChI=1S/C34H36FN3O4/c1-19-13-23(35)14-20(2)30(19)41-28-12-11-22(34(3,4)40)15-24(28)26-18-38(5)33(39)25-16-29(42-31(25)26)27-17-36-32(37-27)21-9-7-6-8-10-21/h11-18,21,40H,6-10H2,1-5H3,(H,36,37)	UCJMBWXOKLINTN-UHFFFAOYSA-N	50604625	CHEMBL5204783	Bromodomain testis-specific protein	Homo sapiens			 195						ChEMBL		10.7270/Q2QJ7NBN	35333526			Li, J; Zhang, C; Xu, H; Wang, C; Dong, R; Shen, H; Zhuang, X; Chen, X; Li, Q; Lu, J; Zhang, M; Wu, X; Loomes, KM; Zhou, Y; Zhang, Y; Liu, J; Xu, Y	Chinese Academy of Sciences	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50604625	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50604625&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			168295310	482615476							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51496623	CO[C@H]1CC[C@@H](CC1)n1c(nc2cc(ccc12)-c1c(C)noc1C)[C@@H]1CCCC(=O)N1c1ccc(F)c(F)c1	InChI=1S/C30H32F2N4O3/c1-17-29(18(2)39-34-17)19-7-14-26-25(15-19)33-30(36(26)20-8-11-22(38-3)12-9-20)27-5-4-6-28(37)35(27)21-10-13-23(31)24(32)16-21/h7,10,13-16,20,22,27H,4-6,8-9,11-12H2,1-3H3/t20-,22-,27-/m0/s1	SKDNDJWEBPQKCS-CLHVYKLBSA-N	50602864	CCS-1477::CCS1477::Ccs 1477::Ccs1477::INOBRODIB::Inobrodib	Bromodomain testis-specific protein	Homo sapiens			 1120						ChEMBL		10.7270/Q2VT1X5F	34962793			Xiang, Q; Wang, C; Wu, T; Zhang, C; Hu, Q; Luo, G; Hu, J; Zhuang, X; Zou, L; Shen, H; Wu, X; Zhang, Y; Kong, X; Liu, J; Xu, Y	Guangzhou Medical University	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50602864	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50602864&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	JHL		134457551	482613715							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529016	COc1cc(ccc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(C)(C)O	InChI=1S/C21H24N2O3/c1-5-6-11-23-13-17(16-9-10-22-19(16)20(23)24)15-8-7-14(21(2,3)25)12-18(15)26-4/h5-10,12-13,22,25H,11H2,1-4H3/b6-5+	GVJYOLRRZZUUOE-AATRIKPKSA-N	50615275	CHEMBL5282240	Bromodomain testis-specific protein	Homo sapiens			 830						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615275&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335254	494505023							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529017	COc1cc(c(OC)cc1-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12)C(C)(C)O	InChI=1S/C23H28N2O4/c1-7-8-9-25-13-17(16-10-14(2)24-21(16)22(25)26)15-11-20(29-6)18(23(3,4)27)12-19(15)28-5/h7-8,10-13,24,27H,9H2,1-6H3/b8-7+	QVMOJFHRHLLSOT-BQYQJAHWSA-N	321437	(E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-2,5-dimethoxyphenyl)-2-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one::US10183009, Example 119	Bromodomain testis-specific protein	Homo sapiens			 2100						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375311	384224526							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529018	C\C=C\Cn1cc(-c2ccc(cc2)C(=O)N2CCOCC2)c2cc[nH]c2c1=O	InChI=1S/C22H23N3O3/c1-2-3-10-25-15-19(18-8-9-23-20(18)22(25)27)16-4-6-17(7-5-16)21(26)24-11-13-28-14-12-24/h2-9,15,23H,10-14H2,1H3/b3-2+	JGOZUFGBTSAWEI-NSCUHMNNSA-N	50615276	CHEMBL5270178	Bromodomain testis-specific protein	Homo sapiens			 2500						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615276&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335206	494505024							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529019	COc1cc(c(OC)cc1C(=O)N1CCOCC1)-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12	InChI=1S/C25H29N3O5/c1-5-6-7-28-15-20(18-12-16(2)26-23(18)25(28)30)17-13-22(32-4)19(14-21(17)31-3)24(29)27-8-10-33-11-9-27/h5-6,12-15,26H,7-11H2,1-4H3/b6-5+	FWTDDBIMDSVPTR-AATRIKPKSA-N	321424	6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-4-carbonyl)phenyl]-2-methyl-1H-pyrrolo[2,3-c]pyridin-7-one::US10183009, Example 108	Bromodomain testis-specific protein	Homo sapiens			>10000						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321424	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321424&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375299	384224513							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529020	COc1cc(ccc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(C)(C)O	InChI=1S/C21H24N2O3/c1-5-6-11-23-13-17(16-9-10-22-19(16)20(23)24)15-8-7-14(21(2,3)25)12-18(15)26-4/h5-10,12-13,22,25H,11H2,1-4H3/b6-5+	GVJYOLRRZZUUOE-AATRIKPKSA-N	50615275	CHEMBL5282240	Bromodomain testis-specific protein	Homo sapiens			 1200						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615275&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335254	494505023							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529021	COc1cc(c(OC)cc1-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12)C(C)(C)O	InChI=1S/C23H28N2O4/c1-7-8-9-25-13-17(16-10-14(2)24-21(16)22(25)26)15-11-20(29-6)18(23(3,4)27)12-19(15)28-5/h7-8,10-13,24,27H,9H2,1-6H3/b8-7+	QVMOJFHRHLLSOT-BQYQJAHWSA-N	321437	(E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-2,5-dimethoxyphenyl)-2-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one::US10183009, Example 119	Bromodomain testis-specific protein	Homo sapiens			 6200						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375311	384224526							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529022	C\C=C\Cn1cc(-c2ccc(cc2)C(=O)N2CCOCC2)c2cc[nH]c2c1=O	InChI=1S/C22H23N3O3/c1-2-3-10-25-15-19(18-8-9-23-20(18)22(25)27)16-4-6-17(7-5-16)21(26)24-11-13-28-14-12-24/h2-9,15,23H,10-14H2,1H3/b3-2+	JGOZUFGBTSAWEI-NSCUHMNNSA-N	50615276	CHEMBL5270178	Bromodomain testis-specific protein	Homo sapiens			 2900						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615276&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335206	494505024							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529023	COc1cc(c(OC)cc1C(=O)N1CCOCC1)-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12	InChI=1S/C25H29N3O5/c1-5-6-7-28-15-20(18-12-16(2)26-23(18)25(28)30)17-13-22(32-4)19(14-21(17)31-3)24(29)27-8-10-33-11-9-27/h5-6,12-15,26H,7-11H2,1-4H3/b6-5+	FWTDDBIMDSVPTR-AATRIKPKSA-N	321424	6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-4-carbonyl)phenyl]-2-methyl-1H-pyrrolo[2,3-c]pyridin-7-one::US10183009, Example 108	Bromodomain testis-specific protein	Homo sapiens			>10000						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321424	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321424&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375299	384224513							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529024	COc1cc(ccc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(C)(C)O	InChI=1S/C21H24N2O3/c1-5-6-11-23-13-17(16-9-10-22-19(16)20(23)24)15-8-7-14(21(2,3)25)12-18(15)26-4/h5-10,12-13,22,25H,11H2,1-4H3/b6-5+	GVJYOLRRZZUUOE-AATRIKPKSA-N	50615275	CHEMBL5282240	Bromodomain testis-specific protein	Homo sapiens			 2600						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615275	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615275&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335254	494505023							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529025	COc1cc(c(OC)cc1-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12)C(C)(C)O	InChI=1S/C23H28N2O4/c1-7-8-9-25-13-17(16-10-14(2)24-21(16)22(25)26)15-11-20(29-6)18(23(3,4)27)12-19(15)28-5/h7-8,10-13,24,27H,9H2,1-6H3/b8-7+	QVMOJFHRHLLSOT-BQYQJAHWSA-N	321437	(E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-2,5-dimethoxyphenyl)-2-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one::US10183009, Example 119	Bromodomain testis-specific protein	Homo sapiens			 6600						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321437	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321437&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375311	384224526							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529026	C\C=C\Cn1cc(-c2ccc(cc2)C(=O)N2CCOCC2)c2cc[nH]c2c1=O	InChI=1S/C22H23N3O3/c1-2-3-10-25-15-19(18-8-9-23-20(18)22(25)27)16-4-6-17(7-5-16)21(26)24-11-13-28-14-12-24/h2-9,15,23H,10-14H2,1H3/b3-2+	JGOZUFGBTSAWEI-NSCUHMNNSA-N	50615276	CHEMBL5270178	Bromodomain testis-specific protein	Homo sapiens			 3500						ChEMBL		10.7270/Q2TF02MF	28606761			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50615276	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50615276&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			121335206	494505024							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51529027	COc1cc(c(OC)cc1C(=O)N1CCOCC1)-c1cn(C\C=C\C)c(=O)c2[nH]c(C)cc12	InChI=1S/C25H29N3O5/c1-5-6-7-28-15-20(18-12-16(2)26-23(18)25(28)30)17-13-22(32-4)19(14-21(17)31-3)24(29)27-8-10-33-11-9-27/h5-6,12-15,26H,7-11H2,1-4H3/b6-5+	FWTDDBIMDSVPTR-AATRIKPKSA-N	321424	6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-4-carbonyl)phenyl]-2-methyl-1H-pyrrolo[2,3-c]pyridin-7-one::US10183009, Example 108	Bromodomain testis-specific protein	Homo sapiens			>10000						ChEMBL		10.7270/Q2TF02MF	28606761			Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D	Genentech	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=321424	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=321424&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			138375299	384224513							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525306	O=c1cc(oc2c(cccc12)-c1cccc2sc3ccccc3c12)N1CCOCC1	InChI=1S/C25H19NO3S/c27-20-15-23(26-11-13-28-14-12-26)29-25-17(7-3-8-18(20)25)16-6-4-10-22-24(16)19-5-1-2-9-21(19)30-22/h1-10,15H,11-14H2	LSUVJEUFZJPDTK-UHFFFAOYSA-N	50613679	CHEMBL5287725	Bromodomain testis-specific protein	Homo sapiens		 1000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50613679	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50613679&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			171349036	494503427							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525307	Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H36N6O3S/c1-20-19-28-26(30-21-10-12-23(13-11-21)36-17-16-33-14-5-6-15-33)31-25(20)29-22-8-7-9-24(18-22)37(34,35)32-27(2,3)4/h7-13,18-19,32H,5-6,14-17H2,1-4H3,(H2,28,29,30,31)	JOOXLOJCABQBSG-UHFFFAOYSA-N	50332294	CHEMBL1287853::N-tert-butyl-3-(5-methyl-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)pyrimidin-4-ylamino)benzenesulfonamide::US10112907, Example 00018::US10730860, TABLE 1.3::US10766894, Compound TABLE 1.3::US11203595, TABLE 1.3::US11384069, Example T-5	Bromodomain testis-specific protein	Homo sapiens			 164						ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50332294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50332294&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2TA	4OGJ,4PS5,6VNE	16722836	123111409		CHEMBL1287853		5716		ZINC19862646	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525308	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(c3)S(=O)(=O)NC(C)(C)C)n2)cc1	InChI=1S/C26H35N7O2S/c1-19-18-27-25(29-20-9-11-22(12-10-20)33-15-13-32(5)14-16-33)30-24(19)28-21-7-6-8-23(17-21)36(34,35)31-26(2,3)4/h6-12,17-18,31H,13-16H2,1-5H3,(H2,27,28,29,30)	JVDOKQYTTYUYDV-UHFFFAOYSA-N	192755	TG101209::US11279703, TABLE 6.171::US11643396, Example TG101209	Bromodomain testis-specific protein	Homo sapiens			 123						ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=192755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=192755&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1M3	5HEZ,4O76,4JI9	16722832	317230231							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525309	Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1	InChI=1S/C20H14FN3O/c21-16-5-1-13(2-6-16)18-19(14-9-11-22-12-10-14)24-20(23-18)15-3-7-17(25)8-4-15/h1-12,25H,(H,23,24)	QHKYPYXTTXKZST-UHFFFAOYSA-N	50044784	CHEBI:79090::SB-202190::US10865384, Compound SB202190	Bromodomain testis-specific protein	Homo sapiens			 3424						ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044784	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044784&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RE	4O77	5353940	313068337							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525310	Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C	InChI=1S/C27H36N6O3S/c1-20-19-28-26(30-21-10-12-23(13-11-21)36-17-16-33-14-5-6-15-33)31-25(20)29-22-8-7-9-24(18-22)37(34,35)32-27(2,3)4/h7-13,18-19,32H,5-6,14-17H2,1-4H3,(H2,28,29,30,31)	JOOXLOJCABQBSG-UHFFFAOYSA-N	50332294	CHEMBL1287853::N-tert-butyl-3-(5-methyl-2-(4-(2-(pyrrolidin-1-yl)ethoxy)phenylamino)pyrimidin-4-ylamino)benzenesulfonamide::US10112907, Example 00018::US10730860, TABLE 1.3::US10766894, Compound TABLE 1.3::US11203595, TABLE 1.3::US11384069, Example T-5	Bromodomain testis-specific protein	Homo sapiens		 290							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50332294	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50332294&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2TA	4OGJ,4PS5,6VNE	16722836	123111409		CHEMBL1287853		5716		ZINC19862646	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525311	CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl	InChI=1S/C21H20ClNO5/c1-23-7-6-12(17(27)10-23)19-14(24)8-15(25)20-16(26)9-18(28-21(19)20)11-4-2-3-5-13(11)22/h2-5,8-9,12,17,24-25,27H,6-7,10H2,1H3/t12-,17+/m0/s1	BIIVYFLTOXDAOV-YVEFUNNKSA-N	5655	2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]-4H-chromen-4-one::CHEMBL428690::Flavopiridol::US10294218, Example Flavopiridol::US9617225, Flavopiridol	Bromodomain testis-specific protein	Homo sapiens		 18000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=5655	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=5655&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	CPB	1C8K,1E1Y,3BLR,3EBP,4O71	5287969	8035270		CHEMBL428690	DB03496	5680		ZINC21288966	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525312	CCc1cnn2c(NCc3ccc[n+]([O-])c3)cc(nc12)N1CCCC[C@H]1CCO	InChI=1S/C21H28N6O2/c1-2-17-14-23-27-19(22-13-16-6-5-9-25(29)15-16)12-20(24-21(17)27)26-10-4-3-7-18(26)8-11-28/h5-6,9,12,14-15,18,22,28H,2-4,7-8,10-11,13H2,1H3/t18-/m0/s1	PIMQWRZWLQKKBJ-SFHVURJKSA-N	50139171	Dinaciclib::MK-7965::SCH-727965::US11643396, Example Dinaciclib::US20230416221, Compound Dinaciclib	Bromodomain testis-specific protein	Homo sapiens		 18700							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50139171	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50139171&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46926350	336952252							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525313	CN1CCN(CC1)c1ccc(Nc2ncc(C)c(Nc3cccc(c3)S(=O)(=O)NC(C)(C)C)n2)cc1	InChI=1S/C26H35N7O2S/c1-19-18-27-25(29-20-9-11-22(12-10-20)33-15-13-32(5)14-16-33)30-24(19)28-21-7-6-8-23(17-21)36(34,35)31-26(2,3)4/h6-12,17-18,31H,13-16H2,1-5H3,(H2,27,28,29,30)	JVDOKQYTTYUYDV-UHFFFAOYSA-N	192755	TG101209::US11279703, TABLE 6.171::US11643396, Example TG101209	Bromodomain testis-specific protein	Homo sapiens		 130							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=192755	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=192755&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	1M3	5HEZ,4O76,4JI9	16722832	317230231							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525314	Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1	InChI=1S/C20H14FN3O/c21-16-5-1-13(2-6-16)18-19(14-9-11-22-12-10-14)24-20(23-18)15-3-7-17(25)8-4-15/h1-12,25H,(H,23,24)	QHKYPYXTTXKZST-UHFFFAOYSA-N	50044784	CHEBI:79090::SB-202190::US10865384, Compound SB202190	Bromodomain testis-specific protein	Homo sapiens		 2500							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50044784	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50044784&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RE	4O77	5353940	313068337							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525315	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 35							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525332	O=NC1Cc2c\c(ccc2=C1)=c1\nc([nH]c1=C1C=CNC=C1)C1CCNCC1	InChI=1S/C22H23N5O/c28-27-19-12-16-1-2-17(11-18(16)13-19)21-20(14-3-7-23-8-4-14)25-22(26-21)15-5-9-24-10-6-15/h1-4,7-8,11-12,15,19,23-24H,5-6,9-10,13H2,(H,25,26)/b21-17+	BYFHOKFVPQCBBK-HEHNFIMWSA-N	50613681	CHEMBL5288660	Bromodomain testis-specific protein	Homo sapiens		 10000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50613681	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50613681&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			171349669	494503429							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525333	Oc1ccc(NC2=C(C(=O)NC2=O)c2cccc(Cl)c2)cc1Cl	InChI=1S/C16H10Cl2N2O3/c17-9-3-1-2-8(6-9)13-14(16(23)20-15(13)22)19-10-4-5-12(21)11(18)7-10/h1-7,21H,(H2,19,20,22,23)	YYGKSMKAYKZSBC-UHFFFAOYSA-N	8246	3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophenyl)-2,5-dihydro-1H-pyrrole-2,5-dione::4-arylmaleimide deriv. 6-c	Bromodomain testis-specific protein	Homo sapiens		 19000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=8246	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=8246&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RF	4O7A	6539478	11108999						ZINC14946002	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525334	COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)N(COP(O)(O)=O)c4n3)n2)cc(OC)c1OC	InChI=1S/C23H26FN6O9P/c1-23(2)21(31)30(11-38-40(32,33)34)20-14(39-23)6-7-17(28-20)27-19-13(24)10-25-22(29-19)26-12-8-15(35-3)18(37-5)16(9-12)36-4/h6-10H,11H2,1-5H3,(H2,32,33,34)(H2,25,26,27,28,29)	GKDRMWXFWHEQQT-UHFFFAOYSA-N	50431381	FOSTAMATINIB::R-788 Free acid::R-935788 Free acid	Bromodomain testis-specific protein	Homo sapiens		 21000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50431381	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50431381&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RC	4O75	11671467	164160256						ZINC43131420	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525335	Oc1cccc(c1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1	InChI=1S/C20H15N3O/c24-17-8-4-7-16(13-17)19-18(14-9-11-21-12-10-14)22-20(23-19)15-5-2-1-3-6-15/h1-13,24H,(H,22,23)	KPDQHNUZQHJLSJ-UHFFFAOYSA-N	50077961	3-(2-Phenyl-5-pyridin-4-yl-1H-imidazol-4-yl)-phenol::3-(2-phenyl-5-(pyridin-4-yl)-1H-imidazol-4-yl)phenol::CHEMBL304624	Bromodomain testis-specific protein	Homo sapiens		 5700							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50077961	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50077961&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RN	4O7E	10638921	103970649		CHEMBL304624				ZINC08536641	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525336	O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1	InChI=1S/C19H17NO3/c21-17-13-18(20-9-11-22-12-10-20)23-19-15(7-4-8-16(17)19)14-5-2-1-3-6-14/h1-8,13H,9-12H2	CZQHHVNHHHRRDU-UHFFFAOYSA-N	12915	2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one::2-(morpholin-4-yl)-8-phenyl-4H-chromen-4-one::CHEMBL98350::LY294002::US10308662, Compound LY294002::US9505780, LY294002	Bromodomain testis-specific protein	Homo sapiens		 12430							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=12915	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=12915&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	LY2	1E7V,1YI3,4AZT,4CFK,6G0D	3973	46509407	65329	CHEMBL98350	DB02656	6004	C15195	ZINC37858693	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51525337	COc1ccccc1Oc1nccc(n1)-c1c(ncn1C1CCNCC1)-c1ccc(F)cc1	InChI=1S/C25H24FN5O2/c1-32-21-4-2-3-5-22(21)33-25-28-15-12-20(30-25)24-23(17-6-8-18(26)9-7-17)29-16-31(24)19-10-13-27-14-11-19/h2-9,12,15-16,19,27H,10-11,13-14H2,1H3	RGWJYCCSHANDCO-UHFFFAOYSA-N	50099334	4-[5-(4-Fluoro-phenyl)-3-piperidin-4-yl-3H-imidazol-4-yl]-2-(2-methoxy-phenoxy)-pyrimidine::CHEMBL417804	Bromodomain testis-specific protein	Homo sapiens		 13000							ChEMBL		10.7270/Q2GX4GVS	27559828			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50099334	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50099334&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	2RQ	4O7F	15872406	103996250		CHEMBL417804				ZINC34753280	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	4KCX,5VBQ,5VBR,7BJY,7L73,7L99,7L9A,7LEJ,7LEK,7LEL,7LEM,7MRC,7MRD,7MRG,7MRH,7UBO,7UUU,8CZA	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51549860	Cc1[nH]c(c2CCCCC(=O)c12)-c1cc(N)ccc1Cl	InChI=1S/C16H17ClN2O/c1-9-15-11(4-2-3-5-14(15)20)16(19-9)12-8-10(18)6-7-13(12)17/h6-8,19H,2-5,18H2,1H3	DGJREYHVQYZTEV-UHFFFAOYSA-N	50623486	CHEMBL5439294	Bromodomain testis-specific protein	Homo sapiens			 240						ChEMBL	10.1016/j.ejmech.2023.115139	10.7270/Q2M61QP9	36736153			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50623486	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50623486&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51549861	CCCc1[nH]c(c2CCCCC(=O)c12)-c1cc(N)ccc1Cl	InChI=1S/C18H21ClN2O/c1-2-5-15-17-12(6-3-4-7-16(17)22)18(21-15)13-10-11(20)8-9-14(13)19/h8-10,21H,2-7,20H2,1H3	YOEMPBAQUPZDDO-UHFFFAOYSA-N	50623487	CHEMBL5398641	Bromodomain testis-specific protein	Homo sapiens			 6100						ChEMBL	10.1016/j.ejmech.2023.115139	10.7270/Q2M61QP9	36736153			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50623487	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50623487&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51549862	CCCCc1[nH]c(c2CCCCC(=O)c12)-c1cc(N)ccc1Cl	InChI=1S/C19H23ClN2O/c1-2-3-7-16-18-13(6-4-5-8-17(18)23)19(22-16)14-11-12(21)9-10-15(14)20/h9-11,22H,2-8,21H2,1H3	IBMWMXLKRQTPOA-UHFFFAOYSA-N	50623488	CHEMBL5433870	Bromodomain testis-specific protein	Homo sapiens			>10000						ChEMBL	10.1016/j.ejmech.2023.115139	10.7270/Q2M61QP9	36736153			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50623488	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50623488&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51549863	CCOC(=O)Nc1cc(nn2c(C)nnc12)-c1ccc(C)c(NS(C)(=O)=O)c1	InChI=1S/C17H20N6O4S/c1-5-27-17(24)18-15-9-14(21-23-11(3)19-20-16(15)23)12-7-6-10(2)13(8-12)22-28(4,25)26/h6-9,22H,5H2,1-4H3,(H,18,24)	UYBRROMMFMPJAN-UHFFFAOYSA-N	50504160	CHEMBL3133807::US11773085, Compound B25	Bromodomain testis-specific protein	Homo sapiens			 40						ChEMBL	10.1016/j.ejmech.2023.115139	10.7270/Q2M61QP9	36736153			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50504160	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50504160&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	BMF    	7LEL,5IGK,5FEA,5IGM,5IGL,7K1P,7LAH,5C7N,7LB4,5TCK,5U9N,7L6D,6V1H,5C4Q,5CZG,6NIM,6V0U	72943187	440712745							1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51551914	CN1CCC(CC1)NC(=O)c1cccc(Cn2c3cccc4c3c(cc3ccccc23)n(C)c4=O)c1	InChI=1S/C30H30N4O2/c1-32-15-13-23(14-16-32)31-29(35)22-9-5-7-20(17-22)19-34-25-11-4-3-8-21(25)18-27-28-24(30(36)33(27)2)10-6-12-26(28)34/h3-12,17-18,23H,13-16,19H2,1-2H3,(H,31,35)	GVCFSBGCJBRHFS-UHFFFAOYSA-N	50624343	CHEMBL5393744	Bromodomain testis-specific protein	Homo sapiens		 527							ChEMBL	10.1021/acs.jmedchem.3c01028	10.7270/Q2RN3D77	37478496			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50624343	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50624343&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51554061	Cc1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(=O)c1n23)C(=O)c1cccc2ccccc12	InChI=1S/C28H23N3O4S/c1-17-12-25-23-13-18(16-36(2,34)35)10-11-24(23)30(15-20-14-29-27(32)26(17)31(20)25)28(33)22-9-5-7-19-6-3-4-8-21(19)22/h3-14H,15-16H2,1-2H3,(H,29,32)	SVWVGWHDUPYUFQ-UHFFFAOYSA-N	50625295	CHEMBL5440806	Bromodomain testis-specific protein	Homo sapiens		 1429							ChEMBL	10.1016/j.ejmech.2022.115023	10.7270/Q28D01PM	36566713			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625295&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HFU    	7DPO,7DPN									1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51554062	Cc1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(=O)c1n23)C(=O)c1ccc2ccccc2c1	InChI=1S/C28H23N3O4S/c1-17-11-25-23-12-18(16-36(2,34)35)7-10-24(23)30(15-22-14-29-27(32)26(17)31(22)25)28(33)21-9-8-19-5-3-4-6-20(19)13-21/h3-14H,15-16H2,1-2H3,(H,29,32)	GZEDEKFDZMUCGJ-UHFFFAOYSA-N	50625296	CHEMBL5437856	Bromodomain testis-specific protein	Homo sapiens		 87							ChEMBL	10.1016/j.ejmech.2022.115023	10.7270/Q28D01PM	36566713			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625296&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51554063	Cc1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(=O)c1n23)C(=O)c1cccc2ccccc12	InChI=1S/C28H23N3O4S/c1-17-12-25-23-13-18(16-36(2,34)35)10-11-24(23)30(15-20-14-29-27(32)26(17)31(20)25)28(33)22-9-5-7-19-6-3-4-8-21(19)22/h3-14H,15-16H2,1-2H3,(H,29,32)	SVWVGWHDUPYUFQ-UHFFFAOYSA-N	50625295	CHEMBL5440806	Bromodomain testis-specific protein	Homo sapiens		 59							ChEMBL	10.1016/j.ejmech.2022.115023	10.7270/Q28D01PM	36566713			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625295	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625295&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	HFU    	7DPO,7DPN									1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51554064	Cc1cc2-c3cc(CS(C)(=O)=O)ccc3N(Cc3c[nH]c(=O)c1n23)C(=O)c1ccc2ccccc2c1	InChI=1S/C28H23N3O4S/c1-17-11-25-23-12-18(16-36(2,34)35)7-10-24(23)30(15-22-14-29-27(32)26(17)31(22)25)28(33)21-9-8-19-5-3-4-6-20(19)13-21/h3-14H,15-16H2,1-2H3,(H,29,32)	GZEDEKFDZMUCGJ-UHFFFAOYSA-N	50625296	CHEMBL5437856	Bromodomain testis-specific protein	Homo sapiens		 43							ChEMBL	10.1016/j.ejmech.2022.115023	10.7270/Q28D01PM	36566713			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625296	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625296&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51566503	Cc1cc(cn(C)c1=O)-c1cc2OCCn3c2c(c1)n(Cc1ccccc1)c3=O	InChI=1S/C23H21N3O3/c1-15-10-18(14-24(2)22(15)27)17-11-19-21-20(12-17)29-9-8-25(21)23(28)26(19)13-16-6-4-3-5-7-16/h3-7,10-12,14H,8-9,13H2,1-2H3	QTVSDAUHDJBCAA-UHFFFAOYSA-N	50629970	CHEMBL5395771	Bromodomain testis-specific protein	Homo sapiens		 68							ChEMBL	10.1016/j.bmc.2023.117461	10.7270/Q2057MCC	37659219			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50629970	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50629970&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51555615	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens			 188						ChEMBL	10.1021/acsmedchemlett.3c00464	10.7270/Q2R215SW	38229743			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51555616	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(CF)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H24ClFN4O2S/c1-12-17(11-25)32-22-19(12)20(14-6-8-15(24)9-7-14)26-16(10-18(30)31-23(3,4)5)21-28-27-13(2)29(21)22/h6-9,16H,10-11H2,1-5H3/t16-/m0/s1	UTRVMZYPPGEUEN-INIZCTEOSA-N	50625919	CHEMBL5431301	Bromodomain testis-specific protein	Homo sapiens			 722						ChEMBL	10.1021/acsmedchemlett.3c00464	10.7270/Q2R215SW	38229743			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625919	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625919&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51555617	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(sc3-n12)C(F)F)c1ccc(Cl)cc1	InChI=1S/C23H23ClF2N4O2S/c1-11-17-18(13-6-8-14(24)9-7-13)27-15(10-16(31)32-23(3,4)5)21-29-28-12(2)30(21)22(17)33-19(11)20(25)26/h6-9,15,20H,10H2,1-5H3/t15-/m0/s1	KDJMZLWFACNZCG-HNNXBMFYSA-N	50625920	CHEMBL5414263	Bromodomain testis-specific protein	Homo sapiens			 3920						ChEMBL	10.1021/acsmedchemlett.3c00464	10.7270/Q2R215SW	38229743			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50625920	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50625920&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51555618	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 124							ChEMBL	10.1021/acsmedchemlett.3c00464	10.7270/Q2R215SW	38229743			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51555619	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 103							ChEMBL	10.1021/acsmedchemlett.3c00464	10.7270/Q2R215SW	38229743			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51532382	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1ncnc(NCCCCCCC(=O)NO)c21	InChI=1S/C23H28N6O4/c1-13-20(14(2)33-29-13)16-10-17-15(11-18(16)32-3)21-22(25-12-26-23(21)27-17)24-9-7-5-4-6-8-19(30)28-31/h10-12,31H,4-9H2,1-3H3,(H,28,30)(H2,24,25,26,27)	OABQDWQBXSGEDG-UHFFFAOYSA-N	50616476	CHEMBL5405779	Bromodomain testis-specific protein	Homo sapiens		 221							ChEMBL	10.1021/acs.jmedchem.2c01191	10.7270/Q26M3C5M	36622852			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50616476	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50616476&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51532383	COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(NCCCCCCC(=O)NO)c21	InChI=1S/C24H30N6O4/c1-13-21(14(2)34-30-13)17-11-18-16(12-19(17)33-4)22-23(26-15(3)27-24(22)28-18)25-10-8-6-5-7-9-20(31)29-32/h11-12,32H,5-10H2,1-4H3,(H,29,31)(H2,25,26,27,28)	BHJOJVLBZYUYGS-UHFFFAOYSA-N	50616481	CHEMBL5422534	Bromodomain testis-specific protein	Homo sapiens		 1109							ChEMBL	10.1021/acs.jmedchem.2c01191	10.7270/Q26M3C5M	36622852			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50616481	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50616481&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51532384	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 534							ChEMBL	10.1021/acs.jmedchem.2c01191	10.7270/Q26M3C5M	36622852			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51531783	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 5.5							ChEMBL	10.1021/acs.jmedchem.2c01770	10.7270/Q2RJ4PS2	36577036			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51531784	CC(=O)OC[C@]12CC[C@H]3[C@@H](C[C@H]4O[C@]44CC=CC(=O)[C@]34C)[C@]1(O)CC[C@@]2(O)[C@@](C)(O)[C@H]1CC(C)=C(C)C(=O)O1	InChI=1S/C30H40O9/c1-16-13-22(38-24(33)17(16)2)26(5,34)30(36)12-11-28(35)20-14-23-29(39-23)9-6-7-21(32)25(29,4)19(20)8-10-27(28,30)15-37-18(3)31/h6-7,19-20,22-23,34-36H,8-15H2,1-5H3/t19-,20+,22+,23+,25-,26-,27+,28+,29+,30+/m0/s1	GKMMNQCWGZRQTN-XVRWHRFDSA-N	50616255	CHEMBL3605565	Bromodomain testis-specific protein	Homo sapiens		 119							ChEMBL	10.1021/acs.jmedchem.2c01770	10.7270/Q2RJ4PS2	36577036			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50616255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50616255&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51531785	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 510							ChEMBL	10.1021/acs.jmedchem.2c01770	10.7270/Q2RJ4PS2	36577036			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51531786	CC(=O)OC[C@]12CC[C@H]3[C@@H](C[C@H]4O[C@]44CC=CC(=O)[C@]34C)[C@]1(O)CC[C@@]2(O)[C@@](C)(O)[C@H]1CC(C)=C(C)C(=O)O1	InChI=1S/C30H40O9/c1-16-13-22(38-24(33)17(16)2)26(5,34)30(36)12-11-28(35)20-14-23-29(39-23)9-6-7-21(32)25(29,4)19(20)8-10-27(28,30)15-37-18(3)31/h6-7,19-20,22-23,34-36H,8-15H2,1-5H3/t19-,20+,22+,23+,25-,26-,27+,28+,29+,30+/m0/s1	GKMMNQCWGZRQTN-XVRWHRFDSA-N	50616255	CHEMBL3605565	Bromodomain testis-specific protein	Homo sapiens		 403							ChEMBL	10.1021/acs.jmedchem.2c01770	10.7270/Q2RJ4PS2	36577036			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50616255	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50616255&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51533939	CCC(C)n1ccc2c(cc(cc12)-c1cn(C)c(=O)c2[nH]ccc12)C(=O)NCc1c(C)cc(C)[nH]c1=O	InChI=1S/C29H31N5O3/c1-6-18(4)34-10-8-20-22(27(35)31-14-23-16(2)11-17(3)32-28(23)36)12-19(13-25(20)34)24-15-33(5)29(37)26-21(24)7-9-30-26/h7-13,15,18,30H,6,14H2,1-5H3,(H,31,35)(H,32,36)	LORVKFYVSXATKW-UHFFFAOYSA-N	50617014	CHEMBL5434556	Bromodomain testis-specific protein	Homo sapiens		 35							ChEMBL	10.1021/acs.jmedchem.2c01607	10.7270/Q2V69PZP	36774555			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50617014	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50617014&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51533940	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 23							ChEMBL	10.1021/acs.jmedchem.2c01607	10.7270/Q2V69PZP	36774555			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51536766	CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCC(=O)OCc2c(no[n+]2[O-])-c2ccccc2)c(C)c1	InChI=1S/C29H27N5O6S/c1-16-11-19(27-30-28(36)24-20-9-10-33(3)13-22(20)41-29(24)31-27)12-17(2)26(16)39-15-23(35)38-14-21-25(32-40-34(21)37)18-7-5-4-6-8-18/h4-8,11-12H,9-10,13-15H2,1-3H3,(H,30,31,36)	SUMJFWHWPZJWDQ-UHFFFAOYSA-N	50618174	CHEMBL5427713	Bromodomain testis-specific protein	Homo sapiens		>20000							ChEMBL	10.1016/j.ejmech.2022.114970	10.7270/Q2WQ0841	36470106			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50618174	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50618174&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search											1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
51536767	Cc1nnc2[C@H](CC(=O)OC(C)(C)C)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1	InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m0/s1	DNVXATUJJDPFDM-KRWDZBQOSA-N	50365262	(+)-JQ1::(S)-JQ1 (1)::CHEMBL1957266::JQ1::US10124009, Compound (S)-JQ1::US10202360, Example JQ-1::US10308662, Compound JQ-1::US10407441, Compound (S)-JQ1::US10617680, Example JQ-1::US10881668, Compound JQ1::US10925881, Name (S)-JQ1::US11020380, Example JQ-1::US11078188, Example (+)-JQ1::US11279703, TABLE 6.180::US11427593, Compound JQ1::US11466034, Example (+)-JQ1::US9320741, (S)-JQ1::US9695172, JQ1	Bromodomain testis-specific protein	Homo sapiens		 134							ChEMBL	10.1016/j.ejmech.2022.114970	10.7270/Q2WQ0841	36470106			n/a	n/a	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50365262	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50004931&target=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50365262&enzyme=Bromodomain+testis-specific+protein&column=ki&startPg=0&Increment=50&submit=Search			46907787	136969324		CHEMBL1957266				ZINC57318556	1	MSLPSRQTAIIVNPPPPEYINTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQVVGVKERIKKGTQQNIAVSSAKEKSSPSATEKVFKQQEIPSVFPKTSISPLNVVQGASVNSSSQTAAQVTKGVKRKADTTTPATSAVKASSEFSPTFTEKSVALPPIKENMPKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVESMPLCYIKTDITETTGRENTNEASSEGNSSDDSEDERVKRLAKLQEQLKAVHQQLQVLSQVPFRKLNKKKEKSKKEKKKEKVNNSNENPRKMCEQMRLKEKSKRNQPKKRKQQFIGLKSEDEDNAKPMNYDEKRQLSLNINKLPGDKLGRVVHIIQSREPSLSNSNPDEIEIDFETLKASTLRELEKYVSACLRKRPLKPPAKKIMMSKEELHSQKKQELEKRLLDVNNQLNSRKRQTKSDKTQPSKAVENVSRLSESSSSSSSSSESESSSSDLSSSDSSDSESEMFPKFTEVKPNDSPSKENVKKMKNECIPPEGRTGVTQIGYCVQDTTSANTTLVHQTTPSHVMPPNHHQLAFNYQELEHLQTVKNISPLQILPPSGDSEQLSNGITVMHPSGDSDTTMLESECQAPVQKDIKIKNADSWKSLGKPVKPSGVMKSSDELFNQFRKAAIEKEVKARTQELIRKHLEQNTKELKASQENQRDLGNGLTVESFSNKIQNKCSGEEQKEHQQSSEAQDKSKLWLLKDRDLARQKEQERRRREAMVGTIDMTLQSDIMTMFENNFD	8YHS,4KCX,7LEJ,7LEL,7LEK,7L9A,7L99,7UBO,8CZA,7UUU,7MRH,7MRG,7MRD,7MRC,7LEM,7L73,7BJY,5VBR,5VBQ	Bromodomain testis-specific protein	BRDT_HUMAN	Q58F21	A6NF68 B7Z811 B7Z890 B7ZAX7 D3DT32 O14789 Q05DQ4 Q6P5T1 Q7Z4A6 Q8IWI6						
