Compile Data Set for Download or QSAR
Report error Found 53 of kd for UniProtKB: P48039
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470001BDBM50470001(CHEMBL322339)
Affinity DataKd:  0.000270nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408578BDBM50408578(CHEMBL417151)
Affinity DataKd:  0.000418nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230659BDBM50230659(CHEMBL37549)
Affinity DataKd:  0.000453nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470007BDBM50470007(CHEMBL322269)
Affinity DataKd:  0.000800nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230663BDBM50230663(CHEMBL34349)
Affinity DataKd:  0.00343nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230657BDBM50230657(CHEMBL290493)
Affinity DataKd:  0.00615nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470004BDBM50470004(CHEMBL111458)
Affinity DataKd:  0.0155nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469993BDBM50469993(CHEMBL320267)
Affinity DataKd:  0.0164nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408556BDBM50408556(CHEMBL37771)
Affinity DataKd:  0.0219nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470009BDBM50470009(CHEMBL109842)
Affinity DataKd:  0.0405nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470000BDBM50470000(CHEMBL111599)
Affinity DataKd:  0.0410nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKd:  0.0915nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50035179BDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408555BDBM50408555(CHEMBL322762)
Affinity DataKd:  0.201nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037253BDBM50037253(2-Iodo-N-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-aceta...)
Affinity DataKd:  0.520nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037219BDBM50037219(N-[2-(5-Methoxy-benzo[b]thiophen-3-yl)-ethyl]-acet...)
Affinity DataKd:  0.560nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037242BDBM50037242(N-[2-(5-Methoxy-benzofuran-3-yl)-ethyl]-acetamide ...)
Affinity DataKd:  0.859nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037222BDBM50037222(Cyclopropanecarboxylic acid [2-(5-methoxy-benzo[b]...)
Affinity DataKd:  1.90nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037228BDBM50037228(2-Iodo-N-[2-(5-methoxy-benzo[b]thiophen-3-yl)-ethy...)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408649BDBM50408649(CHEMBL37703)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037249BDBM50037249(Cyclopropanecarboxylic acid [2-(6-fluoro-5-methoxy...)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037247BDBM50037247(Cyclopropanecarboxylic acid [2-(5-methoxy-benzofur...)
Affinity DataKd:  4.10nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470006BDBM50470006(CHEMBL325593)
Affinity DataKd:  7.10nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469998BDBM50469998(CHEMBL325341)
Affinity DataKd:  7.30nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230662BDBM50230662(CHEMBL285005)
Affinity DataKd:  8.70nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470002BDBM50470002(CHEMBL109323)
Affinity DataKd:  14nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037240BDBM50037240(Pentanoic acid [2-(5-methoxy-benzofuran-3-yl)-ethy...)
Affinity DataKd:  17nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469990BDBM50469990(CHEMBL111063)
Affinity DataKd:  20nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230661BDBM50230661(CHEMBL288301)
Affinity DataKd:  24nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037236BDBM50037236(Cyclobutanecarboxylic acid [2-(5-methoxy-benzo[b]t...)
Affinity DataKd:  46nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470010BDBM50470010(CHEMBL109595)
Affinity DataKd:  49nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037220BDBM50037220(1-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-pyrrolidin...)
Affinity DataKd:  53nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037233BDBM50037233(Cyclobutanecarboxylic acid [2-(6-methoxy-naphthale...)
Affinity DataKd:  59nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469991BDBM50469991(CHEMBL109784)
Affinity DataKd:  65nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469992BDBM50469992(CHEMBL108762)
Affinity DataKd:  71nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469999BDBM50469999(CHEMBL109190)
Affinity DataKd:  80nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470005BDBM50470005(CHEMBL418825)
Affinity DataKd:  91nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469995BDBM50469995(CHEMBL324078)
Affinity DataKd:  120nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230660BDBM50230660(CHEMBL290646)
Affinity DataKd:  160nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470008BDBM50470008(CHEMBL111464)
Affinity DataKd:  160nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469994BDBM50469994(CHEMBL111062)
Affinity DataKd:  170nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469989BDBM50469989(CHEMBL419024)
Affinity DataKd:  190nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408572BDBM50408572(CHEMBL35017)
Affinity DataKd:  280nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470003BDBM50470003(CHEMBL111748)
Affinity DataKd:  960nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469996BDBM50469996(CHEMBL111673)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469988BDBM50469988(CHEMBL419566)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037234BDBM50037234(1H-Indole-2-carboxylic acid [2-(7-methoxy-naphthal...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037224BDBM50037224(N-[2-(6-Methoxy-benzoimidazol-1-yl)-ethyl]-acetami...)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230658BDBM50230658(CHEMBL37721)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037245BDBM50037245(Heptanoic acid [2-(7-methoxy-naphthalen-1-yl)-ethy...)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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