Compile Data Set for Download or QSAR
maximum 50k data
Found 116 of kd for UniProtKB: P24941
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91782(CS260)
Affinity DataKd:  8nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7772(5-({[(12Z)-11-oxo-3-thia-5,10-diazatricyclo[7.3.0....)
Affinity DataKd:  36nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91736(CS11)
Affinity DataKd:  44nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8068(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 39 | 2...)
Affinity DataKd:  45nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91761(CS19)
Affinity DataKd:  62nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91749(CS16)
Affinity DataKd:  73nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7163(3-Phenylacetamidoaminopyrazole deriv. 40 | CS10 | ...)
Affinity DataKd:  79nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7722((3Z)-N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-s...)
Affinity DataKd:  82nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  94nMAssay Description:Binding affinity to recombinant human full-length N-terminal GST-tagged CDK2/cyclin A2 expressed in baculovirus expression system using modified Hist...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8046((4-Fluorophenyl)-[4-(2,4-dimethylthiazol-5-yl)pyri...)
Affinity DataKd:  121nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8043((4-chlorophenyl)-[4-(2,4-dimethylthiazol-5-yl)pyri...)
Affinity DataKd:  151nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKd:  161nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91736(CS11)
Affinity DataKd:  171nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8069(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 40 | 4...)
Affinity DataKd:  190nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7742(4-[2-(7-Oxo-6,7-dihydro[1,2,3]triazolo[4,5-e]indol...)
Affinity DataKd:  191nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91780(CS246)
Affinity DataKd:  207nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7765(3-{[4-({[(3Z)-2-oxo-2,3-dihydro-1H-indol-3-ylidene...)
Affinity DataKd:  210nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91779(CS244)
Affinity DataKd:  333nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91782(CS260)
Affinity DataKd:  334nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7126(3-Propylaminopyrazole deriv. 3 | CHEMBL112442 | CS...)
Affinity DataKd:  360nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7132(1-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzene-1,4-dic...)
Affinity DataKd:  362nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7132(1-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzene-1,4-dic...)
Affinity DataKd:  388nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7157(3-Phenylacetamidoaminopyrazole deriv. 34 | CHEMBL1...)
Affinity DataKd:  463nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7126(3-Propylaminopyrazole deriv. 3 | CHEMBL112442 | CS...)
Affinity DataKd:  537nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM50511927(CHEMBL4517803)
Affinity DataKd:  720nMAssay Description:Binding affinity to recombinant human CDK2/CyclinA by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91781(CS248)
Affinity DataKd:  840nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)
Affinity DataKd:  1.31E+3nMAssay Description:Binding affinity to recombinant human CDK2/CyclinA by SPR assayMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7145(3-Benzamidoaminopyrazole deriv. 22 | 4-bromo-N-(5-...)
Affinity DataKd:  4.09E+3nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7145(3-Benzamidoaminopyrazole deriv. 22 | 4-bromo-N-(5-...)
Affinity DataKd:  5.55E+3nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8037(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 8 | 4-...)
Affinity DataKd:  3.03E+4nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91784(CS27)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91794(CS46)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91806(CS69)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91795(CS47)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91797(CS53)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91791(CS38)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91817(CS82)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91821(CS95)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91759(CS188)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91762(CS196)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7144(3-Benzamidoaminopyrazole deriv. 21 | 4-bromo-N-(5-...)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91793(CS41)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91810(CS73)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91735(CS109)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM7144(3-Benzamidoaminopyrazole deriv. 21 | 4-bromo-N-(5-...)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91803(CS66)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91739(CS115)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91801(CS64)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91786(CS32)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM91774(CS232)
Affinity DataKd: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
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