Compile Data Set for Download or QSAR
Report error Found 5 of ec50 for monomerid = 50015318
TargetVitamin D3 receptor(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)
Affinity DataEC50:  0.0700nMAssay Description:Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)
Affinity DataEC50:  0.400nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)
Affinity DataEC50:  0.5nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)
Affinity DataEC50:  0.600nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)
Affinity DataEC50:  1.5nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed