Compile Data Set for Download or QSAR
Report error Found 3 of ic50 for monomerid = 238373
LigandPNGBDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 640nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandPNGBDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Assays were realized on 96-well plates, as described for yeast FTase but octyl-D-glucopyranoside (0.18%) was used instead of CHAPS and the solution c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
TargetProtein farnesyltransferase alpha subunit/subunit beta(Trypanosoma brucei brucei)
Centre De Recherche De Gif

LigandPNGBDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 5.40E+3nMAssay Description:Assays were realized on 96-well plates, as described for human FTase with the dansylated peptide Dansyl-GCAIM and the solution contains 15 μL of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed