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Report error Found 6 of ic50 for monomerid = 50310922
TargetAdenosine receptor A2b(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 7.10nMAssay Description:The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details
US Patent

TargetAdenosine receptor A2b(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3 [I248L](Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 233nMAssay Description:The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 1.10E+3nMAssay Description:The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 1.40E+3nMAssay Description:The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM50310922({6-Amino-2-[(pyridin-3-ylmethyl)-amino]-thieno[3,2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed