Compile Data Set for Download or QSAR
Report error Found 3 of ki for monomerid = 142083
TargetProtein O-GlcNAcase(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM142083(US8933040, 7)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM142083(US8933040, 7)
Affinity DataKi:  13nM ΔG°:  -45.0kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions were carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2015
Entry Details
US Patent

TargetBeta-hexosaminidase subunit beta(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM142083(US8933040, 7)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human beta hexosaminidase assessed as inhibitory constant using 4-methylumbelliferyl N-acetyl-beta-D-glucosaminide dihydrate as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed