Compile Data Set for Download or QSAR
Report error Found 3 of ki for monomerid = 50200546
TargetCaspase-1(Human)
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200546(CHEMBL3939229)
Affinity DataKi:  75nMAssay Description:Inhibition of human recombinant N-terminal His-tagged DTT-activated caspase-1 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2018
Entry Details Article
PubMed
TargetCaspase-5(Human)
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200546(CHEMBL3939229)
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2018
Entry Details Article
PubMed
TargetCaspase-4(Human)
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200546(CHEMBL3939229)
Affinity DataKi:  276nMAssay Description:Inhibition of human recombinant N-terminal His-tagged DTT-activated caspase-4 expressed in Escherichia coli using Ac-LEVD-AMC as substrate preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2018
Entry Details Article
PubMed