Compile Data Set for Download or QSAR
Report error Found 6 of koff for monomerid = 50163859
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.00620M-1s-1pH: 8.0Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as dissociation rate constant at pH 8 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.00720M-1s-1pH: 7.0Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as dissociation rate constant at pH 7 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.00770M-1s-1Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as dissociation rate constant after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.00790M-1s-1pH: 6.0Assay Description:Binding affinity to human recombinant CA9 catalytic domain assessed as dissociation rate constant at pH 6 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 7(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.0100M-1s-1Assay Description:Binding affinity to human recombinant CA7 assessed as dissociation rate constant after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50163859(carbonic anhydrase (CA) inhibitors, benzenesulphon...)
Affinity DataKon:  0.0500M-1s-1Assay Description:Binding affinity to human recombinant CA12 catalytic domain assessed as dissociation rate constant after 30 secs by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/10/2017
Entry Details Article
PubMed