Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50161628'
Target5-hydroxytryptamine receptor 2B(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161628(8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)
Affinity DataEC50:  1.10E+3nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2B receptors transfected in HEK293 cells was determined by measuring [3H]phosphoinositol releaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161628(8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as intracellular IP3 accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed