Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50291267'
Target5-hydroxytryptamine receptor 6(Human)
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Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50291267BDBM50291267(CHEMBL4161308)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LSD from human 5HT6R expressed in HEK293 cell membranes after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50291267BDBM50291267(CHEMBL4161308)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at 5HT6R (unknown origin) transfected in NG108-15 cells co-transfected with CAMYEL assessed as reduction in cAMP levels after 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2020
Entry Details Article
PubMed