Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase' and Ligand = 'BDBM92445'
Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandChemical structure of BindingDB Monomer ID 92445BDBM92445(US8691753, 105 | Inhibitor, 10)
Affinity DataKi:  377nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
US Patent

Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandChemical structure of BindingDB Monomer ID 92445BDBM92445(US8691753, 105 | Inhibitor, 10)
Affinity DataKi:  377nM ΔG°:  -36.7kJ/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2012
Entry Details Article
PubMed