Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Acyl-protein thioesterase 1' and Ligand = 'BDBM50543969'
TargetAcyl-protein thioesterase 1(Rat)
Peking University First Hospital

Curated by ChEMBL
LigandPNGBDBM50543969(CHEMBL4640030)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant N-terminal FLAG-tagged FAP (unknown origin) (38 to 760 residues) expressed in HEK293 cells using AMCC as substrate by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Peking University First Hospital

Curated by ChEMBL
LigandPNGBDBM50543969(CHEMBL4640030)
Affinity DataIC50: 663nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed