Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50368792'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 0.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataEC50:  794nMAssay Description:Photoaffinity labelling of purified human A2AR (1 to 316 residues) by SDS-PAGE analaysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed