Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM82022'
TargetAdenosine receptor A2a(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKd:  9.10nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as dissociation constant by surface plasmon resonance...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2a(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKi:  76nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAdenosine receptor A2a(Rat)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKi:  83nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain membranes using [3H]cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKi:  100nMAssay Description:Binding affinity to rat recombinant adenosine receptor A2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKi:  119nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
TargetAdenosine receptor A2a(Rat)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82022BDBM82022(N6-Phenylado | 2-[6-Amino-2-(3-cyclohexyl-propylam...)
Affinity DataKi:  663nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed