Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50170191'
TargetAlpha-2A adrenergic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50170191(N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cycloh...)
Affinity DataIC50: 104nMAssay Description:Displacement of [3H]MK-912 from human adrenergic alpha2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50170191(N-[4-(4-Dimethylamino-quinazolin-2-ylamino)-cycloh...)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed