Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM86779'
TargetAmine oxidase [flavin-containing] A(Human)
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86779(Phthalonitrile analogue, 4h)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86779(Phthalonitrile analogue, 4h)
Affinity DataIC50: 642nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed