Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with Target = 'Appetite-regulating hormone' and Ligand = 'BDBM50517283'
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataEC50:  2nMAssay Description:Displacement of C-terminal Cys-tagged NanoLuc luciferase from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataEC50:  1.90nMAssay Description:Displacement of C-terminal Cys-tagged NanoLuc luciferase from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 2.20nMAssay Description:Displacement of C-terminal Cys-tagged SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader based Nan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 2.20nMAssay Description:Displacement of C-terminal Cys-tagged SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader based Nan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 3.5nMAssay Description:Displacement of C-terminal Cys-tagged human LEAP2-SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 3.60nMAssay Description:Displacement of C-terminal Cys-tagged human LEAP2-SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate read...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 12nMAssay Description:Binding affinity to Ghrelin in human serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based micropl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Human)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 12nMAssay Description:Binding affinity to Ghrelin in human serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based micropl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Bovine)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 12nMAssay Description:Binding affinity to Ghrelin in fetal bovine serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetAppetite-regulating hormone(Bovine)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50517283(CHEMBL425281)
Affinity DataIC50: 12nMAssay Description:Binding affinity to Ghrelin in fetal bovine serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed