Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Bcl-2-like protein 1' and Ligand = 'BDBM21429'
TargetBcl-2-like protein 1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 21429BDBM21429(4-{4-[(2-cyanophenyl)methylidene]piperidin-1-yl}-N...)
Affinity DataKi: <0.5nM ΔG°: <-53.1kJ/mole IC50: 520nM EC50:  1.10E+3nMpH: 7.4 T: 2°CAssay Description:The binding affinities (Ki) of compounds were determined using fluorescence polarization assays (FPA) that measure their ability to competitively dis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 21429BDBM21429(4-{4-[(2-cyanophenyl)methylidene]piperidin-1-yl}-N...)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of Bcl-XLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed