Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'CDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7' and Ligand = 'BDBM50526803'
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent