Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM50459792'
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459792BDBM50459792(CHEMBL4206032)
Affinity DataIC50: 59nMAssay Description:Displacement of Histone H4 peptide (1-21) K5/8/12/16Ac-Biotin from recombinant human N-terminal His-tagged CBP bromodomain expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50459792BDBM50459792(CHEMBL4206032)
Affinity DataKd:  85nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length CBP bromodomain (R1081 to G1197 residues) expressed in bacteria...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed