Report error Found 4 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK1' and Ligand = 'BDBM50623175'
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human CLK1 using GRSRSRSRSRSRSRS as substrate incubated for 15 mins in presence of ATP by gamma32P-ATP based analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 51nMAssay Description:Binding affinity to NanoLuc-fused CLK1 (unknown origin) transfected in HEK293T cells assessed as target engagement by measuring inhibition constant i...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 250nMAssay Description:Binding affinity to NanoLuc-fused CLK1 (unknown origin) transfected in HEK293T cells assessed as target engagement incubated for 3 hrs by tracer K5 b...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of NanoLuc-fused CLK1 (unknown origin) transfected in HEK293T cells incubated for 3 hrs in presence of ATP by tracer K5 based NanoBRET ass...More data for this Ligand-Target Pair
Ligand InfoSimilars
