Report error Found 3 Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum chaperone BiP' and Ligand = 'BDBM50617261'
TargetEndoplasmic reticulum chaperone BiP(Human)
The First Affiliated Hospital of Henan University
Curated by ChEMBL
The First Affiliated Hospital of Henan University
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to GRP78 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum chaperone BiP(Human)
The First Affiliated Hospital of Henan University
Curated by ChEMBL
The First Affiliated Hospital of Henan University
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of His-tagged human recombinant GRP78 expressed in Escherichia coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum chaperone BiP(Human)
The First Affiliated Hospital of Henan University
Curated by ChEMBL
The First Affiliated Hospital of Henan University
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
