Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 1' and Ligand = 'BDBM27775'
TargetHistone deacetylase 1(Human)
Merck Research Laboratories

LigandChemical structure of BindingDB Monomer ID 27775BDBM27775(N-[2-amino-5-(thiophen-3-yl)phenyl]-4-{1,8-diazasp...)
Affinity DataIC50: 8nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2009
Entry Details Article
PubMed