Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2 [2-746,Y641N]' and Ligand = 'BDBM435642'
LigandPNGBDBM435642(US10570121, Example 150 | US10570121, Example 151 ...)
Affinity DataIC50: 3nMAssay Description:A. Compound preparation1. Prepare 10 mM stock solutions in 100% DMSO from solid material2. Serial dilute 10 mM compound stocks either 2 or 3-fold in ...More data for this Ligand-Target Pair
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Date in BDB:
11/30/2020
Entry Details
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LigandPNGBDBM435642(US10570121, Example 150 | US10570121, Example 151 ...)
Affinity DataIC50: 9nMAssay Description:A. Compound preparation1. Prepare 10 mM stock solutions in 100% DMSO from solid material2. Serial dilute 10 mM compound stocks either 2 or 3-fold in ...More data for this Ligand-Target Pair
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Date in BDB:
11/30/2020
Entry Details
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LigandPNGBDBM435642(US10570121, Example 150 | US10570121, Example 151 ...)
Affinity DataIC50: 439nMAssay Description:A. Compound preparation1. Prepare 10 mM stock solutions in 100% DMSO from solid material2. Serial dilute 10 mM compound stocks either 2 or 3-fold in ...More data for this Ligand-Target Pair
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Date in BDB:
11/30/2020
Entry Details
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LigandPNGBDBM435642(US10570121, Example 150 | US10570121, Example 151 ...)
Affinity DataIC50: 2.27E+3nMAssay Description:A. Compound preparation1. Prepare 10 mM stock solutions in 100% DMSO from solid material2. Serial dilute 10 mM compound stocks either 2 or 3-fold in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2020
Entry Details
Go to US Patent