Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Ileal sodium/bile acid cotransporter' and Ligand = 'BDBM50140282'
TargetIleal sodium/bile acid cotransporter(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50140282(CHEMBL363392 | CHEMBL17879 | 1-{4-[4-((4R,5R)-3,3-...)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of human IBATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50140282(CHEMBL363392 | CHEMBL17879 | 1-{4-[4-((4R,5R)-3,3-...)
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibition of ASBT mediated uptake of [14C]taurocholate (5 uM) in baby hamster cells expressing human IBATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetIleal sodium/bile acid cotransporter(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50140282(CHEMBL363392 | CHEMBL17879 | 1-{4-[4-((4R,5R)-3,3-...)
Affinity DataIC50: 890nMAssay Description:In vitro Inhibition of apical sodium-dependent bile acid transporter by measuring the uptake of [3H]taurocholate in hamster ileal ringMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed