Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Lactoylglutathione lyase' and Ligand = 'BDBM54705'
TargetLactoylglutathione lyase(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM54705(calcium;2-(3-phenoxyphenyl)propanoic acid;hydrate ...)
Affinity DataKi:  3.83E+5nMAssay Description:Inhibition of human recombinant His-tagged glyoxalase 1 expressed in Escherichia coli BL21 (DE3) preincubated for 20 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM54705(calcium;2-(3-phenoxyphenyl)propanoic acid;hydrate ...)
Affinity DataKi:  3.83E+5nMAssay Description:Inhibition of human glyoxalase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM54705(calcium;2-(3-phenoxyphenyl)propanoic acid;hydrate ...)
Affinity DataKi:  4.00E+5nMAssay Description:Inhibition of glyoxalase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed