Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM8864'
TargetMast/stem cell growth factor receptor Kit(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 8864BDBM8864(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-3-methox...)
Affinity DataIC50: 180nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2006
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 8864BDBM8864(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-3-methox...)
Affinity DataIC50: 180nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Abbott Laboratories

LigandChemical structure of BindingDB Monomer ID 8864BDBM8864(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-3-methox...)
Affinity DataIC50: 182nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed