Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM206343'
TargetMitogen-activated protein kinase 1(Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 206343BDBM206343(US9259470, 167)
Affinity DataIC50: 3.10nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 206343BDBM206343(US9259470, 167)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Array Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 206343BDBM206343(US9259470, 167)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed