Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50000655'
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataIC50: 460nMAssay Description:Inhibitory concentration of compound against mu opioid receptor in guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  52nMAssay Description:Binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  52nMAssay Description:Binding affinity against mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  107nMAssay Description:Binding affinity against opioid receptor mu in guinea pig brain homogenates, using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50000655(CHEMBL39192 | 10-[2-Amino-3-(4-hydroxy-phenyl)-pro...)
Affinity DataKi:  107nMAssay Description:Compound was tested for the inhibition of [3H]- [D-Ala2, N-MePhe4, Gly5-ol]-enkephalin (DAMGO) binding to Opioid receptor mu 1 in guinea pig brain ho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed