Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50061567'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50061567(DMPP | cid_5911 | CHEMBL134752 | CHEMBL47814 | 1,1...)
Affinity DataEC50:  2.50E+3nMAssay Description:Compound was evaluated for functional potencies and efficacies at human Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Georgetown University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50061567(DMPP | cid_5911 | CHEMBL134752 | CHEMBL47814 | 1,1...)
Affinity DataKi:  90nMAssay Description:Binding affinity towards rat Nicotinic acetylcholine receptor alpha4-beta2 expressed in HEK293 cells using [3H]EB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Georgetown University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50061567(DMPP | cid_5911 | CHEMBL134752 | CHEMBL47814 | 1,1...)
Affinity DataKi:  250nMAssay Description:Binding affinity towards nicotinic receptor in rat brain using [3H]cytisine ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2014
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Georgetown University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50061567(DMPP | cid_5911 | CHEMBL134752 | CHEMBL47814 | 1,1...)
Affinity DataKi:  250nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Georgetown University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50061567(DMPP | cid_5911 | CHEMBL134752 | CHEMBL47814 | 1,1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed