Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50324039'
TargetPeroxisome proliferator-activated receptor gamma(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324039BDBM50324039(4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biph...)
Affinity DataEC50:  1.90E+3nMAssay Description:Activation of Gal4-tagged human PPARgamma expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324039BDBM50324039(4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biph...)
Affinity DataEC50:  4.17E+3nMAssay Description:Transactivation at Gal4 fused PPARgamma LBD (unknown origin) expressed in African green monkey COS7 cells after 42 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324039BDBM50324039(4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biph...)
Affinity DataEC50:  6.44E+3nMAssay Description:Transactivation of Gal4 fused human PPARgamma LBD expressed in African green monkey COS7 cells after 42 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324039BDBM50324039(4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biph...)
Affinity DataEC50:  7.22E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed