Report error Found 5 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50490819'
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at GST-tagged PPAR-gamma ligand binding domain (unknown origin) assessed as recruitment of fluorescein-labeled SRC1 coactiva...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at GST-tagged PPAR-gamma ligand binding domain (unknown origin) assessed as recruitment of fluorescein-labeled SRC3 coactiva...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataEC50: 1.73E+4nMAssay Description:Partial agonist activity at GST-tagged PPAR-gamma ligand binding domain (unknown origin) assessed as recruitment of fluorescein-labeled PRIP/RAP250 c...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataEC50: 2.58E+4nMAssay Description:Partial agonist activity at PPARgamma in human BMMSC cells assessed as promotion of adiponectin secretion by measuring increase in adiponectin level ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataKi: 1.07E+4nMAssay Description:Displacement of fluormone pan-PPARgreen from GST-tagged human PPARgamma ligand binding domain by LanthaScreen TR-FRET competitive binding assayMore data for this Ligand-Target Pair
