Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50062429'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50062429(5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...)
Affinity DataKi:  0.490nMAssay Description:The binding affinity measured using baculovirus-expressed hPR-A in sf21 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50062429(5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity for human progesterone receptor isoform A expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50062429(5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...)
Affinity DataEC50:  2.70nMAssay Description:Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50062429(5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...)
Affinity DataEC50:  2.70nMAssay Description:Agonistic activity was measured for modulation of hPR-B (human progesterone receptor) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed