Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM238373'
LigandChemical structure of BindingDB Monomer ID 238373BDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 640nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238373BDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Assays were realized on 96-well plates, as described for yeast FTase but octyl-D-glucopyranoside (0.18%) was used instead of CHAPS and the solution c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed